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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-{7-[2-(2-hydroxy-1-methyl-ethylamino)-pyridin-4-yl]-2-morpholin-4-yl-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-4-yl}-phenol trifluoroacetate 1007214-95-0 C2HF3O2*C24H28N6O3
3-{7-[2-(2-hydroxy-1-methyl-ethylamino)-pyridin-4-yl]-2-morpholin-4-yl-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-4-yl}-phenol trifluoroacetate
—— {1-[1-(3,5-difluorobenzyl)piperidin-4-yl]-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]azetidin-3-yl}acetonitrile 1334301-17-5 C26H26F2N8
{1-[1-(3,5-difluorobenzyl)piperidin-4-yl]-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]azetidin-3-yl}acetonitrile
—— ethyl 3-[(4,5-diisopropylfuran-2-carbonyl)amino]benzoate 1116091-28-1 C20H25NO4
ethyl 3-[(4,5-diisopropylfuran-2-carbonyl)amino]benzoate
—— 5-(3,4-dimethyl-phenyl)-2-methyl-thiazole-4-carboxylic acid cyclopropylmethyl-[2-(4-hydroxy-3-methoxy-phenyl)-ethyl]-amide 1223584-55-1 C26H30N2O3S
5-(3,4-dimethyl-phenyl)-2-methyl-thiazole-4-carboxylic acid cyclopropylmethyl-[2-(4-hydroxy-3-methoxy-phenyl)-ethyl]-amide
—— N-carbamoylmethyl-3-(2-morpholin-4-yl-7-pyridin-3-yl-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-4-yl)-benzamide trifluoroacetate 1007214-13-2 C2HF3O2*C24H25N7O3
N-carbamoylmethyl-3-(2-morpholin-4-yl-7-pyridin-3-yl-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-4-yl)-benzamide trifluoroacetate
—— methyl (2S,3S,4S,5R)-6-(benzylamino)-4,5-bis(benzyloxy)-2,3-dihydroxy-6-oxohexanoate 1354635-21-4 C28H31NO7
methyl (2S,3S,4S,5R)-6-(benzylamino)-4,5-bis(benzyloxy)-2,3-dihydroxy-6-oxohexanoate
—— 2-[6-fluoro-3-(2,3,6-trifluorobenzyl)imidazo[1,5-a]pyridin-1-yl]-5-(1-methyl-1H-imidazol-5-yl)pyrimidin-4-amine 1337565-32-8 C22H15F4N7
2-[6-fluoro-3-(2,3,6-trifluorobenzyl)imidazo[1,5-a]pyridin-1-yl]-5-(1-methyl-1H-imidazol-5-yl)pyrimidin-4-amine
—— (R)-3-({2-butyl-1-[2'-(1-trityl-1H-tetrazol-5-yl)biphenyl-4-ylmethyl]-1H-imidazole-4-carbonyl}amino)-4-phenylbutyric acid 1206696-93-6 C51H47N7O3
(R)-3-({2-butyl-1-[2'-(1-trityl-1H-tetrazol-5-yl)biphenyl-4-ylmethyl]-1H-imidazole-4-carbonyl}amino)-4-phenylbutyric acid
—— 2-[3-(cyclopropylmethylcarbamoyl)phenyl]-5H-pyrrolo[2,3-b]pyrazine-7-carboxylic acid [(R)-2-(3-cyanoazetidin-1-yl)-1-methyl-2-oxoethyl]amide 1334674-32-6 C25H25N7O3
2-[3-(cyclopropylmethylcarbamoyl)phenyl]-5H-pyrrolo[2,3-b]pyrazine-7-carboxylic acid [(R)-2-(3-cyanoazetidin-1-yl)-1-methyl-2-oxoethyl]amide
—— ethyl 2-(4-fluorophenyl)-6-((2-(methyl(phenyl)amino)ethyl)(methylsulfonyl)amino)-5-phenyl-1-benzofuran-3-carboxylate 1333225-26-5 C33H31FN2O5S
