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中文名称 英文名称 CAS号 化学式 结构式图片
—— pyridin-4-carboxylic acid (26-difluorophenyl)amide 1220348-99-1 C12H8F2N2O
pyridin-4-carboxylic acid (26-difluorophenyl)amide
—— US10266493, Example 2K 1352792-82-5 C17H19NO2S
US10266493, Example 2K
—— 2-(4-fluorophenyl)-5-(2-(4-hydroxyphenethoxy)-5-(isobutylcarbamoyl)phenyl)-N-methylbenzofuran-3-carboxamide 1217337-05-7 C35H33FN2O5
2-(4-fluorophenyl)-5-(2-(4-hydroxyphenethoxy)-5-(isobutylcarbamoyl)phenyl)-N-methylbenzofuran-3-carboxamide
—— 8-(2-chloro-5-methoxy-3,6-dimethyl-phenyl)-quinoxaline-5-carboxylic acid [5-(4-ethyl-piperazin-1-ylmethyl)-pyridin-2-yl]-amide 1197330-90-7 C30H33ClN6O2
8-(2-chloro-5-methoxy-3,6-dimethyl-phenyl)-quinoxaline-5-carboxylic acid [5-(4-ethyl-piperazin-1-ylmethyl)-pyridin-2-yl]-amide
—— 3-[4-{[(3R)-3-aminopyrrolidin-1-yl]sulfonyl}-2-(3-hydroxy-2,2-dimethylpropyl)-1-oxo-1,2-dihydroisoquinolin-6-yl]-N-cyclopropyl-5-fluoro-4-methylbenzamide 1220228-86-3 C29H35FN4O5S
3-[4-{[(3R)-3-aminopyrrolidin-1-yl]sulfonyl}-2-(3-hydroxy-2,2-dimethylpropyl)-1-oxo-1,2-dihydroisoquinolin-6-yl]-N-cyclopropyl-5-fluoro-4-methylbenzamide
—— 4-tert-butyl-N-(5-chloro-2-(4-chloro-1H-pyrazol-1-yl)pyridin-3-yl)benzenesulfonamide 1094758-15-2 C18H18Cl2N4O2S
4-tert-butyl-N-(5-chloro-2-(4-chloro-1H-pyrazol-1-yl)pyridin-3-yl)benzenesulfonamide
—— 4-(2-(4-(trifluoromethyl)phenyl)quinazolin-4-yl)morpholine 1093983-08-4 C19H16F3N3O
4-(2-(4-(trifluoromethyl)phenyl)quinazolin-4-yl)morpholine
—— 6-methyl-imidazo[2,1-b]thiazole-5-carboxylic acid [(S)-1-(2-cyclopropyl-5-m-tolyl-thiazole-4-carbonyl)-piperidin-2-ylmethyl]amide 1083280-53-8 C27H29N5O2S2
6-methyl-imidazo[2,1-b]thiazole-5-carboxylic acid [(S)-1-(2-cyclopropyl-5-m-tolyl-thiazole-4-carbonyl)-piperidin-2-ylmethyl]amide
—— —— 1067245-10-6 C13H11N3
—— [1-(4-chloro-3,5-diethoxy-benzyl)-piperidin-4-yl]-(4-phenyl-oxazol-2-yl)-amine 1092464-83-9 C25H30ClN3O3
[1-(4-chloro-3,5-diethoxy-benzyl)-piperidin-4-yl]-(4-phenyl-oxazol-2-yl)-amine
—— 6-{4-[(2-aminoethyl)amino]-2-methylphenyl}-4-(1H-indazol-5-yl)pyrimidin-2(1H)-one 1086626-11-0 C20H20N6O
6-{4-[(2-aminoethyl)amino]-2-methylphenyl}-4-(1H-indazol-5-yl)pyrimidin-2(1H)-one
—— 1-(1,3-Benzodioxol-5-ylmethyl)-3-[4-(4-methylimidazol-1-yl)phenyl]urea 1079170-42-5 C19H18N4O3
1-(1,3-Benzodioxol-5-ylmethyl)-3-[4-(4-methylimidazol-1-yl)phenyl]urea
