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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-(sec-butylsulfonyl)-8-cyclohexyl-11-methoxy-1a-((3-(methylamino)-8-azabicyclo[3.2.1]oct-8-yl)carbonyl)-1,1a,2,12b-tetrahydrocyclopropa[d]indolo[2,1-a][2]benzazepine-5-carboxamide 1058165-83-5 C39H50N4O5S
N-(sec-butylsulfonyl)-8-cyclohexyl-11-methoxy-1a-((3-(methylamino)-8-azabicyclo[3.2.1]oct-8-yl)carbonyl)-1,1a,2,12b-tetrahydrocyclopropa[d]indolo[2,1-a][2]benzazepine-5-carboxamide
—— 2-[(2-cyclopropylethyl)oxy]-8-(methyloxy)-9-[2-(tetrahydro-2H-pyran-2-yl)ethyl]-9H-purin-6-amine 1050498-00-4 C18H27N5O3
2-[(2-cyclopropylethyl)oxy]-8-(methyloxy)-9-[2-(tetrahydro-2H-pyran-2-yl)ethyl]-9H-purin-6-amine
—— 2-(4-(4-((6-(1H-tetrazol-1-yl)pyridin-3-yloxy)methyl)-2H-1,2,3-triazol-2-yl)piperidin-1-yl)pyrimidine-5-carboxylic acid 1108165-10-1 C19H19N11O3
2-(4-(4-((6-(1H-tetrazol-1-yl)pyridin-3-yloxy)methyl)-2H-1,2,3-triazol-2-yl)piperidin-1-yl)pyrimidine-5-carboxylic acid
—— tert-butyl 2-chloro-4-(6-chloro-8-methoxy-4-oxo-4,5-dihydrothieno[2,3-c]quinolin-9-yl)phenethylcarbamate 1338544-52-7 C25H24Cl2N2O4S
tert-butyl 2-chloro-4-(6-chloro-8-methoxy-4-oxo-4,5-dihydrothieno[2,3-c]quinolin-9-yl)phenethylcarbamate
—— 10-azetidin-1-yl-3-methyl-6,7,8,9-tetrahydro-5H-1,4,7,10a-tetraaza-cyclohepta[f]indene 1228220-29-8 C14H19N5
10-azetidin-1-yl-3-methyl-6,7,8,9-tetrahydro-5H-1,4,7,10a-tetraaza-cyclohepta[f]indene
—— (S)-N-(2-oxopiperidin-3-yl)-2-(trifluoromethyl)benzamide 1352127-87-7 C13H13F3N2O2
(S)-N-(2-oxopiperidin-3-yl)-2-(trifluoromethyl)benzamide
—— US10202379, Reference Example 318 1370240-50-8 C26H27N3O5S
US10202379, Reference Example 318
—— N2-butyl-9-[3-(2,2-dimethyltetrahydro-2H-pyran-4-yl)propyl]-8-(methyloxy)-9H-purine-2,6-diamine 1050497-50-1 C20H34N6O2
N2-butyl-9-[3-(2,2-dimethyltetrahydro-2H-pyran-4-yl)propyl]-8-(methyloxy)-9H-purine-2,6-diamine
—— cycloprop[d]indolo[2,1-a][2]benzazepine-5-carboxamide, 8-cyclohexyl-N-[(dimethylamino)sulfonyl]-1,1a,2,12b-tetrahydro-11-methoxy-1a-(3-oxa-9-azabicyclo[3.3.1]non-9-ylcarbonyl)- 1058166-10-1 C36H44N4O6S
cycloprop[d]indolo[2,1-a][2]benzazepine-5-carboxamide, 8-cyclohexyl-N-[(dimethylamino)sulfonyl]-1,1a,2,12b-tetrahydro-11-methoxy-1a-(3-oxa-9-azabicyclo[3.3.1]non-9-ylcarbonyl)-
—— N-(2,4-ditrifluoromethylphenyl)anthranilic acid 1146634-06-1 C15H9F6NO2
N-(2,4-ditrifluoromethylphenyl)anthranilic acid
—— 5-methoxy-1-[6-[3-methyl-2-[[5-methyl-2-[(3R)-oxan-3-yl]-3,4-dihydro-1H-isoquinolin-6-yl]methoxy]phenyl]pyridin-2-yl]pyrazole-4-carboxylic acid 1579514-54-7 C33H36N4O5
5-methoxy-1-[6-[3-methyl-2-[[5-methyl-2-[(3R)-oxan-3-yl]-3,4-dihydro-1H-isoquinolin-6-yl]methoxy]phenyl]pyridin-2-yl]pyrazole-4-carboxylic acid