ethyl 2-(4-fluorophenyl)-6-((2-(methyl(phenyl)amino)ethyl)(methylsulfonyl)amino)-5-phenyl-1-benzofuran-3-carboxylate
—— 3-(2-thiazolyl)phenyl 2,3,4-tri-O-acetyl-5-thio-β-D-xylopyranoside 1011720-43-6 C20H21NO7S2
3-(2-thiazolyl)phenyl 2,3,4-tri-O-acetyl-5-thio-β-D-xylopyranoside
—— {1-[1-(3-fluoro-4-isoquinolin-5-ylbenzoyl)piperidin-4-yl]-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]azetidin-3-yl}acetonitrile 1334300-29-6 C35H30FN9O
{1-[1-(3-fluoro-4-isoquinolin-5-ylbenzoyl)piperidin-4-yl]-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]azetidin-3-yl}acetonitrile
—— tert-butyl N-tert-butoxycarbonyl-N-[3-(4-fluoro-1,3-benzoxazol-2-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2-pyridyl]carbamate 1146951-58-7 C28H35BFN3O7
tert-butyl N-tert-butoxycarbonyl-N-[3-(4-fluoro-1,3-benzoxazol-2-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2-pyridyl]carbamate
—— ethyl 2-(4-methoxyphenyl)allyl carbonate 1639790-31-0 C13H16O4
ethyl 2-(4-methoxyphenyl)allyl carbonate
—— —— 1315481-20-9 C8H5F3O2S*C12H35N7P2
—— —— 142838-93-5 C23H25ClN2O3
—— (2S,3E)-2-(iodomethyl)-5-methylhex-3-enyl acetate 1321534-43-3 C10H17IO2
(2S,3E)-2-(iodomethyl)-5-methylhex-3-enyl acetate
—— 2-[6-(3-Fluoropyridin-4-yl)pyridin-2-yl]quinazoline 1376449-85-2 C18H11FN4
2-[6-(3-Fluoropyridin-4-yl)pyridin-2-yl]quinazoline
—— —— 190974-47-1 C62H54N2O8
—— methyl 4-hydroxythieno[3,4-d]pyrimidine-7-carboxylate 1269667-48-2 C8H6N2O3S
methyl 4-hydroxythieno[3,4-d]pyrimidine-7-carboxylate
—— 6-methoxy-4-methyl-8-phthalimido-5-<<3-(trifluoromethyl)benzyl>oxy>quinoline 1-oxide 121963-24-4 C27H19F3N2O5
6-methoxy-4-methyl-8-phthalimido-5-<<3-(trifluoromethyl)benzyl>oxy>quinoline 1-oxide
—— Benzyl 6-benzyl-7-oxo-2,6-diazabicyclo[3.2.1]octane-2-carboxylate 1001857-33-5 C21H22N2O3
Benzyl 6-benzyl-7-oxo-2,6-diazabicyclo[3.2.1]octane-2-carboxylate
—— (6-Hydroxy-4-iodopyridin-2-YL)acetic acid 1393541-74-6 C7H6INO3
(6-Hydroxy-4-iodopyridin-2-YL)acetic acid
—— 6-chloro-2,3-dihydro-1H-pyrrolo[3,4-c]pyridin-1-one 1393555-72-0 C7H5ClN2O
6-chloro-2,3-dihydro-1H-pyrrolo[3,4-c]pyridin-1-one
—— 4,6-Dichloro-1,3-dihydro-2H-pyrrolo[3,2-C]pyridin-2-one 1260672-68-1 C7H4Cl2N2O
4,6-Dichloro-1,3-dihydro-2H-pyrrolo[3,2-C]pyridin-2-one
—— N-(7-methoxy-4-(3-methoxy-4-phenoxyphenylamino)quinazolin-6-yl)-2-(piperidin-4-ylidene)acetamide 1005195-65-2 C29H29N5O4
N-(7-methoxy-4-(3-methoxy-4-phenoxyphenylamino)quinazolin-6-yl)-2-(piperidin-4-ylidene)acetamide
—— (4S,5R)-2-(6-tert-butyl-4-ethoxy-pyridin-3-yl)-4,5-bis-(4-chloro-phenyl)-4,5-dimethyl-4,5-dihydro-imidazole-1-carboxylic acid bis-(2-methoxy-ethyl)-amide 1143522-49-9 C35H44Cl2N4O4
