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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[3-(3-amino-4,5,7-triazatricyclo[7.3.0.02,6]dodeca-1(9),2,5,7-tetraen-8-yl)phenyl]-3-(trifluoromethyl)benzamide 1225068-51-8 C23H18F3N5O
N-[3-(3-amino-4,5,7-triazatricyclo[7.3.0.02,6]dodeca-1(9),2,5,7-tetraen-8-yl)phenyl]-3-(trifluoromethyl)benzamide
—— 4-({[6-(2,6-dimethoxy-4-{(E)-3-oxo-3-[4-(4-{2-[3-(propan-2-yl)phenoxy]ethyl}benzyl)-piperazin-1-yl]prop-1-en-1-yl}phenoxy)pyridin-3-yl]oxy}methyl)benzonitrile 1322777-52-5 C46H48N4O6
4-({[6-(2,6-dimethoxy-4-{(E)-3-oxo-3-[4-(4-{2-[3-(propan-2-yl)phenoxy]ethyl}benzyl)-piperazin-1-yl]prop-1-en-1-yl}phenoxy)pyridin-3-yl]oxy}methyl)benzonitrile
—— 4-(2,2-dimethyl-[1,3]dioxolan-4-yl)-2,2-dimethyl-2-oxo-2-phenyl-tetrahydro-6λ*5*-[1,3]dioxolo[4,5-d][1,2]oxaphosphinan-3-oxy-3,4-dinitrophenyl 1096143-85-9 C24H27N2O11P
4-(2,2-dimethyl-[1,3]dioxolan-4-yl)-2,2-dimethyl-2-oxo-2-phenyl-tetrahydro-6λ*5*-[1,3]dioxolo[4,5-d][1,2]oxaphosphinan-3-oxy-3,4-dinitrophenyl
—— 2-butylamino-1-(5-tert-butyl-2-methoxy-phenyl)-1-quinoxalin-6-yl-ethanol 1097730-17-0 C25H33N3O2
2-butylamino-1-(5-tert-butyl-2-methoxy-phenyl)-1-quinoxalin-6-yl-ethanol
—— N-(3-amino-1-benzyl-2,3-dioxopropyl)-5-chloro-2-(4-phenyl-1H-imidazol-1-yl)nicotinamide hydrochloride 1037826-61-1 C25H20ClN5O3*ClH
N-(3-amino-1-benzyl-2,3-dioxopropyl)-5-chloro-2-(4-phenyl-1H-imidazol-1-yl)nicotinamide hydrochloride
—— 2-[(6-fluoro-3-oxo-1,2-dihydroisoindol-5-yl)amino]-2-[3-methoxy-4-[(2R)-1-[[3-(methylaminomethyl)phenyl]carbamoyloxy]propan-2-yl]phenyl]acetic acid 1037085-94-1 C29H31FN4O6
2-[(6-fluoro-3-oxo-1,2-dihydroisoindol-5-yl)amino]-2-[3-methoxy-4-[(2R)-1-[[3-(methylaminomethyl)phenyl]carbamoyloxy]propan-2-yl]phenyl]acetic acid
—— tert-butyl {3-[(6'-chloro-4'-oxo-3',4'-dihydro-1H-spiro[piperidine-4,2'-thiochromen]-1-yl)carbonyl]-6-methoxy-1-benzothiophen-2-yl}carbamate 1051386-48-1 C28H29ClN2O5S2
tert-butyl {3-[(6'-chloro-4'-oxo-3',4'-dihydro-1H-spiro[piperidine-4,2'-thiochromen]-1-yl)carbonyl]-6-methoxy-1-benzothiophen-2-yl}carbamate
—— 2-[5-Chloro-2-(2-methoxyethoxy)phenyl]propan-2-ol 1073436-00-6 C12H17ClO3
2-[5-Chloro-2-(2-methoxyethoxy)phenyl]propan-2-ol
—— tert-butyl {3-[(6-chloro-4-oxo-3,4-dihydro-1'H-spiro[chromene-2,4'-piperidin]-1'-yl)carbonyl]-6-(trifluoromethyl)thieno[2,3-b]pyridin-2-yl}carbamate 1051386-87-8 C27H25ClF3N3O5S
