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中文名称 英文名称 CAS号 化学式 结构式图片
—— (RS)-(E)-3-(2,6-dichloro-4-{4-[3-(2,2-dimethylpropyl-1-ethoxy)-2-methyloxyphenyl]thiazol-2-ylcarbamoyl}phenyl)-2-methylacrylic acid 1110767-41-3 C28H30Cl2N2O5S
(RS)-(E)-3-(2,6-dichloro-4-{4-[3-(2,2-dimethylpropyl-1-ethoxy)-2-methyloxyphenyl]thiazol-2-ylcarbamoyl}phenyl)-2-methylacrylic acid
—— 3,3-dimethyl-6-[8-(1,3,5-trimethyl-1H-pyrazol-4-yl)-[1,2,4]triazolo[1,5-a]pyrazin-2-ylamino]-1,3-dihydro-indol-2-one 1451386-68-7 C21H22N8O
3,3-dimethyl-6-[8-(1,3,5-trimethyl-1H-pyrazol-4-yl)-[1,2,4]triazolo[1,5-a]pyrazin-2-ylamino]-1,3-dihydro-indol-2-one
—— 2-({4-cyclopropyl-6'-[(3S)-3-hydroxypyrrolidin-1-yl]-2,3'-bipyridin-6-yl}amino)pyridine-4-carbonitrile hydrochloride 1374140-30-3 C23H22N6O*ClH
2-({4-cyclopropyl-6'-[(3S)-3-hydroxypyrrolidin-1-yl]-2,3'-bipyridin-6-yl}amino)pyridine-4-carbonitrile hydrochloride
—— 2-[[(E)-2-(4-bromophenyl)ethenyl]sulfonylamino]-5-fluoro-benzenesulfonamide 1161943-48-1 C14H12BrFN2O4S2
2-[[(E)-2-(4-bromophenyl)ethenyl]sulfonylamino]-5-fluoro-benzenesulfonamide
—— 4-[2-(4-Chlorophenyl)-4-methyl-1,3-thiazol-5-yl]-2,2,6,6-tetramethyloxane-3,5-dione 1094621-49-4 C19H20ClNO3S
4-[2-(4-Chlorophenyl)-4-methyl-1,3-thiazol-5-yl]-2,2,6,6-tetramethyloxane-3,5-dione
—— 5-[1-ethyl-2-(3-fluorophenyl)-1H-benzimidazol-5-yl]-3,6-dihydro-2H-1,3,4-thiadiazin-2-one 1151821-22-5 C18H15FN4OS
5-[1-ethyl-2-(3-fluorophenyl)-1H-benzimidazol-5-yl]-3,6-dihydro-2H-1,3,4-thiadiazin-2-one
—— (6S,9aS)-8-(1,3-benzoxazol-6-ylmethyl)-N-benzyl-6-[(4-hydroxyphenyl)methyl]-4,7-dioxo-2-prop-2-enyl-3,6,9,9a-tetrahydropyrazino[2,1-c][1,2,4]triazine-1-carboxamide 1145673-74-0 C32H32N6O5
(6S,9aS)-8-(1,3-benzoxazol-6-ylmethyl)-N-benzyl-6-[(4-hydroxyphenyl)methyl]-4,7-dioxo-2-prop-2-enyl-3,6,9,9a-tetrahydropyrazino[2,1-c][1,2,4]triazine-1-carboxamide
—— methyl 4-{3-[(2-tert-butylphenoxy)methyl]azetidin-1-yl}-4-oxobutanoate 1146959-06-9 C19H27NO4
methyl 4-{3-[(2-tert-butylphenoxy)methyl]azetidin-1-yl}-4-oxobutanoate
—— N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-2-pyrimidin-2-yl-4-(trifluoromethyl)-1,3-thiazole-5-carboxamide 1104273-54-2 C22H21F3N4O2S
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-2-pyrimidin-2-yl-4-(trifluoromethyl)-1,3-thiazole-5-carboxamide
—— methyl (2R)-2-[3-cyclopropyl-4-(cyclopropylsulfonyl)phenyl]-3-(4-oxocyclohexyl)propanoate 1174229-58-3 C22H28O5S
methyl (2R)-2-[3-cyclopropyl-4-(cyclopropylsulfonyl)phenyl]-3-(4-oxocyclohexyl)propanoate
—— 1-[4-[3-[1-(Difluoromethyl)benzimidazol-2-yl]phenyl]piperazin-1-yl]-2-piperidin-1-ylethanone 1160831-21-9 C25H29F2N5O
1-[4-[3-[1-(Difluoromethyl)benzimidazol-2-yl]phenyl]piperazin-1-yl]-2-piperidin-1-ylethanone
