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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-chloro-N2-(3,5-dimethyl-4-ethoxyphenyl)-N4-[2-methyl-4-(ethylaminosulfonylamino)methylphenyl]-2,4-pyrimidinediamine 1065083-62-6 C24H31ClN6O3S
5-chloro-N2-(3,5-dimethyl-4-ethoxyphenyl)-N4-[2-methyl-4-(ethylaminosulfonylamino)methylphenyl]-2,4-pyrimidinediamine
—— sodium 6-chloro-7-(4-(4-(2-chlorophenyl)butylcarbamoyl)phenoxy)chroman-4-carboxylate 1202886-98-3 C27H24Cl2NO5*Na
sodium 6-chloro-7-(4-(4-(2-chlorophenyl)butylcarbamoyl)phenoxy)chroman-4-carboxylate
—— 9-(4-{4-[(3,4-dichlorophenyl)-acetyl]-piperazino}-butyl)-9H-fluorene-9-carboxylic acid-(2,2,2-trifluoro-ethyl)-amide 1099094-45-7 C32H32Cl2F3N3O2
9-(4-{4-[(3,4-dichlorophenyl)-acetyl]-piperazino}-butyl)-9H-fluorene-9-carboxylic acid-(2,2,2-trifluoro-ethyl)-amide
—— 2-(6-isopropenyl-2-methoxy-3-methyl-phenoxy)-2-methyl-propionic acid methyl ester 1384950-13-3 C16H22O4
2-(6-isopropenyl-2-methoxy-3-methyl-phenoxy)-2-methyl-propionic acid methyl ester
—— 7-Ethyl-2,4-dimethyl-6,7-dihydro-4H-indeno[5,6-b][1,4]oxazine-3,8-dione 139197-61-8 C15H17NO3
7-Ethyl-2,4-dimethyl-6,7-dihydro-4H-indeno[5,6-b][1,4]oxazine-3,8-dione
—— 2-Bromo-3-butyl-bicyclo[2.2.2]oct-2-ene 131010-67-8 C12H19Br
2-Bromo-3-butyl-bicyclo[2.2.2]oct-2-ene
—— 5-Benzyloxy-2,2-difluoro-pent-3-ynoic acid methyl ester 109872-98-2 C13H12F2O3
5-Benzyloxy-2,2-difluoro-pent-3-ynoic acid methyl ester
—— 1-tert-butyl-4-(di-isopropylamino)-2,2-dimethyl-3-phenyl-1,3,2,4-azaarsasilaboretidine 112795-14-9 C18H34AsBN2Si
1-tert-butyl-4-(di-isopropylamino)-2,2-dimethyl-3-phenyl-1,3,2,4-azaarsasilaboretidine
—— 2-Iodo-3,4,5-trimethoxy-benzoic acid 2-(2-iodo-4,5-dimethoxy-benzoyloxymethyl)-phenyl ester 139058-91-6 C26H24I2O9
2-Iodo-3,4,5-trimethoxy-benzoic acid 2-(2-iodo-4,5-dimethoxy-benzoyloxymethyl)-phenyl ester
—— (3S)-3-<(1'S)-1'-<<(3''-azido-5''-O-(3-chlorobenzoyl)-2'',3''-dideoxy-α-D-ribo-hexaro-1'',4''-lactone)-6''-oyl>amino>-3'-methylbutyl>-3,4-dihydro-8-hydroxy-1H-2-benzopyran-1-one 147804-74-8 C27H27ClN4O8
(3S)-3-<(1'S)-1'-<<(3''-azido-5''-O-(3-chlorobenzoyl)-2'',3''-dideoxy-α-D-ribo-hexaro-1'',4''-lactone)-6''-oyl>amino>-3'-methylbutyl>-3,4-dihydro-8-hydroxy-1H-2-benzopyran-1-one
—— 5-{3-[4-(5-bromo-2-chlorophenoxy)phenyl]-1,2,4-oxadiazol-5-yl}-1H-tetrazole 1161026-03-4 C15H8BrClN6O2
5-{3-[4-(5-bromo-2-chlorophenoxy)phenyl]-1,2,4-oxadiazol-5-yl}-1H-tetrazole
—— p-Nitrophenyl 3-O-(N-propyl-carbamoylmethyl)-β-D-galactopyranoside 183880-39-9 C17H24N2O9
p-Nitrophenyl 3-O-(N-propyl-carbamoylmethyl)-β-D-galactopyranoside
—— N-(2-(N-benzyloxycarbonyl-L-leucinamido)-2-deoxy-β-D-galactopyranosyl)-N-octadecyl-dodecanoamide 113483-91-3 C50H89N3O8
