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—— (5(S)-(((5-chloropyridin-2-yl)amino)methyl)-6-azaspiro[2.5]octan-6-yl)(2-(pyrimidin-2-yl)phenyl)methanone 1262395-97-0 C24H23ClFN5O
(5(S)-(((5-chloropyridin-2-yl)amino)methyl)-6-azaspiro[2.5]octan-6-yl)(2-(pyrimidin-2-yl)phenyl)methanone
—— 2-[[3-(3,4-difluorophenyl)-3,3-difluoropropyl]sulfanyl]-N-[(4-fluorophenyl)methyl]pyridine-3-carboxylic acid amide 1242642-90-5 C22H17F5N2OS
2-[[3-(3,4-difluorophenyl)-3,3-difluoropropyl]sulfanyl]-N-[(4-fluorophenyl)methyl]pyridine-3-carboxylic acid amide
—— (3R,4R,5R)-5-(Hydroxymethyl)-1-(4-pyridinylmethyl)-3,4-piperidinediol 1347751-17-0 C12H18N2O3
(3R,4R,5R)-5-(Hydroxymethyl)-1-(4-pyridinylmethyl)-3,4-piperidinediol
—— 5-(4-chloro-phenyl)-6-(2-pyridin-2-yl-ethyl)-nicotinic acid 1018783-18-0 C19H15ClN2O2
5-(4-chloro-phenyl)-6-(2-pyridin-2-yl-ethyl)-nicotinic acid
—— 2-[(6,7-dichloroquinazolin-4-yl)amino]-1-[(3R)-3-[[(2S)-2,6-diphenylthian-4-yl]amino]pyrrolidin-1-yl]ethanone 1028062-70-5 C31H31Cl2N5OS
2-[(6,7-dichloroquinazolin-4-yl)amino]-1-[(3R)-3-[[(2S)-2,6-diphenylthian-4-yl]amino]pyrrolidin-1-yl]ethanone
—— (S)-4-(3-amino-piperidin-1-yl)-6-methoxymethyl-pyrimidin-2-ylamine 1046450-28-5 C11H19N5O
(S)-4-(3-amino-piperidin-1-yl)-6-methoxymethyl-pyrimidin-2-ylamine
—— 3,4-dichloro-N-[2-oxo-2-[3-(4-pyrimidin-2-ylpiperidin-1-yl)pyrrolidin-1-yl]ethyl]benzamide 1027771-81-8 C22H25Cl2N5O2
3,4-dichloro-N-[2-oxo-2-[3-(4-pyrimidin-2-ylpiperidin-1-yl)pyrrolidin-1-yl]ethyl]benzamide
—— N-(bicyclo[2.2.1]heptan-2-yl)-N-(1H-pyrazol-5-yl)-3-p-tolylpropanamide 1374762-37-4 C20H25N3O
N-(bicyclo[2.2.1]heptan-2-yl)-N-(1H-pyrazol-5-yl)-3-p-tolylpropanamide
—— (3S,4R)-4-(tert-butyldimethylsilyloxy)-7-(5-(3-phenyl-4-(trifluoromethyl)isoxazol-5-yl)-1,2,4-oxadiazol-3-yl)chroman-3-amine 1374445-27-8 C27H29F3N4O4Si
(3S,4R)-4-(tert-butyldimethylsilyloxy)-7-(5-(3-phenyl-4-(trifluoromethyl)isoxazol-5-yl)-1,2,4-oxadiazol-3-yl)chroman-3-amine
—— 6-(4-(dimethylcarbamoyl)phenylamino)-4-(pyrimidin-4-ylmethylamino)nicotinamide 1374213-16-7 C20H21N7O2
6-(4-(dimethylcarbamoyl)phenylamino)-4-(pyrimidin-4-ylmethylamino)nicotinamide
—— (R)-N-(5-bromo-6-fluoropyridin-2-yl)-4H-1'-azaspiro[oxazole-5,3'-bicyclo[2.2.2]octan]-2-amine 1346215-69-7 C14H16BrFN4O
(R)-N-(5-bromo-6-fluoropyridin-2-yl)-4H-1'-azaspiro[oxazole-5,3'-bicyclo[2.2.2]octan]-2-amine
—— N-(5-chloro-3-fluoropyridin-2-yl)-2-((2-chloro-6-fluorophenyl)amino)-7,7-dimethyl-7,8-dihydro-1H-benzofuro[4,5-d]imidazole-5-carboxamide 1374297-21-8 C23H17Cl2F2N5O2
N-(5-chloro-3-fluoropyridin-2-yl)-2-((2-chloro-6-fluorophenyl)amino)-7,7-dimethyl-7,8-dihydro-1H-benzofuro[4,5-d]imidazole-5-carboxamide