(4S,5R)-2-(6-tert-butyl-4-ethoxy-pyridin-3-yl)-4,5-bis-(4-chloro-phenyl)-4,5-dimethyl-4,5-dihydro-imidazole-1-carboxylic acid bis-(2-methoxy-ethyl)-amide
—— 4-bromo-3-chloropyridin-2(1H)-one 1227511-48-9 C5H3BrClNO
4-bromo-3-chloropyridin-2(1H)-one
—— N-(5-chlorothiazol-2-yl)-3-cyclohexyl-2-(6-methyl-4-(oxazol-2-yl)-2-oxopyridin-1(2H)-yl)propanamide 1036207-90-5 C21H23ClN4O3S
N-(5-chlorothiazol-2-yl)-3-cyclohexyl-2-(6-methyl-4-(oxazol-2-yl)-2-oxopyridin-1(2H)-yl)propanamide
—— (2-benzylpiperazin-1-yl)(2-phenylcyclopropyl)methanone 1144508-05-3 C21H24N2O
(2-benzylpiperazin-1-yl)(2-phenylcyclopropyl)methanone
—— 1-[2-methyl-5-[4-(4-sulfamoylphenyl)piperidine-1-carbonyl]phenyl]-3-propan-2-yl-urea 1034469-41-4 C23H30N4O4S
1-[2-methyl-5-[4-(4-sulfamoylphenyl)piperidine-1-carbonyl]phenyl]-3-propan-2-yl-urea
—— (2-Amino-5-benzylpyridin-3-yl)-[6-(1,4-diazepan-1-yl)pyridin-2-yl]methanone 1042983-45-8 C23H25N5O
(2-Amino-5-benzylpyridin-3-yl)-[6-(1,4-diazepan-1-yl)pyridin-2-yl]methanone
—— (2-Aminopyridin-3-yl)-[6-(pyrrolidin-3-ylamino)-3-(trifluoromethyl)pyridin-2-yl]methanone 1042985-43-2 C16H16F3N5O
(2-Aminopyridin-3-yl)-[6-(pyrrolidin-3-ylamino)-3-(trifluoromethyl)pyridin-2-yl]methanone
—— (2-Aminopyridin-3-yl)-(3-phenyl-6-piperazin-1-ylpyridin-2-yl)methanone 1042985-87-4 C21H21N5O
(2-Aminopyridin-3-yl)-(3-phenyl-6-piperazin-1-ylpyridin-2-yl)methanone
—— (S)-4-[(2-chloro-phenylamino)-methyl]-2,2-dimethyl-oxazolidine-3-carboxylic acid tert-butyl ester 1048351-18-3 C17H25ClN2O3
(S)-4-[(2-chloro-phenylamino)-methyl]-2,2-dimethyl-oxazolidine-3-carboxylic acid tert-butyl ester
—— N-[5-[4-(4-cyanophenyl)piperidine-1-carbonyl]-2-methyl-phenyl]-3-(1,3-dioxoisoindol-2-yl)propane-1-sulfonamide 1035169-74-4 C31H30N4O5S
N-[5-[4-(4-cyanophenyl)piperidine-1-carbonyl]-2-methyl-phenyl]-3-(1,3-dioxoisoindol-2-yl)propane-1-sulfonamide
—— 1-[4-[6-(2-Amino-5-bromopyridine-3-carbonyl)pyridin-2-yl]-1,4-diazepan-1-yl]-2-methylpropan-1-one 1042982-18-2 C20H24BrN5O2
1-[4-[6-(2-Amino-5-bromopyridine-3-carbonyl)pyridin-2-yl]-1,4-diazepan-1-yl]-2-methylpropan-1-one
—— (2-aminopyridin-3-yl)-[3-benzyl-6-[(3S)-3-(2-methylpropyl)piperazin-1-yl]pyridin-2-yl]methanone 1042985-89-6 C26H31N5O
(2-aminopyridin-3-yl)-[3-benzyl-6-[(3S)-3-(2-methylpropyl)piperazin-1-yl]pyridin-2-yl]methanone
—— 3-(2-methanesulfonamidoethyl)-1-[2-methyl-5-[4-[4-(trifluoromethyl)phenyl]piperidine-1-carbonyl]phenyl]urea 1034469-22-1 C24H29F3N4O4S
3-(2-methanesulfonamidoethyl)-1-[2-methyl-5-[4-[4-(trifluoromethyl)phenyl]piperidine-1-carbonyl]phenyl]urea
