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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-(4-(5-trifluoromethyl-2-(3-methoxyphenylamino)pyrimidin-4-ylamino)phenyl)methylacrylamide 1202758-38-0 C22H20F3N5O2
N-(4-(5-trifluoromethyl-2-(3-methoxyphenylamino)pyrimidin-4-ylamino)phenyl)methylacrylamide
—— 2-(2,2-dichloro-acetylamino)-2-methyl-3-(4-nitro-phenyl)-propionic acid 100122-46-1 C12H12Cl2N2O5
2-(2,2-dichloro-acetylamino)-2-methyl-3-(4-nitro-phenyl)-propionic acid
—— 2-[5-(4-fluoro-benzyl)-oxazol-2-yl]-3-hydroxy-7-methyl-pyrido[1,2-a]pyrimidin-4-one 1036646-59-9 C19H14FN3O3
2-[5-(4-fluoro-benzyl)-oxazol-2-yl]-3-hydroxy-7-methyl-pyrido[1,2-a]pyrimidin-4-one
—— 2-hydroxy-N-[2,3,5-tris(trifluoromethyl)phenyl]benzamide 17636-70-3 C16H8F9NO2
2-hydroxy-N-[2,3,5-tris(trifluoromethyl)phenyl]benzamide
—— N-[5-(2,4-dichlorophenyl)-1H-pyrazol-3-yl]-4-(1,4-oxazepan-4-yl)butanamide 1040720-21-5 C18H22Cl2N4O2
N-[5-(2,4-dichlorophenyl)-1H-pyrazol-3-yl]-4-(1,4-oxazepan-4-yl)butanamide
—— (R)-4'-(N-(3-(1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-ylamino)-2-hydroxypropyl)-N-methylsulfamoyl)-2'-methylbiphenyl-3-carboxylic acid 1198609-35-6 C31H38N2O5S
(R)-4'-(N-(3-(1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-ylamino)-2-hydroxypropyl)-N-methylsulfamoyl)-2'-methylbiphenyl-3-carboxylic acid
—— (S)-3-ethyl-2-(methoxycarbonylamino)pentanoic acid 1007884-67-4 C9H17NO4
(S)-3-ethyl-2-(methoxycarbonylamino)pentanoic acid
—— N-((S)-3-amino-4-fluorobutyl)-N-((1R)-1-(1-benzyl-3-(2,5-difluorophenyl)-1H-1,2,4-triazol-5-yl)-2,2-dimethylpropyl)-2-methoxyacetamide 1029622-88-5 C27H34F3N5O2
N-((S)-3-amino-4-fluorobutyl)-N-((1R)-1-(1-benzyl-3-(2,5-difluorophenyl)-1H-1,2,4-triazol-5-yl)-2,2-dimethylpropyl)-2-methoxyacetamide
—— 4-[(4-ethoxy-3-methoxyphenyl)(pyrimidin-5-ylmethyl)amino]benzoic acid 1203594-31-3 C21H21N3O4
4-[(4-ethoxy-3-methoxyphenyl)(pyrimidin-5-ylmethyl)amino]benzoic acid
—— 5-{3-[2-chloro-5-methyl-3'-(methylsulfonyl)biphenyl-4-yl]-4-hydroxy-2-oxo-1-oxa-8-azaspiro[4.5]-dec-3-en-8-yl}-5-oxopentanoic acid 1008779-72-3 C27H28ClNO8S
5-{3-[2-chloro-5-methyl-3'-(methylsulfonyl)biphenyl-4-yl]-4-hydroxy-2-oxo-1-oxa-8-azaspiro[4.5]-dec-3-en-8-yl}-5-oxopentanoic acid
—— N-(4-(5-fluoro-2-(3-fluoro-4-(2-methoxyethoxy)phenylamino)pyrimidin-4-ylamino)phenyl)acrylamide 1202759-41-8 C22H21F2N5O3
N-(4-(5-fluoro-2-(3-fluoro-4-(2-methoxyethoxy)phenylamino)pyrimidin-4-ylamino)phenyl)acrylamide
—— 2-(11,11-difluoroundecyl)isoindoline-1,3-dione 1131620-23-9 C19H25F2NO2
2-(11,11-difluoroundecyl)isoindoline-1,3-dione