—— N-(adamantan-1-ylmethyl)-3-cyclopropyl-1-pyrimidin-2-yl-1H-pyrazole-4-carboxamide 1104269-93-3 C22H27N5O
N-(adamantan-1-ylmethyl)-3-cyclopropyl-1-pyrimidin-2-yl-1H-pyrazole-4-carboxamide
—— 3-{4-[(2-tert-butyl-4-fluorophenoxy)methyl]piperidin-1-yl}-3-oxopropanoic acid 1146958-46-4 C19H26FNO4
3-{4-[(2-tert-butyl-4-fluorophenoxy)methyl]piperidin-1-yl}-3-oxopropanoic acid
—— (R)-5-[4-(2-hydroxy-ethoxy)-phenyl]-3-[(1R,2R)-1-(5-iodo-1H-benzoimidazol-2-yl)-2-methoxy-propyl]-imidazolidine-2,4-dione 1116600-68-0 C22H23IN4O5
(R)-5-[4-(2-hydroxy-ethoxy)-phenyl]-3-[(1R,2R)-1-(5-iodo-1H-benzoimidazol-2-yl)-2-methoxy-propyl]-imidazolidine-2,4-dione
—— ((S)-4-(4-(3-fluoro-4-methylphenyl)phthalazin-1-yl)-2-methylpiperazin-1-yl)(phenyl)methanone 1095638-06-4 C27H25FN4O
((S)-4-(4-(3-fluoro-4-methylphenyl)phthalazin-1-yl)-2-methylpiperazin-1-yl)(phenyl)methanone
—— 2-amino-N-(3-difluoromethoxy-phenyl)-2-phenyl-N-[2-(4-trifluoromethyl-phenyl)-ethyl]-acetamide 1111731-55-5 C24H21F5N2O2
2-amino-N-(3-difluoromethoxy-phenyl)-2-phenyl-N-[2-(4-trifluoromethyl-phenyl)-ethyl]-acetamide
—— methyl 2-[[(1R,2R,11R,14R,15S,18S,23S)-2,10,10,14,15,21,21-heptamethyl-5,8-diazahexacyclo[12.12.0.02,11.04,9.015,24.018,23]hexacosa-4,6,8,24-tetraene-18-carbonyl]amino]acetate 1084775-66-5 C35H51N3O3
methyl 2-[[(1R,2R,11R,14R,15S,18S,23S)-2,10,10,14,15,21,21-heptamethyl-5,8-diazahexacyclo[12.12.0.02,11.04,9.015,24.018,23]hexacosa-4,6,8,24-tetraene-18-carbonyl]amino]acetate
—— 4-fluoro-2-[[(E)-2-naphthalen-2-ylethenyl]sulfonylamino]benzenesulfonamide 1161943-37-8 C18H15FN2O4S2
4-fluoro-2-[[(E)-2-naphthalen-2-ylethenyl]sulfonylamino]benzenesulfonamide
—— 1-methyl-3-[6-(1-methyl-1H-pyrrol-2-yl)imidazo[1,2-b]pyridazin-8-yl]urea 1161846-65-6 C13H14N6O
1-methyl-3-[6-(1-methyl-1H-pyrrol-2-yl)imidazo[1,2-b]pyridazin-8-yl]urea
—— N-[3,5-di(morpholin-4-yl)phenyl]-N'-methyl-N'-(5-methylpyridin-2-yl)pyrimidine-2,4-diamine 1104455-22-2 C25H31N7O2
N-[3,5-di(morpholin-4-yl)phenyl]-N'-methyl-N'-(5-methylpyridin-2-yl)pyrimidine-2,4-diamine
—— 2-Pent-4-ynyl-cyclohepta-2,4,6-trienone 109459-03-2 C12H12O
2-Pent-4-ynyl-cyclohepta-2,4,6-trienone
—— (1R,4S,4aR,5R,8aS)-3-cyclohexyl-5-hydroxy-1-methyl-1,4,4a,5,6,7,8,8a-octahydrobenzo[d]oxazine-4-carbonitrile 106625-95-0 C16H26N2O2
(1R,4S,4aR,5R,8aS)-3-cyclohexyl-5-hydroxy-1-methyl-1,4,4a,5,6,7,8,8a-octahydrobenzo[d]oxazine-4-carbonitrile
—— (2R,3R)-2,3-Bis-(2-hydroxy-5-methoxy-phenyl)-1,2,3,4-tetrahydro-benzo[g]quinoxaline-5,10-dione 108059-20-7 C26H22N2O6
(2R,3R)-2,3-Bis-(2-hydroxy-5-methoxy-phenyl)-1,2,3,4-tetrahydro-benzo[g]quinoxaline-5,10-dione
