| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | 15-(4-Methylpiperazin-1-yl)-17-oxa-1,5,7,9,11,22-hexazapentacyclo[20.2.2.13,6.112,16.010,28]octacosa-3,6(28),7,9,12(27),13,15-heptaen-21-one | 1111233-57-8 | C26H34N8O2 |
| —— | 4-(9-benzyl-2-morpholin-4-ylpurin-6-yl)-1H-pyridin-2-one | 1138157-95-5 | C21H20N6O2 |
| —— | (5Z)-N-(5-{[2-(benzotriazol-5-ylazamethylene)-4-oxo-1,3-thiazolidin-5-ylidene]methyl}-1,3-thiazol-2-yl)acetamide | 1253116-25-4 | C15H11N7O2S2 |
| —— | 4-[(3,5-dimethylpyrrol-2-yl)methylene]-3-(2-thienyl)-2-pyrazolin-5-one | 324549-00-0 | C14H13N3OS |
| —— | (E)-(+/-)-6-(3-chloroindol-7-yl)-5,7-difluoro-2,3-dihydro-3-hydroxy-2,2-dimethyl-1H-quinolin-4-one O-ethyl oxime | 1181821-18-0 | C21H20ClF2N3O2 |
| —— | 4-cyclopropyl-N-{2-hydroxymethyl-3-[1-methyl-5-(1-methyl-1H-pyrazol-3-ylamino)-6-oxo-1,6-dihydro-pyridazin-3-yl]-phenyl}-benzamide | 1147529-70-1 | C26H26N6O3 |
| —— | 3-[5-Chloro-6-[4-[5-[3-[[methyl-[2-[(2-methylpropan-2-yl)oxycarbonylamino]acetyl]amino]methyl]phenyl]pyrimidin-2-yl]piperazin-1-yl]pyridin-3-yl]prop-2-enoic acid | 1279031-68-3 | C31H36ClN7O5 |
| —— | 3-[(2-{[2-(methyloxy)-4-(1-propyl-1,2,5,6-tetrahydro-3-pyridinyl)phenyl]amino}-1H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-2-naphthalenecarboxamide | 1116234-13-9 | C32H33N7O2 |
| —— | 2-hydroxy-7,7-dimethyl-6,7,8,9-tetrahydro-4H-pyrimido[1,2-a]pyrimidin-4-one | 1383777-82-9 | C9H13N3O2 |
| —— | 2-fluoro-6-[(2-{[6-(methyloxy)-1,2,3,4-tetrahydro-7-quinolinyl]amino}-1H-pyrrolo[2,3-d]pyrimidin-4-yl)amino]benzamide | 1116238-73-3 | C23H22FN7O2 |
| —— | 6-formyl-1,3,5-trimethyl-2,4-dioxo-2,3,4,5-tetrahydro-1<i>H</i>-pyrrolo[3,2-<i>d</i>]pyrimidine-7-carboxylic acid methyl ester | 71411-53-5 | C12H13N3O5 |
| —— | (+/-)-4-benzyl-N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-N-isobutyl-2-methylmorpholine-2-carboxamide | 941709-40-6 | C27H36N2O4 |
| —— | 2-amino-2-(3-(2-benzylpiperidin-1-yl)propyl)-6-boronohexanoic acid | 1384297-22-6 | C21H35BN2O4 |
| —— | N-(5-benzo[1,3]dioxol-5-ylmethyl-4-methylthiazol-2-yl)-3-pyridin-3-ylpropionamide | 1384184-01-3 | C20H19N3O3S |
| —— | (R)-5-(2-(2,5-difluorophenyl)pyrrolidin-1-yl)-N-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide | 1260840-28-5 | C18H17F2N5O |
| —— | 7-methoxy-8-{4-[(5-(5-(4-trifluoromethylphenyl)-1,3,4-oxadiazol-2-yl)-2-methoxyphenyl)oxy]butyloxy}-(11aS)-1,2,3,11a-tetrahydro-5H-pyrrolo[2,1-c][1,4]benzodiazepin-5-one | 1251485-26-3 | C33H31F3N4O6 |
| —— | 3-heptyl-6-methyl-3,4-dihydroquinazolin-2(1H)-one | 1244766-22-0 | C16H24N2O |
| —— | N-(3-(2-ethoxyphenyl)-1-(2-hydroxy-2-methylpropyl)-1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide | 1260166-04-8 | C22H24N6O3 |
| —— | 1-(4-chlorophenyl)-N-(3-(4-(2,3-dichlorophenyl)piperazin-1-yl)propyl)-2-ethyl-5-methyl-1H-imidazole-4-carboxamide | 1261175-44-3 | C26H30Cl3N5O |
| —— | 1-(4-Indolyl)-4-[1-[(2S)-5-oxopyrrolidine-2-ylcarbonyl]-1,2,3,4-tetrahydroquinoline-2-ylmethyl]piperazine | 511232-95-4 | C27H31N5O2 |
| —— | 7-[(4-phenyl-1-piperidinyl)carbonyl]-3-[6-(trifluoromethyl)-3-pyridinyl]-2-quinoxalinepentanoic acid | 1383694-57-2 | C31H29F3N4O3 |
| —— | 1-[2-(1,3-benzodioxol-5-yl)ethyl]-3-[3-[[5-cyano-4-(3-methoxyphenyl)-6-oxo-1H-pyrimidin-2-yl]sulfanylmethyl]phenyl]urea | 879870-75-4 | C29H25N5O5S |