—— 4-Cyclopropoxy-3-(trifluoromethyl)benzonitrile 1228582-01-1 C11H8F3NO
4-Cyclopropoxy-3-(trifluoromethyl)benzonitrile
—— (2R,3R,4R,4aR,6R,8aR)-4-(methoxymethoxy)-2-(oxan-2-yloxymethyl)spiro[3,4,4a,7,8,8a-hexahydro-2H-pyrano[3,2-b]pyran-6,2'-oxolane]-3-ol 115369-18-1 C19H32O8
(2R,3R,4R,4aR,6R,8aR)-4-(methoxymethoxy)-2-(oxan-2-yloxymethyl)spiro[3,4,4a,7,8,8a-hexahydro-2H-pyrano[3,2-b]pyran-6,2'-oxolane]-3-ol
—— 4-Methyl-3-[2-oxo-prop-(E)-ylidene]-1-propyl-azetidin-2-one 111390-81-9 C10H15NO2
4-Methyl-3-[2-oxo-prop-(E)-ylidene]-1-propyl-azetidin-2-one
—— 6-morpholinopicolinohydrazide 1338375-35-1 C10H14N4O2
6-morpholinopicolinohydrazide
—— N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-1-isopropyl-6-(4-(4-isopropylpiperazin-1-yl)phenyl)-3-methyl-1H-indole-4-carboxamide 1346572-39-1 C34H43N5O2
N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-1-isopropyl-6-(4-(4-isopropylpiperazin-1-yl)phenyl)-3-methyl-1H-indole-4-carboxamide
—— (4R,5R)-5-ethyl-4-methyl-6-(2-phenyl-benzoxazol-6-yl)-4,5-dihydro-2H-pyridazin-3-one 1346699-92-0 C20H19N3O2
(4R,5R)-5-ethyl-4-methyl-6-(2-phenyl-benzoxazol-6-yl)-4,5-dihydro-2H-pyridazin-3-one
—— 3,5-dimethyl-1-oxo-2-phenyl-1,2-dihydro-isoquinoline-4-carboxylic acid 1075715-27-3 C18H15NO3
3,5-dimethyl-1-oxo-2-phenyl-1,2-dihydro-isoquinoline-4-carboxylic acid
—— 2-[2-amino-1-(3H-1,3-benzothiazol-2-ylidene)-2-oxoethyl]-6-methylpyrimidine-4-carboxylic acid 1219482-35-5 C15H12N4O3S
2-[2-amino-1-(3H-1,3-benzothiazol-2-ylidene)-2-oxoethyl]-6-methylpyrimidine-4-carboxylic acid
—— (1H-imidazol-4-ylmethyl)-isopropyl-(1-phenyl-1H-pyrazol-3-yl)-amine 1020817-85-9 C16H19N5
(1H-imidazol-4-ylmethyl)-isopropyl-(1-phenyl-1H-pyrazol-3-yl)-amine
—— {4-[8-(4-ethyl-phenyl)-6-methoxycarbamoyl-5-oxo-5,8-dihydro-pyrido[2,3-d]pyrimidin-2-ylamino]-phenyl}-acetic acid 1023276-68-7 C25H23N5O5
{4-[8-(4-ethyl-phenyl)-6-methoxycarbamoyl-5-oxo-5,8-dihydro-pyrido[2,3-d]pyrimidin-2-ylamino]-phenyl}-acetic acid
—— N-(1-methylethyl)-5-[2-methyl-8-(4-morpholinyl)imidazo[1,2-b]pyridazin-3-yl]-2-pyridinamine 1298031-23-8 C19H24N6O
N-(1-methylethyl)-5-[2-methyl-8-(4-morpholinyl)imidazo[1,2-b]pyridazin-3-yl]-2-pyridinamine
—— 1-methyl-1H-indazole-3-carboxylic acid (2-{cyclopropylmethyl-[2-methyl-5-(3-trifluoromethyl-phenyl)-thiazole-4-carbonyl]-amino}-ethyl)-amide 1117695-78-9 C27H26F3N5O2S
1-methyl-1H-indazole-3-carboxylic acid (2-{cyclopropylmethyl-[2-methyl-5-(3-trifluoromethyl-phenyl)-thiazole-4-carbonyl]-amino}-ethyl)-amide
—— ((2S,4R)-4-(4-octylphenoxy)pyrrolidin-2-yl)methyl dihydrogen phosphate 1046158-44-4 C19H32NO5P
((2S,4R)-4-(4-octylphenoxy)pyrrolidin-2-yl)methyl dihydrogen phosphate
—— 1-[5-[4-[6-(trifluoromethyl)-1H-benzimidazol-2-yl]phenyl]pyridin-2-yl]piperidine-4-carbonitrile 1388143-86-9 C25H20F3N5