—— ((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(2-isopropoxynaphthalen-1-yl)pyrazolo[1,5-a]pyrimidin-7-ylamino)cyclopentyl)methyl sulfamate 1450834-53-3 C25H29N5O6S
((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(2-isopropoxynaphthalen-1-yl)pyrazolo[1,5-a]pyrimidin-7-ylamino)cyclopentyl)methyl sulfamate
—— 2-[1-(2,2-dimethylpropyl)-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-4-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}benzonitrile 1352422-90-2 C28H34N8O
2-[1-(2,2-dimethylpropyl)-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-4-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}benzonitrile
—— 15-[[N-[N-[(1,1-dimethylethoxy)carbonyl]-L-Leucyl]-O-(phenylmethyl)-D-glutamyl]amino]-2,3,5,6,8,9,11,12-octahydro-1,4,7,10,13-benzopentaoxacyclopentadecin 149674-03-3 C37H53N3O11
15-[[N-[N-[(1,1-dimethylethoxy)carbonyl]-L-Leucyl]-O-(phenylmethyl)-D-glutamyl]amino]-2,3,5,6,8,9,11,12-octahydro-1,4,7,10,13-benzopentaoxacyclopentadecin
—— —— 1606589-58-5 C22H34BrNO2Si
—— (S)-2-(3-oxo-3-(pyridin-2-yl)-1-(4-(trifluoromethyl)phenyl)propyl)malononitrile 1394363-87-1 C18H12F3N3O
(S)-2-(3-oxo-3-(pyridin-2-yl)-1-(4-(trifluoromethyl)phenyl)propyl)malononitrile
—— (3R,4R,6S)-1-benzyl-6-[(1S)-1,2-dihydroxyethyl]-3,4-dihydroxyazepan-2-one 1587637-33-9 C15H21NO5
(3R,4R,6S)-1-benzyl-6-[(1S)-1,2-dihydroxyethyl]-3,4-dihydroxyazepan-2-one
—— —— 1384972-96-6 C18H16N6O2S
—— —— 1395878-13-3 C19H27NO6
—— (R)-diethyl 2-(4-(3-fluorophenyl)-1-nitrobut-3-yn-2-yl)malonate 1432626-36-2 C17H18FNO6
(R)-diethyl 2-(4-(3-fluorophenyl)-1-nitrobut-3-yn-2-yl)malonate
—— C5a-n-butoxymethylminocycline trifluoroacetate 1352457-55-6 C2HF3O2*C28H37N3O8
C5a-n-butoxymethylminocycline trifluoroacetate
—— 6,7,9-trimethoxy-10,11-dihydrodibenz[b,f]oxepin-10-one 182321-85-3 C17H16O5
6,7,9-trimethoxy-10,11-dihydrodibenz[b,f]oxepin-10-one
—— 1-(1-ethyl-propyl)-4,7-dimethyl-5-(2,4,6-trimethyl-phenoxy)-1,4-dihydro-2H-pyrimido[4,5-d][1,3]oxazine 1348515-62-7 C22H31N3O2
1-(1-ethyl-propyl)-4,7-dimethyl-5-(2,4,6-trimethyl-phenoxy)-1,4-dihydro-2H-pyrimido[4,5-d][1,3]oxazine
—— 2-methanesulfonyl-4-[5-azabenzimidazol-1-yl]pyrimidine 1426231-51-7 C11H9N5O2S
2-methanesulfonyl-4-[5-azabenzimidazol-1-yl]pyrimidine
—— 4'-methyl-5-(4-methyl-imidazol-1-yl)-biphenyl-3-carboxylic acid (2-methoxy-1-methyl-ethyl)-amide 1161830-27-8 C22H25N3O2
4'-methyl-5-(4-methyl-imidazol-1-yl)-biphenyl-3-carboxylic acid (2-methoxy-1-methyl-ethyl)-amide
—— N-[2-(dimethylamino)ethyl]-4-({[4-(5-methyl-4-morpholin-4-yl-5H-pyrrolo[3,2-d]pyrimidin-2-yl)phenyl]carbamoyl}amino)-N-methylbenzamide 1155811-59-8 C30H36N8O3
N-[2-(dimethylamino)ethyl]-4-({[4-(5-methyl-4-morpholin-4-yl-5H-pyrrolo[3,2-d]pyrimidin-2-yl)phenyl]carbamoyl}amino)-N-methylbenzamide