N-(2-(N-benzyloxycarbonyl-L-leucinamido)-2-deoxy-β-D-galactopyranosyl)-N-octadecyl-dodecanoamide
—— Ethyl 3-[5-[3-[(1-methylpyrazol-3-yl)carbamoyl]-5-propan-2-yloxyphenoxy]pyridin-2-yl]-1,2,4-oxadiazole-5-carboxylate 1310808-84-4 C24H24N6O6
Ethyl 3-[5-[3-[(1-methylpyrazol-3-yl)carbamoyl]-5-propan-2-yloxyphenoxy]pyridin-2-yl]-1,2,4-oxadiazole-5-carboxylate
—— N-(1-methyl-1H-benzimidazol-2-yl)-1-oxo-2,3,4,5-tetrahydro-1H-[1,4]diazepino[1,2-a]benzimidazole-8-carboxamide 1311567-93-7 C20H18N6O2
N-(1-methyl-1H-benzimidazol-2-yl)-1-oxo-2,3,4,5-tetrahydro-1H-[1,4]diazepino[1,2-a]benzimidazole-8-carboxamide
—— (3,4-dichlorophenyl)-1-((1'R)-phenylethyl)tetrahydro-1H-4-imidazolone 1004755-08-1 C17H16Cl2N2O
(3,4-dichlorophenyl)-1-((1'R)-phenylethyl)tetrahydro-1H-4-imidazolone
—— 2-cyano-1-(6-(morpholinosulfonyl)hexyl)-3-(pyridin-4-yl)guanidine 1225285-70-0 C17H26N6O3S
2-cyano-1-(6-(morpholinosulfonyl)hexyl)-3-(pyridin-4-yl)guanidine
—— 1-(2-deoxy-β-D-erythro-pentofuranosyl)-5-tert-butyldiphenylsilyloxymethyl-1H,3H-pyrimidine-2,4-dione 1234711-52-4 C26H32N2O6Si
1-(2-deoxy-β-D-erythro-pentofuranosyl)-5-tert-butyldiphenylsilyloxymethyl-1H,3H-pyrimidine-2,4-dione
—— 5-Methoxy-1-(6-methoxypyridin-3-yl)-2-pyridin-2-ylbenzimidazole 1312309-80-0 C19H16N4O2
5-Methoxy-1-(6-methoxypyridin-3-yl)-2-pyridin-2-ylbenzimidazole
—— (2S,4R,5R)-5-(3-carboxypropyl)-4-[7-methoxy-8-methyl-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-1-[(2-methylpropan-2-yl)oxycarbonyl]pyrrolidine-2-carboxylic acid 1310552-33-0 C31H39N3O8S
(2S,4R,5R)-5-(3-carboxypropyl)-4-[7-methoxy-8-methyl-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-1-[(2-methylpropan-2-yl)oxycarbonyl]pyrrolidine-2-carboxylic acid
—— (S)-1-methyl-3-(1-propionylpiperidin-3-yl)-5-(pyrazolo[1,5-a]pyridin-3-yl)-1H-imidazo[4,5-b]pyridin-2(3H)-one 1299419-68-3 C22H24N6O2
(S)-1-methyl-3-(1-propionylpiperidin-3-yl)-5-(pyrazolo[1,5-a]pyridin-3-yl)-1H-imidazo[4,5-b]pyridin-2(3H)-one
—— 4-benzyl-N-((R)-1-(3-methoxyphenyl)ethyl)-5-oxomorpholine-3-carboxamide 1398395-10-2 C21H24N2O4
4-benzyl-N-((R)-1-(3-methoxyphenyl)ethyl)-5-oxomorpholine-3-carboxamide
—— N-[3-{1-[3-(dimethylamino)cyclobutyl]piperidin-4-yl}-1-(5-methylpyridin-2-yl)-1H-pyrazol-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide 1401220-91-4 C27H33N9O
N-[3-{1-[3-(dimethylamino)cyclobutyl]piperidin-4-yl}-1-(5-methylpyridin-2-yl)-1H-pyrazol-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (RS)-(4-morpholin-2-yl-phenyl)-(1H-pyrazol-3-yl)-amine 1400996-49-7 C13H16N4O
(RS)-(4-morpholin-2-yl-phenyl)-(1H-pyrazol-3-yl)-amine
—— 2-(3,5-difluoro-4-(trifluoromethyl)phenyl)quinoline 1447730-06-4 C16H8F5N
