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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(13S,19S)-23-(acetylamino)-4,8-dimethyl-7,14-dioxo-21-oxa-3,8,15,27-tetraazatetracyclo[20.2.2.1<sup>2,6</sup>.0<sup>15,19</sup>]heptacosa-1(24),2(27),3,5,22,25-hexaen-13-yl]-2-phenylacetamide trifluoroacetate 1460305-09-2 C2HF3O2*C34H40N6O5
N-[(13S,19S)-23-(acetylamino)-4,8-dimethyl-7,14-dioxo-21-oxa-3,8,15,27-tetraazatetracyclo[20.2.2.1<sup>2,6</sup>.0<sup>15,19</sup>]heptacosa-1(24),2(27),3,5,22,25-hexaen-13-yl]-2-phenylacetamide trifluoroacetate
—— (4-methoxyphenyl)methyl 2-iodopropanoate 1612216-62-2 C11H13IO3
(4-methoxyphenyl)methyl 2-iodopropanoate
—— (S,S)-(2-ethyl-3-[4-(methylsulfonyl)phenyl]oxiran-2-yl)methanol 1246268-49-4 C12H16O4S
(S,S)-(2-ethyl-3-[4-(methylsulfonyl)phenyl]oxiran-2-yl)methanol
—— S-ethyl-2-(pyridin-2-yl)ethylcarbamothioate 1248568-83-3 C10H14N2OS
S-ethyl-2-(pyridin-2-yl)ethylcarbamothioate
—— naphthalen-2-ylcarboxylic acid 2-methyl-3-(4-methylbenzoyl)-1,1-dioxo-2H-benzo[e][1,2]thiazin-4-yl ester 1242051-23-5 C28H21NO5S
naphthalen-2-ylcarboxylic acid 2-methyl-3-(4-methylbenzoyl)-1,1-dioxo-2H-benzo[e][1,2]thiazin-4-yl ester
—— (S)-6-chloro-3-nitro-2-phenyl-1-(2,4,6-triisopropylphenylsulfonyl)-1,2-dihydroquinoline 1245022-93-8 C30H33ClN2O4S
(S)-6-chloro-3-nitro-2-phenyl-1-(2,4,6-triisopropylphenylsulfonyl)-1,2-dihydroquinoline
—— (Endo)-3-(2-methoxybenzyloxy)-8-methyl-8-azabicyclo[3.2.1]octane 1182356-60-0 C16H23NO2
(Endo)-3-(2-methoxybenzyloxy)-8-methyl-8-azabicyclo[3.2.1]octane
—— N-[5-butyl-4-(4-hydroxyphenyl)-1,3-selenazol-2-yl]-3,4,5-trihydroxybenzamide 1245904-78-2 C20H20N2O5Se
N-[5-butyl-4-(4-hydroxyphenyl)-1,3-selenazol-2-yl]-3,4,5-trihydroxybenzamide
—— 3-(benzyloxycarbonyl-L-leucylamino)-N-(2-(dimethylamino)ethyl)-2-oxophenylbutanamide 1241981-31-6 C28H38N4O5
3-(benzyloxycarbonyl-L-leucylamino)-N-(2-(dimethylamino)ethyl)-2-oxophenylbutanamide
—— 7-(3-chlorophenyl)-2-(pyridin-2-yl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyrazine 1247880-29-0 C16H14ClN5
7-(3-chlorophenyl)-2-(pyridin-2-yl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyrazine
—— 6-benzyl-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2,6,7,8-tetrahydro-1,2,3,5,6-pentaazaacenaphthylen-4-amine 1246670-06-3 C23H22N6O2
6-benzyl-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2,6,7,8-tetrahydro-1,2,3,5,6-pentaazaacenaphthylen-4-amine
—— 4-(3-cycloheptyl-6-methoxy-7-methyl-2-oxoindolin-3-yl)phenyl dihydroqenphosphate 1246452-63-0 C23H28NO6P
4-(3-cycloheptyl-6-methoxy-7-methyl-2-oxoindolin-3-yl)phenyl dihydroqenphosphate
—— (R)-5-(4-methyl-5-(1-(2-m-tolyl-2H-tetrazol-5-yl)ethylthio)-4H-1,2,4-triazol-3-yl)pyridazin-3(2H)-one 1253375-87-9 C17H17N9OS
