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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-{(1R)-1-[3-(2-methylpyrimidin-4-yl)azetidin-1-yl]ethyl}-1-(tetrahydro-2H-pyran-4-yl)-1,5-dihydro-4H-pyrazolo[3,4-d]pyrimidin-4-one 1236858-41-5 C20H25N7O2
6-{(1R)-1-[3-(2-methylpyrimidin-4-yl)azetidin-1-yl]ethyl}-1-(tetrahydro-2H-pyran-4-yl)-1,5-dihydro-4H-pyrazolo[3,4-d]pyrimidin-4-one
—— 2-methoxy-4-(7-pyridin-4-yl-imidazo[1,2-b]pyridazin-3-yl)-phenol 1107654-72-7 C18H14N4O2
2-methoxy-4-(7-pyridin-4-yl-imidazo[1,2-b]pyridazin-3-yl)-phenol
—— 5-((R)-2-((S)-2-amino-5-(bis(2-aminoethyl)amino)-5-oxopentanamido)-4-(4-(trifluoromethyl)phenyl)butanamido)-2,3-difluorophenylboronic acid hydrochloride 1393476-16-8 C26H34BF5N6O5*ClH
5-((R)-2-((S)-2-amino-5-(bis(2-aminoethyl)amino)-5-oxopentanamido)-4-(4-(trifluoromethyl)phenyl)butanamido)-2,3-difluorophenylboronic acid hydrochloride
—— —— 1421964-46-6 C28H25F3N6O3
—— 1-(trans-3-((5-(trifluoromethyl)pyrimidin-2-yl)amino)cyclobutyl)-3,3-dimethyl-1H-pyrrolo[2,3-b]pyridin-2(3H)-one 1452552-10-1 C18H18F3N5O
1-(trans-3-((5-(trifluoromethyl)pyrimidin-2-yl)amino)cyclobutyl)-3,3-dimethyl-1H-pyrrolo[2,3-b]pyridin-2(3H)-one
—— —— 1381951-06-9 C19H19BrCl2N2O7S
—— (R)-3-({5-[(2-chlorobenzyl)carbamoyl]-2-cyclopropyl-1',1'-dioxido-2',3',5',6'-tetrahydrospiro[indole-3,4'-thiopyran]-1(2H)-yl}sulfonyl)benzoic acid 1448040-63-8 C30H29ClN2O7S2
(R)-3-({5-[(2-chlorobenzyl)carbamoyl]-2-cyclopropyl-1',1'-dioxido-2',3',5',6'-tetrahydrospiro[indole-3,4'-thiopyran]-1(2H)-yl}sulfonyl)benzoic acid
—— —— 1332453-28-7 C29H30ClF3N4O2
—— 3-(n-hexylcarboxy)-4,5α-epoxy-17-methylmorphinan-6-one 1261158-59-1 C24H31NO4
3-(n-hexylcarboxy)-4,5α-epoxy-17-methylmorphinan-6-one
—— —— 1192349-93-1 C28H23N5O3S
—— —— 1193395-27-5 C26H31F2N3O5S3
—— tert-butyl (8aS)-8a-(3-bromo-4-fluorophenyl)-4,4a,5,7,8,8a-hexahydropyrano[4,3-d][1,3]thiazin-2-ylcarbamate 1262038-38-9 C18H22BrFN2O3S
tert-butyl (8aS)-8a-(3-bromo-4-fluorophenyl)-4,4a,5,7,8,8a-hexahydropyrano[4,3-d][1,3]thiazin-2-ylcarbamate
—— —— 111201-21-9 C20H18Br2CoCuN2O6
—— bistrimethylsilyl N<sub>1</sub>-acetyl N<sub>2</sub>-paranitrobenzoylhydrazine 126713-69-7 C15H25N3O4Si2
bistrimethylsilyl N<sub>1</sub>-acetyl N<sub>2</sub>-paranitrobenzoylhydrazine
—— 5-(3,5-dibromo-4-hydroxyphenyl)-N-methyl-N-(3-(trifluoromethyl)benzyl)isoxazole-3-carboxamide 1191243-52-3 C19H13Br2F3N2O3
5-(3,5-dibromo-4-hydroxyphenyl)-N-methyl-N-(3-(trifluoromethyl)benzyl)isoxazole-3-carboxamide
—— N-benzyl-3-(1-cyclohexyl-4-oxo-4,5-dihydro-1H-pyrazolo[3,4-d]pyrimidin-6-yl)azetidine-1-carboxamide 1025709-98-1 C22H26N6O2
N-benzyl-3-(1-cyclohexyl-4-oxo-4,5-dihydro-1H-pyrazolo[3,4-d]pyrimidin-6-yl)azetidine-1-carboxamide
—— 5-[4-(benzothiazol-2-yl)-3-hydroxyphenyl]-3,3-dimethyl-2,3-dihydrofuran 1225265-80-4 C19H17NO2S
