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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2,2-Difluoro-1-(trifluoromethyl)cyclopropane-1-carboxylic acid 1378809-21-2 C5H3F5O2
2,2-Difluoro-1-(trifluoromethyl)cyclopropane-1-carboxylic acid
—— (R)-1-(5-(2-(2,5-difluorophenyl)pyrrolidin-1-yl)pyrazolo[1,5-a]pyrimidin-3-yl)-3-(4-methoxyphenyl)urea 1223403-66-4 C24H22F2N6O2
(R)-1-(5-(2-(2,5-difluorophenyl)pyrrolidin-1-yl)pyrazolo[1,5-a]pyrimidin-3-yl)-3-(4-methoxyphenyl)urea
—— (S)-1-benzyl-3-[5-chloro-2-[1-(3-trifluoromethyl-phenyl)-ethoxy]-phenoxy]-azetidine 1227620-42-9 C25H23ClF3NO2
(S)-1-benzyl-3-[5-chloro-2-[1-(3-trifluoromethyl-phenyl)-ethoxy]-phenoxy]-azetidine
—— (S)-3-{4-chloro-3-[(1S,2S)-6-chloro-4-fluoro-2((R)-3-hydroxypyrrolidin-1-yl)indan-1-yloxy]phenyl}-4-isopropyloxazolidin-2-one 1215273-40-7 C25H27Cl2FN2O4
(S)-3-{4-chloro-3-[(1S,2S)-6-chloro-4-fluoro-2((R)-3-hydroxypyrrolidin-1-yl)indan-1-yloxy]phenyl}-4-isopropyloxazolidin-2-one
—— N-[(1R,6R)-6-amino-2,2-difluorocyclohexyl]-5-ethynyl-4-pyrazolo[1,5-a]pyridin-3-yl-1,3-thiazole-2-carboxamide 1207556-85-1 C19H17F2N5OS
N-[(1R,6R)-6-amino-2,2-difluorocyclohexyl]-5-ethynyl-4-pyrazolo[1,5-a]pyridin-3-yl-1,3-thiazole-2-carboxamide
—— N-[3-((4aS,5S,8aS)-2-amino-5-fluoro-4,4a,5,6-tetrahydro-7-oxa-3-thia-1-azanaphthalen-8a-yl)-4-fluorophenyl]-5-difluoromethylpyrazine-2-carboxamide 1220325-65-4 C19H17F4N5O2S
N-[3-((4aS,5S,8aS)-2-amino-5-fluoro-4,4a,5,6-tetrahydro-7-oxa-3-thia-1-azanaphthalen-8a-yl)-4-fluorophenyl]-5-difluoromethylpyrazine-2-carboxamide
—— 2-chloro-6-[4-(1-methylimidazole-4-sulfonyl)-piperazin-1-ylmethyl]-4-morpholin-4-yl-thieno[3,2-d]pyrimidine 1032758-05-6 C19H24ClN7O3S2
2-chloro-6-[4-(1-methylimidazole-4-sulfonyl)-piperazin-1-ylmethyl]-4-morpholin-4-yl-thieno[3,2-d]pyrimidine
—— ethyl (2E)-4-[3-(2-tert-butyl-4-fluorophenoxy)azetidin-1-yl]-4-oxobut-2-enoate 1146957-95-0 C19H24FNO4
ethyl (2E)-4-[3-(2-tert-butyl-4-fluorophenoxy)azetidin-1-yl]-4-oxobut-2-enoate
—— 4-{[2-ethyl-4-(ethylsulfonyl)-3-fluorophenyl]carbonyl}-7-[5-(1H-imidazol-2-yl)-3-thienyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine 1251162-04-5 C27H26FN3O4S2
4-{[2-ethyl-4-(ethylsulfonyl)-3-fluorophenyl]carbonyl}-7-[5-(1H-imidazol-2-yl)-3-thienyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
—— 5,6-dimethyl-1-(pentan-3-yl)-1H-imidazo[4,5-b]pyridin-2-ol 1064781-31-2 C13H19N3O
5,6-dimethyl-1-(pentan-3-yl)-1H-imidazo[4,5-b]pyridin-2-ol
—— N-(4-(1H-1,2,4-triazol-1-yl)phenyl)-4-(3-morpholinophenyl)pyrimidin-2-amine 1128095-78-2 C22H21N7O