(R)-5-(4-methyl-5-(1-(2-m-tolyl-2H-tetrazol-5-yl)ethylthio)-4H-1,2,4-triazol-3-yl)pyridazin-3(2H)-one
—— 5-ethyl-2-(5-isopropyl-5-methyl-4-oxo-imidazolin-2-yl)-6-methoxymethylpyridine-3-carboxylic acid methyl ester 120680-57-1 C18H25N3O4
5-ethyl-2-(5-isopropyl-5-methyl-4-oxo-imidazolin-2-yl)-6-methoxymethylpyridine-3-carboxylic acid methyl ester
—— 20-(4-(thiophene-3-yl)-1H-1,2,3-triazol-1-yl)-20-deoxodesmycosin 1438281-53-8 C45H70N4O13S
20-(4-(thiophene-3-yl)-1H-1,2,3-triazol-1-yl)-20-deoxodesmycosin
—— methyl 5-(2-aminoethyl)-2-fluoro-benzoate hydrochloride 1072438-59-5 C10H12FNO2*ClH
methyl 5-(2-aminoethyl)-2-fluoro-benzoate hydrochloride
—— —— 1257062-01-3 C20H22ClN5O2
—— N-(1-(6-methoxypyridin-3-yl)-3-methyl-8-(pyridin-4-yl)-1H-imidazo[4,5-c]quinolin-2(3H)-ylidene)cyanamide 1356033-69-6 C23H17N7O
N-(1-(6-methoxypyridin-3-yl)-3-methyl-8-(pyridin-4-yl)-1H-imidazo[4,5-c]quinolin-2(3H)-ylidene)cyanamide
—— —— 1616354-34-7 C31H32BF2N7O
—— 3-methyl-4-pyrazin-2-yl-1H-pyrazolo[4,3-c]pyridine 1246347-25-0 C11H9N5
3-methyl-4-pyrazin-2-yl-1H-pyrazolo[4,3-c]pyridine
—— 4-{6-[2-fluoro-1-(fluoromethyl)ethoxy]-2,4-dioxo-3-(4-(thiophen-2-yl)-benzyl)-3,4-dihydroquinazolin-1(2H)-yl}piperidine-1-carbaldehyde 1162649-85-5 C28H27F2N3O4S
4-{6-[2-fluoro-1-(fluoromethyl)ethoxy]-2,4-dioxo-3-(4-(thiophen-2-yl)-benzyl)-3,4-dihydroquinazolin-1(2H)-yl}piperidine-1-carbaldehyde
—— 2-[[2-[(4-methoxy-2,6-dimethylphenyl)sulfonyl]-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-1-yl]methoxy]-1-(3-pyridin-4-yloxypyrrolidin-1-yl)ethanone 1242847-66-0 C28H34N4O6S
2-[[2-[(4-methoxy-2,6-dimethylphenyl)sulfonyl]-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-1-yl]methoxy]-1-(3-pyridin-4-yloxypyrrolidin-1-yl)ethanone
—— N-(Cyclobutylmethyl)-2-(2-chloro-5-{[(tert-butylcarbonyl)-amino]-methyl}-phenylamino)-6-(2,2-difluoro-ethoxy)-1-methyl-1H-benzimidazole-5-carboxylic acid amide 1242269-92-6 C28H34ClF2N5O3
N-(Cyclobutylmethyl)-2-(2-chloro-5-{[(tert-butylcarbonyl)-amino]-methyl}-phenylamino)-6-(2,2-difluoro-ethoxy)-1-methyl-1H-benzimidazole-5-carboxylic acid amide
—— N-[4-(trifluoromethyl)benzyl]-9H-dipyrido[2,3-b:4',3'-f]pyrimido[4,5-d]azepin-2-amine 1246546-61-1 C22H15F3N6
N-[4-(trifluoromethyl)benzyl]-9H-dipyrido[2,3-b:4',3'-f]pyrimido[4,5-d]azepin-2-amine
—— 5-[7-(5-{4-[bis(9,9-dimethyl-9H-fluoren-2-yl)-amino]phenyl}thiophen-2-yl)benzo[1,2,-5]thiadiazol-4-yl]thiophene-2-carbaldehyde 1093862-59-9 C51H37N3OS3
5-[7-(5-{4-[bis(9,9-dimethyl-9H-fluoren-2-yl)-amino]phenyl}thiophen-2-yl)benzo[1,2,-5]thiadiazol-4-yl]thiophene-2-carbaldehyde
—— (2R,3S)-2-naphthalen-1-yl-1-(4-nitrophenyl)sulfonyl-3-phenylsulfanylpiperidine 1429866-93-2 C27H24N2O4S2
(2R,3S)-2-naphthalen-1-yl-1-(4-nitrophenyl)sulfonyl-3-phenylsulfanylpiperidine
