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中文名称 英文名称 CAS号 化学式 结构式图片
—— Boc-Phe-Ser-N3 110338-47-1 C17H23N5O5
Boc-Phe-Ser-N3
—— N-(1-hydroxy-3,4-dihydro-1H-benzo[c][1,2]oxaborinin-7-yl)-2-trifluoromethyl-benzamide 1335094-76-2 C16H13BF3NO4
N-(1-hydroxy-3,4-dihydro-1H-benzo[c][1,2]oxaborinin-7-yl)-2-trifluoromethyl-benzamide
—— 3-((1H-pyrrolo[2,3-b]pyridin-4-yl)ethynyl)-N-phenylaniline 1174297-33-6 C21H15N3
3-((1H-pyrrolo[2,3-b]pyridin-4-yl)ethynyl)-N-phenylaniline
—— (2S,3S)-3-hydroxy-N-((2-octylbenzofuran-5-yl)methyl)pyrrolidine-2-carboxamide 1218816-89-7 C22H32N2O3
(2S,3S)-3-hydroxy-N-((2-octylbenzofuran-5-yl)methyl)pyrrolidine-2-carboxamide
—— 2-chloro-4-[[5-chloro-4-[[(1S)-1,2-dimethyl-3-oxo-1H-isoindol-4-yl]oxy]pyrimidin-2-yl]amino]-5-methoxy-N-[(3R,4S)-3-methoxy-1-methylpiperidin-4-yl]benzamide 1227949-64-5 C29H32Cl2N6O5
2-chloro-4-[[5-chloro-4-[[(1S)-1,2-dimethyl-3-oxo-1H-isoindol-4-yl]oxy]pyrimidin-2-yl]amino]-5-methoxy-N-[(3R,4S)-3-methoxy-1-methylpiperidin-4-yl]benzamide
—— 4-[3-(2-Hydroxy-3,3,5,5-tetramethyl-4,6-dioxocyclohexen-1-yl)-4-methylphenyl]benzaldehyde 1033760-12-1 C24H24O4
4-[3-(2-Hydroxy-3,3,5,5-tetramethyl-4,6-dioxocyclohexen-1-yl)-4-methylphenyl]benzaldehyde
—— 3-[[4-oxo-3-phenyl-6-[6-(trifluoromethyl)-1H-benzimidazol-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]sulfanylmethyl]benzonitrile 1240708-89-7 C29H21F3N6OS
3-[[4-oxo-3-phenyl-6-[6-(trifluoromethyl)-1H-benzimidazol-2-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]sulfanylmethyl]benzonitrile
—— 6-chloro-8-(cyclopropanecarboxamidomethyl)-2-oxo-1,2-dihydroquinoline-3-carboxylic acid 1415593-78-0 C15H13ClN2O4
6-chloro-8-(cyclopropanecarboxamidomethyl)-2-oxo-1,2-dihydroquinoline-3-carboxylic acid
—— 6-chloro-8-{[2-(2,6-difluoro-phenyl)-acetylamino]-methyl}-2-methoxy-quinoline-3-carboxylic acid methyl ester 1415595-44-6 C21H17ClF2N2O4
6-chloro-8-{[2-(2,6-difluoro-phenyl)-acetylamino]-methyl}-2-methoxy-quinoline-3-carboxylic acid methyl ester
—— (S)-2-(2-chloro-5-((5-(((S)-1-(3-isopropylphenyl)ethyl)carbamoyl)-2,3-dimethyl-1H-indol-1-yl)methyl)phenoxy)-3-methylbutanoic acid 1415321-98-0 C34H39ClN2O4
(S)-2-(2-chloro-5-((5-(((S)-1-(3-isopropylphenyl)ethyl)carbamoyl)-2,3-dimethyl-1H-indol-1-yl)methyl)phenoxy)-3-methylbutanoic acid
—— (2R,3R)-4-(2-chlorophenyl)-3-[4-ethyl-3-(3-methyl-5-oxo-4,5-dihydro-pyrazol-1-yl)-benzoylamino]-2-hydroxy-butyric acid 1415482-15-3 C23H24ClN3O5