N-(4-(1H-1,2,4-triazol-1-yl)phenyl)-4-(3-morpholinophenyl)pyrimidin-2-amine
—— 4-(1H-Imidazol-1-yl)-2-(6-morpholin-4-ylpyrimidin-4-yl)-1,2-dihydro-3H-pyrazol-3-on 1154028-86-0 C14H15N7O2
4-(1H-Imidazol-1-yl)-2-(6-morpholin-4-ylpyrimidin-4-yl)-1,2-dihydro-3H-pyrazol-3-on
—— N-[2-hydroxy-1-(hydroxymethyl)ethyl]-4-({4-[({2-[methyl(methylsulfonyl)amino]pyridin-3-yl}methyl)amino]-5-(trifluoromethyl)pyrimidin-2-yl}amino)benzamide 1073157-92-2 C23H26F3N7O5S
N-[2-hydroxy-1-(hydroxymethyl)ethyl]-4-({4-[({2-[methyl(methylsulfonyl)amino]pyridin-3-yl}methyl)amino]-5-(trifluoromethyl)pyrimidin-2-yl}amino)benzamide
—— N-[4-(4-{[2-ethyl-3-fluoro-4-(methylsulfonyl)-phenyl]carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)phenyl]-2,2,2-trifluoroacetamide 1251161-59-7 C27H24F4N2O5S
N-[4-(4-{[2-ethyl-3-fluoro-4-(methylsulfonyl)-phenyl]carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)phenyl]-2,2,2-trifluoroacetamide
—— (1R,2R,4R)-N,N'-bis(benzyloxycarbonyl)-4-methyl-1,2-cyclohexanediamine 1246967-38-3 C23H28N2O4
(1R,2R,4R)-N,N'-bis(benzyloxycarbonyl)-4-methyl-1,2-cyclohexanediamine
—— —— 1638188-55-2 C8H12O5
—— —— 1399850-20-4 C16H25NO3*ClH
—— —— 1569076-60-3 C31H30N2O3S2
—— —— 1445004-77-2 C45H27IrN12
—— —— 1246195-71-0 C19H18F3NO4
—— 3-Fluoro-2-hydroxy-5-[3-(4-methylpiperazine-1-carbonyl)phenyl]benzaldehyde 1093119-07-3 C19H19FN2O3
3-Fluoro-2-hydroxy-5-[3-(4-methylpiperazine-1-carbonyl)phenyl]benzaldehyde
—— 8-N-[(2-amino-1,3-benzothiazol-6-yl)methyl]-3-N-(2-hydroxy-2-pyridin-4-ylethyl)-2-thiophen-3-ylimidazo[1,2-a]pyridine-3,8-dicarboxamide 1038692-90-8 C28H23N7O3S2
8-N-[(2-amino-1,3-benzothiazol-6-yl)methyl]-3-N-(2-hydroxy-2-pyridin-4-ylethyl)-2-thiophen-3-ylimidazo[1,2-a]pyridine-3,8-dicarboxamide
—— 4-[3-(3,5-dimethoxybenzyl)-6-[2-fluoro-1-(fluoromethyl)ethoxy]-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl]piperidine-1-carbaldehyde 1162651-20-8 C26H29F2N3O6
4-[3-(3,5-dimethoxybenzyl)-6-[2-fluoro-1-(fluoromethyl)ethoxy]-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl]piperidine-1-carbaldehyde
—— 3-(3-fluoro-5-formyl-4-hydroxyphenyl)-N-propan-2-ylbenzamide 1093118-99-0 C17H16FNO3
3-(3-fluoro-5-formyl-4-hydroxyphenyl)-N-propan-2-ylbenzamide
—— 4-N-cyclopropyl-6-N-[4-(diethylamino)phenyl]-3-methylsulfonyl-2H-pyrazolo[3,4-d]pyrimidine-4,6-diamine 1037475-61-8 C19H25N7O2S
4-N-cyclopropyl-6-N-[4-(diethylamino)phenyl]-3-methylsulfonyl-2H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
—— 4-oxo-4,5-dihydropyrrolo[1,2-a]quinoxaline-7-carboxamide 1255927-11-7 C12H9N3O2