—— 6-(2,5-dichlorophenyl)-9,9-dimethyl-6,8,10,11-tetrahydro-5H-pyrido[3,4-b][1,4]benzodiazepin-7-one 1047618-93-8 C20H19Cl2N3O
6-(2,5-dichlorophenyl)-9,9-dimethyl-6,8,10,11-tetrahydro-5H-pyrido[3,4-b][1,4]benzodiazepin-7-one
—— 1-[5-[4-[(3,4-Difluorophenyl)methoxy]-2-fluoro-phenyl]-10-hydroxy-2,2-dimethyl-4,4-dioxo-1,3,5,11-tetrahydrothiopyrano[2,3-c][1,5]benzodiazepin-6-yl]-2-(o-tolyl)ethanone 1049092-61-6 C36H33F3N2O5S
1-[5-[4-[(3,4-Difluorophenyl)methoxy]-2-fluoro-phenyl]-10-hydroxy-2,2-dimethyl-4,4-dioxo-1,3,5,11-tetrahydrothiopyrano[2,3-c][1,5]benzodiazepin-6-yl]-2-(o-tolyl)ethanone
—— N-[(1R,2S)-1-(5-fluoro-2-methyl-phenyl)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-propan-2-yl]-1-methyl-cyclopropane-1-carboxamide 1034151-37-5 C28H27F2N3O2
N-[(1R,2S)-1-(5-fluoro-2-methyl-phenyl)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-propan-2-yl]-1-methyl-cyclopropane-1-carboxamide
—— 3-[1-{4-[(4-fluorophenoxy)methyl]phenyl}-3-(2-pyridin-2-ylethyl)-1H-indol-5-yl]propanoic acid 1069045-35-7 C31H27FN2O3
3-[1-{4-[(4-fluorophenoxy)methyl]phenyl}-3-(2-pyridin-2-ylethyl)-1H-indol-5-yl]propanoic acid
—— [(3-benzylcarbamoyl-1H-indol-6-yl)-(3,5-dichloro-phenylsulphonyl)-amino]-acetic acid 1058741-25-5 C24H19Cl2N3O5S
[(3-benzylcarbamoyl-1H-indol-6-yl)-(3,5-dichloro-phenylsulphonyl)-amino]-acetic acid
—— N-[3-[(1S)-1-[[6-[4-(ethylcarbamoylamino)phenyl]pyrazin-2-yl]amino]ethyl]phenyl]pyridine-3-carboxamide 1027252-92-1 C27H27N7O2
N-[3-[(1S)-1-[[6-[4-(ethylcarbamoylamino)phenyl]pyrazin-2-yl]amino]ethyl]phenyl]pyridine-3-carboxamide
—— N-(2-(1H-1,2,3-triazol-1-yl)ethyl)-4-(7-(2-fluoro-5-methylpyridin-4-yl)benzo[b]thiophen-2-yl)pyrimidin-2-amine 1087077-00-6 C22H18FN7S
N-(2-(1H-1,2,3-triazol-1-yl)ethyl)-4-(7-(2-fluoro-5-methylpyridin-4-yl)benzo[b]thiophen-2-yl)pyrimidin-2-amine
—— [4-(5-ethanesulfonyl-pyridin-2-yloxy)-6-fluoro-1-methyl-naphthalen-2-yl]-acetic acid 1227384-58-8 C20H18FNO5S
[4-(5-ethanesulfonyl-pyridin-2-yloxy)-6-fluoro-1-methyl-naphthalen-2-yl]-acetic acid
—— tert-butyl (3-propanesulfonylaminobenzyl)-[2-[6-fluoro-3-(4-fluorobenzyl)-3,4-dihydroisoquinolin-2(1H)-yl]ethyl]carbamate 1070670-84-6 C33H41F2N3O4S
tert-butyl (3-propanesulfonylaminobenzyl)-[2-[6-fluoro-3-(4-fluorobenzyl)-3,4-dihydroisoquinolin-2(1H)-yl]ethyl]carbamate
—— tert-butyl pent-4-en-1-yl(phenyl)carbamate 1428904-08-8 C16H23NO2
tert-butyl pent-4-en-1-yl(phenyl)carbamate
—— (4-methoxyphenyl)methyl (2R)-2-[2-(1,3-benzothiazol-2-yldisulfanyl)-4-oxoazetidin-1-yl]-3-methylbut-3-enoate 118331-41-2 C23H22N2O4S3
(4-methoxyphenyl)methyl (2R)-2-[2-(1,3-benzothiazol-2-yldisulfanyl)-4-oxoazetidin-1-yl]-3-methylbut-3-enoate
—— 3-neopentyl-1-p-tolyltriazene 127316-77-2 C12H19N3
3-neopentyl-1-p-tolyltriazene