(2R,3R)-4-(2-chlorophenyl)-3-[4-ethyl-3-(3-methyl-5-oxo-4,5-dihydro-pyrazol-1-yl)-benzoylamino]-2-hydroxy-butyric acid
—— 6-(3-amino-4-chlorophenyl)-N-[(4R)-3,4-dihydro-2H-chromen-4-yl]-2-methylpyrimidin-4-amine 1404106-99-5 C20H19ClN4O
6-(3-amino-4-chlorophenyl)-N-[(4R)-3,4-dihydro-2H-chromen-4-yl]-2-methylpyrimidin-4-amine
—— N-[[2-[(2R,6S)-2,6-dimethyl-4-morpholinyl]-5-(6-methyl-3-pyridinyl)-4-thiazolyl]methyl]-2-fluoro-benzamide 1309443-90-0 C23H25FN4O2S
N-[[2-[(2R,6S)-2,6-dimethyl-4-morpholinyl]-5-(6-methyl-3-pyridinyl)-4-thiazolyl]methyl]-2-fluoro-benzamide
—— N-diethyl-2-amino-6-(1-ethylcarbamoylcyclobutyl)quinazoline-4-carboxamide 1309355-53-0 C20H27N5O2
N-diethyl-2-amino-6-(1-ethylcarbamoylcyclobutyl)quinazoline-4-carboxamide
—— 4-[2-amino-6-ethyl-5-(6-methyl-pyridin-3-ylethynyl)-pyrimidin-4-yl]-2-fluoro-benzoic acid methyl ester 1207351-53-8 C22H19FN4O2
4-[2-amino-6-ethyl-5-(6-methyl-pyridin-3-ylethynyl)-pyrimidin-4-yl]-2-fluoro-benzoic acid methyl ester
—— 2-(3-chloropyridin-2-yl)-N-[4-iodo-2-methyl-6-[[(2S)-1-methylsulfanylpropan-2-yl]carbamoyl]phenyl]-5-[[4-(trifluoromethyl)triazol-1-yl]methyl]pyrazole-3-carboxamide 1339950-40-1 C25H23ClF3IN8O2S
2-(3-chloropyridin-2-yl)-N-[4-iodo-2-methyl-6-[[(2S)-1-methylsulfanylpropan-2-yl]carbamoyl]phenyl]-5-[[4-(trifluoromethyl)triazol-1-yl]methyl]pyrazole-3-carboxamide
—— 5-[4-[(4-chloro-2-fluorophenyl)methoxy]-2-methoxyphenyl]-2-(4-methylphenyl)-1H-imidazole 1239261-34-7 C24H20ClFN2O2
5-[4-[(4-chloro-2-fluorophenyl)methoxy]-2-methoxyphenyl]-2-(4-methylphenyl)-1H-imidazole
—— N-(4-bromo-1-(2-(3-hydroxyoxetan-3-yl)ethyl)-1H-indol-3-yl)-2-adamantane-1-ylacetamide 1415461-37-8 C25H31BrN2O3
N-(4-bromo-1-(2-(3-hydroxyoxetan-3-yl)ethyl)-1H-indol-3-yl)-2-adamantane-1-ylacetamide
—— (R)-tert-butyl 4'-((5-((1-(6-cyclopropylpyridin-3-yl)ethyl)carbamoyl)-2,3-dimethyl-1H-indol-1-yl)methyl)-[1,1'-biphenyl]-2-carboxylate 1415257-51-0 C39H41N3O3
(R)-tert-butyl 4'-((5-((1-(6-cyclopropylpyridin-3-yl)ethyl)carbamoyl)-2,3-dimethyl-1H-indol-1-yl)methyl)-[1,1'-biphenyl]-2-carboxylate
—— 4-chloro-N-(adamantane-1-yl-methyl)-1-(2-(3-hydroxyoxetan-3-yl)ethyl)-1H-indole-3-carboxamide 1415459-94-7 C25H31ClN2O3
4-chloro-N-(adamantane-1-yl-methyl)-1-(2-(3-hydroxyoxetan-3-yl)ethyl)-1H-indole-3-carboxamide
