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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-(1-Methyl-2-oxo-1,2-dihydropyridin-4-yl)propanoicacid 1784875-09-7 C9H11NO3
3-(1-Methyl-2-oxo-1,2-dihydropyridin-4-yl)propanoicacid
—— 2-(3,4-dichlorophenyl)-4-methyl[1]benzothiopyrano[4,3-c ]pyrazol-3(2 H)-one 128789-98-0 C17H10Cl2N2OS
2-(3,4-dichlorophenyl)-4-methyl[1]benzothiopyrano[4,3-c ]pyrazol-3(2 H)-one
—— (1H-imidazol-4-ylmethyl)-isopropyl-(4-methyl-6-phenyl-pyrimidin-2-yl)-amine 1020817-00-8 C18H21N5
(1H-imidazol-4-ylmethyl)-isopropyl-(4-methyl-6-phenyl-pyrimidin-2-yl)-amine
—— N-[5-[4-[2-(2-chlorophenyl)-4-oxoquinazolin-3-yl]phenyl]-1,3,4-thiadiazol-2-yl]-2-phenylacetamide 1009361-20-9 C30H20ClN5O2S
N-[5-[4-[2-(2-chlorophenyl)-4-oxoquinazolin-3-yl]phenyl]-1,3,4-thiadiazol-2-yl]-2-phenylacetamide
—— —— 1278523-77-5 C54H57NO6
—— N-((1S,4r)-4-((S)-5,5-dimethyl-2-oxo-4-phenyloxazolidin-3-yl)cyclohexyl)benzo[d]thiazole-5-carboxamide 1456506-10-7 C25H27N3O3S
N-((1S,4r)-4-((S)-5,5-dimethyl-2-oxo-4-phenyloxazolidin-3-yl)cyclohexyl)benzo[d]thiazole-5-carboxamide
—— 2-allyl-N-((5-methylfuran-2-yl)methyl)-4-(trifluoromethoxy)aniline 1383957-03-6 C16H16F3NO2
2-allyl-N-((5-methylfuran-2-yl)methyl)-4-(trifluoromethoxy)aniline
—— 2,3-di-O-benzyl-4,6-O-benzylidene-α-D-galactopyranosyl acetate 1454689-81-6 C29H30O7
2,3-di-O-benzyl-4,6-O-benzylidene-α-D-galactopyranosyl acetate
—— trans-4-[(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)amino]cyclohexanol 1388890-07-0 C14H19N3OS
trans-4-[(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)amino]cyclohexanol
—— 4-(4-{4-[3-(2-ethoxyethyl)ureido]-2-fluorophenyl}cyclohexylideneaminooxy)piperidine-1-carboxylic acid isopropyl ester 1393684-66-6 C26H39FN4O5
4-(4-{4-[3-(2-ethoxyethyl)ureido]-2-fluorophenyl}cyclohexylideneaminooxy)piperidine-1-carboxylic acid isopropyl ester
—— 2-cyclobutyl-5-[4-[(1R,2S)-2-[2-(5-methylsulfonylpyridin-2-yl)oxyethyl]cyclopropyl]piperidin-1-yl]-1,3,4-oxadiazole 1402554-35-1 C22H30N4O4S
2-cyclobutyl-5-[4-[(1R,2S)-2-[2-(5-methylsulfonylpyridin-2-yl)oxyethyl]cyclopropyl]piperidin-1-yl]-1,3,4-oxadiazole
—— tert-Butyl-((S)-3-ethyl-heptyloxy)-dimethyl-silane 165334-51-0 C15H34OSi
tert-Butyl-((S)-3-ethyl-heptyloxy)-dimethyl-silane
—— [(2R)-2-aminopropyl](butyl)methylamine 1418293-61-4 C8H20N2
[(2R)-2-aminopropyl](butyl)methylamine
—— [3-chloro-4-(4-chloro-phenoxy)-phenyl]-(1H-imidazol-4-ylmethyl)-isopropyl-amine 1020815-80-8 C19H19Cl2N3O
