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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-(4-(5-ethoxycarbonyl-[1,2,4]oxadiazol-3-yl)-2-fluorophenyl)piperazine-1-carboxylic acid tert-butyl ester 1163247-98-0 C20H25FN4O5
4-(4-(5-ethoxycarbonyl-[1,2,4]oxadiazol-3-yl)-2-fluorophenyl)piperazine-1-carboxylic acid tert-butyl ester
—— 5-(2-(3-(1-(benzylamino)ethyl)phenylamino)-5-methylpyrimidin-4-ylamino)benzo[d]oxazol-2(3H)-one 1236665-27-2 C27H26N6O2
5-(2-(3-(1-(benzylamino)ethyl)phenylamino)-5-methylpyrimidin-4-ylamino)benzo[d]oxazol-2(3H)-one
—— 4-[2-amino-5-(trifluoromethyl)thieno[2,3-d]pyrimidin-4-yl]piperazine-1-carboxylic acid (4-methoxy-2-methylphenyl)amide 1423163-30-7 C20H21F3N6O2S
4-[2-amino-5-(trifluoromethyl)thieno[2,3-d]pyrimidin-4-yl]piperazine-1-carboxylic acid (4-methoxy-2-methylphenyl)amide
—— 1-cyclopropyl-6-fluoro-8-methoxy-4-oxo-7-(7-oxo-8H-1,8-naphthyridin-3-yl)quinoline-3-carboxylic acid 1426216-12-7 C22H16FN3O5
1-cyclopropyl-6-fluoro-8-methoxy-4-oxo-7-(7-oxo-8H-1,8-naphthyridin-3-yl)quinoline-3-carboxylic acid
—— tert-butyl N-[(2S)-1-[(2S,4R)-4-[[9-chloro-2-[2-(2-hydroxypropan-2-yl)-1,3-thiazol-4-yl]-8-methoxy-[1]benzofuro[3,2-b]pyridin-4-yl]oxy]-2-[[(1R,2S)-1-(cyclopropylsulfonylcarbamoyl)-2-ethenylcyclopropyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]carbamate 1421605-23-3 C43H53ClN6O11S2
tert-butyl N-[(2S)-1-[(2S,4R)-4-[[9-chloro-2-[2-(2-hydroxypropan-2-yl)-1,3-thiazol-4-yl]-8-methoxy-[1]benzofuro[3,2-b]pyridin-4-yl]oxy]-2-[[(1R,2S)-1-(cyclopropylsulfonylcarbamoyl)-2-ethenylcyclopropyl]carbamoyl]pyrrolidin-1-yl]-3,3-dimethyl-1-oxobutan-2-yl]carbamate
—— N-[2-(2-amino-3H-benzimidazol-5-ylcarbamoyl)-1-(3,5-dimethoxyphenyl)-2-hydroxyethyl]-4-diethyl-aminobenzamide 1013416-54-0 C29H34N6O5
N-[2-(2-amino-3H-benzimidazol-5-ylcarbamoyl)-1-(3,5-dimethoxyphenyl)-2-hydroxyethyl]-4-diethyl-aminobenzamide
—— 5-[1-[3-(trifluoromethyl)phenyl]-1H-benzimidazol-6-yl]-1,3,4-oxadiazol-2-amine 1005204-59-0 C16H10F3N5O
5-[1-[3-(trifluoromethyl)phenyl]-1H-benzimidazol-6-yl]-1,3,4-oxadiazol-2-amine
—— methyl 3-chloro-4-[5-(5-methyl-1,3,4-oxadiazol-2-yl)-1-benzofuran-3-yl]benzoate 1005203-44-0 C19H13ClN2O4
methyl 3-chloro-4-[5-(5-methyl-1,3,4-oxadiazol-2-yl)-1-benzofuran-3-yl]benzoate
—— 2-[[5-(2,3-dihydro-1-benzofuran-5-yl)-1,3,4-oxadiazol-2-yl]thio]-N,N-diethylacetamide 1005200-68-9 C16H19N3O3S
2-[[5-(2,3-dihydro-1-benzofuran-5-yl)-1,3,4-oxadiazol-2-yl]thio]-N,N-diethylacetamide
—— 1-(2-(4-(4-(1,2,2,6,6-pentamethylpiperidin-4-ylamino)-5-fluoropyrimidin-2-ylamino)-2-(difluoromethoxy)phenoxy)ethyl)pyrrolidin-2-one 1239593-61-3 C27H37F3N6O3
1-(2-(4-(4-(1,2,2,6,6-pentamethylpiperidin-4-ylamino)-5-fluoropyrimidin-2-ylamino)-2-(difluoromethoxy)phenoxy)ethyl)pyrrolidin-2-one