4-oxo-4,5-dihydropyrrolo[1,2-a]quinoxaline-7-carboxamide
—— N-(4-(1H-tetrazol-1-yl)phenyl)-4-(3-morpholinophenyl)pyrimidin-2-amine 1128096-82-1 C21H20N8O
N-(4-(1H-tetrazol-1-yl)phenyl)-4-(3-morpholinophenyl)pyrimidin-2-amine
—— (R)-1-[rac-trans-(1,2)-4-chloro-6-fluoro-1-(3-methyl-4-trifluoromethanesulfonylphenoxy)indan-2-yl]piperidin-3-ylamine 1215272-20-0 C22H23ClF4N2O3S
(R)-1-[rac-trans-(1,2)-4-chloro-6-fluoro-1-(3-methyl-4-trifluoromethanesulfonylphenoxy)indan-2-yl]piperidin-3-ylamine
—— 1-[(2,2,3-trimethylcyclopent-3-enyl)methoxy]butan-2-ol 1020411-24-8 C13H24O2
1-[(2,2,3-trimethylcyclopent-3-enyl)methoxy]butan-2-ol
—— (R)-7-(2-(3-((4-(2,6-dimethylimidazo[1,2-a]pyridine-3-carbonyl)-1-oxa-4,9-diazaspiro[5.5]undecan-9-yl)methyl)-5-fluorophenethylamino)-1-hydroxyethyl)-4-hydroxybenzo[d]thiazol-2(3H)-one 1179334-36-1 C36H41FN6O5S
(R)-7-(2-(3-((4-(2,6-dimethylimidazo[1,2-a]pyridine-3-carbonyl)-1-oxa-4,9-diazaspiro[5.5]undecan-9-yl)methyl)-5-fluorophenethylamino)-1-hydroxyethyl)-4-hydroxybenzo[d]thiazol-2(3H)-one
—— N'-[4-(6-methoxy-4-morpholin-4-yl-2-naphthyl)pyrimidin-2-yl]-n,N-dimethylethane-1,2-diamine 1313486-02-0 C23H29N5O2
N'-[4-(6-methoxy-4-morpholin-4-yl-2-naphthyl)pyrimidin-2-yl]-n,N-dimethylethane-1,2-diamine
—— (R)-4-(4-(dimethylamino)phenyl)-5-nitropentan-2-one 1160841-00-8 C13H18N2O3
(R)-4-(4-(dimethylamino)phenyl)-5-nitropentan-2-one
—— (Z)-3-(ethylidene-1-d)-4-methyl-1-tosylpyrrolidine 1165841-57-5 C14H19NO2S
(Z)-3-(ethylidene-1-d)-4-methyl-1-tosylpyrrolidine
—— 8-(2-chloro-benzenesulfonyl)-2-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-phenyl]-2,8-diaza-spiro[4.5]decan-1-one 1255713-46-2 C23H21ClF6N2O4S
8-(2-chloro-benzenesulfonyl)-2-[4-(2,2,2-trifluoro-1-hydroxy-1-trifluoromethyl-ethyl)-phenyl]-2,8-diaza-spiro[4.5]decan-1-one
—— 5-hexyl-3-(4-methoxy-3-methylphenyl)-1,3-oxazolidin-2-one 1174336-68-5 C17H25NO3
5-hexyl-3-(4-methoxy-3-methylphenyl)-1,3-oxazolidin-2-one
—— tert-butyl 4-[(2-tert-butyl-4-fluorophenoxy)methyl]piperidine-1-carboxylate 1146960-30-6 C21H32FNO3
tert-butyl 4-[(2-tert-butyl-4-fluorophenoxy)methyl]piperidine-1-carboxylate
—— 2-[[trans-4-(1,1-Dimethylethyl)cyclohexyl]methyl]-1,4-naphthalenedione 1184761-65-6 C21H26O2
2-[[trans-4-(1,1-Dimethylethyl)cyclohexyl]methyl]-1,4-naphthalenedione
—— 6-(benzyloxy)-N-(2-fluorophenyl)-3-nitropyridin-2-amine 1217350-67-8 C18H14FN3O3
6-(benzyloxy)-N-(2-fluorophenyl)-3-nitropyridin-2-amine
—— (S)-2-(6-(4-(2,6-difluorobenzamido)phenyl)-1-oxoisoindolin-2-yl)-3-methylbutanoic acid 1313576-91-8 C26H22F2N2O4