—— (S)-6-chloro-2-hydroxy-N-methoxy-3-(2-(1-methoxy-3-phenylpropan-2-ylamino)-3,4-dioxocyclobut-1-enylamino)-N-methylbenzenesulfonamide 1206896-07-2 C22H24ClN3O7S
(S)-6-chloro-2-hydroxy-N-methoxy-3-(2-(1-methoxy-3-phenylpropan-2-ylamino)-3,4-dioxocyclobut-1-enylamino)-N-methylbenzenesulfonamide
—— Ethyl 2-[3-chloro-4-[[2-chloro-5-[(2-chlorophenyl)methoxy]benzoyl]amino]phenyl]acetate 1034026-39-5 C24H20Cl3NO4
Ethyl 2-[3-chloro-4-[[2-chloro-5-[(2-chlorophenyl)methoxy]benzoyl]amino]phenyl]acetate
—— (+/-)-1-methylethyl 4-[1-({6-[4-(methylsulfonyl)phenyl]-3-pyridinyl}oxy)propyl]-1-piperidinecarboxylate 1032824-27-3 C24H32N2O5S
(+/-)-1-methylethyl 4-[1-({6-[4-(methylsulfonyl)phenyl]-3-pyridinyl}oxy)propyl]-1-piperidinecarboxylate
—— 6-((S)-2-hydroxymethyl-pyrrolidin-1-yl)-pyridine-2-carboxylic acid [3-(3-fluoro-benzoylamino)-adamantan-1-yl]-amide 1206459-39-3 C28H33FN4O3
6-((S)-2-hydroxymethyl-pyrrolidin-1-yl)-pyridine-2-carboxylic acid [3-(3-fluoro-benzoylamino)-adamantan-1-yl]-amide
—— 2-[5-(2,4-Difluorophenyl)-4-methyl-3-phenylpyrazol-1-yl]-1,3-thiazole-4-carboxylic acid 1204747-05-6 C20H13F2N3O2S
2-[5-(2,4-Difluorophenyl)-4-methyl-3-phenylpyrazol-1-yl]-1,3-thiazole-4-carboxylic acid
—— 3'-[4-(4-Chlorophenyl)-2,5-dimethylphenyl]-4'-hydroxyspiro[1,2,3,3a,4,5,7,7a-octahydroindene-6,5'-furan]-2'-one 1008777-86-3 C26H27ClO3
3'-[4-(4-Chlorophenyl)-2,5-dimethylphenyl]-4'-hydroxyspiro[1,2,3,3a,4,5,7,7a-octahydroindene-6,5'-furan]-2'-one
—— (4S,5R)-2,2,5-trimethyl-4-propyl-1,3-dioxane 170207-76-8 C10H20O2
(4S,5R)-2,2,5-trimethyl-4-propyl-1,3-dioxane
—— 5-[4-[4-Hydroxy-1-methyl-5-(3,5,6,7-tetrahydropyrrolo[3,4-f]benzimidazol-2-yl)pyrazol-3-yl]phenyl]pyridine-2-carbonitrile 1197339-60-8 C25H19N7O
5-[4-[4-Hydroxy-1-methyl-5-(3,5,6,7-tetrahydropyrrolo[3,4-f]benzimidazol-2-yl)pyrazol-3-yl]phenyl]pyridine-2-carbonitrile
—— 1-ethyl-3-(3-(4-(4-(methylsulfonyl)phenylsulfonyl)piperazine-1-carbonyl)benzo[b]thiophen-2-yl)urea 1067907-92-9 C23H26N4O6S3
1-ethyl-3-(3-(4-(4-(methylsulfonyl)phenylsulfonyl)piperazine-1-carbonyl)benzo[b]thiophen-2-yl)urea
—— 1-(1-((2R,3R)-3-(2,4-difluorophenyl)-3-hydroxy-4-(1H-1,2,4-triazol-1-yl)butan-2-yl)-1H-pyrazol-4-yl)-1H-(3-(4-trifluoromethyl)phenyl)imidazole-2(3H)-one 1037784-75-0 C25H20F5N7O2
1-(1-((2R,3R)-3-(2,4-difluorophenyl)-3-hydroxy-4-(1H-1,2,4-triazol-1-yl)butan-2-yl)-1H-pyrazol-4-yl)-1H-(3-(4-trifluoromethyl)phenyl)imidazole-2(3H)-one
—— 4-[4-(4-tetrazol-1-ylphenoxymethyl)thiazol-2-yl]piperidine-1-carboxylic acid 2-fluoroethyl ester 1037792-02-1 C19H21FN6O3S
4-[4-(4-tetrazol-1-ylphenoxymethyl)thiazol-2-yl]piperidine-1-carboxylic acid 2-fluoroethyl ester
—— 3-((3-(isoquinolin-5-ylamino)piperidin-1-yl)methyl)benzonitrile 1035096-23-1 C22H22N4