—— 2-{[(2R)-5-amino-2,3-dihydro-1H-inden-2-yl](methyl)amino}ethanol 1092794-24-5 C12H18N2O
2-{[(2R)-5-amino-2,3-dihydro-1H-inden-2-yl](methyl)amino}ethanol
—— 3-methyl-N-(3-morpholinopropyl)imidazo[1,2-b]pyridazin-6-amine fumarate 1034622-11-1 C4H4O4*C14H21N5O
3-methyl-N-(3-morpholinopropyl)imidazo[1,2-b]pyridazin-6-amine fumarate
—— [5-(4-bromo-phenyl)-3-methyl-isoxazol-4-yl]-carbamic acid 1-(3-cyano-phenyl)-ethyl ester 1257213-91-4 C20H16BrN3O3
[5-(4-bromo-phenyl)-3-methyl-isoxazol-4-yl]-carbamic acid 1-(3-cyano-phenyl)-ethyl ester
—— (S)-1-(2-(carboxymethoxy)-5-chlorophenyl)-6-fluoro-3,4-dihydro-1H-isoquinoline-2-carboxylic acid benzooxazol-2-ylmethyl ester 1355057-20-3 C26H20ClFN2O6
(S)-1-(2-(carboxymethoxy)-5-chlorophenyl)-6-fluoro-3,4-dihydro-1H-isoquinoline-2-carboxylic acid benzooxazol-2-ylmethyl ester
—— (1R,2R,3S,5R)-2-(5-chloro-2-((3,4-dihydro-4-(2-(dimethylamino)ethyl)-2H-benzo[b][1,4]oxazin-7-yl)amino)pyrimidin-4-ylamino)-N,2,6,6-tetramethylbicyclo[3.1.1]heptane-3-carboxamide 1019639-92-9 C28H40ClN7O2
(1R,2R,3S,5R)-2-(5-chloro-2-((3,4-dihydro-4-(2-(dimethylamino)ethyl)-2H-benzo[b][1,4]oxazin-7-yl)amino)pyrimidin-4-ylamino)-N,2,6,6-tetramethylbicyclo[3.1.1]heptane-3-carboxamide
—— N4-(3-n-propylbenzo[d]oxazol-2(3H)-on-5-yl)-N2-((3-methylsulfonyl)phenyl)-5-methylpyrimidine-2,4-diamine 1236662-56-8 C22H23N5O4S
N4-(3-n-propylbenzo[d]oxazol-2(3H)-on-5-yl)-N2-((3-methylsulfonyl)phenyl)-5-methylpyrimidine-2,4-diamine
—— tert-butyl 3-{6-[(2-methylphenyl)sulfanyl]-2H-spiro[1-benzofuran-3,4'-piperidine]-1'-yl}propanoate 1355090-05-9 C26H33NO3S
tert-butyl 3-{6-[(2-methylphenyl)sulfanyl]-2H-spiro[1-benzofuran-3,4'-piperidine]-1'-yl}propanoate
—— (S)-tert-butyl (1-(benzyloxy)-5-((tertbutyldimethylsilyl)oxy)pentan-2-yl)carbamate 1400659-38-2 C23H41NO4Si
(S)-tert-butyl (1-(benzyloxy)-5-((tertbutyldimethylsilyl)oxy)pentan-2-yl)carbamate
—— (S)-2-((R)-(4-chlorophenyl)(hydroxy)methyl)cycloheptanone 1413142-52-5 C14H17ClO2
(S)-2-((R)-(4-chlorophenyl)(hydroxy)methyl)cycloheptanone
—— 7-(2-cyano-3-(pyridin-4-yl)guanidino)-N-(tetrahydrofuran-3-yloxy)heptanamide 1170234-93-1 C18H26N6O3
7-(2-cyano-3-(pyridin-4-yl)guanidino)-N-(tetrahydrofuran-3-yloxy)heptanamide
—— 7-hydroxy-1-isopropyl-6-methoxy-1,2,3,4-tetrahydroisoquinoline 1032822-09-5 C13H19NO2
7-hydroxy-1-isopropyl-6-methoxy-1,2,3,4-tetrahydroisoquinoline
—— 5-fluoro-N4-(1,2,2,6,6-pentamethylpiperidin-4-yl)-N2-(3,4,5-trifluorophenyl)-2,4-pyrimidinediamine 1105123-02-1 C20H25F4N5
5-fluoro-N4-(1,2,2,6,6-pentamethylpiperidin-4-yl)-N2-(3,4,5-trifluorophenyl)-2,4-pyrimidinediamine
—— 4-(imidazo[1,2-a]pyridin-2-ylmethoxy)-1-(9-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-7-yl)pyridin-2(1H)-one hydrochloride 1173153-13-3 C25H23N5O2*ClH