—— 2-[2-methoxy-4-[3-(4-methoxyphenyl)-3-oxoprop-1-enyl]phenoxy]acetic acid 1373337-14-4 C19H18O6
2-[2-methoxy-4-[3-(4-methoxyphenyl)-3-oxoprop-1-enyl]phenoxy]acetic acid
—— 7-Cyano-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxylic acid 1030019-30-7 C7H3N5O2
7-Cyano-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxylic acid
—— 4-cyclopentyloxy-5-difluoromethoxy-2-hydroxymethylpyridine 166742-56-9 C12H15F2NO3
4-cyclopentyloxy-5-difluoromethoxy-2-hydroxymethylpyridine
—— (1R)-1-[(3R)-2,2-dioxido-1-phenyl-3,4-dihydro-1H-2,1-benzothiazin-3-yl]-3-(methylamino)propan-1-ol 1033628-55-5 C18H22N2O3S
(1R)-1-[(3R)-2,2-dioxido-1-phenyl-3,4-dihydro-1H-2,1-benzothiazin-3-yl]-3-(methylamino)propan-1-ol
—— 1-Amino-3-(2-methyl-6-prop-2-enylphenoxy)propan-2-ol 1008456-35-6 C13H19NO2
1-Amino-3-(2-methyl-6-prop-2-enylphenoxy)propan-2-ol
—— 5-Tert-butylpiperazin-2-one 1509510-94-4 C8H16N2O
5-Tert-butylpiperazin-2-one
—— [3-(naphthalen-2-ylmethylamino)pyrrolidin-1-yl]-[3-(trifluoromethyl)-7,8-dihydro-5H-1,6-naphthyridin-6-yl]methanone 1027770-69-9 C25H25F3N4O
[3-(naphthalen-2-ylmethylamino)pyrrolidin-1-yl]-[3-(trifluoromethyl)-7,8-dihydro-5H-1,6-naphthyridin-6-yl]methanone
—— 4-(benzo[b]thiophen-7-ylmethylamino)-6-(4-((3,3-dimethylureido)methyl)phenylamino)nicotinamide 1374213-72-5 C25H26N6O2S
4-(benzo[b]thiophen-7-ylmethylamino)-6-(4-((3,3-dimethylureido)methyl)phenylamino)nicotinamide
—— 4-((1H-indol-4-yl)methylamino)-6-(4-(trifluoromethoxy)phenylamino)nicotinamide 1374213-39-4 C22H18F3N5O2
4-((1H-indol-4-yl)methylamino)-6-(4-(trifluoromethoxy)phenylamino)nicotinamide
—— 5-(hydroxymethyl)-6-(2,2,2-trifluoroethoxy)nicotinic acid 1373863-88-7 C9H8F3NO4
5-(hydroxymethyl)-6-(2,2,2-trifluoroethoxy)nicotinic acid
—— 1H-Indene, 1-chloro-2,3-dihydro-5,6,7-trimethoxy- 1082562-98-8 C12H15ClO3
1H-Indene, 1-chloro-2,3-dihydro-5,6,7-trimethoxy-
—— 1-(3-chloro-1-(pyridin-3-yl)-1H-pyrazol-4-yl)imidazolidin-2-one 1374314-47-2 C11H10ClN5O
1-(3-chloro-1-(pyridin-3-yl)-1H-pyrazol-4-yl)imidazolidin-2-one
—— 5-((R)-2-(2-ethyl-5-fluoropyridin-3-yl)pyrrolidin-1-yl)-N-((1S,3S)-3-hydroxycyclopentyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide 1260844-68-5 C23H27FN6O2
5-((R)-2-(2-ethyl-5-fluoropyridin-3-yl)pyrrolidin-1-yl)-N-((1S,3S)-3-hydroxycyclopentyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 3-{4-chloro-3-[2-(4-methoxy-phenyl)-ethyl]-phenyl}-5-methanesulfonyl-1-(3-morpholin-4-yl-propyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine 1049808-21-0 C29H37ClN4O4S
3-{4-chloro-3-[2-(4-methoxy-phenyl)-ethyl]-phenyl}-5-methanesulfonyl-1-(3-morpholin-4-yl-propyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine
—— tert-butyl N-[3-[2-[(2S,3R)-3-hydroxybutan-2-yl]oxyphenyl]propyl]carbamate 1047665-45-1 C18H29NO4