tert-butyl {3-[(6-chloro-4-oxo-3,4-dihydro-1'H-spiro[chromene-2,4'-piperidin]-1'-yl)carbonyl]-6-(trifluoromethyl)thieno[2,3-b]pyridin-2-yl}carbamate
—— (E)-3-(4-methoxybenzylidene)heptan-2-one 1065850-27-2 C15H20O2
(E)-3-(4-methoxybenzylidene)heptan-2-one
—— 8-(cyclopropylamino)-6-((3-(4-hydroxy-1-piperidinyl)phenyl)amino)imidazo[1,2-b]pyridazine-3-carbonitrile 1220629-51-5 C21H23N7O
8-(cyclopropylamino)-6-((3-(4-hydroxy-1-piperidinyl)phenyl)amino)imidazo[1,2-b]pyridazine-3-carbonitrile
—— (3RS)-(4RS)-4-azidomethyl-pyrrolidin-3-ol 1072827-70-3 C5H10N4O
(3RS)-(4RS)-4-azidomethyl-pyrrolidin-3-ol
—— 1-(4-trifluoromethoxy-3,5-difluorophenylethynyl)-4-(2,6-difluoro-4-n-butylphenylethynyl)naphthalene 1296203-55-8 C31H19F7O
1-(4-trifluoromethoxy-3,5-difluorophenylethynyl)-4-(2,6-difluoro-4-n-butylphenylethynyl)naphthalene
—— 5-[(4,6-dioxo-2-sulfanylidene-1,3-diazinan-5-yl)-(4-methylphenyl)sulfamoyl]-2-hydroxybenzoic acid 118509-77-6 C18H15N3O7S2
5-[(4,6-dioxo-2-sulfanylidene-1,3-diazinan-5-yl)-(4-methylphenyl)sulfamoyl]-2-hydroxybenzoic acid
—— 3-[4-(spiro[5.5]undec-2-ylmethoxy)-phenyl]-pentanoic acid 1147730-77-5 C23H34O3
3-[4-(spiro[5.5]undec-2-ylmethoxy)-phenyl]-pentanoic acid
—— N-hydroxy-2-(4-methoxyphenoxy)-2-phenylacetamide 1070700-51-4 C15H15NO4
N-hydroxy-2-(4-methoxyphenoxy)-2-phenylacetamide
—— 5-(4-Benzylsulfonylpiperazin-1-yl)-2-(3,5-difluorophenyl)-4-(8-hydroxyoctoxy)pyridazin-3-one 1062081-40-6 C29H36F2N4O5S
5-(4-Benzylsulfonylpiperazin-1-yl)-2-(3,5-difluorophenyl)-4-(8-hydroxyoctoxy)pyridazin-3-one
—— 2-(3-Chlorophenyl)-5-(4-propan-2-ylsulfonylpiperazin-1-yl)-4-(5,6,7,8-tetrahydroquinolin-5-yloxy)pyridazin-3-one 1062081-43-9 C26H30ClN5O4S
2-(3-Chlorophenyl)-5-(4-propan-2-ylsulfonylpiperazin-1-yl)-4-(5,6,7,8-tetrahydroquinolin-5-yloxy)pyridazin-3-one
—— (S)-5-cyclopropyl-1-(3-(3-fluorophenoxy)-2-hydroxypropyl)-8-methoxy-2,3,5,6-tetrahydrobenzo[b][1,5]diazocin-4(1H)-one 1307894-53-6 C23H27FN2O4
(S)-5-cyclopropyl-1-(3-(3-fluorophenoxy)-2-hydroxypropyl)-8-methoxy-2,3,5,6-tetrahydrobenzo[b][1,5]diazocin-4(1H)-one
—— N-(1-((2,4-dimethylphenyl)sulfonyl)-1H-pyrazol-4-yl)picolinamide 1296784-30-9 C17H16N4O3S
N-(1-((2,4-dimethylphenyl)sulfonyl)-1H-pyrazol-4-yl)picolinamide
—— Tyr-Asp-Phe-Gly-Val-NH2 1273019-63-8 C29H38N6O8