—— N-((1R,2R)-1-(2,3-dihydrobenzo[β][1,4]dioxin-6-yl)-1-hydroxy-3-(pyrrolidin-1-yl)propan-2-yl)biphenyl-4-carboxamide 1092465-34-3 C28H30N2O4
N-((1R,2R)-1-(2,3-dihydrobenzo[β][1,4]dioxin-6-yl)-1-hydroxy-3-(pyrrolidin-1-yl)propan-2-yl)biphenyl-4-carboxamide
—— 2-(2,7-diaza-spiro[3.5]non-2-ylmethyl)-5-(5-fluoro-1H-indol-4-yl)-7-morpholin-4-yl-thiazolo[5,4-d]pyrimidine 1093075-30-9 C25H28FN7OS
2-(2,7-diaza-spiro[3.5]non-2-ylmethyl)-5-(5-fluoro-1H-indol-4-yl)-7-morpholin-4-yl-thiazolo[5,4-d]pyrimidine
—— 2-{(8'-chloro-2'-oxo-2',3'-dihydro-1'H-spiro[cyclopentane-1,4'-quinazolin]-5'-yl)oxy}-3-fluorobenzoic acid 1086424-20-5 C19H16ClFN2O4
2-{(8'-chloro-2'-oxo-2',3'-dihydro-1'H-spiro[cyclopentane-1,4'-quinazolin]-5'-yl)oxy}-3-fluorobenzoic acid
—— methyl N-[4-[3-(5-chloroindol-1-yl)propanoylamino]phenyl]sulfonylcarbamate 1086445-20-6 C19H18ClN3O5S
methyl N-[4-[3-(5-chloroindol-1-yl)propanoylamino]phenyl]sulfonylcarbamate
—— β-naphthylamine dithiocarbamate 102828-95-5 C11H9NS2
β-naphthylamine dithiocarbamate
—— —— 145758-48-1 C16H12F2O2
—— —— 1412452-62-0 C18H28N2O6
—— —— 183255-81-4 C17H16O6SW
—— 2-Carboxy-benzoyl-D-phenylalanin 101399-64-8 C17H15NO5
2-Carboxy-benzoyl-D-phenylalanin
—— 1-(2-O-acetylnaphthyl)-2,3,4-tri-O-acetyl-β-D-xylopyranoside 1155676-58-6 C23H24O10
1-(2-O-acetylnaphthyl)-2,3,4-tri-O-acetyl-β-D-xylopyranoside
—— 2-methoxy-2-methylindeno<1,2,3-cd>pyreno<4,5-d>-1,3-dioxole 102434-58-2 C25H18O3
2-methoxy-2-methylindeno<1,2,3-cd>pyreno<4,5-d>-1,3-dioxole
—— —— 1186603-50-8 C20H19NO3
—— 1,2,3,4,4a,4bα,5,6,7,8,10,10aα-Dodecahydro-2β,4aβ,8,8-tetramethyl-phenanthren-2α-carboxaldehyd 1910-13-0 C19H30O
1,2,3,4,4a,4bα,5,6,7,8,10,10aα-Dodecahydro-2β,4aβ,8,8-tetramethyl-phenanthren-2α-carboxaldehyd
—— 4-{[(2-chlorophenyl)imino]methyl-N-(p-methoxyphenyl)-N-phenyl}benzenamine 105276-33-3 C26H21ClN2O
4-{[(2-chlorophenyl)imino]methyl-N-(p-methoxyphenyl)-N-phenyl}benzenamine
—— (R)-2-((S)-1,2-Bis-benzyloxy-ethyl)-but-3-ene-1,2-diol 153096-81-2 C20H24O4
(R)-2-((S)-1,2-Bis-benzyloxy-ethyl)-but-3-ene-1,2-diol
—— (Z)-3-Isopropylamino-2-pentafluorobenzoyl-acrylic acid ethyl ester 119877-52-0 C15H14F5NO3
(Z)-3-Isopropylamino-2-pentafluorobenzoyl-acrylic acid ethyl ester
—— 6,7,8-Trifluoro-1-(4-fluoro-phenyl)-5-(4-methyl-piperazin-1-yl)-4-oxo-1,4-dihydro-quinoline-3-carboxylic acid ethyl ester 113846-25-6 C23H21F4N3O3