2-(3,5-difluoro-4-(trifluoromethyl)phenyl)quinoline
—— N4-(4-Fluorophenyl)-7-methoxyquinazoline-4,6-diamine (Dacomitinib Impurity) 1562180-31-7 C15H13FN4O
N4-(4-Fluorophenyl)-7-methoxyquinazoline-4,6-diamine (Dacomitinib Impurity)
—— N-(4-Bromo-phenyl)-2-(2-chloro-5-{[(2-chloro-6-fluorophenylcarbonyl)-amino]-methyl}-phenylamino)-6-(2,2-difluoro-ethoxy)-1-methyl-1H-benzimidazole-5-carboxylic acid amide 1242269-65-3 C31H23BrCl2F3N5O3
N-(4-Bromo-phenyl)-2-(2-chloro-5-{[(2-chloro-6-fluorophenylcarbonyl)-amino]-methyl}-phenylamino)-6-(2,2-difluoro-ethoxy)-1-methyl-1H-benzimidazole-5-carboxylic acid amide
—— 2-(3-cyano-5-fluorophenyl)-4-((3-fluoro-4-methoxyphenylsulfonamido)methyl)phenoxyacetic acid 1242846-39-4 C23H18F2N2O6S
2-(3-cyano-5-fluorophenyl)-4-((3-fluoro-4-methoxyphenylsulfonamido)methyl)phenoxyacetic acid
—— (1aR,12bS)-8-cyclohexyl-N-(dimethylsulfamoyl)-11-methoxy-1a-((10-(methylcarbarnoyl)-3-oxa-7,10-diazatricyclo[3.3.3.0(1,5)]undec-7-yl)carbonyl)-1,1a,2,12b-tetrahydrocyclopropa[d]indolo[2,1-a][2]benzazepine-5-carboxamide 1241621-39-5 C39H48N6O7S
(1aR,12bS)-8-cyclohexyl-N-(dimethylsulfamoyl)-11-methoxy-1a-((10-(methylcarbarnoyl)-3-oxa-7,10-diazatricyclo[3.3.3.0(1,5)]undec-7-yl)carbonyl)-1,1a,2,12b-tetrahydrocyclopropa[d]indolo[2,1-a][2]benzazepine-5-carboxamide
—— N-[(3,4-difluorophenyl)-methyl]-2-ethylsulfanyl-4-methyl-7-(trifluoromethyl)-quinoline-3-carboxamide 1242552-02-8 C21H17F5N2OS
N-[(3,4-difluorophenyl)-methyl]-2-ethylsulfanyl-4-methyl-7-(trifluoromethyl)-quinoline-3-carboxamide
—— 5-{5-[4-(2-ethylpiperidin-1-yl)-3-(methoxymethyl)phenyl]-1,2,4-oxadiazol-3-yl}pyridin-2-amine 1243557-73-4 C22H27N5O2
5-{5-[4-(2-ethylpiperidin-1-yl)-3-(methoxymethyl)phenyl]-1,2,4-oxadiazol-3-yl}pyridin-2-amine
—— ((1Z,3R,4R,5E,7Z)-1-bromo-8-iodo-4,6-dimethylocta-1,5,7-trien-3-yloxy)triethylsilane 1239951-19-9 C16H28BrIOSi
((1Z,3R,4R,5E,7Z)-1-bromo-8-iodo-4,6-dimethylocta-1,5,7-trien-3-yloxy)triethylsilane
—— 2-cyclopentyl-N-{3-[2-(6-morpholin-4-yl-pyridin-3-ylamino)-pyrrolo[2,3-d]pyrimidin-7-yl]-propyl}-acetamide 1243268-30-5 C25H33N7O2
2-cyclopentyl-N-{3-[2-(6-morpholin-4-yl-pyridin-3-ylamino)-pyrrolo[2,3-d]pyrimidin-7-yl]-propyl}-acetamide
—— 2-aminophenyl diphenylphosphinite 1187833-36-8 C18H16NOP
2-aminophenyl diphenylphosphinite
—— 5-bromo-3-[1-(5-bromo-2-nitrophenyl)-2-nitroethyl]-1H-indole 1240076-51-0 C16H11Br2N3O4
5-bromo-3-[1-(5-bromo-2-nitrophenyl)-2-nitroethyl]-1H-indole
—— 4-bromo-2-[4,4,4-trifluoro-3-hydroxy-1,1-dimethyl-3-(1H-pyrrolo[2,3-c]pyridin-2-ylmethyl)butyl]phenol 1245526-93-5 C20H20BrF3N2O2
4-bromo-2-[4,4,4-trifluoro-3-hydroxy-1,1-dimethyl-3-(1H-pyrrolo[2,3-c]pyridin-2-ylmethyl)butyl]phenol