—— 4-methyl-3,4,5,6-tetrahydro-2H-[1,2']bipyridinyl-5'-carboxylicacid (3-chloro-phenyl)-amide 1110781-33-3 C18H20ClN3O
4-methyl-3,4,5,6-tetrahydro-2H-[1,2']bipyridinyl-5'-carboxylicacid (3-chloro-phenyl)-amide
—— 5H-indolo[2,1-a][2]benzazepine-10-carboxamide, 13-cyclohexyl-N-[(dimethylamino)sulfonyl]-6,7-dihydro-3-methoxy-6-[6-(4-morpholinyl)-2-pyridinyl]- 1112187-63-9 C36H43N5O5S
5H-indolo[2,1-a][2]benzazepine-10-carboxamide, 13-cyclohexyl-N-[(dimethylamino)sulfonyl]-6,7-dihydro-3-methoxy-6-[6-(4-morpholinyl)-2-pyridinyl]-
—— (6-{5-[(5-bromopyridine-2-carbonyl)amino]-2-fluorophenyl}-4,6-dimethyl-3,4,5,6-tetrahydropyrazin-2-yl)carbamic acid tert-butyl ester 1313525-79-9 C23H27BrFN5O3
(6-{5-[(5-bromopyridine-2-carbonyl)amino]-2-fluorophenyl}-4,6-dimethyl-3,4,5,6-tetrahydropyrazin-2-yl)carbamic acid tert-butyl ester
—— 2-bromo-N-(adamantan-2-yl)-2-methyl-N'-(4-nitrophenyl)propane hydrazide 1224513-58-9 C20H26BrN3O3
2-bromo-N-(adamantan-2-yl)-2-methyl-N'-(4-nitrophenyl)propane hydrazide
—— 4-[4-(3-Chloro-4-methoxyphenyl)-2-ethylphenyl]-5-hydroxy-2,2,6,6-tetramethylpyran-3-one 1160560-00-8 C24H27ClO4
4-[4-(3-Chloro-4-methoxyphenyl)-2-ethylphenyl]-5-hydroxy-2,2,6,6-tetramethylpyran-3-one
—— 4-[3-(1H-benzimidazol-2-yl)-4-chlorophenyl]-N-(2-morpholin-4-ylethyl)-1,4-diazepane-1-carboxamide 1160833-78-2 C25H31ClN6O2
4-[3-(1H-benzimidazol-2-yl)-4-chlorophenyl]-N-(2-morpholin-4-ylethyl)-1,4-diazepane-1-carboxamide
—— 2-[3-(1-amino-cyclopropyl)-1-methyl-azetidin-3-yl]-8-[4-(3-morpholin-4-yl-propyl)-phenyl]-4,5-dihydro-1H-pyrrolo[2,3-f]isoquinoline-3-carboxylic acid lactam 1105660-90-9 C32H37N5O2
2-[3-(1-amino-cyclopropyl)-1-methyl-azetidin-3-yl]-8-[4-(3-morpholin-4-yl-propyl)-phenyl]-4,5-dihydro-1H-pyrrolo[2,3-f]isoquinoline-3-carboxylic acid lactam
—— 2-(3,5-dimethyl-pyrazol-1-yl)-1-{4-[2-(1H-imidazo[4,5-c]pyridin-2-yl)phenyl]piperazin-1-yl}ethanone 1253936-88-7 C23H25N7O
2-(3,5-dimethyl-pyrazol-1-yl)-1-{4-[2-(1H-imidazo[4,5-c]pyridin-2-yl)phenyl]piperazin-1-yl}ethanone
—— 2-Hydroxy-5-(4-isoquinolinyl)-3-methoxybenzaldehyde 1093118-40-1 C17H13NO3
2-Hydroxy-5-(4-isoquinolinyl)-3-methoxybenzaldehyde
—— (+/-)-(2-{[4-(10-{[4-(trifluoromethyl)phenyl]sulfonyl}-4,5,6,7,8,9-hexahydro-1H-4,8-epiminocycloocta[c]pyrazol-6-yl)phenyl]amino}ethoxy)acetic acid 1215182-14-1 C26H27F3N4O5S
(+/-)-(2-{[4-(10-{[4-(trifluoromethyl)phenyl]sulfonyl}-4,5,6,7,8,9-hexahydro-1H-4,8-epiminocycloocta[c]pyrazol-6-yl)phenyl]amino}ethoxy)acetic acid
—— 6-ethoxy-2-(2,3,6-trichloro-benzylsulfanyl)-benzothiazole 133043-87-5 C16H12Cl3NOS2
6-ethoxy-2-(2,3,6-trichloro-benzylsulfanyl)-benzothiazole
—— —— 102764-28-3 C36H30N4O2S2Zn