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吖庚因类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-(2,4-difluorophenyl)-3-pyridin-3-yl-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C18H16F2N4
1-(2,4-difluorophenyl)-3-pyridin-3-yl-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 3-(3-bromophenyl)-1-(3-chloro-2-methylphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C20H19BrClN3
3-(3-bromophenyl)-1-(3-chloro-2-methylphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 1-(4-chlorophenyl)-3-(1-ethylpiperidin-3-yl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C20H27ClN4
1-(4-chlorophenyl)-3-(1-ethylpiperidin-3-yl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 3-[(2-fluorophenyl)methyl]-1-(2-methylphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C21H22FN3
3-[(2-fluorophenyl)methyl]-1-(2-methylphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 1-(4-chlorophenyl)-3-pentan-3-yl-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C18H24ClN3
1-(4-chlorophenyl)-3-pentan-3-yl-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 1-(3-methylphenyl)-3-propyl-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C17H23N3
1-(3-methylphenyl)-3-propyl-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 3-(4-methylthiophen-2-yl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine-1-carbothioamide —— C13H16N4S2
3-(4-methylthiophen-2-yl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine-1-carbothioamide
—— 3-(3-bromophenyl)-4,5,6,7-tetrahydro-2H-[1,2]oxazolo[5,4-b]azepine —— C13H13BrN2O
3-(3-bromophenyl)-4,5,6,7-tetrahydro-2H-[1,2]oxazolo[5,4-b]azepine
—— 3-pyridin-2-yl-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine-1-carboxamide —— C13H15N5O
3-pyridin-2-yl-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine-1-carboxamide
—— N-(3-oxo-2,5,6,7,8,9-hexahydro-3H-[1,2,4]triazolo[4,3-a]azepin-7-yl)-3-(1,3,5-trimethyl-1H-pyrazol-4-yl)propanamide —— C16H24N6O2
N-(3-oxo-2,5,6,7,8,9-hexahydro-3H-[1,2,4]triazolo[4,3-a]azepin-7-yl)-3-(1,3,5-trimethyl-1H-pyrazol-4-yl)propanamide
—— 3-(2-chloro-4-fluorophenyl)-1-(4-chlorophenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C19H16Cl2FN3
3-(2-chloro-4-fluorophenyl)-1-(4-chlorophenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 3-(methylsulfanylmethyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine-1-carbothioamide —— C10H16N4S2
3-(methylsulfanylmethyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine-1-carbothioamide
—— 2-[(3-Bromophenyl)methyl]-4-(5-methyl-1,2,4-oxadiazol-3-YL)-1H,2H,3H,5H,6H,7H,8H,9H-pyrimido[1,6-A]azepine-1,3-dione —— C19H19BrN4O3
2-[(3-Bromophenyl)methyl]-4-(5-methyl-1,2,4-oxadiazol-3-YL)-1H,2H,3H,5H,6H,7H,8H,9H-pyrimido[1,6-A]azepine-1,3-dione
—— 1-(3-bromophenyl)-3-(4-bromophenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C19H17Br2N3
1-(3-bromophenyl)-3-(4-bromophenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 3-cyclopentyl-1-(2-fluorophenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C18H22FN3
3-cyclopentyl-1-(2-fluorophenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— N-benzyl-2-[4-(5-ethyl-1,2,4-oxadiazol-3-yl)-1,3-dioxo-3,5,6,7,8,9-hexahydropyrimido[1,6-a]azepin-2(1H)-yl]acetamide —— C22H25N5O4
N-benzyl-2-[4-(5-ethyl-1,2,4-oxadiazol-3-yl)-1,3-dioxo-3,5,6,7,8,9-hexahydropyrimido[1,6-a]azepin-2(1H)-yl]acetamide
—— 3-tert-butyl-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine-1-carboximidamide —— C12H21N5