6,7,8-Trifluoro-1-(4-fluoro-phenyl)-5-(4-methyl-piperazin-1-yl)-4-oxo-1,4-dihydro-quinoline-3-carboxylic acid ethyl ester
—— —— 117985-27-0 C13H8FeO5S
—— (1S,4aR,8aS,10aR)-1,4a-Dimethyl-6-oxo-tetradecahydro-phenanthrene-1-carboxylic acid methyl ester 19954-86-0 C18H28O3
(1S,4aR,8aS,10aR)-1,4a-Dimethyl-6-oxo-tetradecahydro-phenanthrene-1-carboxylic acid methyl ester
—— —— 1160587-17-6 C9H12F4
—— 3-(perfluorohexyl)pyridazine 136949-46-7 C10H3F13N2
3-(perfluorohexyl)pyridazine
—— 4-(Morpholino)-3-(3',4'-dihydro-1'-isoquinolyl)-8-methoxyquinoline 104386-22-3 C23H23N3O2
4-(Morpholino)-3-(3',4'-dihydro-1'-isoquinolyl)-8-methoxyquinoline
—— 2-(4-fluorophenyl)-5-[3-[(3-hydroxyphenyl)carbamoyl]phenyl]-N-methyl-1-benzofuran-3-carboxamide 1217334-98-9 C29H21FN2O4
2-(4-fluorophenyl)-5-[3-[(3-hydroxyphenyl)carbamoyl]phenyl]-N-methyl-1-benzofuran-3-carboxamide
—— (S)-pyrrolidine-1,2-dicarboxylic acid 2-amide 1-({5-[2-(1-d3-methyl-cyclobutyl)-pyridin-4-yl]-thiazol-2-yl}-amide) 1217486-88-8 C19H23N5O2S
(S)-pyrrolidine-1,2-dicarboxylic acid 2-amide 1-({5-[2-(1-d3-methyl-cyclobutyl)-pyridin-4-yl]-thiazol-2-yl}-amide)
—— 2-aminocarbonylamino-5-[5-fluoro-2-[2-(4-hydroxypiperidin-1-yl)ethyloxy]phenyl]pyrrole-3-carboxamide 1052080-25-7 C19H24FN5O4
2-aminocarbonylamino-5-[5-fluoro-2-[2-(4-hydroxypiperidin-1-yl)ethyloxy]phenyl]pyrrole-3-carboxamide
—— tert-butyl [(3,5-dichloro-phenylsulphonyl)-(1-imidazo[1,2-a]pyrazin-6-yl-1H-indol-5-yl)-amino]-acetate 1049025-06-0 C26H23Cl2N5O4S
tert-butyl [(3,5-dichloro-phenylsulphonyl)-(1-imidazo[1,2-a]pyrazin-6-yl-1H-indol-5-yl)-amino]-acetate
—— 4-fluoro-N-{3-[3-(4-methyl-benzo[b]thiophen-3-ylmethyl)-2-oxo-2,3-dihydro-benzimidazol-1-yl]-hexanoyl}-benzenesulfonamide 1090895-66-1 C29H28FN3O4S2
4-fluoro-N-{3-[3-(4-methyl-benzo[b]thiophen-3-ylmethyl)-2-oxo-2,3-dihydro-benzimidazol-1-yl]-hexanoyl}-benzenesulfonamide
—— 1-{(R)-2-[2-(1H-indazol-3-yl)-thiazol-4-yl]-piperidin-1-yl}-2-phenoxy-ethanone 1089729-51-0 C23H22N4O2S
1-{(R)-2-[2-(1H-indazol-3-yl)-thiazol-4-yl]-piperidin-1-yl}-2-phenoxy-ethanone
—— 4-methoxyphenyl 4-(4-(3,5-dichloropyridin-4-ylamino)-7,8-dihydropyrimido[5,4-b][1,4]oxazepin-9(6H)-yl)piperidine-1-carboxylate 1079052-90-6 C25H26Cl2N6O4
4-methoxyphenyl 4-(4-(3,5-dichloropyridin-4-ylamino)-7,8-dihydropyrimido[5,4-b][1,4]oxazepin-9(6H)-yl)piperidine-1-carboxylate