5-[4-(benzothiazol-2-yl)-3-hydroxyphenyl]-3,3-dimethyl-2,3-dihydrofuran
—— N'-[(3,5-dihexoxyphenyl)methyl]ethane-1,2-diamine 1217553-40-6 C21H38N2O2
N'-[(3,5-dihexoxyphenyl)methyl]ethane-1,2-diamine
—— (5R)-5-methyl-3-{[4'-(trifluoromethyl)biphenyl-4-yl]methyl}-1,3-oxazolidin-2-one 1095984-96-5 C18H16F3NO2
(5R)-5-methyl-3-{[4'-(trifluoromethyl)biphenyl-4-yl]methyl}-1,3-oxazolidin-2-one
—— (3aR,5s,6aS)-5-(4-chloro-3-fluorophenoxy)octahydrocyclopenta[c]pyrrole 1256240-55-7 C13H15ClFNO
(3aR,5s,6aS)-5-(4-chloro-3-fluorophenoxy)octahydrocyclopenta[c]pyrrole
—— —— 1416223-95-4 C27H25N5O5S
—— —— 1448541-23-8 C19H15F3N4O3
—— N-[2-(dimethylamino)ethyl]-5,6-dihydroxy-2-(naphthalen-1-ylmethyl)pyrimidine-4-carboxamide 1407174-29-1 C20H22N4O3
N-[2-(dimethylamino)ethyl]-5,6-dihydroxy-2-(naphthalen-1-ylmethyl)pyrimidine-4-carboxamide
—— —— 1193350-44-5 C18H15ClF2N2O
—— (E)-3-[(1α,3α,4α)-3,4-difluorocyclopentyl]-N-(3-ethyl-1,2,4-thiadiazol-5-yl)-2-(4-(methylsulfonyl)phenyl)acrylamide 1193393-59-7 C19H21F2N3O3S2
(E)-3-[(1α,3α,4α)-3,4-difluorocyclopentyl]-N-(3-ethyl-1,2,4-thiadiazol-5-yl)-2-(4-(methylsulfonyl)phenyl)acrylamide
—— —— 1187064-21-6 C19H18F3N5O4S
—— (S)-3-[(S)-1-(2,4-dichlorophenoxy)butyl]pyrrolidine monotrifluoroacetate 1261123-91-4 C2HF3O2*C14H19Cl2NO
(S)-3-[(S)-1-(2,4-dichlorophenoxy)butyl]pyrrolidine monotrifluoroacetate
—— (S)-3-[(R)-1-(4-chlorophenoxy)butyl]pyrrolidine monotrifluoroacetate 1261123-38-9 C2HF3O2*C14H20ClNO
(S)-3-[(R)-1-(4-chlorophenoxy)butyl]pyrrolidine monotrifluoroacetate
—— —— 1329426-64-3 C34H50Cl3NO21
—— —— 1404435-81-9 C28H17ClN2O6S
—— —— 1404436-30-1 C34H21ClN2O7
—— N,N'-Bis(4-chinazolyl)-α, δ-diamino-butan 1051-83-8 C20H20N6
N,N'-Bis(4-chinazolyl)-α, δ-diamino-butan
—— 4-(4-hydroxy-3-methylphenyl)-6-(4-{[2-(3-methylpiperidin-1-yl)-2-oxoethyl]oxy}phenyl)pyrimidin-2(1H)-one 1076184-87-6 C25H27N3O4
4-(4-hydroxy-3-methylphenyl)-6-(4-{[2-(3-methylpiperidin-1-yl)-2-oxoethyl]oxy}phenyl)pyrimidin-2(1H)-one
—— 1-(5-(1-(2,4-difluorophenyl)-1H-pyrazolo[3,4-b]pyridin-4-yl)pyrimidin-4-yl)azetidin-3-ol 1356054-23-3 C19H14F2N6O
1-(5-(1-(2,4-difluorophenyl)-1H-pyrazolo[3,4-b]pyridin-4-yl)pyrimidin-4-yl)azetidin-3-ol
—— tris(5-butyl-1-phenyl-1H-1,2,3-triazol-4-yl)phpsphane 1283071-90-8 C36H42N9P
tris(5-butyl-1-phenyl-1H-1,2,3-triazol-4-yl)phpsphane
—— 1-(3-chloro-4-hydroxyphenyl)-3-(2-(3-(4-(2-(cyclopentyloxy)ethoxy)phenoxy)-2-hydroxypropylamino)ethyl)urea 1354967-32-0 C25H34ClN3O6
1-(3-chloro-4-hydroxyphenyl)-3-(2-(3-(4-(2-(cyclopentyloxy)ethoxy)phenoxy)-2-hydroxypropylamino)ethyl)urea
—— 3-(6-(1-(3-fluoropropyl)piperidin-4-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-iodopyridin-2(1H)-one 1054315-52-4 C21H24FIN4O
3-(6-(1-(3-fluoropropyl)piperidin-4-yl)-4-methyl-1H-benzo[d]imidazol-2-yl)-4-iodopyridin-2(1H)-one