—— 3-(2-dimethylaminoethyl)-1-[2-methyl-5-[4-[4-(trifluoromethyl)phenyl]piperidine-1-carbonyl]phenyl]urea 1034469-15-2 C25H31F3N4O2
3-(2-dimethylaminoethyl)-1-[2-methyl-5-[4-[4-(trifluoromethyl)phenyl]piperidine-1-carbonyl]phenyl]urea
—— (2-Amino-5-ethylpyridin-3-yl)-[6-(4-methyl-1,4-diazepan-1-yl)pyridin-2-yl]methanone 1042983-07-2 C19H25N5O
(2-Amino-5-ethylpyridin-3-yl)-[6-(4-methyl-1,4-diazepan-1-yl)pyridin-2-yl]methanone
—— 2-(4-hydroxy-1-methyl-2-oxo-6-propyl-1,2-dihydro-1,8-naphthyridine-3-carboxamido)acetic acid 1034130-39-6 C15H17N3O5
2-(4-hydroxy-1-methyl-2-oxo-6-propyl-1,2-dihydro-1,8-naphthyridine-3-carboxamido)acetic acid
—— (S)-4-{[ethyl-(3-oxazol-5-yl-phenyl)-amino]-methyl}-4,5-dihydro-oxazol-2-ylamine 1048348-94-2 C15H18N4O2
(S)-4-{[ethyl-(3-oxazol-5-yl-phenyl)-amino]-methyl}-4,5-dihydro-oxazol-2-ylamine
—— (2-aminopyridin-3-yl)-[3-(difluoromethoxy)-6-[(3S)-3-(2-methylpropyl)piperazin-1-yl]pyridin-2-yl]methanone 1042985-23-8 C20H25F2N5O2
(2-aminopyridin-3-yl)-[3-(difluoromethoxy)-6-[(3S)-3-(2-methylpropyl)piperazin-1-yl]pyridin-2-yl]methanone
—— (3S)-N-[3-(2-cyclopropylpyridin-4-yl)-1H-indazol-5-yl]-3-methoxy-1-[2-[4-(3-methoxy-4-pyrimidin-2-ylphenyl)-3,6-dihydro-2H-pyridin-1-yl]-2-oxoethyl]pyrrolidine-3-carboxamide 1093062-07-7 C39H40N8O4
(3S)-N-[3-(2-cyclopropylpyridin-4-yl)-1H-indazol-5-yl]-3-methoxy-1-[2-[4-(3-methoxy-4-pyrimidin-2-ylphenyl)-3,6-dihydro-2H-pyridin-1-yl]-2-oxoethyl]pyrrolidine-3-carboxamide
—— N-{3-[2,2,2-trifluoro-1-(pyridin-3-yl)ethoxy]quinoxalin-2-yl}cyclopentanesulfonamide 1226504-60-4 C20H19F3N4O3S
N-{3-[2,2,2-trifluoro-1-(pyridin-3-yl)ethoxy]quinoxalin-2-yl}cyclopentanesulfonamide
—— 3-{2-chloro-5-[5-methanesulfonyl-1-(3-morpholin-4-yl-propyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]-phenyl}-N-phenyl-propionamide 1048036-88-9 C29H36ClN5O4S
3-{2-chloro-5-[5-methanesulfonyl-1-(3-morpholin-4-yl-propyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]-phenyl}-N-phenyl-propionamide
—— 4-[(2R)-4-benzyl-1-(2-chloro-4-hydroxyphenyl)piperazin-2-yl]benzonitrile 1097210-81-5 C24H22ClN3O
4-[(2R)-4-benzyl-1-(2-chloro-4-hydroxyphenyl)piperazin-2-yl]benzonitrile
—— 1-[5-[4-(4-cyanophenyl)piperidine-1-carbonyl]-2-methyl-phenyl]-3-[(1S)-1-phenylethyl]urea 1034465-04-7 C29H30N4O2
1-[5-[4-(4-cyanophenyl)piperidine-1-carbonyl]-2-methyl-phenyl]-3-[(1S)-1-phenylethyl]urea
—— (3S)-1-[2-[4-(3-fluorophenyl)-3,6-dihydro-2H-pyridin-1-yl]-2-oxoethyl]-N-[3-(6-fluoropyridin-3-yl)-1H-indazol-5-yl]-3-methoxypyrrolidine-3-carboxamide 1093062-47-5 C31H30F2N6O3
(3S)-1-[2-[4-(3-fluorophenyl)-3,6-dihydro-2H-pyridin-1-yl]-2-oxoethyl]-N-[3-(6-fluoropyridin-3-yl)-1H-indazol-5-yl]-3-methoxypyrrolidine-3-carboxamide