1-[5-[4-[6-(trifluoromethyl)-1H-benzimidazol-2-yl]phenyl]pyridin-2-yl]piperidine-4-carbonitrile
—— 5-isopropyl-2,4-dimethoxy-N-(1-methyl-1H-indol-5-yl)benzamide 1003046-17-0 C21H24N2O3
5-isopropyl-2,4-dimethoxy-N-(1-methyl-1H-indol-5-yl)benzamide
—— (1S,14R)-23-benzyl-17-methoxy-11,23-diazahexacyclo[12.7.4.01,14.03,12.05,10.015,20]pentacosa-3,5,7,9,11,15(20),16,18-octaene 1613036-99-9 C31H30N2O
(1S,14R)-23-benzyl-17-methoxy-11,23-diazahexacyclo[12.7.4.01,14.03,12.05,10.015,20]pentacosa-3,5,7,9,11,15(20),16,18-octaene
—— N-[1-(3,5-dimethylphenyl)-3-trimethylsilyl-2-propinylidene]-4-methylaniline 1140916-17-1 C21H25NSi
N-[1-(3,5-dimethylphenyl)-3-trimethylsilyl-2-propinylidene]-4-methylaniline
—— N-[1-(4-methoxyphenyl)-3-(4-nitrophenylthio)-2-propenylidene]aniline 1140913-91-2 C22H18N2O3S
N-[1-(4-methoxyphenyl)-3-(4-nitrophenylthio)-2-propenylidene]aniline
—— N-[2-(4-methylphenyl)ethenyl]aniline 111383-05-2 C15H15N
N-[2-(4-methylphenyl)ethenyl]aniline
—— [(S)-4-oxo-1-(2,2,2-trifluoro-ethyl)-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-3-yl]-carbamic acid tert-butyl ester 1015085-59-2 C16H20F3N3O3
[(S)-4-oxo-1-(2,2,2-trifluoro-ethyl)-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-3-yl]-carbamic acid tert-butyl ester
—— 6-methyl-4-oxo-1-(tetrahydro-furan-3-yl)-1,4-dihydro-pyridine-3-carboxylic acid 1569651-00-8 C11H13NO4
6-methyl-4-oxo-1-(tetrahydro-furan-3-yl)-1,4-dihydro-pyridine-3-carboxylic acid
—— 1-methyl-1H-indazole-3-carboxylic acid {2-[cyclopropyl-(4'-methyl-biphenyl-2-carbonyl)-amino]-ethyl}-amide 1117695-17-6 C28H28N4O2
1-methyl-1H-indazole-3-carboxylic acid {2-[cyclopropyl-(4'-methyl-biphenyl-2-carbonyl)-amino]-ethyl}-amide
—— 6-{2-[(E)-2-(2-pentyloxy-3-methoxyphenyl)vinyl]-4-oxo-3H-imidazo[4,5-b]pyridin-3-yl}nicotinonitrile 1233449-25-6 C26H25N5O3
6-{2-[(E)-2-(2-pentyloxy-3-methoxyphenyl)vinyl]-4-oxo-3H-imidazo[4,5-b]pyridin-3-yl}nicotinonitrile
—— ethyl 2,2-dimethyl-3-(1-methanesulfonyloxy-2,2-dichloro-3,3,3trifluoropropyl)cyclopropanecarboxylate 117065-02-8 C12H17Cl2F3O5S
ethyl 2,2-dimethyl-3-(1-methanesulfonyloxy-2,2-dichloro-3,3,3trifluoropropyl)cyclopropanecarboxylate
—— 5-Chloro-1-methyl-1H-pyrazole-4-carboxylic acid 2-acetylhydrazide 110763-10-5 C7H9ClN4O2
5-Chloro-1-methyl-1H-pyrazole-4-carboxylic acid 2-acetylhydrazide
—— 5-Acetoxy-7-methoxynaphtho<1,2-b>thiophene 114987-60-9 C15H12O3S
5-Acetoxy-7-methoxynaphtho<1,2-b>thiophene
—— 2-(4-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)-1,4-diazepan-1-yl)nicotinic acid 1227170-71-9 C20H23N3O4
2-(4-((2,3-dihydrobenzo[b][1,4]dioxin-2-yl)methyl)-1,4-diazepan-1-yl)nicotinic acid
—— diethyl 2-(1-(4-(2-(5-((tert-butoxycarbonyl(2-methoxyethyl)amino)methyl)-pyridin-2-yl)thieno[3,2-b]pyridin-7-yloxy)-3-fluorophenylamino)-2,2,2-trifluoroethyl)-malonate 1342834-02-9 C36H40F4N4O8S