tert-butyl N-[3-[2-[(2S,3R)-3-hydroxybutan-2-yl]oxyphenyl]propyl]carbamate
—— 3,4-dichloro-N-[1-oxo-1-[3-(4-phenylpiperidin-1-yl)pyrrolidin-1-yl]propan-2-yl]benzamide 1027772-39-9 C25H29Cl2N3O2
3,4-dichloro-N-[1-oxo-1-[3-(4-phenylpiperidin-1-yl)pyrrolidin-1-yl]propan-2-yl]benzamide
—— 5-ethyl-N-[5-(ethylcarbamoyl)-2-methylphenyl]-3-methyl-4-oxo-1,6-dihydropyrrolo[3,4-b]pyrrole-2-carboxamide 1026765-53-6 C20H24N4O3
5-ethyl-N-[5-(ethylcarbamoyl)-2-methylphenyl]-3-methyl-4-oxo-1,6-dihydropyrrolo[3,4-b]pyrrole-2-carboxamide
—— 4-(dibenzo[b,f][1,4]oxazepin-10(11H)-yl)-N-hydroxybenzamide 1024009-99-1 C20H16N2O3
4-(dibenzo[b,f][1,4]oxazepin-10(11H)-yl)-N-hydroxybenzamide
—— 3-(4-{2-chloro-5-[5-methanesulfonyl-1-(3-morpholin-4-yl-propyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]-phenylethynyl}-phenyl)-propionic acid 1049807-16-0 C31H35ClN4O5S
3-(4-{2-chloro-5-[5-methanesulfonyl-1-(3-morpholin-4-yl-propyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]-phenylethynyl}-phenyl)-propionic acid
—— N-[2-[3-[4-(2-amino-1,3-benzothiazol-4-yl)-3,6-dihydro-2H-pyridin-1-yl]pyrrolidin-1-yl]-2-oxoethyl]-3,4-dichlorobenzamide 1027771-80-7 C25H25Cl2N5O2S
N-[2-[3-[4-(2-amino-1,3-benzothiazol-4-yl)-3,6-dihydro-2H-pyridin-1-yl]pyrrolidin-1-yl]-2-oxoethyl]-3,4-dichlorobenzamide
—— N-hydroxy-2-(4-((11-oxodibenzo[b,f][1,4]oxazepin-10(11H)-yl)methyl)phenyl)acetamide 1024009-61-7 C22H18N2O4
N-hydroxy-2-(4-((11-oxodibenzo[b,f][1,4]oxazepin-10(11H)-yl)methyl)phenyl)acetamide
—— 2-[2-Oxo-2-[3-(4-phenylpiperidin-1-yl)pyrrolidin-1-yl]ethyl]-3,4-dihydroisoquinolin-1-one 1027772-42-4 C26H31N3O2
2-[2-Oxo-2-[3-(4-phenylpiperidin-1-yl)pyrrolidin-1-yl]ethyl]-3,4-dihydroisoquinolin-1-one
—— 5-(2-(piperidin-1-yl)ethoxy)-1H-pyrrolo[2,3-b]pyridine 1029053-04-0 C14H19N3O
5-(2-(piperidin-1-yl)ethoxy)-1H-pyrrolo[2,3-b]pyridine
—— 12-(2-hydroxy-2-(4-(trifluoromethyl)phenyl)acetamido)dodecanoic acid 1033777-61-5 C21H30F3NO4
12-(2-hydroxy-2-(4-(trifluoromethyl)phenyl)acetamido)dodecanoic acid
—— 4-(1-carboxy-cyclobutylcarbamoyl)-2-pyridin-4-yl-thiazolidine-3-carboxylic acid benzyl ester 1029799-62-9 C22H23N3O5S
4-(1-carboxy-cyclobutylcarbamoyl)-2-pyridin-4-yl-thiazolidine-3-carboxylic acid benzyl ester
—— (Z)-6-(5H-dibenzo[b,f]azepin-5-yl)-N-hydroxyhexanamide 1024009-27-5 C20H22N2O2
(Z)-6-(5H-dibenzo[b,f]azepin-5-yl)-N-hydroxyhexanamide
—— N-{3-[2-chloro-5-(5-methanesulfonyl-1-{3-[4-(2-oxo-pyrrolidin-1-yl)-piperidin-1-yl]-propyl}-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl)-phenyl]-propyl}-3-nitro-benzenesulfonamide 1049808-91-4 C34H44ClN7O7S2