[3-chloro-4-(4-chloro-phenoxy)-phenyl]-(1H-imidazol-4-ylmethyl)-isopropyl-amine
—— 9α-chloro-11β,17α,21-trihydroxy-16α-methylpregna-1,4-diene-3,20-dione 17-butyrate 21-valerate 103466-76-8 C31H43ClO7
9α-chloro-11β,17α,21-trihydroxy-16α-methylpregna-1,4-diene-3,20-dione 17-butyrate 21-valerate
—— Methyl 5-[3,4-di(4-fluorophenyl)-6-isopropylpyridazin-5-yl]-3(S)-hydroxy-4(E)-pentenoate 124278-75-7 C25H24F2N2O3
Methyl 5-[3,4-di(4-fluorophenyl)-6-isopropylpyridazin-5-yl]-3(S)-hydroxy-4(E)-pentenoate
—— 5'-d(AGGT(Dew)C*GGC)-3' 1218784-60-1 C79H100N33O46P7
5'-d(AGGT(Dew)C*GGC)-3'
—— (4-chloro-pyrimidin-2-yl)-ethyl-(3H-imidazol-4-ylmethyl)-amine 1020816-59-4 C10H12ClN5
(4-chloro-pyrimidin-2-yl)-ethyl-(3H-imidazol-4-ylmethyl)-amine
—— —— 1217889-87-6 C60H76N25O35P5
—— (S)-tert-butyl 1-(4-oxo-3-(1H-pyrazol-3-yl)-3,4-dihydropyrrolo[1,2-f][1,2,4]triazin-2-yl)ethylcarbamate 1403942-98-2 C16H20N6O3
(S)-tert-butyl 1-(4-oxo-3-(1H-pyrazol-3-yl)-3,4-dihydropyrrolo[1,2-f][1,2,4]triazin-2-yl)ethylcarbamate
—— (R)-N-((5-((2-(pyridin-3-yl)phenoxy)methyl)-4,5-dihydroisoxazol-3-yl) methyl)imidazo[1,2-a]pyridine-6-carboxamide 1620291-79-3 C24H21N5O3
(R)-N-((5-((2-(pyridin-3-yl)phenoxy)methyl)-4,5-dihydroisoxazol-3-yl) methyl)imidazo[1,2-a]pyridine-6-carboxamide
—— —— 1229444-18-1 C21H26O3
—— (2-chloro-pyrimidin-4-yl)-ethyl-(3H-imidazol-4-ylmethyl)-amine 1020816-60-7 C10H12ClN5
(2-chloro-pyrimidin-4-yl)-ethyl-(3H-imidazol-4-ylmethyl)-amine
—— 1-(4'-(1-oxyl-3-oxide-4,4,5,5-tetramethylimidazolin-2-yl)biphenyl)-4-(p-(1-oxyl-3-oxide-4,4,5,5-tetramethylimidazolin-2-yl)phenyl)bicyclo[2.2.2]octane 1253571-32-2 C40H48N4O4
1-(4'-(1-oxyl-3-oxide-4,4,5,5-tetramethylimidazolin-2-yl)biphenyl)-4-(p-(1-oxyl-3-oxide-4,4,5,5-tetramethylimidazolin-2-yl)phenyl)bicyclo[2.2.2]octane
—— —— 1214711-82-6 C10H11ClO3
—— 1-(4-bromopyridin-2-yl)-2-fluoroethan-1-one 1404489-43-5 C7H5BrFNO
1-(4-bromopyridin-2-yl)-2-fluoroethan-1-one
—— [(1S,2R,5R,6R,7S,8R,10R)-10-[(2R)-2-hydroxypent-4-ynoyl]oxy-1,5-dimethyl-8-propan-2-yl-11-oxatricyclo[6.2.1.02,6]undecan-7-yl] naphthalene-2-carboxylate 1383567-91-6 C31H36O6
[(1S,2R,5R,6R,7S,8R,10R)-10-[(2R)-2-hydroxypent-4-ynoyl]oxy-1,5-dimethyl-8-propan-2-yl-11-oxatricyclo[6.2.1.02,6]undecan-7-yl] naphthalene-2-carboxylate
—— US10138229, Example 112 1558037-43-6 C22H25N5O3
US10138229, Example 112