—— 4-[3-(1H-benzimidazol-2-yl)-1H-indazol-5-yl]-1,4-dihydro-2,6-dimethyl-3,5-pyridinedicarbonitrile 1033768-89-6 C23H17N7
4-[3-(1H-benzimidazol-2-yl)-1H-indazol-5-yl]-1,4-dihydro-2,6-dimethyl-3,5-pyridinedicarbonitrile
—— {5-methyl-4-[2-(3-methyl-1,2,4-oxadiazol-5-yl)-1H-indol-5-yl]-1H-imidazol-2-yl}(pyrrolidin-1-yl)methanone 1222174-02-8 C20H20N6O2
{5-methyl-4-[2-(3-methyl-1,2,4-oxadiazol-5-yl)-1H-indol-5-yl]-1H-imidazol-2-yl}(pyrrolidin-1-yl)methanone
—— 3-[7-chloro-5-(2-fluoro-phenyl)-1H-benzoimidazol-2-yl]-1-oxa-2-aza-spiro[4.5]dec-2-ene 1221349-75-2 C21H19ClFN3O
3-[7-chloro-5-(2-fluoro-phenyl)-1H-benzoimidazol-2-yl]-1-oxa-2-aza-spiro[4.5]dec-2-ene
—— 1-cyclopentyl-6-{(1R)-1-[3-(4-methylpyrimidin-2-yl)azetidin-1-yl]ethyl}-1,5-dihydro-4H-pyrazolo[3,4-d]pyrimidin-4-one 1236858-75-5 C20H25N7O
1-cyclopentyl-6-{(1R)-1-[3-(4-methylpyrimidin-2-yl)azetidin-1-yl]ethyl}-1,5-dihydro-4H-pyrazolo[3,4-d]pyrimidin-4-one
—— 2-({4-[6-(4-hydroxy-3-methylphenyl)-2-oxo-2,3-dihydropyrimidin-4-yl]phenyl}oxy)-N-[3-(methyloxy)propyl]acetamide 1076186-90-7 C23H25N3O5
2-({4-[6-(4-hydroxy-3-methylphenyl)-2-oxo-2,3-dihydropyrimidin-4-yl]phenyl}oxy)-N-[3-(methyloxy)propyl]acetamide
—— tris(dimethylamino)-[(2S)-octan-2-yl]sulfanylphosphanium 103514-67-6 C14H35N3PS
tris(dimethylamino)-[(2S)-octan-2-yl]sulfanylphosphanium
—— (1-Methylpiperidin-3-yl)methanamine;hydrochloride 1260783-75-2 C7H17ClN2
(1-Methylpiperidin-3-yl)methanamine;hydrochloride
—— methyl N-[(2S)-1-[(2S)-2-[5-[1-fluoro-6-[5-(1-fluoropropan-2-yl)thiophen-2-yl]-3-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate 1620447-84-8 C50H57F2N9O7S
methyl N-[(2S)-1-[(2S)-2-[5-[1-fluoro-6-[5-(1-fluoropropan-2-yl)thiophen-2-yl]-3-[2-[(2S)-1-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]pyrrolidin-2-yl]-1H-imidazol-5-yl]-6H-indolo[1,2-c][1,3]benzoxazin-10-yl]-1H-imidazol-2-yl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]carbamate
—— 1-{4-[4-(2-phenylacetyl)piperazine-1-sulfonyl]phenyl}-3-(pyridin-3-ylmethyl)urea 1363152-62-8 C25H27N5O4S
1-{4-[4-(2-phenylacetyl)piperazine-1-sulfonyl]phenyl}-3-(pyridin-3-ylmethyl)urea
—— [(5-phenylamino-pyridine-2-carbonyl)-amino]-acetic acid ethyl ester 1188374-67-5 C16H17N3O3
[(5-phenylamino-pyridine-2-carbonyl)-amino]-acetic acid ethyl ester
—— US10266493, Example 2ZZ 1352793-21-5 C17H16N2O3S
US10266493, Example 2ZZ
—— 10-allyl-9-(4-chloro-phenyl)-7-methyl-6-phenyl-5,6-dihydro-2H-benzo[b][1,4]oxazocine-8-carboxylic acid ethyl ester 1190367-24-8 C29H28ClNO3
10-allyl-9-(4-chloro-phenyl)-7-methyl-6-phenyl-5,6-dihydro-2H-benzo[b][1,4]oxazocine-8-carboxylic acid ethyl ester
—— N-(2-bromo-4,6-difluorophenyl)-4-(2-bromo-4-fluorophenyl)-1,3-dimethyl-1H-pyrazol-5-amine 1242533-56-7 C17H12Br2F3N3
N-(2-bromo-4,6-difluorophenyl)-4-(2-bromo-4-fluorophenyl)-1,3-dimethyl-1H-pyrazol-5-amine