(S)-2-(6-(4-(2,6-difluorobenzamido)phenyl)-1-oxoisoindolin-2-yl)-3-methylbutanoic acid
—— 4-[2-(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthalen-2-yl)thiazol-5-yl]piperidine 1314084-19-9 C22H30N2S
4-[2-(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthalen-2-yl)thiazol-5-yl]piperidine
—— pyridine-3-sulfonic acid (4-chloro-benzyl)-[3-(3-hydroxy-piperidine-1-carbonyl)-phenyl]-amide 1214251-23-6 C24H24ClN3O4S
pyridine-3-sulfonic acid (4-chloro-benzyl)-[3-(3-hydroxy-piperidine-1-carbonyl)-phenyl]-amide
—— 3-chloro-4-(4-phenylpyrimidin-2-ylamino)benzamide 1128097-07-3 C17H13ClN4O
3-chloro-4-(4-phenylpyrimidin-2-ylamino)benzamide
—— 5-[(tert-butoxycarbonyl)amino]-2-{[7-(1-propen-2-yl)-4,5-dihydroimidazo[1,5-a]quinolin-3-yl]methyl}pentanoic acid 1224849-22-2 C25H33N3O4
5-[(tert-butoxycarbonyl)amino]-2-{[7-(1-propen-2-yl)-4,5-dihydroimidazo[1,5-a]quinolin-3-yl]methyl}pentanoic acid
—— N-[3-methoxy-4-(4-methyl-5-oxazolyl)phenyl]-8-[2-(trifluoromethyl)phenyl]-[1,2,4]triazolo[1,5-a]pyridin-2-amine 1314786-32-7 C24H18F3N5O2
N-[3-methoxy-4-(4-methyl-5-oxazolyl)phenyl]-8-[2-(trifluoromethyl)phenyl]-[1,2,4]triazolo[1,5-a]pyridin-2-amine
—— ethyl (E)-3-[4-[[4-[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperazin-1-yl]methyl]phenyl]prop-2-enoate 1166811-84-2 C22H23F3N6O2
ethyl (E)-3-[4-[[4-[3-(trifluoromethyl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]piperazin-1-yl]methyl]phenyl]prop-2-enoate
—— tert-butyl 3-[(7-cyclohexyl-4,5-dihydroimidazo[1,5-a]quinolin-3-yl)methyl]-2-oxopiperidine-1-carboxylate 1224849-04-0 C28H37N3O3
tert-butyl 3-[(7-cyclohexyl-4,5-dihydroimidazo[1,5-a]quinolin-3-yl)methyl]-2-oxopiperidine-1-carboxylate
—— (E)-N-(1-(1H-benzo[d][1,2,3]triazol-1-yl)propylidene)aniline 1244768-88-4 C15H14N4
(E)-N-(1-(1H-benzo[d][1,2,3]triazol-1-yl)propylidene)aniline
—— 4-(3,5-Dimethoxyphenyl)-4-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]butan-2-one 1380311-70-5 C24H24N4O3
4-(3,5-Dimethoxyphenyl)-4-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]butan-2-one
—— N-tosyl-5-bromo-2-phenylindole-3-carboxylic acid 1374753-82-8 C22H16BrNO4S
N-tosyl-5-bromo-2-phenylindole-3-carboxylic acid
—— [(2,6-Me<sub>2</sub>C<sub>6</sub>H<sub>3</sub>NPPh<sub>2</sub>NPh<sub>2</sub>PNC<sub>6</sub>H<sub>3</sub>Me<sub>2</sub>-2,6)Sc(CH<sub>2</sub>SiMe<sub>3</sub>)<sub>2</sub>] 1415036-20-2 C48H60N3P2ScSi2
[(2,6-Me<sub>2</sub>C<sub>6</sub>H<sub>3</sub>NPPh<sub>2</sub>NPh<sub>2</sub>PNC<sub>6</sub>H<sub>3</sub>Me<sub>2</sub>-2,6)Sc(CH<sub>2</sub>SiMe<sub>3</sub>)<sub>2</sub>]