—— 2-(2-bromo-4-(3-(4-cyclopropylphenoxy)-2-oxo-2,5-dihydro-1H-pyrrol-1-yl)phenoxy)ethyl methanesulfonate 1574542-07-6 C22H22BrNO6S
2-(2-bromo-4-(3-(4-cyclopropylphenoxy)-2-oxo-2,5-dihydro-1H-pyrrol-1-yl)phenoxy)ethyl methanesulfonate
—— 8-(4-ethyl-phenyl)-2-(1-methanesulfonyl-2,3-dihydro-1H-indol-5-ylamino)-5-oxo-5,8-dihydro-pyrido[2,3-d]pyrimidine-6-carboxylic acid methoxy-amide 1023275-63-9 C26H26N6O5S
8-(4-ethyl-phenyl)-2-(1-methanesulfonyl-2,3-dihydro-1H-indol-5-ylamino)-5-oxo-5,8-dihydro-pyrido[2,3-d]pyrimidine-6-carboxylic acid methoxy-amide
—— 8-indan-5-yl-5-oxo-2-(4-piperidin-2-yl-phenylamino)-5,8-dihydro-pyrido[2,3-d]pyrimidine-6-carboxylic acid methoxy-amide 1023275-29-7 C29H30N6O3
8-indan-5-yl-5-oxo-2-(4-piperidin-2-yl-phenylamino)-5,8-dihydro-pyrido[2,3-d]pyrimidine-6-carboxylic acid methoxy-amide
—— 3-hydroxy-3,4,4-trimethylpentyl p-tolyl sulfone 126665-31-4 C15H24O3S
3-hydroxy-3,4,4-trimethylpentyl p-tolyl sulfone
—— 4-chloro-6-((2-(4-(((2-(tetrahydro-2H-pyran-4-yl)ethyl)amino)methyl)phenyl)pyrrolidin-1-yl)carbonyl)benzene-1,3-diol 1023887-58-2 C25H31ClN2O4
4-chloro-6-((2-(4-(((2-(tetrahydro-2H-pyran-4-yl)ethyl)amino)methyl)phenyl)pyrrolidin-1-yl)carbonyl)benzene-1,3-diol
—— (5-fluoro-2-methoxy-phenyl)-(1H-imidazol-4-ylmethyl)-isopropyl-amine 1020815-33-1 C14H18FN3O
(5-fluoro-2-methoxy-phenyl)-(1H-imidazol-4-ylmethyl)-isopropyl-amine
—— (3H-imidazol-4-ylmethyl)-isopropyl-[3-(2-methoxy-phenoxy)-phenyl]-amine 1020815-82-0 C20H23N3O2
(3H-imidazol-4-ylmethyl)-isopropyl-[3-(2-methoxy-phenoxy)-phenyl]-amine
—— 8-(2,6-dichlorophenyl)-9-[[(3R)-piperidin-3-yl]methyl]-N-[(5-pyridin-2-ylthiophen-2-yl)methyl]purin-2-amine 1021696-63-8 C27H25Cl2N7S
8-(2,6-dichlorophenyl)-9-[[(3R)-piperidin-3-yl]methyl]-N-[(5-pyridin-2-ylthiophen-2-yl)methyl]purin-2-amine
—— (2R,3S,4S,5R)-1,6-Bis-(3,5-dimethoxy-phenyl)-3,4-bis-(2-trimethylsilanyl-ethoxymethoxy)-hexane-2,5-diamine 1054658-78-4 C34H60N2O8Si2
(2R,3S,4S,5R)-1,6-Bis-(3,5-dimethoxy-phenyl)-3,4-bis-(2-trimethylsilanyl-ethoxymethoxy)-hexane-2,5-diamine
—— —— 1422052-87-6 C31H28N2O3
—— —— 1365548-90-8 C36H24BN3O2
—— (10S)-N-(4-methoxyphenyl)-N-methyl-12-oxo-9,10,11,12,13,18-hexahydro-1H-8,4-(metheno)[1 ,7]thiazacyclopentadecino[3,4-b]indole-10(3H)-carboxamide trifluoromethanesulfonate 1620083-91-1 C2HF3O2*C29H29N3O3S
(10S)-N-(4-methoxyphenyl)-N-methyl-12-oxo-9,10,11,12,13,18-hexahydro-1H-8,4-(metheno)[1 ,7]thiazacyclopentadecino[3,4-b]indole-10(3H)-carboxamide trifluoromethanesulfonate