—— 2-Amino-5-[[4-(2,6-difluorophenyl)-5-oxotetrazole-1-carbonyl]-propan-2-ylamino]benzoic acid 1346564-50-8 C18H16F2N6O4
2-Amino-5-[[4-(2,6-difluorophenyl)-5-oxotetrazole-1-carbonyl]-propan-2-ylamino]benzoic acid
—— 2-(1-pyrenyl)-5,5-di(hydroxymethyl)-1,3-dioxane 1234562-92-5 C22H20O4
2-(1-pyrenyl)-5,5-di(hydroxymethyl)-1,3-dioxane
—— N-[2-(tert-butylcarbamoyl)-4-cyano-6-methylphenyl]-2-(3-chloropyridin-2-yl)-5-[(4,5,6,7-tetrachlorobenzotriazol-1-yl)methyl]pyrazole-3-carboxamide 1339949-21-1 C29H22Cl5N9O2
N-[2-(tert-butylcarbamoyl)-4-cyano-6-methylphenyl]-2-(3-chloropyridin-2-yl)-5-[(4,5,6,7-tetrachlorobenzotriazol-1-yl)methyl]pyrazole-3-carboxamide
—— 3-{1-[(4-chlorophenyl)carbonyl]-3-(2,2-dimethylpropanoyl)-6-[(2-methyl-1,3-thiazol-4-yl)methoxy]indolizin-2-yl}-2,2-dimethylpropanoic acid 1215281-77-8 C30H31ClN2O5S
3-{1-[(4-chlorophenyl)carbonyl]-3-(2,2-dimethylpropanoyl)-6-[(2-methyl-1,3-thiazol-4-yl)methoxy]indolizin-2-yl}-2,2-dimethylpropanoic acid
—— 2-[5-[4-Chloro-3-(trifluoromethyl)phenyl]-2-ethylphenyl]-3-hydroxycyclopent-2-en-1-one 1235109-85-9 C20H16ClF3O2
2-[5-[4-Chloro-3-(trifluoromethyl)phenyl]-2-ethylphenyl]-3-hydroxycyclopent-2-en-1-one
—— 5-((4-(benzyloxy)benzyl)(4H-1,2,4-triazol-4-yl)amino)-4'-methoxy-biphenyl-2-carbonitrile 1260389-58-9 C30H25N5O2
5-((4-(benzyloxy)benzyl)(4H-1,2,4-triazol-4-yl)amino)-4'-methoxy-biphenyl-2-carbonitrile
—— N-[4-(5-{[(1S)-1-cyclohexyl-2-(methylamino)-2-oxoethyl]carbamoyl}furan-2-yl)benzyl]-3-methylfuran-2-carboxamide 1227191-98-1 C27H31N3O5
N-[4-(5-{[(1S)-1-cyclohexyl-2-(methylamino)-2-oxoethyl]carbamoyl}furan-2-yl)benzyl]-3-methylfuran-2-carboxamide
—— 5-[1-[[2-[(4-Chlorophenyl)methyl]benzoyl]amino]ethyl]thiophene-2-carboxylic acid 1097195-37-3 C21H18ClNO3S
5-[1-[[2-[(4-Chlorophenyl)methyl]benzoyl]amino]ethyl]thiophene-2-carboxylic acid
—— N-{(1S)-1-[(3-(((cyclopropylsulfonyl)amino)methyl)azetidin-1-yl)carbonyl]-2,2-dimethylpropyl}-1-(4-fluorobenzyl)-1H-indazole-3-carboxamide 1185285-60-2 C28H34FN5O4S
N-{(1S)-1-[(3-(((cyclopropylsulfonyl)amino)methyl)azetidin-1-yl)carbonyl]-2,2-dimethylpropyl}-1-(4-fluorobenzyl)-1H-indazole-3-carboxamide
—— 8-(S)-8-(tert-butyl-dimethyl-silanyloxy)-9-cyclopentyl-6,6-dimethyl-1-(4-trifluoromethyl-phenyl)-1,3,5,6,7,8-hexahydro-furo[3,4-b]quinoline 1186525-78-9 C31H42F3NO2Si
8-(S)-8-(tert-butyl-dimethyl-silanyloxy)-9-cyclopentyl-6,6-dimethyl-1-(4-trifluoromethyl-phenyl)-1,3,5,6,7,8-hexahydro-furo[3,4-b]quinoline