3-((3-(isoquinolin-5-ylamino)piperidin-1-yl)methyl)benzonitrile
—— 7,9-dichloro-N-(3,4-dichlorophenyl)-3-oxo-2,3,4,5-tetrahydro-1,4-benzoxazepine-5-carboxamide 1067226-50-9 C16H10Cl4N2O3
7,9-dichloro-N-(3,4-dichlorophenyl)-3-oxo-2,3,4,5-tetrahydro-1,4-benzoxazepine-5-carboxamide
—— N-((1S,3R)-3-(6H-pyrrolo[2,3-e][1,2,4]triazolo[4,3-a]pyrazin-1-yl)cyclopentyl)-2-(4-cyanophenyl)ethanamide 1310723-29-5 C21H19N7O
N-((1S,3R)-3-(6H-pyrrolo[2,3-e][1,2,4]triazolo[4,3-a]pyrazin-1-yl)cyclopentyl)-2-(4-cyanophenyl)ethanamide
—— {5-[5-(1-methyl-1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-3-yl]-1,3,4-oxadiazol-2-yl}phenylmethanol 1379669-97-2 C20H16N6O2
{5-[5-(1-methyl-1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridin-3-yl]-1,3,4-oxadiazol-2-yl}phenylmethanol
—— 2,3,3a,6,7,7a-hexahydro-7-methyl-3-oxo-isothiazolo[4,5-c]pyridine-5(4H)-carboxylic acid 1,1-dimethylethyl ester 126737-86-8 C12H20N2O3S
2,3,3a,6,7,7a-hexahydro-7-methyl-3-oxo-isothiazolo[4,5-c]pyridine-5(4H)-carboxylic acid 1,1-dimethylethyl ester
—— tris(4-(but-1-en-1-yl)phenyl)stibane 19629-37-9 C30H33Sb
tris(4-(but-1-en-1-yl)phenyl)stibane
—— 3-(2-methoxycarbonylmethoxy-3,4-dimethoxy-phenyl)-trans(?)-crotonic acid methyl ester 107059-00-7 C16H20O7
3-(2-methoxycarbonylmethoxy-3,4-dimethoxy-phenyl)-trans(?)-crotonic acid methyl ester
—— 2-bromo-N-(4-((tert-butyldimethylsilyl)oxy)-2-(4-carbamoyl-4-(methylamino)piperidin-1-yl)phenyl)thiazole-4-carboxamide 1374113-36-6 C23H34BrN5O3SSi
2-bromo-N-(4-((tert-butyldimethylsilyl)oxy)-2-(4-carbamoyl-4-(methylamino)piperidin-1-yl)phenyl)thiazole-4-carboxamide
—— triisopropyl(6-methyl-1H-inden-2-yl)silane 1352210-87-7 C19H30Si
triisopropyl(6-methyl-1H-inden-2-yl)silane
—— 1,3-dimethyl-6-(3-methoxyphenyl)uracil 105202-44-6 C13H14N2O3
1,3-dimethyl-6-(3-methoxyphenyl)uracil
—— 3-<5-Oxo-5,6,7,8-tetrahydro-phenanthryl-(2)>-buttersaeure 1576-02-9 C18H18O3
3-<5-Oxo-5,6,7,8-tetrahydro-phenanthryl-(2)>-buttersaeure
—— 6,6-dioxo-5,7-dihydro-6λ6-dibenzo[c,e]thiepin-3,9-dicarboxylic acid diethyl ester 111413-77-5 C20H20O6S
6,6-dioxo-5,7-dihydro-6λ6-dibenzo[c,e]thiepin-3,9-dicarboxylic acid diethyl ester
—— Ethyl (Z)-2-(N-benzoylamino)-4(R),5(R)-bis<(p-methoxybenzyl)oxy>-5-<N-(monomethoxytrityl)-2'(S)-aziridinyl>-2-pentenoate 139559-29-8 C52H52N2O8
Ethyl (Z)-2-(N-benzoylamino)-4(R),5(R)-bis<(p-methoxybenzyl)oxy>-5-<N-(monomethoxytrityl)-2'(S)-aziridinyl>-2-pentenoate
—— 3(R)4(S)5(S)-3-methyl-4-benzylthio-5-(d-menthyloxy)-butyrolactone 141643-08-5 C22H32O3S
3(R)4(S)5(S)-3-methyl-4-benzylthio-5-(d-menthyloxy)-butyrolactone
