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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-methoxyethyl (Z)-2-cyano-3-isopropyl-3-{[(5-methylthio-1,3,4-thiadiazol-2-yl)methyl]amino}acrylate 1322098-35-0 C14H20N4O3S2
2-methoxyethyl (Z)-2-cyano-3-isopropyl-3-{[(5-methylthio-1,3,4-thiadiazol-2-yl)methyl]amino}acrylate
—— 1,2,4,5-tetrakis(3,5-ditertbutylpyrazol-1-ylmethyl)benzene 172606-29-0 C30H38N8
1,2,4,5-tetrakis(3,5-ditertbutylpyrazol-1-ylmethyl)benzene
—— 6-methoxyquinoxalin-2-yl 4-methylbenzenesulfonate 1315336-89-0 C16H14N2O4S
6-methoxyquinoxalin-2-yl 4-methylbenzenesulfonate
—— N3,N3,N5,N5-tetraethyl-[1,2,4,3,5]dithiazadiborolo[3,4-c][1,2,4,3,5]dithiazadiborole-3,5-diamine 124665-21-0 C8H20B3N3S4
N3,N3,N5,N5-tetraethyl-[1,2,4,3,5]dithiazadiborolo[3,4-c][1,2,4,3,5]dithiazadiborole-3,5-diamine
—— —— 1245576-26-4 C28H30F3FeN3O3S2
—— (CH(C(CF3)N(C6H3(CH3)2))2)2Cu2(μ-oxo-(18)O)2 1149343-44-1 C42H38Cu2F12N4O2
(CH(C(CF3)N(C6H3(CH3)2))2)2Cu2(μ-oxo-(18)O)2
—— methyl 3-picolinoylbenzoate 1374650-42-6 C14H11NO3
methyl 3-picolinoylbenzoate
—— isopropyl 5'-isopropoxy-4,6-dimethyl-2-oxo-2H,3'H-spiro[benzofuran-3,2'-[1,3,4]oxadiazole]-3'-carboxylate 1453085-70-5 C18H22N2O6
isopropyl 5'-isopropoxy-4,6-dimethyl-2-oxo-2H,3'H-spiro[benzofuran-3,2'-[1,3,4]oxadiazole]-3'-carboxylate
—— (3S,1'R)-N-(1'-phenylethyl)-2-(1-methyl-3-ethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamide 1203474-47-8 C21H24N2O2
(3S,1'R)-N-(1'-phenylethyl)-2-(1-methyl-3-ethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamide
—— [(3S,7R,8R)-8-butyl-3-[(3-formamido-2-methoxybenzoyl)amino]-4,9-dioxo-1,5-dioxonan-7-yl] 3-methylbutanoate 1058162-25-6 C25H34N2O9
[(3S,7R,8R)-8-butyl-3-[(3-formamido-2-methoxybenzoyl)amino]-4,9-dioxo-1,5-dioxonan-7-yl] 3-methylbutanoate
—— 1,1-di-tert-butyl-2,5-bis[(2,2'-bithiophen)-5-yl]-3,4-diphenylsilole 1089758-36-0 C40H38S4Si
1,1-di-tert-butyl-2,5-bis[(2,2'-bithiophen)-5-yl]-3,4-diphenylsilole
—— 4-C-methyl-D-glucono-1,4-lactone 1202752-41-7 C7H12O6
4-C-methyl-D-glucono-1,4-lactone
—— (-)-(3,5-dimethyl-1H-pyrazol-1-yl)(6-methoxy-3,3-dimethylbicyclo[4.2.0]octa-4,7-dien-7-yl)methanone 1033604-13-5 C17H22N2O2
(-)-(3,5-dimethyl-1H-pyrazol-1-yl)(6-methoxy-3,3-dimethylbicyclo[4.2.0]octa-4,7-dien-7-yl)methanone
—— methyl (3aR,4R,6S,7aS)-3-(2-acetyloxyacetyl)-6-[(2R,3S,4S,5R,6R)-5-benzoyloxy-2-(benzoyloxymethyl)-3-hydroxy-6-[[(2R,3R,4S,5R,6R)-6-methoxy-3,4,5-tris(phenylmethoxy)oxan-2-yl]methoxy]oxan-4-yl]oxy-2-oxo-4-[(1S,2R)-1,2,3-triacetyloxypropyl]-3a,4,7,7a-tetrahydropyrano[3,4-d][1,3]oxazole-6-carboxylate 1057491-43-6 C69H75NO27
