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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-<1-(6,7-Dimethoxy-4-quinazolinyl)-4-piperidinyl>-3-(2-acetoxyethyl)-2-imidazolidinone 130819-16-8 C22H29N5O5
1-<1-(6,7-Dimethoxy-4-quinazolinyl)-4-piperidinyl>-3-(2-acetoxyethyl)-2-imidazolidinone
—— 5-[N-(4,5-dimethoxy-2-ethoxycarbonylphenyl)carbamoylmethyl]-2-isopropylidenehydrazonothiazolidin-4-one 163108-30-3 C19H24N4O6S
5-[N-(4,5-dimethoxy-2-ethoxycarbonylphenyl)carbamoylmethyl]-2-isopropylidenehydrazonothiazolidin-4-one
—— 4-chloro-N-(pyridin-2-ylmethyl)-N-[2-[4-(2H-tetrazol-5-yl)phenyl]ethyl]benzenesulfonamide 1191068-89-9 C21H19ClN6O2S
4-chloro-N-(pyridin-2-ylmethyl)-N-[2-[4-(2H-tetrazol-5-yl)phenyl]ethyl]benzenesulfonamide
—— N-hydroxy-4-phenyl-2-(thiophen-2-yl)thiazole-5-carboxamide 1148158-32-0 C14H10N2O2S2
N-hydroxy-4-phenyl-2-(thiophen-2-yl)thiazole-5-carboxamide
—— 4-[1-[4-(oxan-4-ylamino)-5-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]piperidin-4-yl]-N-[(1,3,5-trimethylpyrazol-4-yl)methyl]benzamide 1146359-79-6 C30H39N7O3S
4-[1-[4-(oxan-4-ylamino)-5-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]piperidin-4-yl]-N-[(1,3,5-trimethylpyrazol-4-yl)methyl]benzamide
—— tert-butyl 6,6,6-trifluoro-4-methyl-2-{4-[(5-oxo-2-phenyl-5,6-dihydro-4H-1,3,4-oxadiazin-4-yl)methyl]phenyl}hexanoate 1192040-24-6 C27H31F3N2O4
tert-butyl 6,6,6-trifluoro-4-methyl-2-{4-[(5-oxo-2-phenyl-5,6-dihydro-4H-1,3,4-oxadiazin-4-yl)methyl]phenyl}hexanoate
—— 3-[5-[[(5S)-5-[4-(trifluoromethoxy)phenyl]-4,5-dihydro-1,2-oxazol-3-yl]oxy]pyridin-2-yl]propanoic acid 1256369-38-6 C18H15F3N2O5
3-[5-[[(5S)-5-[4-(trifluoromethoxy)phenyl]-4,5-dihydro-1,2-oxazol-3-yl]oxy]pyridin-2-yl]propanoic acid
—— 3-[[(5R)-5-(4-phenoxyphenyl)-4,5-dihydro-1,2-oxazol-3-yl]oxy]benzoic acid 1256369-73-9 C22H17NO5
3-[[(5R)-5-(4-phenoxyphenyl)-4,5-dihydro-1,2-oxazol-3-yl]oxy]benzoic acid
—— (2R,6R,11S)-6,11-dimethyl-8-pyridin-3-yl-1,2,5,6-tetrahydro-4H-2,6-methano-benzo[d]azocine-3-carboxylic acid tert-butyl ester 1155855-34-7 C24H30N2O2
(2R,6R,11S)-6,11-dimethyl-8-pyridin-3-yl-1,2,5,6-tetrahydro-4H-2,6-methano-benzo[d]azocine-3-carboxylic acid tert-butyl ester
—— N-[(1S)-1-carbamoyl-2,2-dimethylpropyl]-1-(4-cyano-2-fluorobenzyl)-7-fluoro-1H-indazole-3-carboxamide 1185285-83-9 C22H21F2N5O2
N-[(1S)-1-carbamoyl-2,2-dimethylpropyl]-1-(4-cyano-2-fluorobenzyl)-7-fluoro-1H-indazole-3-carboxamide
