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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-Cyclopropylthiopyrano[3,2-b][1]benzothiol-4-one 1207479-47-7 C14H10OS2
2-Cyclopropylthiopyrano[3,2-b][1]benzothiol-4-one
—— 1-(4-{7-[2-(isopropylamino)ethyl]-4-morpholin-4-yl-7H-pyrrolo[2,3-d]pyrimidin-2-yl}phenyl)-3-pyridin-4-ylurea 1202884-75-0 C27H32N8O2
1-(4-{7-[2-(isopropylamino)ethyl]-4-morpholin-4-yl-7H-pyrrolo[2,3-d]pyrimidin-2-yl}phenyl)-3-pyridin-4-ylurea
—— 1-ethyl-3-[4-fluoro-5-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-7-(pyridin-2-yl)-1,3-benzothiazol-2-yl]urea 1202806-21-0 C27H27FN6O2S
1-ethyl-3-[4-fluoro-5-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-7-(pyridin-2-yl)-1,3-benzothiazol-2-yl]urea
—— (R,S)-9-cyclopentyl-2-(1-(2-fluorophenyl)ethylamino)-5,7,7-trimethyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1204831-41-3 C23H30FN5O
(R,S)-9-cyclopentyl-2-(1-(2-fluorophenyl)ethylamino)-5,7,7-trimethyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one
—— 1-(2,4-difluorobenzyl)-3-(3-fluorophenyl)cinnolin-4(1H)-one 1204652-52-7 C21H13F3N2O
1-(2,4-difluorobenzyl)-3-(3-fluorophenyl)cinnolin-4(1H)-one
—— 2-[4-[4-(2-methyl-10H-thieno[2,3-b][1,5]benzodiazepin-4-yl)piperazin-1-yl]butyl]-2-azaspiro[4.4]nonane-1,3-dione 1417032-29-1 C28H35N5O2S
2-[4-[4-(2-methyl-10H-thieno[2,3-b][1,5]benzodiazepin-4-yl)piperazin-1-yl]butyl]-2-azaspiro[4.4]nonane-1,3-dione
—— 3-Ethyl-2-methylthio-7-[4-(4-morpholinoethoxybenzoyl)benzyl]-7H-pyrrolo[2,3-d]pyrimidin-4-one-hydrochloride 183170-00-5 C29H32N4O4S*ClH
3-Ethyl-2-methylthio-7-[4-(4-morpholinoethoxybenzoyl)benzyl]-7H-pyrrolo[2,3-d]pyrimidin-4-one-hydrochloride
—— 5-(4-cyclohexylthiazol-2-yl)-6-ethyl-4-(4-hydroxyphenyl)-3,4-dihydropyrimidin-2(1H)-one 1224736-10-0 C21H25N3O2S
5-(4-cyclohexylthiazol-2-yl)-6-ethyl-4-(4-hydroxyphenyl)-3,4-dihydropyrimidin-2(1H)-one
—— (3R)-1-diazo-3-methyl-7-phenylmethoxyheptan-2-one 1424403-33-7 C15H20N2O2
(3R)-1-diazo-3-methyl-7-phenylmethoxyheptan-2-one
—— ((1S,2R,3R)-2-iodo-1-methyl-3-phenethylcyclopropyl)methyl 3,5-dinitrobenzoate 1433964-32-9 C20H19IN2O6
((1S,2R,3R)-2-iodo-1-methyl-3-phenethylcyclopropyl)methyl 3,5-dinitrobenzoate
—— —— 1195780-72-3 C28H46O3
—— 2-(2-(3-fluorophenyl)piperidin-1-yl)pyridine 1478114-68-9 C16H17FN2
2-(2-(3-fluorophenyl)piperidin-1-yl)pyridine
—— <i>O</i><sup>2</sup>,<i>O</i><sup>4</sup>;<i>O</i><sup>3</sup>,<i>O</i><sup>5</sup>-((<i>R,S</i>)-diethylLiDene)-D-xylose-dibutyldithioacetal 101592-24-9 C17H32O4S2
<i>O</i><sup>2</sup>,<i>O</i><sup>4</sup>;<i>O</i><sup>3</sup>,<i>O</i><sup>5</sup>-((<i>R,S</i>)-diethylLiDene)-D-xylose-dibutyldithioacetal
—— 1-ethyl-5-[5-(1H-indol-2-yl)-1,2,4-oxadiazol-3-yl]-1H-benzimidazole 1185150-36-0 C19H15N5O