4-(imidazo[1,2-a]pyridin-2-ylmethoxy)-1-(9-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-7-yl)pyridin-2(1H)-one hydrochloride
—— 2-fluoro-iodo-phenyl acetic acid 1261675-21-1 C8H6FIO2
2-fluoro-iodo-phenyl acetic acid
—— Arylpyrazole, 24 1174985-66-0 C22H24F3N5
Arylpyrazole, 24
—— 3-[4-chloro-5-({isopropyl[(3R)-piperidin-3-yl]amino}carbonyl)-2-methoxyphenoxy]propanoic acid hydrochloride 1044559-41-2 C19H27ClN2O5*ClH
3-[4-chloro-5-({isopropyl[(3R)-piperidin-3-yl]amino}carbonyl)-2-methoxyphenoxy]propanoic acid hydrochloride
—— 5-(2-(3-fluoro-5-morpholinophenylamino)-5-methylpyrimidin-4-ylamino)benzo[d]oxazol-2(3H)-one 1236665-54-5 C22H21FN6O3
5-(2-(3-fluoro-5-morpholinophenylamino)-5-methylpyrimidin-4-ylamino)benzo[d]oxazol-2(3H)-one
—— N4-(benzoxazolin-2-on-5-yl)-N2-(3,4,5-trimethoxyphenyl)-5-fluoropyrimidine-2,4-diamine 1236664-30-4 C20H18FN5O5
N4-(benzoxazolin-2-on-5-yl)-N2-(3,4,5-trimethoxyphenyl)-5-fluoropyrimidine-2,4-diamine
—— 1-cyano-cyclopropanecarboxylic acid {5-[3-(5-chloro-thiophen-2-ylmethyl)-ureido]-[1,2,4]thiadiazol-3-ylmethyl}-methyl-amide 1108711-49-4 C15H15ClN6O2S2
1-cyano-cyclopropanecarboxylic acid {5-[3-(5-chloro-thiophen-2-ylmethyl)-ureido]-[1,2,4]thiadiazol-3-ylmethyl}-methyl-amide
—— Ethyl 2-[[2-[1-[(4-hydroxy-3-propan-2-ylphenyl)methyl]-2-methylindol-3-yl]acetyl]amino]acetate 1170718-93-0 C25H30N2O4
Ethyl 2-[[2-[1-[(4-hydroxy-3-propan-2-ylphenyl)methyl]-2-methylindol-3-yl]acetyl]amino]acetate
—— (6-bromo-pyrazolo[1,5-a]pyrimidin-2-yl)-(1,6-dimethyl-3,4-dihydro-1H-furo[3,2-c]pyridazin-2-yl)-methanone 1174648-91-9 C15H14BrN5O2
(6-bromo-pyrazolo[1,5-a]pyrimidin-2-yl)-(1,6-dimethyl-3,4-dihydro-1H-furo[3,2-c]pyridazin-2-yl)-methanone
—— N-[3-(10H-dipyrido[3,4-b:3',4'-e][1,4]thiazin-10-yl)propyl]methanesulfonamide 1320136-91-1 C14H16N4O2S2
N-[3-(10H-dipyrido[3,4-b:3',4'-e][1,4]thiazin-10-yl)propyl]methanesulfonamide
—— cyclopropyl-[5"-(3-methoxy-phenyl)-[2,2';4',3'']terpyridin-6'-yl]-amine 1171040-21-3 C25H22N4O
cyclopropyl-[5"-(3-methoxy-phenyl)-[2,2';4',3'']terpyridin-6'-yl]-amine
—— O-((4-chlorobiphenyl-2-yl)methyl)hydroxylamine 1160488-30-1 C13H12ClNO
O-((4-chlorobiphenyl-2-yl)methyl)hydroxylamine
—— 3-(4-(trifluoromethoxy)phenethyl)-2-(3,4-dichlorophenyl)-1-methylimidazolidin-4-one 1162339-66-3 C19H17Cl2F3N2O2
3-(4-(trifluoromethoxy)phenethyl)-2-(3,4-dichlorophenyl)-1-methylimidazolidin-4-one
—— 3-(5-chloro-2-fluorophenyl)-5-(4-methoxyphenoxy)-1,3,4-oxadiazol-2(3H)-one 1169938-41-3 C15H10ClFN2O4
3-(5-chloro-2-fluorophenyl)-5-(4-methoxyphenoxy)-1,3,4-oxadiazol-2(3H)-one
—— 5-(2-(3-methoxy-5-methylphenylamino)-5-methylpyrimidin-4-ylamino)benzo[d]oxazol-2(3H)-one 1236665-73-8 C20H19N5O3