—— 5-fluoro-4-[(2-methoxyphenyl)methylcarbamoylamino]-2-oxo-N-pentylpyrimidine-1-carboxamide 1265170-16-8 C19H24FN5O4
5-fluoro-4-[(2-methoxyphenyl)methylcarbamoylamino]-2-oxo-N-pentylpyrimidine-1-carboxamide
—— N-(2,5-dichlorophenyl)iminodiacetic acid 1190891-83-8 C10H9Cl2NO4
N-(2,5-dichlorophenyl)iminodiacetic acid
—— (4R,5S)-4-methyl-5-(4-phenoxyphenyl)-3-pyridin-3-yloxy-4,5-dihydro-1,2-oxazole 1256368-62-3 C21H18N2O3
(4R,5S)-4-methyl-5-(4-phenoxyphenyl)-3-pyridin-3-yloxy-4,5-dihydro-1,2-oxazole
—— N-(2-(4,5-dimethylpyridin-3-yl)-1-(m-tolyl)ethyl)-4,5-dihydrooxazol-2-amine 1173171-87-3 C19H23N3O
N-(2-(4,5-dimethylpyridin-3-yl)-1-(m-tolyl)ethyl)-4,5-dihydrooxazol-2-amine
—— N-benzyl-4-chloro-N-[1-[4-(2H-tetrazol-5-yl)phenyl]ethyl]benzenesulfonamide 1191071-08-5 C22H20ClN5O2S
N-benzyl-4-chloro-N-[1-[4-(2H-tetrazol-5-yl)phenyl]ethyl]benzenesulfonamide
—— 1-(4-cyano-2-fluorobenzyl)-N-[(1S)-2,2-dimethyl-1-{[2-(methylsulfonyl)ethyl]carbamoyl}propyl]-7-fluoro-1H-indazole-3-carboxamide 1185285-85-1 C25H27F2N5O4S
1-(4-cyano-2-fluorobenzyl)-N-[(1S)-2,2-dimethyl-1-{[2-(methylsulfonyl)ethyl]carbamoyl}propyl]-7-fluoro-1H-indazole-3-carboxamide
—— (S)-1-[(2R,6S)-6,11,11-trimethyl-1,2,5,6-tetrahydro-4H-2,6-methano-benzo[d]azocine-3-carbonyl]-piperidine-3-carboxylic acid ethyl ester 1181262-63-4 C24H34N2O3
(S)-1-[(2R,6S)-6,11,11-trimethyl-1,2,5,6-tetrahydro-4H-2,6-methano-benzo[d]azocine-3-carbonyl]-piperidine-3-carboxylic acid ethyl ester
—— 10-(3-(1H-pyrazol-1-yl)propylamino)-8-amino-9-fluoro-7-oxo-2,7-dihydrospiro[[1,4]oxazino[2,3,4-ij]quinoline-3,1'-cyclopropane]-6-carbonitrile 1132814-14-2 C20H19FN6O2
10-(3-(1H-pyrazol-1-yl)propylamino)-8-amino-9-fluoro-7-oxo-2,7-dihydrospiro[[1,4]oxazino[2,3,4-ij]quinoline-3,1'-cyclopropane]-6-carbonitrile
—— 1-chloracetyl-4-(4-tert-butyl-phenyl)-piperazine 1163268-93-6 C16H23ClN2O
1-chloracetyl-4-(4-tert-butyl-phenyl)-piperazine
—— US10202379, Reference Example 509 1370242-41-3 C25H24FN3O3S
US10202379, Reference Example 509
—— 1-(Nα-(3-(α,α-Dimethylbenzyl)benzenesulphonyl)-(S)-arginyl)-piperidine-4-acetic acid 154938-57-5 C28H39N5O5S
1-(Nα-(3-(α,α-Dimethylbenzyl)benzenesulphonyl)-(S)-arginyl)-piperidine-4-acetic acid
—— methyl 6-(benzyloxy)-5-oxo-1-(thiazol-2-ylmethyl)-1,5-dihydroimidazo[1,2-a]pyrimidine-7-carboxylate 1202898-32-5 C19H16N4O4S
methyl 6-(benzyloxy)-5-oxo-1-(thiazol-2-ylmethyl)-1,5-dihydroimidazo[1,2-a]pyrimidine-7-carboxylate
—— 3-(3-fluorophenylsulfonamido)-N-[2,4,6-trimethyl-3-(morpholin-4-yl)phenyl]thiophene-2-carboxamide 1138340-91-6 C24H26FN3O4S2