1-ethyl-5-[5-(1H-indol-2-yl)-1,2,4-oxadiazol-3-yl]-1H-benzimidazole
—— 3-(1,3-Benzothiazol-2(3H)-ylidene)anthracen-2(3H)-one 116646-52-7 C21H13NOS
3-(1,3-Benzothiazol-2(3H)-ylidene)anthracen-2(3H)-one
—— N-(4-(-6H-pyrrolo[2,3-e][1,2,4]triazolo[4,3-a]pyrazin-1-yl)bicyclo[2.2.2]octan-1-yl)cyclopropanecarboxamide 1201182-84-4 C19H22N6O
N-(4-(-6H-pyrrolo[2,3-e][1,2,4]triazolo[4,3-a]pyrazin-1-yl)bicyclo[2.2.2]octan-1-yl)cyclopropanecarboxamide
—— 5-[2-(4-Methoxyphenyl)hydrazinylidene]-3-oxo-3,5-dihydronaphthalene-2-carboxylic acid 144337-62-2 C18H14N2O4
5-[2-(4-Methoxyphenyl)hydrazinylidene]-3-oxo-3,5-dihydronaphthalene-2-carboxylic acid
—— Benzoic acid, 3-fluoro-5-(3-piperidinyl)- 1260863-47-5 C12H14FNO2
Benzoic acid, 3-fluoro-5-(3-piperidinyl)-
—— 4-{3-[1-(5-chloro-pyrimidin-2-yl)piperidin-4-yl]propoxy}-N-(2-hydroxy-1-hydroxymethyl-1-methyl-ethyl)-2,6-dimethyl-benzamide 1204335-16-9 C25H35ClN4O4
4-{3-[1-(5-chloro-pyrimidin-2-yl)piperidin-4-yl]propoxy}-N-(2-hydroxy-1-hydroxymethyl-1-methyl-ethyl)-2,6-dimethyl-benzamide
—— KNI-1366 1179355-10-2 C32H36FN3O5S
KNI-1366
—— 1-(3-isopropyl-[1,2,4]oxadiazol-5-yl)-4-{3-[4-(5-methyltetrazol-1-yl)-phenoxy]propyl}piperidine 1204309-49-8 C21H29N7O2
1-(3-isopropyl-[1,2,4]oxadiazol-5-yl)-4-{3-[4-(5-methyltetrazol-1-yl)-phenoxy]propyl}piperidine
—— 3-(hydroxymethyl)-8-morpholino-2-(phenylamino)-4H-pyrido[1,2-a]pyrimidin-4-one 1204420-57-4 C19H20N4O3
3-(hydroxymethyl)-8-morpholino-2-(phenylamino)-4H-pyrido[1,2-a]pyrimidin-4-one
—— 9-[2-(3-methoxy-phenyl)-2-oxo-ethyl]-2-pyrimidin-4-yl-9,10-dihydro-1,4a,9-triaza-anthracen-4-one 1202406-29-8 C24H19N5O3
9-[2-(3-methoxy-phenyl)-2-oxo-ethyl]-2-pyrimidin-4-yl-9,10-dihydro-1,4a,9-triaza-anthracen-4-one
—— 2,7-bis(5-(2-methoxybenzylamino)pentyl)benzo[lmn][3,8]phenanthroline-1,3,6,8(2H,7H)-tetraone 1191058-82-8 C40H44N4O6
2,7-bis(5-(2-methoxybenzylamino)pentyl)benzo[lmn][3,8]phenanthroline-1,3,6,8(2H,7H)-tetraone
—— 1-N-[4-(2-fluorophenyl)piperazin-1-yl]carbonylethyl-2-phenylimidazole 1202777-98-7 C22H23FN4O
1-N-[4-(2-fluorophenyl)piperazin-1-yl]carbonylethyl-2-phenylimidazole
—— (2S,3R)-N,3-dihydroxy-2-[3-oxo-7-[[4-(2-phenylethynyl)phenyl]methyl]-5,6,8,8a-tetrahydro-1H-imidazo[1,5-a]pyrazin-2-yl]butanamide 1202236-53-0 C25H28N4O4
(2S,3R)-N,3-dihydroxy-2-[3-oxo-7-[[4-(2-phenylethynyl)phenyl]methyl]-5,6,8,8a-tetrahydro-1H-imidazo[1,5-a]pyrazin-2-yl]butanamide
—— (S)-2-(3-(2,5-difluorophenyl)-5-ethyl-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine-1-carboxamido)-3,3-dimethylbutanoic acid 1231909-33-3 C21H26F2N4O3
(S)-2-(3-(2,5-difluorophenyl)-5-ethyl-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridine-1-carboxamido)-3,3-dimethylbutanoic acid