3-tert-butyl-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine-1-carboximidamide
—— 6-[(tetrahydro-2H-pyran-2-ylmethoxy)acetyl]-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepin-3(2H)-one —— C15H23N3O4
6-[(tetrahydro-2H-pyran-2-ylmethoxy)acetyl]-1,4,5,6,7,8-hexahydropyrazolo[3,4-d]azepin-3(2H)-one
—— 3-(5-bromopyridin-3-yl)-1-(2-methylphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C19H19BrN4
3-(5-bromopyridin-3-yl)-1-(2-methylphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 3-cyclobutyl-1-(4-fluorophenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C17H20FN3
3-cyclobutyl-1-(4-fluorophenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 3-(5-chlorothiophen-2-yl)-4,5,6,7-tetrahydro-2H-[1,2]oxazolo[5,4-b]azepine —— C11H11ClN2OS
3-(5-chlorothiophen-2-yl)-4,5,6,7-tetrahydro-2H-[1,2]oxazolo[5,4-b]azepine
—— 1-(2,4-difluorophenyl)-3-(2-ethoxyethyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C17H21F2N3O
1-(2,4-difluorophenyl)-3-(2-ethoxyethyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 1-(4-ethylphenyl)-3-pyridin-4-yl-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C20H22N4
1-(4-ethylphenyl)-3-pyridin-4-yl-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 3-(4-fluorophenyl)-4,5,6,7-tetrahydro-2H-[1,2]oxazolo[5,4-b]azepine —— C13H13FN2O
3-(4-fluorophenyl)-4,5,6,7-tetrahydro-2H-[1,2]oxazolo[5,4-b]azepine
—— 2-(3,5-difluorobenzyl)-4-(5-ethyl-1,2,4-oxadiazol-3-yl)-6,7,8,9-tetrahydropyrimido[1,6-a]azepine-1,3(2H,5H)-dione —— C20H20F2N4O3
2-(3,5-difluorobenzyl)-4-(5-ethyl-1,2,4-oxadiazol-3-yl)-6,7,8,9-tetrahydropyrimido[1,6-a]azepine-1,3(2H,5H)-dione
—— 2-(3-chlorobenzyl)-4-(5-methyl-1,2,4-oxadiazol-3-yl)-6,7,8,9-tetrahydropyrimido[1,6-a]azepine-1,3(2H,5H)-dione —— C19H19ClN4O3
2-(3-chlorobenzyl)-4-(5-methyl-1,2,4-oxadiazol-3-yl)-6,7,8,9-tetrahydropyrimido[1,6-a]azepine-1,3(2H,5H)-dione
—— 2-[4-(5-ethyl-1,2,4-oxadiazol-3-yl)-1,3-dioxo-3,5,6,7,8,9-hexahydropyrimido[1,6-a]azepin-2(1H)-yl]-N-(2-thienylmethyl)acetamide —— C20H23N5O4S
2-[4-(5-ethyl-1,2,4-oxadiazol-3-yl)-1,3-dioxo-3,5,6,7,8,9-hexahydropyrimido[1,6-a]azepin-2(1H)-yl]-N-(2-thienylmethyl)acetamide
—— N-(4-chlorobenzyl)-2-[4-(5-methyl-1,2,4-oxadiazol-3-yl)-1,3-dioxo-3,5,6,7,8,9-hexahydropyrimido[1,6-a]azepin-2(1H)-yl]acetamide —— C21H22ClN5O4
N-(4-chlorobenzyl)-2-[4-(5-methyl-1,2,4-oxadiazol-3-yl)-1,3-dioxo-3,5,6,7,8,9-hexahydropyrimido[1,6-a]azepin-2(1H)-yl]acetamide
—— N-(4-fluorobenzyl)-2-[4-(5-methyl-1,2,4-oxadiazol-3-yl)-1,3-dioxo-3,5,6,7,8,9-hexahydropyrimido[1,6-a]azepin-2(1H)-yl]acetamide —— C21H22FN5O4
N-(4-fluorobenzyl)-2-[4-(5-methyl-1,2,4-oxadiazol-3-yl)-1,3-dioxo-3,5,6,7,8,9-hexahydropyrimido[1,6-a]azepin-2(1H)-yl]acetamide
—— 4-(5-ethyl-1,2,4-oxadiazol-3-yl)-2-(2-fluorobenzyl)-6,7,8,9-tetrahydropyrimido[1,6-a]azepine-1,3(2H,5H)-dione —— C20H21FN4O3
4-(5-ethyl-1,2,4-oxadiazol-3-yl)-2-(2-fluorobenzyl)-6,7,8,9-tetrahydropyrimido[1,6-a]azepine-1,3(2H,5H)-dione
—— N-cyclopentyl-2-[4-(5-ethyl-1,2,4-oxadiazol-3-yl)-1,3-dioxo-3,5,6,7,8,9-hexahydropyrimido[1,6-a]azepin-2(1H)-yl]acetamide —— C20H27N5O4
N-cyclopentyl-2-[4-(5-ethyl-1,2,4-oxadiazol-3-yl)-1,3-dioxo-3,5,6,7,8,9-hexahydropyrimido[1,6-a]azepin-2(1H)-yl]acetamide
—— 2-(2-chlorobenzyl)-4-(5-methyl-1,2,4-oxadiazol-3-yl)-6,7,8,9-tetrahydropyrimido[1,6-a]azepine-1,3(2H,5H)-dione —— C19H19ClN4O3
2-(2-chlorobenzyl)-4-(5-methyl-1,2,4-oxadiazol-3-yl)-6,7,8,9-tetrahydropyrimido[1,6-a]azepine-1,3(2H,5H)-dione
—— 2-(4-methylbenzyl)-4-(5-methyl-1,2,4-oxadiazol-3-yl)-6,7,8,9-tetrahydropyrimido[1,6-a]azepine-1,3(2H,5H)-dione —— C20H22N4O3