3-(3-fluorophenylsulfonamido)-N-[2,4,6-trimethyl-3-(morpholin-4-yl)phenyl]thiophene-2-carboxamide
—— 4-Amino-5-fluoro-1-thiophen-2-ylsulfonylpyrimidin-2-one 1263302-42-6 C8H6FN3O3S2
4-Amino-5-fluoro-1-thiophen-2-ylsulfonylpyrimidin-2-one
—— N-hydroxy-6-(quinoline-8-carbonyl)-4,5,6,7-tetrahydrothieno[2,3-c]pyridine-2-carboxamide 1259287-08-5 C18H15N3O3S
N-hydroxy-6-(quinoline-8-carbonyl)-4,5,6,7-tetrahydrothieno[2,3-c]pyridine-2-carboxamide
—— 13-(4-Fluoranthen-3-ylphenyl)pentacyclo[10.7.1.02,7.08,20.014,19]icosa-1(20),2,4,6,8,10,12,14,16,18-decaene 1080632-75-2 C42H24
13-(4-Fluoranthen-3-ylphenyl)pentacyclo[10.7.1.02,7.08,20.014,19]icosa-1(20),2,4,6,8,10,12,14,16,18-decaene
—— 1-adamantyl N,N-dibenzylcarbamate 1145659-64-8 C25H29NO2
1-adamantyl N,N-dibenzylcarbamate
—— tert-butyl 3-[3-(benzylamino)-5-fluorophenyl]-propanoate 1192040-05-3 C20H24FNO2
tert-butyl 3-[3-(benzylamino)-5-fluorophenyl]-propanoate
—— 4-(9-cyclohexyl-8-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoic acid 1137206-15-5 C22H27N5O4
4-(9-cyclohexyl-8-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoic acid
—— 5-fluoro-4-[(2-methoxyphenyl)methylcarbamoylamino]-2-oxo-N-propan-2-ylpyrimidine-1-carboxamide 1265170-12-4 C17H20FN5O4
5-fluoro-4-[(2-methoxyphenyl)methylcarbamoylamino]-2-oxo-N-propan-2-ylpyrimidine-1-carboxamide
—— 8-(4-fluorophenyl)-N-[(2-fluorophenyl)methyl]-9-(2-piperidin-4-ylethyl)purin-2-amine 1021696-15-0 C25H26F2N6
8-(4-fluorophenyl)-N-[(2-fluorophenyl)methyl]-9-(2-piperidin-4-ylethyl)purin-2-amine
—— 8-(2-chlorophenyl)-N-[(3-fluorophenyl)methyl]-9-(2-piperidin-4-ylethyl)purin-2-amine 1021694-74-5 C25H26ClFN6
8-(2-chlorophenyl)-N-[(3-fluorophenyl)methyl]-9-(2-piperidin-4-ylethyl)purin-2-amine
—— N-(2-(5-tert-butyloxazol-2-yl)phenyl)-4-(ethyl(2-methoxyethyl)amino)-6-phenylpicolinamide 1148121-13-4 C30H34N4O3
N-(2-(5-tert-butyloxazol-2-yl)phenyl)-4-(ethyl(2-methoxyethyl)amino)-6-phenylpicolinamide
—— (2-Chlorophenyl)methyl 4-amino-5-fluoro-2-oxopyrimidine-1-carboxylate 1263295-40-4 C12H9ClFN3O3
(2-Chlorophenyl)methyl 4-amino-5-fluoro-2-oxopyrimidine-1-carboxylate
—— 2-[(5-chloro-1-benzofuran-2-yl)carbonyl]-N-hydroxy-2,3,4,5-tetrahydro-1H-2-benzazepine-7-carboxamide 1259297-62-5 C20H17ClN2O4
2-[(5-chloro-1-benzofuran-2-yl)carbonyl]-N-hydroxy-2,3,4,5-tetrahydro-1H-2-benzazepine-7-carboxamide
—— 8,10-dimethoxy-1-thiophen-3-yl-5,6-dihydropyrrolo[2,1-a]isoquinoline-3-carboxylic acid tert-butylmethylamide 1177017-06-9 C24H28N2O3S