—— N-methyl-N-[(1S)-1-[5-[5-[6-[2-[(1S)-1-[methyl[(2R)-2-phenyl-2-(1-piperidinyl)acetyl]amino]ethyl]-1H-imidazol-5-yl]-1,3,5-hexatriynyl]-2-thienyl]-1H-imidazol-2-yl]ethyl]-α-phenyl-(αR)-1-piperidineacetamide 1380291-84-8 C48H52N8O2S
N-methyl-N-[(1S)-1-[5-[5-[6-[2-[(1S)-1-[methyl[(2R)-2-phenyl-2-(1-piperidinyl)acetyl]amino]ethyl]-1H-imidazol-5-yl]-1,3,5-hexatriynyl]-2-thienyl]-1H-imidazol-2-yl]ethyl]-α-phenyl-(αR)-1-piperidineacetamide
—— N,4,5-Trimethyl-I+/--3-thienyl-2-thiazolemethanamine 1249298-71-2 C11H14N2S2
N,4,5-Trimethyl-I+/--3-thienyl-2-thiazolemethanamine
—— methyl 2-[5-chloro-2-[2-[(2-methylpropan-2-yl)oxycarbonylamino]acetyl]-3,4-dihydro-1H-2,6-naphthyridin-1-yl]acetate 1571146-07-0 C18H24ClN3O5
methyl 2-[5-chloro-2-[2-[(2-methylpropan-2-yl)oxycarbonylamino]acetyl]-3,4-dihydro-1H-2,6-naphthyridin-1-yl]acetate
—— 4-[5-fluoro-4-(4-methoxyphenyl)-2-oxopyridin-1(2H)-yl]-N-hydroxy-2-methyl-2-(methylsulfonyl)butanamide 1398502-28-7 C18H21FN2O6S
4-[5-fluoro-4-(4-methoxyphenyl)-2-oxopyridin-1(2H)-yl]-N-hydroxy-2-methyl-2-(methylsulfonyl)butanamide
—— US10202379, Reference Example 406 1370241-38-5 C24H19F4N3O4
US10202379, Reference Example 406
—— 5-chloro-N-[1-(2-hydroxyphenyl)ethylideneamino]thiophene-2-carboxamide 1360865-30-0 C13H11ClN2O2S
5-chloro-N-[1-(2-hydroxyphenyl)ethylideneamino]thiophene-2-carboxamide
—— 6-{[1-(cyclopropylcarbonyl)azetidin-3-yl]methyl}-5-[4-(1-methyl-1H-pyrazol-5-yl)phenyl]-4,6-diazaspiro[2.4]hept-4-en-7-one 1579512-84-7 C23H25N5O2
6-{[1-(cyclopropylcarbonyl)azetidin-3-yl]methyl}-5-[4-(1-methyl-1H-pyrazol-5-yl)phenyl]-4,6-diazaspiro[2.4]hept-4-en-7-one
—— 2-hydroxyethyl 3-[[3-(1H-indazol-5-ylamino)piperidin-1-yl]methyl]benzoate 1404375-36-5 C22H26N4O3
2-hydroxyethyl 3-[[3-(1H-indazol-5-ylamino)piperidin-1-yl]methyl]benzoate
—— N-[[4-(N-cyano-S-propan-2-ylsulfonimidoyl)phenyl]methyl]-5-[3-(difluoromethyl)phenyl]-6-methyl-1-(2-methylpyrazol-3-yl)-4-oxopyridine-3-carboxamide 1570076-48-0 C29H28F2N6O3S
N-[[4-(N-cyano-S-propan-2-ylsulfonimidoyl)phenyl]methyl]-5-[3-(difluoromethyl)phenyl]-6-methyl-1-(2-methylpyrazol-3-yl)-4-oxopyridine-3-carboxamide
—— (E)-6-(3-oxo-3-(4-((4-(trifluoromethoxy)phenoxy)methyl)-5,6-dihydropyridin-1(2H)-yl)prop-1-en-1-yl)-3,4-dihydro-1,8-naphthyridin-2(1H)-one 1441351-24-1 C24H22F3N3O4
(E)-6-(3-oxo-3-(4-((4-(trifluoromethoxy)phenoxy)methyl)-5,6-dihydropyridin-1(2H)-yl)prop-1-en-1-yl)-3,4-dihydro-1,8-naphthyridin-2(1H)-one