Tyr-Asp-Phe-Gly-Val-NH2
—— (3S,6S)-4-[4-((S)-4-hydroxy-6-aza-spiro[2.5]oct-6-yl)-4-oxo-butyl]-6-methyl-5-oxo-piperazine-1,3-dicarboxylic acid 3-amide 1-[(3,4-bis-trifluoromethyl-phenyl)-amide] 1290050-76-8 C26H31F6N5O5
(3S,6S)-4-[4-((S)-4-hydroxy-6-aza-spiro[2.5]oct-6-yl)-4-oxo-butyl]-6-methyl-5-oxo-piperazine-1,3-dicarboxylic acid 3-amide 1-[(3,4-bis-trifluoromethyl-phenyl)-amide]
—— 1-(4-(2-(cyclopropylmethyl)-1-oxoisoindolin-5-yl)benzyl)-3-ethylimidazolidine-2,4-dione 1295301-69-7 C24H25N3O3
1-(4-(2-(cyclopropylmethyl)-1-oxoisoindolin-5-yl)benzyl)-3-ethylimidazolidine-2,4-dione
—— 1-(3-{3-[2-(4-chloro-phenyl)-ethyl]-4-trifluoromethyl-phenyl}-5-methanesulfonyl-4,5,6,7-tetrahydro-pyrazolo[4,3-c]pyridin-1-yl)-3-morpholin-4-yl-propan-2-ol 1049809-70-2 C29H34ClF3N4O4S
1-(3-{3-[2-(4-chloro-phenyl)-ethyl]-4-trifluoromethyl-phenyl}-5-methanesulfonyl-4,5,6,7-tetrahydro-pyrazolo[4,3-c]pyridin-1-yl)-3-morpholin-4-yl-propan-2-ol
—— 7-Thiomethoxy-thiochromanon 13735-15-4 C10H10OS2
7-Thiomethoxy-thiochromanon
—— —— 102697-65-4 C78H66O24
—— (R)-3-{(1S,2S)-1-[5-(2-chloro-4-iodo-phenyl)-1H-imidazol-2-yl]-2-phenyl-propyl}-5-[4-(2-hydroxy-ethoxy)-phenyl]-imidazolidine-2,4-dione 1165869-37-3 C29H26ClIN4O4
(R)-3-{(1S,2S)-1-[5-(2-chloro-4-iodo-phenyl)-1H-imidazol-2-yl]-2-phenyl-propyl}-5-[4-(2-hydroxy-ethoxy)-phenyl]-imidazolidine-2,4-dione
—— (R)-3-{(1R,2R)-1-[5-(2-fluoro-4-iodophenyl)-4-methyl-1H-imidazol-2-yl]-2-methoxypropyl}-5-[4-(2-hydroxyethoxy)phenyl]imidazolidine-2,4-dione 1165870-35-8 C25H26FIN4O5
(R)-3-{(1R,2R)-1-[5-(2-fluoro-4-iodophenyl)-4-methyl-1H-imidazol-2-yl]-2-methoxypropyl}-5-[4-(2-hydroxyethoxy)phenyl]imidazolidine-2,4-dione
—— (3R,6S,9R,12R,15S)-6-cyclopropyl-12-[(4-hydroxyphenyl)methyl]-3,8,9,15-tetramethyl-2-oxa-5,8,11,14,19-pentazabicyclo[16.4.0]docosa-1(18),19,21-triene-7,10,13-trione 1047667-38-8 C30H41N5O5
(3R,6S,9R,12R,15S)-6-cyclopropyl-12-[(4-hydroxyphenyl)methyl]-3,8,9,15-tetramethyl-2-oxa-5,8,11,14,19-pentazabicyclo[16.4.0]docosa-1(18),19,21-triene-7,10,13-trione
—— 4-[4-(2-morpholin-4-yl-ethylcarbamoyl)-phenylcarbamoyl]-2-pyridin-4-yl-thiazolidine-3-carboxylic acid benzyl ester 1029799-65-2 C30H33N5O5S
4-[4-(2-morpholin-4-yl-ethylcarbamoyl)-phenylcarbamoyl]-2-pyridin-4-yl-thiazolidine-3-carboxylic acid benzyl ester