8,10-dimethoxy-1-thiophen-3-yl-5,6-dihydropyrrolo[2,1-a]isoquinoline-3-carboxylic acid tert-butylmethylamide
—— methyl (1R,3S)-3-[(cyclopentyl{4-[(5-oxo-2-phenyl-5,6-dihydro-4H-1,3,4-oxadiazin-4-yl)methyl]phenyl}-acetyl)amino]cyclopentanecarboxylate 1191413-80-5 C30H35N3O5
methyl (1R,3S)-3-[(cyclopentyl{4-[(5-oxo-2-phenyl-5,6-dihydro-4H-1,3,4-oxadiazin-4-yl)methyl]phenyl}-acetyl)amino]cyclopentanecarboxylate
—— —— 1415632-24-4 C25H33N3O5
—— —— 1425792-88-6 C66H81N2O4P2Y
—— 4-((1-methyl-1H-indol-5-yl)sulfonyl)-6-(2-methylpyridin-4-yl)-3,4-dihydro-2H-benzo[b][1,4]oxazine 1401774-76-2 C23H21N3O3S
4-((1-methyl-1H-indol-5-yl)sulfonyl)-6-(2-methylpyridin-4-yl)-3,4-dihydro-2H-benzo[b][1,4]oxazine
—— tert-butyl 4-[2-(2-fluoro-4-methanesulfonylphenoxymethyl)pyridin-5-yl]piperidine-1-carboxylate 1206967-81-8 C23H29FN2O5S
tert-butyl 4-[2-(2-fluoro-4-methanesulfonylphenoxymethyl)pyridin-5-yl]piperidine-1-carboxylate
—— —— 19635-42-8 C16H17Cl4N2OPS
—— ethyl (3S)-{6-fluoro-3-[ethyl-(4-nitrobenzenesulfonyl)-amino]-1,2,3,4-tetrahydro-9H-carbazol-9-yl}-acetate 1007204-14-9 C24H26FN3O6S
ethyl (3S)-{6-fluoro-3-[ethyl-(4-nitrobenzenesulfonyl)-amino]-1,2,3,4-tetrahydro-9H-carbazol-9-yl}-acetate
—— 6-Methyl-4-oxo-9-[1-phenylamino-meth-(Z)-ylidene]-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidine-3-carbonitrile 101478-36-8 C17H16N4O
6-Methyl-4-oxo-9-[1-phenylamino-meth-(Z)-ylidene]-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidine-3-carbonitrile
—— (1R,2S)-1-((3aR,5R,6S,6aR)-6-Hydroxy-2,2-dimethyl-tetrahydro-furo[2,3-d][1,3]dioxol-5-yl)-2-phenyl-ethane-1,2-diol 183371-84-8 C15H20O6
(1R,2S)-1-((3aR,5R,6S,6aR)-6-Hydroxy-2,2-dimethyl-tetrahydro-furo[2,3-d][1,3]dioxol-5-yl)-2-phenyl-ethane-1,2-diol
—— (2-phenoxybenzoato)triphenyltin 136661-09-1 C31H24O3Sn
(2-phenoxybenzoato)triphenyltin
—— (3R,5S)-7-chloro-3,5-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepine 1345731-82-9 C11H14ClNO
(3R,5S)-7-chloro-3,5-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
—— 2-(2-Methoxy-benzyl)-3H-imidazo[4,5-b]pyridine 142590-54-3 C14H13N3O
2-(2-Methoxy-benzyl)-3H-imidazo[4,5-b]pyridine
—— 3-[({3-[5-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-3-yl]propanoyl}amino)methyl]benzoic acid 1353542-48-9 C27H24FN3O4
3-[({3-[5-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-3-yl]propanoyl}amino)methyl]benzoic acid
—— —— 1429661-32-4 C19H26FNO4