5-(2-(3-methoxy-5-methylphenylamino)-5-methylpyrimidin-4-ylamino)benzo[d]oxazol-2(3H)-one
—— 4-[[[9-(4-Chlorobutyl)purin-6-yl]amino]methyl]-2-methoxyphenol 1167446-64-1 C17H20ClN5O2
4-[[[9-(4-Chlorobutyl)purin-6-yl]amino]methyl]-2-methoxyphenol
—— O-((4’-chlorobiphenyl-2-yl)methyl)hydroxylamine 1160488-08-3 C13H12ClNO
O-((4’-chlorobiphenyl-2-yl)methyl)hydroxylamine
—— 1-methyl-5-[5-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-5,8-diazaspiro[2.6]nonane-8-carbonyl]pyrrole-2-sulfonamide 1354624-14-8 C19H23N7O3S
1-methyl-5-[5-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-5,8-diazaspiro[2.6]nonane-8-carbonyl]pyrrole-2-sulfonamide
—— 3-[5-(cyclohexylmethoxy)-2H-spiro[1-benzofuran-3,4'-piperidine]-1'-yl]propanoic acid hydrochloride 1355084-10-4 C22H31NO4*ClH
3-[5-(cyclohexylmethoxy)-2H-spiro[1-benzofuran-3,4'-piperidine]-1'-yl]propanoic acid hydrochloride
—— 5-(4-chlorophenyl)-3-(1-methylethyl)imino-2-(3-nitro-2-pyridyl)amino-3,5-dihydrophenazine 1353735-05-3 C26H21ClN6O2
5-(4-chlorophenyl)-3-(1-methylethyl)imino-2-(3-nitro-2-pyridyl)amino-3,5-dihydrophenazine
—— 1-methyl-5-[5-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-5,8-diazaspiro[2.6]nonane-8-carbonyl]pyrrole-3-sulfonamide 1354624-15-9 C19H23N7O3S
1-methyl-5-[5-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-5,8-diazaspiro[2.6]nonane-8-carbonyl]pyrrole-3-sulfonamide
—— 6-(4-pyridinyl)-2-pyridinyl 5-thio-β-D-xylopyranoside 1012082-09-5 C15H16N2O4S
6-(4-pyridinyl)-2-pyridinyl 5-thio-β-D-xylopyranoside
—— methyl-[5"-(4-morpholin-4-ylmethyl-phenyl)-[2,2';4',3"]terpyridin-6'-yl]-amine 1171039-79-4 C27H27N5O
methyl-[5"-(4-morpholin-4-ylmethyl-phenyl)-[2,2';4',3"]terpyridin-6'-yl]-amine
—— 4-benzamido-2,5-dimethoxybenzenediazonium;dichlorozinc;dichloride 14726-29-5 C15H14Cl4N3O3Zn-
4-benzamido-2,5-dimethoxybenzenediazonium;dichlorozinc;dichloride
—— 4-(3-(3-(2-ethyl-8-(trifluoromethyl)imidazo[1,2-a]pyridin-3-yl)phenoxy)phenylsulfonyl)-2-methylbutan-2-ol 1167570-93-5 C27H27F3N2O4S
4-(3-(3-(2-ethyl-8-(trifluoromethyl)imidazo[1,2-a]pyridin-3-yl)phenoxy)phenylsulfonyl)-2-methylbutan-2-ol
—— 2-ethyl-3-(3-(3-fluoro-5-(methylsulfonyl)phenoxy)phenyl)-8-(trifluoromethyl)imidazo[1,2-a]pyridine 1167570-95-7 C23H18F4N2O3S
2-ethyl-3-(3-(3-fluoro-5-(methylsulfonyl)phenoxy)phenyl)-8-(trifluoromethyl)imidazo[1,2-a]pyridine
—— 1-[(3,4-dichlorophenyl)methyl]-2-methyl-N-[3-methyl-1-(2-thienyl)butyl]-1H-benzimidazole-5-carboxamide 1168138-31-5 C25H25Cl2N3OS
1-[(3,4-dichlorophenyl)methyl]-2-methyl-N-[3-methyl-1-(2-thienyl)butyl]-1H-benzimidazole-5-carboxamide
—— (R)-6-(1-methyl-1H-pyrazol-4-yl)-2-(3-(piperidin-1-yl)pyrrolidin-1-yl)benzo[d]thiazole 1161730-59-1 C20H25N5S
(R)-6-(1-methyl-1H-pyrazol-4-yl)-2-(3-(piperidin-1-yl)pyrrolidin-1-yl)benzo[d]thiazole