—— 1-(4-amino-6,7-dimethoxy-quinazolin-2-yl)-4-(4-chloro-benzyl)-piperidine-4-carboxylic acid benzylamide 1227168-94-6 C30H32ClN5O3
1-(4-amino-6,7-dimethoxy-quinazolin-2-yl)-4-(4-chloro-benzyl)-piperidine-4-carboxylic acid benzylamide
—— 6-chloro-2-fluoro-3-(3-fluoropropylsulfonamido)-N-(3-(2-methoxyethoxy)-1H-pyrazolo[3,4-b]pyridin-5-yl)benzamide 1186607-77-1 C19H20ClF2N5O5S
6-chloro-2-fluoro-3-(3-fluoropropylsulfonamido)-N-(3-(2-methoxyethoxy)-1H-pyrazolo[3,4-b]pyridin-5-yl)benzamide
—— 3-benzyloxy-5-bromo-2-(4-methanesulfonylphenoxymethyl)pyridine 1206968-87-7 C20H18BrNO4S
3-benzyloxy-5-bromo-2-(4-methanesulfonylphenoxymethyl)pyridine
—— 6-[({5-[(E)-Phenyldiazenyl]pyridin-2-yl}amino)methylidene]cyclohexa-2,4-dien-1-one 140116-13-8 C18H14N4O
6-[({5-[(E)-Phenyldiazenyl]pyridin-2-yl}amino)methylidene]cyclohexa-2,4-dien-1-one
—— 6-[2-(3,5-Di-tert-butyl-4-chloro-2-nitrophenyl)hydrazinylidene]cyclohexa-2,4-dien-1-one 106085-68-1 C20H24ClN3O3
6-[2-(3,5-Di-tert-butyl-4-chloro-2-nitrophenyl)hydrazinylidene]cyclohexa-2,4-dien-1-one
—— {2',6'-dimethyl-4'-[3-(methylthio)propoxy]-6-phenoxybiphenyl-3-yl}methanol 1000414-15-2 C25H28O3S
{2',6'-dimethyl-4'-[3-(methylthio)propoxy]-6-phenoxybiphenyl-3-yl}methanol
—— 2-(carbamoylamino)-N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-(3-methoxyphenyl)propan-2-yl]acetamide 1034152-52-7 C26H26FN5O4
2-(carbamoylamino)-N-[(1R,2S)-1-[1-(4-fluorophenyl)indazol-5-yl]oxy-1-(3-methoxyphenyl)propan-2-yl]acetamide
—— allyl (4R,5S,6S)-3-[(2R,4S)-1-allyloxycarbonyl-2-{2-(pyridin-2-yl)ethyl}pyrrolidin-4-yl]thio-6-[(1R)-1-hydroxyethyl]-4-methyl-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylate 156442-69-2 C28H35N3O6S
allyl (4R,5S,6S)-3-[(2R,4S)-1-allyloxycarbonyl-2-{2-(pyridin-2-yl)ethyl}pyrrolidin-4-yl]thio-6-[(1R)-1-hydroxyethyl]-4-methyl-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylate
—— 2-fluoro-N-(2'-methoxy-5'-(4-methyl-5-oxo-4,5-dihydro-1,3,4-oxadiazol-2-yl)-[1,1'-biphenyl]-4-yl)-6-methylbenzamide 1373938-42-1 C24H20FN3O4
2-fluoro-N-(2'-methoxy-5'-(4-methyl-5-oxo-4,5-dihydro-1,3,4-oxadiazol-2-yl)-[1,1'-biphenyl]-4-yl)-6-methylbenzamide
—— 2,3-dihydro-benzofuran-4-carboxylic acid {(1S,3S,5S)-2-[2-cyclopropyl-5-(4-fluoro-phenyl)-thiazole-4-carbonyl]-2-aza-bicyclo[3.1.0]hex-3-ylmethyl}-amide 1038508-03-0 C28H26FN3O3S
2,3-dihydro-benzofuran-4-carboxylic acid {(1S,3S,5S)-2-[2-cyclopropyl-5-(4-fluoro-phenyl)-thiazole-4-carbonyl]-2-aza-bicyclo[3.1.0]hex-3-ylmethyl}-amide
—— tert-butyl [(3-carbamoyl-1-methyl-1H-indol-6-yl)-(3,5-dichloro-phenylsulphonyl)-amino]-acetate 1058739-11-9 C22H23Cl2N3O5S
tert-butyl [(3-carbamoyl-1-methyl-1H-indol-6-yl)-(3,5-dichloro-phenylsulphonyl)-amino]-acetate
—— (S)-4-[3-methyl-2-(3-trifluoromethylphenyl)butyl]-4,5-dihydrooxazol-2-ylamine 1043494-37-6 C15H19F3N2O