2-(4-methylbenzyl)-4-(5-methyl-1,2,4-oxadiazol-3-yl)-6,7,8,9-tetrahydropyrimido[1,6-a]azepine-1,3(2H,5H)-dione
—— 2-(3,4-difluorobenzyl)-4-(5-ethyl-1,2,4-oxadiazol-3-yl)-6,7,8,9-tetrahydropyrimido[1,6-a]azepine-1,3(2H,5H)-dione —— C20H20F2N4O3
2-(3,4-difluorobenzyl)-4-(5-ethyl-1,2,4-oxadiazol-3-yl)-6,7,8,9-tetrahydropyrimido[1,6-a]azepine-1,3(2H,5H)-dione
—— 2-benzyl-4-(5-ethyl-1,2,4-oxadiazol-3-yl)-6,7,8,9-tetrahydropyrimido[1,6-a]azepine-1,3(2H,5H)-dione —— C20H22N4O3
2-benzyl-4-(5-ethyl-1,2,4-oxadiazol-3-yl)-6,7,8,9-tetrahydropyrimido[1,6-a]azepine-1,3(2H,5H)-dione
—— 1-(2,4-difluorophenyl)-3-ethyl-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C15H17F2N3
1-(2,4-difluorophenyl)-3-ethyl-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 1-(3-chloro-2-methylphenyl)-3-(2-piperidin-1-ylethyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C21H29ClN4
1-(3-chloro-2-methylphenyl)-3-(2-piperidin-1-ylethyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 1-(4-chlorophenyl)-3-(2-methylphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C20H20ClN3
1-(4-chlorophenyl)-3-(2-methylphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 3-(3-fluorophenyl)-1-(2-methylphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C20H20FN3
3-(3-fluorophenyl)-1-(2-methylphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 1-(2-bromophenyl)-3-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C19H16BrF2N3
1-(2-bromophenyl)-3-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 1-(2,4-difluorophenyl)-3-(2-fluorophenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C19H16F3N3
1-(2,4-difluorophenyl)-3-(2-fluorophenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 3-benzyl-1-(3-methylphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C21H23N3
3-benzyl-1-(3-methylphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 3-[(2-chlorophenyl)methyl]-1-(2-ethylphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C22H24ClN3
3-[(2-chlorophenyl)methyl]-1-(2-ethylphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 3-(5-chlorothiophen-2-yl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine-1-carboxamide —— C12H13ClN4OS
3-(5-chlorothiophen-2-yl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine-1-carboxamide
—— 3-(4-chlorophenyl)-1-(4-ethylphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C21H22ClN3
3-(4-chlorophenyl)-1-(4-ethylphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 3-(2-fluorophenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine-1-carbothioamide —— C14H15FN4S
3-(2-fluorophenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine-1-carbothioamide
—— 3-(2-bromophenyl)-1-(5-chloro-2-methylphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C20H19BrClN3
3-(2-bromophenyl)-1-(5-chloro-2-methylphenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 1-(4-bromophenyl)-3-(5-bromopyridin-3-yl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C18H16Br2N4
1-(4-bromophenyl)-3-(5-bromopyridin-3-yl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 3-(2-bromophenyl)-1-(2-chlorophenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine —— C19H17BrClN3
3-(2-bromophenyl)-1-(2-chlorophenyl)-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine
—— 3-pyridin-2-yl-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine-1-carboximidamide —— C13H16N6
3-pyridin-2-yl-4,5,6,7-tetrahydro-2H-pyrazolo[3,4-b]azepine-1-carboximidamide