methyl (3aR,4R,6S,7aS)-3-(2-acetyloxyacetyl)-6-[(2R,3S,4S,5R,6R)-5-benzoyloxy-2-(benzoyloxymethyl)-3-hydroxy-6-[[(2R,3R,4S,5R,6R)-6-methoxy-3,4,5-tris(phenylmethoxy)oxan-2-yl]methoxy]oxan-4-yl]oxy-2-oxo-4-[(1S,2R)-1,2,3-triacetyloxypropyl]-3a,4,7,7a-tetrahydropyrano[3,4-d][1,3]oxazole-6-carboxylate
—— 3-(2-hydroxyphenyl)-4-phenylanthracen-1-ol 1192115-53-9 C26H18O2
3-(2-hydroxyphenyl)-4-phenylanthracen-1-ol
—— N-(4'-methoxy-4,5-dimethyl-biphenyl-2-yl)-acetamide 1227513-43-0 C17H19NO2
N-(4'-methoxy-4,5-dimethyl-biphenyl-2-yl)-acetamide
—— 2',3'-bis-O-acetyl-5'-azido-5'-deoxy-N<sup>6</sup>-(N-phenylcarbamoyl)adenosine 1401415-38-0 C21H21N9O6
2',3'-bis-O-acetyl-5'-azido-5'-deoxy-N<sup>6</sup>-(N-phenylcarbamoyl)adenosine
—— (1R,2S,6R)-2-(pentyloxy)-3-tosyl-7-oxa-3-azabicyclo[4.1.0]heptane 1438279-82-3 C17H25NO4S
(1R,2S,6R)-2-(pentyloxy)-3-tosyl-7-oxa-3-azabicyclo[4.1.0]heptane
—— sec-butyl (4-chlorophenyl)carbamate 115382-09-7 C11H14ClNO2
sec-butyl (4-chlorophenyl)carbamate
—— {Ge(OH)(Hedta)}*H2O 126371-31-1 C10H14GeN2O9*H2O
{Ge(OH)(Hedta)}*H2O
—— dimethyl 3-(2,2-dimethylhydrazono)-2-oxo-3-phenylpropylphosphonate 1151733-58-2 C13H19N2O4P
dimethyl 3-(2,2-dimethylhydrazono)-2-oxo-3-phenylpropylphosphonate
—— N-[2-(1,1-dioxido-2,3-dihydro-1,4-benzothiazepin-4(5H)-yl)-6-methylquinolin-4-yl]-2-hydroxyacetamide 1422500-20-6 C21H21N3O4S
N-[2-(1,1-dioxido-2,3-dihydro-1,4-benzothiazepin-4(5H)-yl)-6-methylquinolin-4-yl]-2-hydroxyacetamide
—— (S)-3-{[1-(2-chloro-phenyl)-5-methyl-1H-[1,2,4]triazole-3-carbonyl]-amino}-3-o-tolyl-propionic acid 1420833-65-3 C20H19ClN4O3
(S)-3-{[1-(2-chloro-phenyl)-5-methyl-1H-[1,2,4]triazole-3-carbonyl]-amino}-3-o-tolyl-propionic acid
—— N-(4-((4-ethylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-4-methyl-3-((2-(methylamino)pyrimidin-4-yl)oxy)benzamide 1315330-08-5 C27H31F3N6O2
N-(4-((4-ethylpiperazin-1-yl)methyl)-3-(trifluoromethyl)phenyl)-4-methyl-3-((2-(methylamino)pyrimidin-4-yl)oxy)benzamide
—— (2S)-N-[4-cyano-3-(trifluoromethyl)phenyl]-13-(hexylthio)-2-hydroxy-2-methyltridecanamide 1019975-01-9 C28H43F3N2O2S
(2S)-N-[4-cyano-3-(trifluoromethyl)phenyl]-13-(hexylthio)-2-hydroxy-2-methyltridecanamide
—— example 111 : 7-fluoro-2-isopropyl-N-(2-pyridin-2-ylethyl)-10,11-dihydrodibenzo[b,f]thiepine-3-sulfonamide 5,5-dioxide 1027348-38-4 C24H25FN2O4S2
example 111 : 7-fluoro-2-isopropyl-N-(2-pyridin-2-ylethyl)-10,11-dihydrodibenzo[b,f]thiepine-3-sulfonamide 5,5-dioxide
—— (S)-3-{[5-(2-fluoro-phenyl)-[1,2,4]oxadiazole-3-carbonyl]-amino}-3-o-tolyl-propionic acid 1420833-12-0 C19H16FN3O4
(S)-3-{[5-(2-fluoro-phenyl)-[1,2,4]oxadiazole-3-carbonyl]-amino}-3-o-tolyl-propionic acid
—— ethyl 5-amino-3-(4-(methylamino)phenyl)-4-oxo-3,4-dihydrothieno[3,4-d]pyridazine-1-carboxylate 1282449-00-6 C16H16N4O3S