(S)-4-[3-methyl-2-(3-trifluoromethylphenyl)butyl]-4,5-dihydrooxazol-2-ylamine
—— methyl 5-[tert-butoxycarbonylmethyl-(3,5-dichloro-phenylsulphonyl)-amino]-benzo[b]thiophen-2-carboxylate 1058738-88-7 C22H21Cl2NO6S2
methyl 5-[tert-butoxycarbonylmethyl-(3,5-dichloro-phenylsulphonyl)-amino]-benzo[b]thiophen-2-carboxylate
—— N-[4-(2,7-diazaspiro[4.5]decan-7-yl)pyridin-3-yl]-2-(5-methoxy-3-oxo-1H-isoindol-2-yl)-1,3-thiazole-4-carboxamide 1023297-67-7 C26H28N6O3S
N-[4-(2,7-diazaspiro[4.5]decan-7-yl)pyridin-3-yl]-2-(5-methoxy-3-oxo-1H-isoindol-2-yl)-1,3-thiazole-4-carboxamide
—— 6-(1-methylpyrazol-4-yl)-7-(pyridin-3-ylmethoxy)-N-[3-(1,2,4-triazol-1-ylmethyl)phenyl]quinazolin-2-amine 1202035-24-2 C27H23N9O
6-(1-methylpyrazol-4-yl)-7-(pyridin-3-ylmethoxy)-N-[3-(1,2,4-triazol-1-ylmethyl)phenyl]quinazolin-2-amine
—— 2,8-dimethyl-5-(3-methoxyphenylethynyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole 1061353-39-6 C22H22N2O
2,8-dimethyl-5-(3-methoxyphenylethynyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
—— N<sup>4</sup>-(6,6-dimethyl-5-{[(2S)-2,4,5,5-tetramethylpiperazin-1-yl]carbonyl}-1,4,5,6-tetrahydropyrrolo[3 ,4-c]pyrazol-3-yl)-N<sup>2</sup>,N<sup>2</sup>-dimethylpyrimidine-2,4-diamine 1046786-66-6 C22H35N9O
N<sup>4</sup>-(6,6-dimethyl-5-{[(2S)-2,4,5,5-tetramethylpiperazin-1-yl]carbonyl}-1,4,5,6-tetrahydropyrrolo[3 ,4-c]pyrazol-3-yl)-N<sup>2</sup>,N<sup>2</sup>-dimethylpyrimidine-2,4-diamine
—— 6-(4-chloro-1H-pyrrolo[2,3-b]pyridin-5-yl)-3-cyclohex-1-en-1-yl-1-[(2S)-1,4-dioxan-2-ylmethyl]-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one 1207626-16-1 C24H24ClN5O3
6-(4-chloro-1H-pyrrolo[2,3-b]pyridin-5-yl)-3-cyclohex-1-en-1-yl-1-[(2S)-1,4-dioxan-2-ylmethyl]-1,3-dihydro-2H-imidazo[4,5-b]pyridin-2-one
—— (+/-)-(3-hydroxyquinoxalin-2-yl)[2-(pyridin-3-ylmethyl)pyrrolidin-1-yl]methanone 1374848-73-3 C19H18N4O2
(+/-)-(3-hydroxyquinoxalin-2-yl)[2-(pyridin-3-ylmethyl)pyrrolidin-1-yl]methanone
—— Methyl 4-[5-chloro-2-(3-methyloxiran-2-yl)benzoyl]benzoate 1370529-43-3 C18H15ClO4
Methyl 4-[5-chloro-2-(3-methyloxiran-2-yl)benzoyl]benzoate
—— 6-(4-hydroxy-phenyl)-1H-pyrazolo[3,4-b]pyridine-4-carboxylic acid (1-aza-bicyclo[2.2.2]oct-3-yl)-amide 1431977-86-4 C20H21N5O2
6-(4-hydroxy-phenyl)-1H-pyrazolo[3,4-b]pyridine-4-carboxylic acid (1-aza-bicyclo[2.2.2]oct-3-yl)-amide
—— N-[(1R)-1-phenylpropyl]-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-12-amine 1226548-37-3 C18H19N3S
N-[(1R)-1-phenylpropyl]-7-thia-9,11-diazatricyclo[6.4.0.02,6]dodeca-1(12),2(6),8,10-tetraen-12-amine
—— 3-[7-(4-fluorophenyl)imidazo[1,2-a]pyridin-3-yl]-N-(2,2,2-trifluoroethylsulfamoyl)aniline 1036985-47-3 C21H16F4N4O2S
3-[7-(4-fluorophenyl)imidazo[1,2-a]pyridin-3-yl]-N-(2,2,2-trifluoroethylsulfamoyl)aniline