N-{3-[2-chloro-5-(5-methanesulfonyl-1-{3-[4-(2-oxo-pyrrolidin-1-yl)-piperidin-1-yl]-propyl}-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl)-phenyl]-propyl}-3-nitro-benzenesulfonamide
—— 5-(4-chlorophenyl)-N-(5-(cyclobutylcarbamoyl)-2-methylphenyl)thiophene-2-carboxamide 1026767-03-2 C23H21ClN2O2S
5-(4-chlorophenyl)-N-(5-(cyclobutylcarbamoyl)-2-methylphenyl)thiophene-2-carboxamide
—— N-(5-(cyclopropylcarbamoyl)-2-methylphenyl)-5-(4-(methylsulfonamido)phenyl)thiophene-2-carboxamide 1026766-64-2 C23H23N3O4S2
N-(5-(cyclopropylcarbamoyl)-2-methylphenyl)-5-(4-(methylsulfonamido)phenyl)thiophene-2-carboxamide
—— (2S,4R)-4-[(4-bromo-2-fluorophenyl)methoxy]-N-[(3-chlorophenyl)methyl]-1-[(2R)-2-(methanesulfonamido)-4-piperidin-4-ylbutanoyl]pyrrolidine-2-carboxamide 1039361-45-9 C29H37BrClFN4O5S
(2S,4R)-4-[(4-bromo-2-fluorophenyl)methoxy]-N-[(3-chlorophenyl)methyl]-1-[(2R)-2-(methanesulfonamido)-4-piperidin-4-ylbutanoyl]pyrrolidine-2-carboxamide
—— N-[5-[4-chloro-1-(1,3-thiazol-2-yl)-3,6-dihydro-2H-pyridin-5-yl]pyridin-2-yl]-2,4-difluorobenzamide 1028699-56-0 C20H15ClF2N4OS
N-[5-[4-chloro-1-(1,3-thiazol-2-yl)-3,6-dihydro-2H-pyridin-5-yl]pyridin-2-yl]-2,4-difluorobenzamide
—— 4-(5-chloro-2-pyridyloxy)indole 111110-73-7 C13H9ClN2O
4-(5-chloro-2-pyridyloxy)indole
—— (3R)-7-({2-chloro-5-[5-(methylsulfonyl)-1-(3-morpholin-4-ylpropyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]phenyl}ethynyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide 1049810-50-5 C32H37ClN6O4S
(3R)-7-({2-chloro-5-[5-(methylsulfonyl)-1-(3-morpholin-4-ylpropyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]phenyl}ethynyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
—— [4-(5-iodo-2-pyridyl)piperazino]-2,5-dichlorophenylmethanone 1029360-09-5 C16H14Cl2IN3O
[4-(5-iodo-2-pyridyl)piperazino]-2,5-dichlorophenylmethanone
—— 2-(2-tert-butylpyrimidin-5-yl)-3-[2-(4-methoxyphenyl)ethyl]-1-methylimidazolidin-4-one 1162341-73-2 C21H28N4O2
2-(2-tert-butylpyrimidin-5-yl)-3-[2-(4-methoxyphenyl)ethyl]-1-methylimidazolidin-4-one
—— N-[4-[5-[3,5-bis(trifluoromethyl)phenyl]-5-trifluoromethyl-4,5-dihydroisoxazol-3-yl]-2-chlorophenyl]methyl-N-ethyl-2-(ethylsulfonyl)acetamide 1132700-86-7 C25H22ClF9N2O4S
N-[4-[5-[3,5-bis(trifluoromethyl)phenyl]-5-trifluoromethyl-4,5-dihydroisoxazol-3-yl]-2-chlorophenyl]methyl-N-ethyl-2-(ethylsulfonyl)acetamide
—— 3-[(3S)-1-(2,5-difluorophenyl)-6-fluoro-2,2-dioxido-3,4-dihydro-1H-2,1-benzothiazin-3-yl]-N-methylpropan-1-amine 1033627-21-2 C18H19F3N2O2S
3-[(3S)-1-(2,5-difluorophenyl)-6-fluoro-2,2-dioxido-3,4-dihydro-1H-2,1-benzothiazin-3-yl]-N-methylpropan-1-amine
—— 1-(4-hydroxyphenyl)-2-[2-(3-methoxyphenyl)pyridin-4-yl]ethane-1,2-dione 1035266-13-7 C20H15NO4
1-(4-hydroxyphenyl)-2-[2-(3-methoxyphenyl)pyridin-4-yl]ethane-1,2-dione