ethyl 5-amino-3-(4-(methylamino)phenyl)-4-oxo-3,4-dihydrothieno[3,4-d]pyridazine-1-carboxylate
—— N-(4-(dimethylamino)phenyl)-4-(5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl)benzamide 1418292-23-5 C18H15F3N4O2
N-(4-(dimethylamino)phenyl)-4-(5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl)benzamide
—— 5'-[2-(5-methoxy-2-methyl-phenylamino)-oxazol-5-yl]-[1,3']bipyridinyl-2-one 1420997-80-3 C21H18N4O3
5'-[2-(5-methoxy-2-methyl-phenylamino)-oxazol-5-yl]-[1,3']bipyridinyl-2-one
—— N-(adamantane-2-yl)-2-methyl-2-(4-chlorophenylsulfonamido)propanamide 1422024-34-7 C20H27ClN2O3S
N-(adamantane-2-yl)-2-methyl-2-(4-chlorophenylsulfonamido)propanamide
—— 3-(3,3-dimethyl-piperidin-4-yl)-5-fluoro-1H-indole 1005744-80-8 C15H19FN2
3-(3,3-dimethyl-piperidin-4-yl)-5-fluoro-1H-indole
—— N6-cyclohexyl-N2-{4-[4-({3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}sulfonyl)piperazin-1-yl]-2-methoxyphenyl}-9H-purine-2,6-diamine 1246531-17-8 C31H48N10O3S
N6-cyclohexyl-N2-{4-[4-({3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}sulfonyl)piperazin-1-yl]-2-methoxyphenyl}-9H-purine-2,6-diamine
—— (3S)-5-(2-pyrrolidin-1-ylethoxy)chroman-3-amine 1074763-84-0 C15H22N2O2
(3S)-5-(2-pyrrolidin-1-ylethoxy)chroman-3-amine
—— cyclopentyl-(5-{[(8,8-dimethoxy-octyl)-methyl-amino]-methyl}-oxazol-2-yl)-phenyl-methanol 1006063-65-5 C27H42N2O4
cyclopentyl-(5-{[(8,8-dimethoxy-octyl)-methyl-amino]-methyl}-oxazol-2-yl)-phenyl-methanol
—— (R)-3-aminocarbonylmethylene-N-[3-methoxy-4-(2-chloro-5-fluoro-phenylcarbonyl)amino-phenylcarbonyl]-spiro[cyclopentane-1,4'-benzo[b]azepane] 1092408-64-4 C31H29ClFN3O4
(R)-3-aminocarbonylmethylene-N-[3-methoxy-4-(2-chloro-5-fluoro-phenylcarbonyl)amino-phenylcarbonyl]-spiro[cyclopentane-1,4'-benzo[b]azepane]
—— 3-[4-(4-aminomethylpiperidin-1-yl)-6-((3R)-hydroxymethyl-3,4-dihydro-1H-isoquinolin-2-yl)-[1,3,5]triazin-2-yl]-phenol 1033594-97-6 C25H30N6O2
3-[4-(4-aminomethylpiperidin-1-yl)-6-((3R)-hydroxymethyl-3,4-dihydro-1H-isoquinolin-2-yl)-[1,3,5]triazin-2-yl]-phenol
—— 4-bromo-N-(1-isonicotinoylpiperidin-4-yl)-2-(trifluoromethyl)benzenesulfonamide 1027007-52-8 C18H17BrF3N3O3S
4-bromo-N-(1-isonicotinoylpiperidin-4-yl)-2-(trifluoromethyl)benzenesulfonamide
—— (S)-[4-(5-cyclopropyl-3-methylpyridin-2-yl)piperazin-1-yl][4-(3-hydroxymethyl-1,1-dioxo-1λ<sup>6</sup>-isothiazolidin-2-yl)phenyl]methanone 1346114-75-7 C24H30N4O4S
(S)-[4-(5-cyclopropyl-3-methylpyridin-2-yl)piperazin-1-yl][4-(3-hydroxymethyl-1,1-dioxo-1λ<sup>6</sup>-isothiazolidin-2-yl)phenyl]methanone
—— 2-(2-((3,5-dimethylisoxazol-4-yl)(2-methoxyethoxy)methyl)benzofuran-5-yl)-N-((2,4-dimethylphenyl)(phenyl)methyl)acetamide 1422168-51-1 C34H36N2O5
