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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-propylphenyl]amino}-4-pyrimidinyl)imidazo-[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide 1089279-32-2 C43H44F2N8O
3-[3-(2-{[4-(1,4'-bipiperidin-1'-yl)-2-propylphenyl]amino}-4-pyrimidinyl)imidazo-[1,2-a]pyridin-2-yl]-N-(2,6-difluorophenyl)benzamide
—— tetraethyl [2-(2,3-dihydro-2-oxoindene-1-yl)ethylidene]bisphosphonate 1353722-33-4 C19H30O7P2
tetraethyl [2-(2,3-dihydro-2-oxoindene-1-yl)ethylidene]bisphosphonate
—— ((1R,2R,3S,4R)-4-(6-benzamido-9H-purin-9-yl)-2-(benzoyloxy)-3-(((trifluoromethyl)sulfonyl)oxy)cyclopentyl)methyl benzoate 118149-20-5 C33H26F3N5O8S
((1R,2R,3S,4R)-4-(6-benzamido-9H-purin-9-yl)-2-(benzoyloxy)-3-(((trifluoromethyl)sulfonyl)oxy)cyclopentyl)methyl benzoate
—— ethyl 3-[4-(1,2,4-triazol-1-yl)phenyl]propanoate 143426-73-7 C13H15N3O2
ethyl 3-[4-(1,2,4-triazol-1-yl)phenyl]propanoate
—— N-(2-(4-(2,3-dichlorophenyl)piperazin-1-yl)ethyl)-2-methyl-5-phenyl-1-propyl-1H-pyrrole-3-carboxamide hydrochloride 1220949-28-9 C27H32Cl2N4O*ClH
N-(2-(4-(2,3-dichlorophenyl)piperazin-1-yl)ethyl)-2-methyl-5-phenyl-1-propyl-1H-pyrrole-3-carboxamide hydrochloride
—— (2S,3R)-2-amino-3-hydroxy-N-(4-(octyloxy)phenyl)butanamide 1218815-87-2 C18H30N2O3
(2S,3R)-2-amino-3-hydroxy-N-(4-(octyloxy)phenyl)butanamide
—— 2-(5-(4-bromophenyl)-1-(2-chlorophenyl)-4-(methylsulfonyl)-1H-pyrazol-3-yl)-5-(1-(4-chlorophenyl)cyclopropyl)-1,3,4-oxadiazole 1219736-76-1 C27H19BrCl2N4O3S
2-(5-(4-bromophenyl)-1-(2-chlorophenyl)-4-(methylsulfonyl)-1H-pyrazol-3-yl)-5-(1-(4-chlorophenyl)cyclopropyl)-1,3,4-oxadiazole
—— 3-[3-(4-bromophenyl)-1-phenyl-1H-pyrazol-4-yl]-5-phenyl-3a,6a-dihydro-pyrrolo[3,4-d]isoxazole-4,6-dione 1174889-25-8 C26H17BrN4O3
3-[3-(4-bromophenyl)-1-phenyl-1H-pyrazol-4-yl]-5-phenyl-3a,6a-dihydro-pyrrolo[3,4-d]isoxazole-4,6-dione
—— 4-((6-(2-chloro-4-fluorophenyl)-5-(ethoxycarbonyl)-2-(thiophen-2-yl)-3,6-dihydropyrimidin-4-yl)methyl)morpholine-3-carboxylic acid 1571216-59-5 C23H23ClFN3O5S
4-((6-(2-chloro-4-fluorophenyl)-5-(ethoxycarbonyl)-2-(thiophen-2-yl)-3,6-dihydropyrimidin-4-yl)methyl)morpholine-3-carboxylic acid
—— 4-({4-[4-(4-fluorophenyl)pyrimidin-2-ylamino]-benzenesulphonyl}(methyl)amino)piperidine-1-carboxylic acid tert-butyl ester 1037899-68-5 C27H32FN5O4S
4-({4-[4-(4-fluorophenyl)pyrimidin-2-ylamino]-benzenesulphonyl}(methyl)amino)piperidine-1-carboxylic acid tert-butyl ester
—— 5-methyl-N2-[(3aS,8aR)-2-oxo-3,3a,8,8a-tetrahydro-2H-indeno[1,2-d]oxazol-5-yl]-N4-[4-(pyridin-3-ylmethoxy)phenyl]-2,4-pyrimidinediamine 1220451-26-2 C27H24N6O3
5-methyl-N2-[(3aS,8aR)-2-oxo-3,3a,8,8a-tetrahydro-2H-indeno[1,2-d]oxazol-5-yl]-N4-[4-(pyridin-3-ylmethoxy)phenyl]-2,4-pyrimidinediamine