—— N-(2(R)-hydroxy-1(S)-indanyl)-5(S)-(2-furanylmethoxycarbonylamino)-4(S)-hydroxy-2(R)-(4-(2-(4-morpholino)-ethoxy)phenyl)methyl-6-cyclohexylhexanamide 138498-20-1 C40H53N3O8
N-(2(R)-hydroxy-1(S)-indanyl)-5(S)-(2-furanylmethoxycarbonylamino)-4(S)-hydroxy-2(R)-(4-(2-(4-morpholino)-ethoxy)phenyl)methyl-6-cyclohexylhexanamide
—— 4-chloro-8,9-dihydro-7H-pyrimido[4,5-b]azepine-6-carboxylic acid monohydrochloride 1428956-08-4 C9H8ClN3O2*ClH
4-chloro-8,9-dihydro-7H-pyrimido[4,5-b]azepine-6-carboxylic acid monohydrochloride
—— ethyl 6-(4-trifluoromethyl-phenyl)-5-phenyl-1,2,4-triazine-3-carboxylate 1011301-64-6 C19H14F3N3O2
ethyl 6-(4-trifluoromethyl-phenyl)-5-phenyl-1,2,4-triazine-3-carboxylate
—— N-(2-(1H-1,2,3-triazol-1-yl)ethyl)-5-fluoro-4-(7-(2-fluoro-5-((isopropyl(methyl)amino)methyl)pyridin-4-yl)benzo[b]thiophen-2-yl)pyrimidin-2-amine 1087077-57-3 C26H26F2N8S
N-(2-(1H-1,2,3-triazol-1-yl)ethyl)-5-fluoro-4-(7-(2-fluoro-5-((isopropyl(methyl)amino)methyl)pyridin-4-yl)benzo[b]thiophen-2-yl)pyrimidin-2-amine
—— 1-(4-amino-6,7-dimethoxy-quinazolin-2-yl)-4-benzyl-piperidine-4-carboxylic acid 3-trifluoromethyl-benzylamide 1227169-13-2 C31H32F3N5O3
1-(4-amino-6,7-dimethoxy-quinazolin-2-yl)-4-benzyl-piperidine-4-carboxylic acid 3-trifluoromethyl-benzylamide
—— 5-[[2,3-Difluoro-6-[(5-methyl-1,2-oxazol-3-yl)methoxy]phenyl]methoxy]-2-fluoroaniline 1075700-91-2 C18H15F3N2O3
5-[[2,3-Difluoro-6-[(5-methyl-1,2-oxazol-3-yl)methoxy]phenyl]methoxy]-2-fluoroaniline
—— N-[3-[(1S)-1-[[6-(3-methylsulfonylphenyl)pyrazin-2-yl]amino]ethyl]phenyl]-3-(trifluoromethyl)benzamide 1027256-20-7 C27H23F3N4O3S
N-[3-[(1S)-1-[[6-(3-methylsulfonylphenyl)pyrazin-2-yl]amino]ethyl]phenyl]-3-(trifluoromethyl)benzamide
—— N-[(2S)-3-amino-1-(hydroxyamino)-3-methyl-1-oxobutan-2-yl]-4-[3-[3-(hydroxymethyl)phenyl]prop-2-ynoxy]benzamide 1219366-39-8 C22H25N3O5
N-[(2S)-3-amino-1-(hydroxyamino)-3-methyl-1-oxobutan-2-yl]-4-[3-[3-(hydroxymethyl)phenyl]prop-2-ynoxy]benzamide
—— 1-[(2-amino-1-benzothiophen-3-yl)carbonyl]spiro[piperidine-4,2'-pyrano[3,2-b]pyridin]-4'(3'H)-one 1051385-13-7 C21H19N3O3S
1-[(2-amino-1-benzothiophen-3-yl)carbonyl]spiro[piperidine-4,2'-pyrano[3,2-b]pyridin]-4'(3'H)-one
—— N-{[1-(dimethylamino)cyclohexyl]methyl}pyridine-3-carboxamide 1427543-91-6 C15H23N3O
N-{[1-(dimethylamino)cyclohexyl]methyl}pyridine-3-carboxamide
—— 6-(4-{[(3,5-dicyclopentyl-4-isoxazolyl)methyl]oxy}phenyl)-2-quinolinecarboxylic acid 1020573-35-6 C30H30N2O4
6-(4-{[(3,5-dicyclopentyl-4-isoxazolyl)methyl]oxy}phenyl)-2-quinolinecarboxylic acid
—— [6-fluoro-3-methyl-4-(4-pyrimidin-2-ylpiperazine-1-carbonyl)naphthalen-2-yl]acetic acid 1227257-20-6 C22H21FN4O3
[6-fluoro-3-methyl-4-(4-pyrimidin-2-ylpiperazine-1-carbonyl)naphthalen-2-yl]acetic acid