| —— | N-hydroxy-2-[(2-methoxyphenoxy)methyl]-4-oxo-3,4-dihydroquinazoline-7-carboxamide | 1372888-41-9 | C17H15N3O5 |
| —— | 4-{3-[(5-hydroxypyridin-2-yl)-1,2,4-oxadiazol-5-yl]propanoyl}amino-1-(3,5-difluorobenzyl)pyrrole-3-carboxylic acid | 1204422-25-2 | C22H17F2N5O5 |
| —— | 4-{3-[2-(5-hydroxypyridin-2-yl)oxazol-5-yl]propanoyl}amino-1-butylpyrrole-3-carboxylic acid | 1204422-21-8 | C20H22N4O5 |
| —— | 2-((R)-1-(4-(dimethylamino)phenyl)ethylamino)-4-(5-(trifluoromethyl)-1H-pyrrolo[2,3-b]pyridin-3-yl)pyrimidine-5-carbonitrile | 1036025-32-7 | C23H20F3N7 |
| —— | 3-{2-[5-chloro-2-(4-trifluoromethyl-benzyloxy)-phenyl]-5-methyl-pyrrol-1-yl}-6-methyl-benzoic acid | 854192-86-2 | C27H21ClF3NO3 |
| —— | Ethyl 3-(3-bromo-7-chloro-5-methylpyrazolo[1,5-a]pyrimidin-6-yl)propanoate | 934297-16-2 | C12H13BrClN3O2 |
| —— | 4-[1-cyclopentyl-7-(trifluromethyl)-1H-indazol-3-yl]benzene-1,3-diol | 680611-89-6 | C19H17F3N2O2 |
| —— | 2-chloro-5-ethyl-4,6-dimethylpyrimidine | 73492-47-4 | C8H11ClN2 |
| —— | 3-(1,3-Dioxan-2-yl)-1-(2-pyridyl)-1-propene | 145912-81-8 | C12H15NO2 |
| —— | 4-amino-3-(6-methyl-5-morpholin-4-yl-1H-benzimidazol-2-yl) quinolin-2(1H)-one | 405168-67-4 | C21H21N5O2 |
| —— | 9-[(5-methyl-2-furanyl)methyl]-N-(4-piperidinyl)-9H-purin-8-amine | 116062-63-6 | C16H20N6O |
| —— | 2-ethyl-4-{3-[2-(ethyl-methyl-amino)-6-methyl-pyridin-4-yl]-[1,2,4]oxadiazol-5-yl}-6-methyl-phenol | 1062670-56-7 | C20H24N4O2 |
| —— | methyl 3-[3-(4-{[5-cyclopropyl-3-(2,6-dichlorophenyl)-1,2-oxazol-4-yl]methoxy}piperidin-1-yl)-1,2,4-oxadiazol-5-yl]benzoate | 1383743-74-5 | C28H26Cl2N4O5 |
| —— | 9-bromo-2-methyl-6H-1,3,3a,6-tetraaza-benzo[e]azulen-5-one | 882517-74-0 | C11H9BrN4O |
| —— | 2-{(5-Methoxy-4-oxospiro[1,2,3,4-tetrahydroquinoline-2,1'-cyclohexan]-7-yl)oxy}acetic acid | 135111-85-2 | C17H21NO5 |
| —— | 3-{8-[(butylamino)methyl]-1,1-dioxido-4H-[1,3]oxazolo[5,4-h][1,2,4]benzothiadiazin-3-yl}-4-hydroxy-1-(isobutylamino)quinolin-2(1H)-one | 691361-01-0 | C26H30N6O5S |
| —— | ethyl 5-[({4-[4-(2-aminopyrimidin-5-yl)phenyl]tetrahydro-2H-pyran-4-yl}carbonyl)amino]-3-methyl-1-benzothiophene-2-carboxylate | 1382482-80-5 | C28H28N4O4S |
| —— | 3-(1,1-dioxido-4H-1,2,4-benzothiadiazin-3-yl)-4-hydroxy-1-[(4-isopropylcyclohexyl)amino]quinolin-2(1H)-one | 686269-35-2 | C25H28N4O4S |
| —— | 6,10a-Diaza-cyclopenta[a]phenalen-7-one oxime | 55852-29-4 | C14H9N3O |
| —— | 5-(2-(4-fluorophenyl)-6-(3-phenylazetidine-1-carbonyl)quinolin-3-yl)pentanoic acid | 1383848-91-6 | C30H27FN2O3 |
| —— | 5-amino-3-(4-chloro-3-methylphenyl)-4-(4-pyridyl)isoxazole | 1000187-82-5 | C15H12ClN3O |
| —— | 4-cyclopropyl-5-methyl-4H-1,2,4-triazole-3-thiol | 854137-73-8 | C6H9N3S |
| —— | 5-phenylsulphonyl-4-piperidino-2H-benzimidazole-2-spirocyclohexane | 94526-22-4 | C23H27N3O2S |
| —— | ethyl 5-amino-2-[(2E)-2-[(4-nitrophenyl)methylidene]hydrazinyl]-4-phenylthieno[2,3-d]pyrimidine-6-carboxylate | 135300-50-4 | C22H18N6O4S |
| —— | 7-acetonyl-5-(methylsulfonyl)-6,7-dihydro-3-phenyl-3H-1,2,3-triazolo<4,5-d>pyrimidine | 124799-22-0 | C14H15N5O3S |
| —— | 6-chloro-5-methanesulfonylindole | 1268816-56-3 | C9H8ClNO2S |
| —— | 2-(5,6-dimethoxypyridin-3-yl)-6-[6-[1,3-dioxolan-2-ylmethyl(methyl)amino]pyridin-3-yl]-7H-pyrrolo[3,4-b]pyridin-5-one | 1315536-36-7 | C24H25N5O5 |
| —— | US8653087, III-387 | 1213246-74-2 | C25H28FN9O2 |