—— N-[N-[5(S)-[[N-(benzyloxycarbonyl)-L-asparaginyl]amino]-6-cyclohexyl-4(S)-hydroxy-2(S)-isopropylhexanoyl]-L-isoleucyl]-L-phenylalanine methyl ester 134015-12-6 C43H63N5O9
N-[N-[5(S)-[[N-(benzyloxycarbonyl)-L-asparaginyl]amino]-6-cyclohexyl-4(S)-hydroxy-2(S)-isopropylhexanoyl]-L-isoleucyl]-L-phenylalanine methyl ester
—— N-(1H-benzo[d]imidazol-2-yl)-3-((3-(6-((dimethylamino)methyl)pyridin-3-yl)-6-oxopyridazin-1(6H)-yl)methyl)benzamide 1621689-38-0 C27H25N7O2
N-(1H-benzo[d]imidazol-2-yl)-3-((3-(6-((dimethylamino)methyl)pyridin-3-yl)-6-oxopyridazin-1(6H)-yl)methyl)benzamide
—— 2-(3-Chlorophenyl)-5-[4-[(2,6-dichlorophenyl)methyl]piperazin-1-yl]-4-(2-ethoxyethoxy)pyridazin-3-one 1062052-29-2 C25H27Cl3N4O3
2-(3-Chlorophenyl)-5-[4-[(2,6-dichlorophenyl)methyl]piperazin-1-yl]-4-(2-ethoxyethoxy)pyridazin-3-one
—— N-(5-methyl-pyrazin-2-ylmethyl)-3-(5-methyl-pyridin-2-yl)-5-(5-trifluoromethyl-pyrazol-1-yl)-benzamide 1162644-34-9 C23H19F3N6O
N-(5-methyl-pyrazin-2-ylmethyl)-3-(5-methyl-pyridin-2-yl)-5-(5-trifluoromethyl-pyrazol-1-yl)-benzamide
—— (2R,5R)-4-[2-(6-cyano-3,3-dimethyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-5-methoxymethyl-2-methyl-piperazine-1-carboxylic acid tert-butyl ester 1403903-38-7 C25H36N4O4
(2R,5R)-4-[2-(6-cyano-3,3-dimethyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-5-methoxymethyl-2-methyl-piperazine-1-carboxylic acid tert-butyl ester
—— (8-tert-butyl-5,6,7,8-tetrahydroquinazolin-2-yl)-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]amine 1172639-16-5 C23H29N5O
(8-tert-butyl-5,6,7,8-tetrahydroquinazolin-2-yl)-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]amine
—— (R)-3-{(1S,2S)-1-[5-(4-bromo-2-methylphenyl)-1H-imidazol-2-yl]-2-phenylpropyl}-5-[4-(2-hydroxyethoxy)phenyl]imidazolidine-2,4-dione 1165868-74-5 C30H29BrN4O4
(R)-3-{(1S,2S)-1-[5-(4-bromo-2-methylphenyl)-1H-imidazol-2-yl]-2-phenylpropyl}-5-[4-(2-hydroxyethoxy)phenyl]imidazolidine-2,4-dione
—— 5-[4-[(2R)-2-aminopropanoyl]piperazin-1-yl]-4-(3-ethoxypropylamino)-2-phenylpyridazin-3-one 1062071-29-7 C22H32N6O3
5-[4-[(2R)-2-aminopropanoyl]piperazin-1-yl]-4-(3-ethoxypropylamino)-2-phenylpyridazin-3-one
—— 5-(2-phenylthiazol-4-yl)indolin-2-one hydrochloride 1129403-60-6 C17H12N2OS*ClH
5-(2-phenylthiazol-4-yl)indolin-2-one hydrochloride