—— (S)-N-(3,3-dimethyl-1-(methylamino)-1-oxobutan-2-yl)-3-(thiophen-3-yl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-1-carboxamide 1094085-45-6 C18H25N5O2S
(S)-N-(3,3-dimethyl-1-(methylamino)-1-oxobutan-2-yl)-3-(thiophen-3-yl)-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-1-carboxamide
—— 7-{6-[2-(7-fluoro-2,4-dimethyl-1H-indol-3-yl)ethylamino]pyrimidin-4-ylamino}-4-methylchromen-2-one 1093165-53-7 C26H24FN5O2
7-{6-[2-(7-fluoro-2,4-dimethyl-1H-indol-3-yl)ethylamino]pyrimidin-4-ylamino}-4-methylchromen-2-one
—— 3-(4-bromobenzyl)-6-(2-cyano-2-phenylbutyl)-3-(4-methylpent-3-en-1-yl)-3-azoniabicyclo[3.1.0]hexane bromide 1065523-51-4 Br*C29H36BrN2
3-(4-bromobenzyl)-6-(2-cyano-2-phenylbutyl)-3-(4-methylpent-3-en-1-yl)-3-azoniabicyclo[3.1.0]hexane bromide
—— 4-methyl-4H-furo[3,2-b]pyrrole-5-carboxylic acid {(S)-1-[2-cyclopropyl-5-(4-fluoro-phenyl)-thiazole-4-carbonyl]-piperidin-2-ylmethyl}amide 1083280-43-6 C27H27FN4O3S
4-methyl-4H-furo[3,2-b]pyrrole-5-carboxylic acid {(S)-1-[2-cyclopropyl-5-(4-fluoro-phenyl)-thiazole-4-carbonyl]-piperidin-2-ylmethyl}amide
—— (R)-N-{(S)-1-[4-(4-cyano-phenylamino)-piperidine-1-carbonyl]-2,2-dimethyl-propyl}-2-cyclopentylmethyl-3-(formyl-hydroxy-amino)-propionamide 1091682-54-0 C28H41N5O4
(R)-N-{(S)-1-[4-(4-cyano-phenylamino)-piperidine-1-carbonyl]-2,2-dimethyl-propyl}-2-cyclopentylmethyl-3-(formyl-hydroxy-amino)-propionamide
—— methyl N-[4-[[(2R)-2-(6-chloro-7-methyl-3,4-dihydro-2H-quinolin-1-yl)propanoyl]amino]phenyl]sulfonylcarbamate 1086444-92-9 C21H24ClN3O5S
methyl N-[4-[[(2R)-2-(6-chloro-7-methyl-3,4-dihydro-2H-quinolin-1-yl)propanoyl]amino]phenyl]sulfonylcarbamate
—— (R)-2-(4-acetylpiperazin-1-yl)-4-(1-(4-ethoxy-2-fluorophenyl)ethylamino)-6-isopropyl-5H-pyrrolo[3,4-d]pyrimidin-7(6H)-one 1079657-26-3 C25H33FN6O3
(R)-2-(4-acetylpiperazin-1-yl)-4-(1-(4-ethoxy-2-fluorophenyl)ethylamino)-6-isopropyl-5H-pyrrolo[3,4-d]pyrimidin-7(6H)-one
—— 8-(3,5-diisopropoxy-benzyl)-2-phenyl-1,3,8-triaza-spiro[4.5]dec-1-en-4-one 1084926-11-3 C26H33N3O3
8-(3,5-diisopropoxy-benzyl)-2-phenyl-1,3,8-triaza-spiro[4.5]dec-1-en-4-one
—— 2-[1,1-dioxo-2-(4-methylsulfanylphenyl)-2,3-dihydro-1H-benzo[d]isothiazol-3-yl]-N-hydroxyacetamide 1087007-50-8 C16H16N2O4S2
2-[1,1-dioxo-2-(4-methylsulfanylphenyl)-2,3-dihydro-1H-benzo[d]isothiazol-3-yl]-N-hydroxyacetamide