—— Methyl 5-[4-(2,2,2-trifluoroethyl)phenyl]piperidine-3-carboxylate 1256841-41-4 C15H18F3NO2
Methyl 5-[4-(2,2,2-trifluoroethyl)phenyl]piperidine-3-carboxylate
—— 2-[3-[[(5S)-5-methyl-5-[4-(trifluoromethoxy)phenyl]-4H-1,2-oxazol-3-yl]oxy]phenyl]-1,3,4-oxadiazole 1256371-48-8 C19H14F3N3O4
2-[3-[[(5S)-5-methyl-5-[4-(trifluoromethoxy)phenyl]-4H-1,2-oxazol-3-yl]oxy]phenyl]-1,3,4-oxadiazole
—— 1-methyl-3-(4-methylpiperazine-1-yl)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indazole 1471258-73-7 C19H29BN4O2
1-methyl-3-(4-methylpiperazine-1-yl)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indazole
—— 4-methoxy-2-(2-methoxy-acetyl)-3-oxo-butyric acid methyl ester 1107660-06-9 C9H14O6
4-methoxy-2-(2-methoxy-acetyl)-3-oxo-butyric acid methyl ester
—— (R)-2-chloro-5-((3-ethylisoxazol-5-yl)methyl)-5,6,6a,7,9,10-hexahydro-[1,4]oxazino[3,4-h]pteridine 1394071-14-7 C15H18ClN5O2
(R)-2-chloro-5-((3-ethylisoxazol-5-yl)methyl)-5,6,6a,7,9,10-hexahydro-[1,4]oxazino[3,4-h]pteridine
—— (2S)-5-(ethanimidoylamino)-2-[({2-oxo-1-[3-(trifluoromethyl)benzyl]-1,2-dihydropyridin-3-yl}carbonyl)amino]pentanoic acid trifluoroacetate 1037089-98-7 C2HF3O2*C21H23F3N4O4
(2S)-5-(ethanimidoylamino)-2-[({2-oxo-1-[3-(trifluoromethyl)benzyl]-1,2-dihydropyridin-3-yl}carbonyl)amino]pentanoic acid trifluoroacetate
—— 1-(4-fluorobenzyl)-N-[(1S)-1-{[2-(hydroxymethyl)morpholin-4-yl]carbonyl}-2,2-dimethylpropyl]-1H-indazole-3-carboxamide 1185284-60-9 C26H31FN4O4
1-(4-fluorobenzyl)-N-[(1S)-1-{[2-(hydroxymethyl)morpholin-4-yl]carbonyl}-2,2-dimethylpropyl]-1H-indazole-3-carboxamide
—— 5-[5-bromo-2-(4-fluorophenyl)-1,3-oxazol-4-yl]pyridine-2-carbonitrile 1207747-33-8 C15H7BrFN3O
5-[5-bromo-2-(4-fluorophenyl)-1,3-oxazol-4-yl]pyridine-2-carbonitrile
—— Ethyl 1-[[4-[[(4-cyanophenyl)sulfonyl-(pyridin-2-ylmethyl)amino]methyl]benzoyl]amino]cyclopropane-1-carboxylate 1191067-59-0 C27H26N4O5S
Ethyl 1-[[4-[[(4-cyanophenyl)sulfonyl-(pyridin-2-ylmethyl)amino]methyl]benzoyl]amino]cyclopropane-1-carboxylate
—— tert-butyl (2S, 6S)-2,6-dimethyl-4-[2-(5-methanesulfonylindol-1-ylmethyl)pyridin-5-yl]-3,6-dihydro-2H-pyridine-1-carboxylate 1268816-08-5 C27H33N3O4S
tert-butyl (2S, 6S)-2,6-dimethyl-4-[2-(5-methanesulfonylindol-1-ylmethyl)pyridin-5-yl]-3,6-dihydro-2H-pyridine-1-carboxylate
—— 2-(2-bromo-3-oxo-propyl)-5-fluoro-benzoic acid methyl ester 1202897-50-4 C11H10BrFO3