diethyl 2-(1-(4-(2-(5-((tert-butoxycarbonyl(2-methoxyethyl)amino)methyl)-pyridin-2-yl)thieno[3,2-b]pyridin-7-yloxy)-3-fluorophenylamino)-2,2,2-trifluoroethyl)-malonate
—— 2-(1-(cyclohexylsulfonyl)-3-(4-(7-(1-methyl-1H-pyrazol-4-yl)imidazo[1,2-c]pyrimidin-5-yl)-1H-pyrazol-1-yl)azetidin-3-yl)acetonitrile 1339889-41-6 C24H27N9O2S
2-(1-(cyclohexylsulfonyl)-3-(4-(7-(1-methyl-1H-pyrazol-4-yl)imidazo[1,2-c]pyrimidin-5-yl)-1H-pyrazol-1-yl)azetidin-3-yl)acetonitrile
—— (3-(2-isobutylthiazol-4-yl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)(4-(thiophen-2-yl)phenyl)methanone 1338374-68-7 C23H23N5OS2
(3-(2-isobutylthiazol-4-yl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)(4-(thiophen-2-yl)phenyl)methanone
—— ethyl 2-(4-(7-azabicyclo[2.2.1]heptan-7-yl)-2-(3-(dimethylamino)prop-1-ynyl)phenylcarbamoyl)-6-cyano-2H-benzo[b][1,4]oxazine-4(3H)-carboxylate 1301756-77-3 C30H33N5O4
ethyl 2-(4-(7-azabicyclo[2.2.1]heptan-7-yl)-2-(3-(dimethylamino)prop-1-ynyl)phenylcarbamoyl)-6-cyano-2H-benzo[b][1,4]oxazine-4(3H)-carboxylate
—— (3-(1-(2-methoxyethyl)-3-phenyl-1H-pyrazol-5-yl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)(4-(thiophen-2-yl)phenyl)methanone 1338374-66-5 C28H26N6O2S
(3-(1-(2-methoxyethyl)-3-phenyl-1H-pyrazol-5-yl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)(4-(thiophen-2-yl)phenyl)methanone
—— N-{1-[4-(p-Fluorophenoxy)butyl]-4-piperidyl}-N-methylamine 149069-31-8 C16H25FN2O
N-{1-[4-(p-Fluorophenoxy)butyl]-4-piperidyl}-N-methylamine
—— N-(2-azidoethyl)-4-propylbenzenesulfonamide 1160749-88-1 C11H16N4O2S
N-(2-azidoethyl)-4-propylbenzenesulfonamide
—— 1-biphenyl-3-yl-3-hydroxy-3-methylbutane-2-sulfonamide 1397770-19-2 C17H21NO3S
1-biphenyl-3-yl-3-hydroxy-3-methylbutane-2-sulfonamide
—— cyclohepta[b]pyrrole-5-carboxylic acid nitrile 105852-69-5 C10H6N2
cyclohepta[b]pyrrole-5-carboxylic acid nitrile
—— 3-[1-(5-tert-butyl-isoxazol-3-ylcarbamoyl)-1-methyl-ethylsulfanylmethyl]-piperidine-1-carboxylic acid tert-butyl ester 1017540-37-2 C22H37N3O4S
3-[1-(5-tert-butyl-isoxazol-3-ylcarbamoyl)-1-methyl-ethylsulfanylmethyl]-piperidine-1-carboxylic acid tert-butyl ester
—— 3-chloro-5-cyano-pyridine-2-carboxylic acid [6-((3R,6R)-5-amino-3,6-dimethyl-6-trifluoromethyl-3,6-dihydro-2H-[1,4]oxazin-3-yl)-pyridin-2-yl]-amide 1387559-84-3 C19H16ClF3N6O2
3-chloro-5-cyano-pyridine-2-carboxylic acid [6-((3R,6R)-5-amino-3,6-dimethyl-6-trifluoromethyl-3,6-dihydro-2H-[1,4]oxazin-3-yl)-pyridin-2-yl]-amide
—— Ethyl 4-[[(3,5-dimethoxy-4-methylbenzoyl)-(3-phenylpropyl)amino]methyl]-1,3-thiazole-2-carboxylate 1282551-78-3 C26H30N2O5S
Ethyl 4-[[(3,5-dimethoxy-4-methylbenzoyl)-(3-phenylpropyl)amino]methyl]-1,3-thiazole-2-carboxylate