—— (2,2,5-trimethyl-1,3-dioxan-5-yl)methyl 4-methylbenzoate 1163693-76-2 C16H22O4
(2,2,5-trimethyl-1,3-dioxan-5-yl)methyl 4-methylbenzoate
—— 5-(2-chloro-phenyl)-2-methyl-thiazole-4-carboxylic acid methyl ester 1007875-60-6 C12H10ClNO2S
5-(2-chloro-phenyl)-2-methyl-thiazole-4-carboxylic acid methyl ester
—— N-[(1S,2S)-2-hydroxycyclohexyl]-4-[(6-(1,3-thiazol-2-yl)pyridin-3-yl)methyl]-quinoline-2-carboxamide 1314142-47-6 C25H24N4O2S
N-[(1S,2S)-2-hydroxycyclohexyl]-4-[(6-(1,3-thiazol-2-yl)pyridin-3-yl)methyl]-quinoline-2-carboxamide
—— 5'-(2,6-dichlorobenzylamino)-5-fluorouridine 1266254-00-5 C16H16Cl2FN3O5
5'-(2,6-dichlorobenzylamino)-5-fluorouridine
—— (4S,5R,6S,7S,8S,9R)-6-azido-8-[[tert-butyl(diphenyl)silyl]oxymethyl]-2-(4-methoxyphenyl)-4,9-dimethyl-7-(3-prop-1-en-2-ylanilino)-3-oxa-1-azaspiro[4.4]non-1-ene-8,9-diol 1295471-25-8 C42H49N5O5Si
(4S,5R,6S,7S,8S,9R)-6-azido-8-[[tert-butyl(diphenyl)silyl]oxymethyl]-2-(4-methoxyphenyl)-4,9-dimethyl-7-(3-prop-1-en-2-ylanilino)-3-oxa-1-azaspiro[4.4]non-1-ene-8,9-diol
—— N-(2-t-butoxycarbonylaminophenyl)-4-[1-(3-t-butoxycarbonylaminopropyl)-3-(2,3-dihydrobenzo[1,4]dioxin-6-yl)ureidomethyl]benzamide 1034494-61-5 C36H45N5O8
N-(2-t-butoxycarbonylaminophenyl)-4-[1-(3-t-butoxycarbonylaminopropyl)-3-(2,3-dihydrobenzo[1,4]dioxin-6-yl)ureidomethyl]benzamide
—— 2-(5-((4-(5-methylthiophen-2-ylcarbonyl)-1-oxa-4,9-diazaspiro[5.5]undecane-9-yl)methyl)thiophen-3-yl)ethanaldehyde 1179336-88-9 C21H26N2O3S2
2-(5-((4-(5-methylthiophen-2-ylcarbonyl)-1-oxa-4,9-diazaspiro[5.5]undecane-9-yl)methyl)thiophen-3-yl)ethanaldehyde
—— (R)-5-(1-(tert-butyldimethylsilanyloxy)-2-((5-(2-(4-(2-methylthiazol-4-ylcarbonyl)-1-oxa-4,9-diazaspiro[5.5]undec-9-yl)ethyl)thiophen-2-yl)methylamino)ethyl)-8-hydroxyquinoline-2(1H)-one 1179338-80-7 C37H51N5O5S2Si
(R)-5-(1-(tert-butyldimethylsilanyloxy)-2-((5-(2-(4-(2-methylthiazol-4-ylcarbonyl)-1-oxa-4,9-diazaspiro[5.5]undec-9-yl)ethyl)thiophen-2-yl)methylamino)ethyl)-8-hydroxyquinoline-2(1H)-one
—— 5-fluoro-2-{4-[4-(2-fluoro-4-tetrazol-1-ylphenoxymethyl)thiazol-2-yl]piperidin-1-yl}pyrimidine 1037797-23-1 C20H18F2N8OS
5-fluoro-2-{4-[4-(2-fluoro-4-tetrazol-1-ylphenoxymethyl)thiazol-2-yl]piperidin-1-yl}pyrimidine
—— 3-hydroxy-4-(3-pyridyl-amino)pyridine 1412913-79-1 C10H9N3O
3-hydroxy-4-(3-pyridyl-amino)pyridine
—— bis-(2-benzenesulfonyl-1,1-dioxo-2H-1λ6-naphtho[1,8-cd]isothiazol-5-yl)-methane 118763-84-1 C33H22N2O8S4
bis-(2-benzenesulfonyl-1,1-dioxo-2H-1λ6-naphtho[1,8-cd]isothiazol-5-yl)-methane
—— N'-(2-(2,4-dichlorophenoxy)acetyl)-4-iodobenzohydrazide 1417515-28-6 C15H11Cl2IN2O3
N'-(2-(2,4-dichlorophenoxy)acetyl)-4-iodobenzohydrazide
—— —— 1307759-57-4 C47H73N5O13