2-(2-((3,5-dimethylisoxazol-4-yl)(2-methoxyethoxy)methyl)benzofuran-5-yl)-N-((2,4-dimethylphenyl)(phenyl)methyl)acetamide
—— (5-bromopyrimidin-2-yl)[4-(3,5-dimethylpyridin-2-yl)piperazin-1-yl]methanone 1346124-31-9 C16H18BrN5O
(5-bromopyrimidin-2-yl)[4-(3,5-dimethylpyridin-2-yl)piperazin-1-yl]methanone
—— 5-[(3-{(Z)-2-[6-(2,6-dimethylmorpholin-4-yl)pyridin-3-yl]-1-fluorovinyl}-5-methyl-1H-pyrazol-1-yl)methyl]-N-methylpyridine-2-amine 1418296-56-6 C24H29FN6O
5-[(3-{(Z)-2-[6-(2,6-dimethylmorpholin-4-yl)pyridin-3-yl]-1-fluorovinyl}-5-methyl-1H-pyrazol-1-yl)methyl]-N-methylpyridine-2-amine
—— (R)-1-(4-(6-(5-isopropyl-2-methylphenyl)-2-(3-methyl-1H-indol-4-yl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-yl)-2-methylpiperazin-1-yl)ethanone 1421250-75-0 C33H40N6O
(R)-1-(4-(6-(5-isopropyl-2-methylphenyl)-2-(3-methyl-1H-indol-4-yl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-yl)-2-methylpiperazin-1-yl)ethanone
—— 3-(1-methylpyrazol-4-yl)-5-phenyl-6-[(1S)-1-(pyrazolo[1,5-a]pyrimidin-7-ylamino)ethyl]thieno[3,2-c]pyridin-4-one 1420621-14-2 C25H21N7OS
3-(1-methylpyrazol-4-yl)-5-phenyl-6-[(1S)-1-(pyrazolo[1,5-a]pyrimidin-7-ylamino)ethyl]thieno[3,2-c]pyridin-4-one
—— [(2S,3aR,6aR)-2-[(4aR,8aS)-hexahydropyrano[3,4-b][1,4]oxazin-1(5H)-yl]hexahydropentalen-3a(1H)-yl][3-(trifluoromethyl)-7,8-dihydro-1,6-naphthyridin-6(5H)-yl]methanone 1421064-21-2 C25H32F3N3O3
[(2S,3aR,6aR)-2-[(4aR,8aS)-hexahydropyrano[3,4-b][1,4]oxazin-1(5H)-yl]hexahydropentalen-3a(1H)-yl][3-(trifluoromethyl)-7,8-dihydro-1,6-naphthyridin-6(5H)-yl]methanone
—— 2-(4-(4-fluorobenzoyl)piperidin-1-yl)-N-((4-oxo-4,5,7,8-tetrahydro-3H-pyrano[4,3-d]pyrimidin-2-yl)methyl)-N-(pyridin-3-ylmethyl)ethanamide 1419949-84-0 C28H30FN5O4
2-(4-(4-fluorobenzoyl)piperidin-1-yl)-N-((4-oxo-4,5,7,8-tetrahydro-3H-pyrano[4,3-d]pyrimidin-2-yl)methyl)-N-(pyridin-3-ylmethyl)ethanamide
—— 1-(2,5-Difluorobenzyl)-N-(1-methyl-1H-pyrazol-3-yl)-1H-pyrazolo[4,3-c]pyridin-6-amine 1421856-80-5 C17H14F2N6
1-(2,5-Difluorobenzyl)-N-(1-methyl-1H-pyrazol-3-yl)-1H-pyrazolo[4,3-c]pyridin-6-amine
—— 2-(1-cyclobutylpiperidin-4-yl)-1-methyl-3-oxo-2,3-dihydro-1H-indazole-4-carboxamide 1421274-89-6 C18H24N4O2
2-(1-cyclobutylpiperidin-4-yl)-1-methyl-3-oxo-2,3-dihydro-1H-indazole-4-carboxamide
—— 8-((4-(3,4-difluorophenoxy)benzyl)oxy)-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one 1420369-92-1 C20H17F2N3O3
8-((4-(3,4-difluorophenoxy)benzyl)oxy)-3,4-dihydro-1H-pyrimido[1,6-a]pyrimidin-6(2H)-one
—— 1-((2-(4-methylpiperidin-1-yl)-6-(trifluoromethyl)pyridin-3-yl)methyl)-3-(2-methylpyrimidin-5-yl)urea 1421474-30-7 C19H23F3N6O
1-((2-(4-methylpiperidin-1-yl)-6-(trifluoromethyl)pyridin-3-yl)methyl)-3-(2-methylpyrimidin-5-yl)urea