2-(2-bromo-3-oxo-propyl)-5-fluoro-benzoic acid methyl ester
—— 1-(4-fluorobenzyl)-N-[(1S)-1-({[(1-hydroxycyclopropyl)methyl]amino}carbonyl)-2,2-dimethylpropyl]-1H-indazole-3-carboxamide 1185283-62-8 C25H29FN4O3
1-(4-fluorobenzyl)-N-[(1S)-1-({[(1-hydroxycyclopropyl)methyl]amino}carbonyl)-2,2-dimethylpropyl]-1H-indazole-3-carboxamide
—— 2-tert-butyl-9-oxo-1,4,9,10-tetrahydro-2H-3-oxa-10-azaphenanthrene-6-carboxylic acid amide 1520891-24-0 C17H20N2O3
2-tert-butyl-9-oxo-1,4,9,10-tetrahydro-2H-3-oxa-10-azaphenanthrene-6-carboxylic acid amide
—— 6-chloro-4-(3-chloro-phenyl)-2-dimethylamino-quinoline-3-carboxylic acid tert-butyl ester 1433903-88-8 C22H22Cl2N2O2
6-chloro-4-(3-chloro-phenyl)-2-dimethylamino-quinoline-3-carboxylic acid tert-butyl ester
—— 4-(3-(tert-butyldimethylsilyloxy)propoxy)-2,6-difluorobenzaldehyde 1239964-38-5 C16H24F2O3Si
4-(3-(tert-butyldimethylsilyloxy)propoxy)-2,6-difluorobenzaldehyde
—— 2-Amino[1,3]thiazolo[5,4-b]pyridin-5-ol dihydrobromide 1174229-36-7 C6H7Br2N3OS
2-Amino[1,3]thiazolo[5,4-b]pyridin-5-ol dihydrobromide
—— (R)-6-(((3-((4-(5-((2-((tert-butyldimethylsilyl)oxy)-2-(5-hydroxy-3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazin-8-yl)ethyl)amino)pent-1-yn-1-yl)-3-methylphenyl)carbamoyl)phenyl)sulfonyl))-4-((3-methoxyphenyl)amino)-8-methylquinoline-3-carboxamide 1346655-91-1 C53H58N6O9SSi
(R)-6-(((3-((4-(5-((2-((tert-butyldimethylsilyl)oxy)-2-(5-hydroxy-3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazin-8-yl)ethyl)amino)pent-1-yn-1-yl)-3-methylphenyl)carbamoyl)phenyl)sulfonyl))-4-((3-methoxyphenyl)amino)-8-methylquinoline-3-carboxamide
—— (2Z,4Z) methyl 2,4-difluoro-12-(2-quinolinyloxy)dodeca-2,4-dienoate 127425-93-8 C22H25F2NO3
(2Z,4Z) methyl 2,4-difluoro-12-(2-quinolinyloxy)dodeca-2,4-dienoate
—— [5-(4-chloro-3-trifluoromethyl-benzyl)-4-methyl-thiazol-2-yl]-[3-methoxy-4-(4-methyl-imidazol-1-yl)-phenyl]-amine 1077629-50-5 C23H20ClF3N4OS
[5-(4-chloro-3-trifluoromethyl-benzyl)-4-methyl-thiazol-2-yl]-[3-methoxy-4-(4-methyl-imidazol-1-yl)-phenyl]-amine
—— 5-butyl-1-(5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl)-N-((4-methyl-4H-1,2,4-triazol-3-yl)methyl)-1H-pyrazole-4-carboxamide 1019253-24-7 C21H24N8OS
5-butyl-1-(5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl)-N-((4-methyl-4H-1,2,4-triazol-3-yl)methyl)-1H-pyrazole-4-carboxamide