—— 2-iodo-5-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl)-1H-pyrrolo[3,2-b]pyridine 1612287-54-3 C12H8F3IN4
2-iodo-5-(1-methyl-3-(trifluoromethyl)-1H-pyrazol-5-yl)-1H-pyrrolo[3,2-b]pyridine
—— (2R)-2-[({6-[4-(ethylsulfanyl)phenyl]-3-fluoropyridin-2-yl}methyl)amino]-3-methylbutan-1-ol 1401166-08-2 C19H25FN2OS
(2R)-2-[({6-[4-(ethylsulfanyl)phenyl]-3-fluoropyridin-2-yl}methyl)amino]-3-methylbutan-1-ol
—— 5-(3-(2-fluoro-5-(1-methylethoxy)phenyl)-1H-pyrrolo[3,2-b]pyridin-5-yl)-1,3,4-oxadiazol-2-amine 1401346-50-6 C18H16FN5O2
5-(3-(2-fluoro-5-(1-methylethoxy)phenyl)-1H-pyrrolo[3,2-b]pyridin-5-yl)-1,3,4-oxadiazol-2-amine
—— [5-(2-methoxy-ethoxy)-pyrimidin-2-yl]((S)-4-morpholin-2-yl-phenyl)-amine 1400996-32-8 C17H22N4O3
[5-(2-methoxy-ethoxy)-pyrimidin-2-yl]((S)-4-morpholin-2-yl-phenyl)-amine
—— 3,4-dichloro-N-(2-methyl-2-(3-(trifluoromethyl)phenylsulfonyl)propyl)benzamide 1276677-12-3 C18H16Cl2F3NO3S
3,4-dichloro-N-(2-methyl-2-(3-(trifluoromethyl)phenylsulfonyl)propyl)benzamide
—— N-[2-(6-fluorobiphenyl-3-yl)propan-2-yl]-1,4-diazabicyclo[3.2.2]nonane-4-carboxamide 1401090-30-9 C23H28FN3O
N-[2-(6-fluorobiphenyl-3-yl)propan-2-yl]-1,4-diazabicyclo[3.2.2]nonane-4-carboxamide
—— tert-butyl 4-(5-cyano-4-{[4-(1H-tetrazol-1-yl)phenoxy]methyl}-1H-pyrazol-1-yl)piperidine-1-carboxylate 1379604-32-6 C22H26N8O3
tert-butyl 4-(5-cyano-4-{[4-(1H-tetrazol-1-yl)phenoxy]methyl}-1H-pyrazol-1-yl)piperidine-1-carboxylate
—— 3-Amino-4-brom-N.N-Diaethyl-benzolsulfonamid 10372-46-0 C10H15BrN2O2S
3-Amino-4-brom-N.N-Diaethyl-benzolsulfonamid
—— 6-[4-[2-(2,2-Dimethylaziridin-1-yl)ethyl]-5-ethyl-2-methoxyphenyl]pyridin-2-amine 1055761-73-3 C20H27N3O
6-[4-[2-(2,2-Dimethylaziridin-1-yl)ethyl]-5-ethyl-2-methoxyphenyl]pyridin-2-amine
—— (5-Cyclopropyl-1,3-oxazol-2-yl)methanol 1889189-26-7 C7H9NO2
(5-Cyclopropyl-1,3-oxazol-2-yl)methanol
—— 2-(2-(2-chlorophenyl)-2-oxoethyl)spiro[cyclopropane-1,2'-indene]-1',3'-dione 1350725-20-0 C19H13ClO3
2-(2-(2-chlorophenyl)-2-oxoethyl)spiro[cyclopropane-1,2'-indene]-1',3'-dione
—— 5-((3,5-dichloropyridin-4-yl)thio)-N-(3-methoxybenzyl)-N-methyl-4-nitrothiophene-2-carboxamide 1247820-64-9 C19H15Cl2N3O4S2
5-((3,5-dichloropyridin-4-yl)thio)-N-(3-methoxybenzyl)-N-methyl-4-nitrothiophene-2-carboxamide
—— 8-ethyl-9-(4-heptyl)-6-(2-trifluoromethyl-4 methoxyphenyl)-9H-purine 1139646-79-9 C22H27F3N4O
8-ethyl-9-(4-heptyl)-6-(2-trifluoromethyl-4 methoxyphenyl)-9H-purine
—— methyl 4-(((2,4-diaminopteridin-6-yl)methyl)(methyl)amino)-2-(2-methoxy-2-oxoethoxy)benzoate 1246636-67-8 C19H21N7O5
methyl 4-(((2,4-diaminopteridin-6-yl)methyl)(methyl)amino)-2-(2-methoxy-2-oxoethoxy)benzoate