—— 5-[5-(1-dimethylamino-ethyl)-[1,2,4]triazol-1-yl]-4'-methyl-biphenyl-3-carboxylic acid (1-pyrazin-2-yl-ethyl)-amide 1161870-03-6 C26H29N7O
5-[5-(1-dimethylamino-ethyl)-[1,2,4]triazol-1-yl]-4'-methyl-biphenyl-3-carboxylic acid (1-pyrazin-2-yl-ethyl)-amide
—— 3-[5-(1,1-difluoro-ethyl)-[1,2,4]triazol-1-yl]-N-((S)-2-hydroxy-1-methyl-ethyl)-5-(5-methyl-pyridin-2-yl)-benzamide 1161870-25-2 C20H21F2N5O2
3-[5-(1,1-difluoro-ethyl)-[1,2,4]triazol-1-yl]-N-((S)-2-hydroxy-1-methyl-ethyl)-5-(5-methyl-pyridin-2-yl)-benzamide
—— 3-[4-(4-methoxyphenoxy)-5-[[(2S)-pyrrolidin-2-yl]methylamino]pyrimidin-2-yl]phenol 1298096-56-6 C22H24N4O3
3-[4-(4-methoxyphenoxy)-5-[[(2S)-pyrrolidin-2-yl]methylamino]pyrimidin-2-yl]phenol
—— 1-[2-amino-4-(isoindoline-2-carbonyl)quinazolin-6-yl]-N,N-dimethylcyclopropanecarboxamide 1309088-52-5 C23H23N5O2
1-[2-amino-4-(isoindoline-2-carbonyl)quinazolin-6-yl]-N,N-dimethylcyclopropanecarboxamide
—— 7-(3,5-dimethyl-4-isoxazolyl)-8-(methyloxy)-2-[2-(methyloxy)ethyl]-1-{2-[(trifluoromethyl)oxy]phenyl}-1H-imidazo[4,5-c]-1,5-naphthyridine 1300737-20-5 C26H23F3N4O4
7-(3,5-dimethyl-4-isoxazolyl)-8-(methyloxy)-2-[2-(methyloxy)ethyl]-1-{2-[(trifluoromethyl)oxy]phenyl}-1H-imidazo[4,5-c]-1,5-naphthyridine
—— N-[1-(3-{1-ethyl-5-[4-(trifluoromethyI)phenoxy]-1H-pyrazol-3-yl}phenyl)-1-methylethyl]-N'-isobutylsulfamide 1289201-71-3 C25H31F3N4O3S
N-[1-(3-{1-ethyl-5-[4-(trifluoromethyI)phenoxy]-1H-pyrazol-3-yl}phenyl)-1-methylethyl]-N'-isobutylsulfamide
—— 3,4-dichloro-N-[2-[3-(3-fluoropiperidin-1-yl)pyrrolidin-1-yl]-2-oxoethyl]benzamide 1027773-55-2 C18H22Cl2FN3O2
3,4-dichloro-N-[2-[3-(3-fluoropiperidin-1-yl)pyrrolidin-1-yl]-2-oxoethyl]benzamide
—— 5-Chlor-2,1,3-benzothiadiazol-4-sulfonsaeureamid 113950-69-9 C6H4ClN3O2S2
5-Chlor-2,1,3-benzothiadiazol-4-sulfonsaeureamid
—— 2-[5-[(E)-2-(4-methoxyphenyl)ethenyl]-1,1-dioxo-3H-thieno[3,2-d][1,2]thiazol-2-yl]butanoic acid 1170194-49-6 C18H19NO5S2
2-[5-[(E)-2-(4-methoxyphenyl)ethenyl]-1,1-dioxo-3H-thieno[3,2-d][1,2]thiazol-2-yl]butanoic acid
—— N-(2-(trifluoromethyl)phenylcarbamoyl)decanamide 1161363-33-2 C18H25F3N2O2
N-(2-(trifluoromethyl)phenylcarbamoyl)decanamide
—— ethyl 2-[3-fluoro-4-(4-methylimidazol-1-yl)phenylamino]-5,6,7,8-tetrahydroquinazoline-8-carboxylate 1172638-90-2 C21H22FN5O2
ethyl 2-[3-fluoro-4-(4-methylimidazol-1-yl)phenylamino]-5,6,7,8-tetrahydroquinazoline-8-carboxylate