—— [4-amino-2-(3-fluoro-phenyl)thieno[2,3-d]pyrimidin-6-yl]-(2-methoxy-phenyl)methanone 1221185-56-3 C20H14FN3O2S
[4-amino-2-(3-fluoro-phenyl)thieno[2,3-d]pyrimidin-6-yl]-(2-methoxy-phenyl)methanone
—— 6-(2-chloro-benzyl)-2-pyrimidin-2-yl-thieno[2,3-d]pyrimidin-4-ylamine 1221430-95-0 C17H12ClN5S
6-(2-chloro-benzyl)-2-pyrimidin-2-yl-thieno[2,3-d]pyrimidin-4-ylamine
—— 2-[(3S)-7-[2-aminoethyl]-3-[benzylsulfonylamino]-4-oxo-3,4-dihydro-1,5-benzothiazepin-5(2H)-yl]-N-{4-[amino(imino)methyl]benzyl}acetamide 1143583-98-5 C28H32N6O4S2
2-[(3S)-7-[2-aminoethyl]-3-[benzylsulfonylamino]-4-oxo-3,4-dihydro-1,5-benzothiazepin-5(2H)-yl]-N-{4-[amino(imino)methyl]benzyl}acetamide
—— t-butyl (3R)-3-{[(R)-tert-butylsulfinyl]amino}-4,4,4-trifluoro-2-methylidenebutanoate 1613583-16-6 C13H22F3NO3S
t-butyl (3R)-3-{[(R)-tert-butylsulfinyl]amino}-4,4,4-trifluoro-2-methylidenebutanoate
—— 6-cyclohexylamino-2-[2-(dimethylamino)ethyl]-1H-benz[de]isoquinoline-1,3(2H)-dione 1000288-28-7 C22H27N3O2
6-cyclohexylamino-2-[2-(dimethylamino)ethyl]-1H-benz[de]isoquinoline-1,3(2H)-dione
—— 6-(4-bromophenyl)-1-butyl-3,5-dichloropyrazin-2(1H)-one 1178895-98-1 C14H13BrCl2N2O
6-(4-bromophenyl)-1-butyl-3,5-dichloropyrazin-2(1H)-one
—— 1-(4-benzamidophenylamino)-N-(2-hydroxyethyl)-6-oxo-5,6-dihydrobenzo[c][1,8]naphthyridine-9-carboxamide 1186377-20-7 C28H23N5O4
1-(4-benzamidophenylamino)-N-(2-hydroxyethyl)-6-oxo-5,6-dihydrobenzo[c][1,8]naphthyridine-9-carboxamide
—— 3-Cyclohexyl-1-[4-[4-[2-(2-propyloxy)phenyl]-1-piperidinyl]butan-1-yl]-2-imidazolidinone 174822-66-3 C27H43N3O2
3-Cyclohexyl-1-[4-[4-[2-(2-propyloxy)phenyl]-1-piperidinyl]butan-1-yl]-2-imidazolidinone
—— N-{[1,6-diethyl-4-(tetrahydro-2H-pyran-4-ylamino)-1H-pyrazolo[3,4-b]pyridin-5-yl]methyl}-N'-[(6-fluoro-3'-{[(3R)-3-methyl-1-piperazinyl]methyl}-3-biphenylyl)methyl]-2,6-pyridinedicarboxamide 1178905-70-8 C42H50FN9O3
N-{[1,6-diethyl-4-(tetrahydro-2H-pyran-4-ylamino)-1H-pyrazolo[3,4-b]pyridin-5-yl]methyl}-N'-[(6-fluoro-3'-{[(3R)-3-methyl-1-piperazinyl]methyl}-3-biphenylyl)methyl]-2,6-pyridinedicarboxamide
—— (1-methyl-piperidin-4-yl)-(3-quinolin-6-ylmethyl-imidazo[1,2-b]pyridazin-6-yl)-amine 1185764-55-9 C22H24N6
(1-methyl-piperidin-4-yl)-(3-quinolin-6-ylmethyl-imidazo[1,2-b]pyridazin-6-yl)-amine
—— 1-[4-(2,5-Dimethyl-pyrrolidin-1-yl)-but-2-ynyl]-pyrrolidine-2,5-dione 18324-97-5 C14H20N2O2
1-[4-(2,5-Dimethyl-pyrrolidin-1-yl)-but-2-ynyl]-pyrrolidine-2,5-dione
—— N-Propyl-N-ethyl-2-methyl-5-nitro-N'-(2,4,6-trimethylphenyl)-pyrimidine-4,6-diamine 175139-14-7 C19H27N5O2
N-Propyl-N-ethyl-2-methyl-5-nitro-N'-(2,4,6-trimethylphenyl)-pyrimidine-4,6-diamine
—— 2-[(benzyloxyimino)]-N-(4-tert-butylphenyl)acetamide 1421739-78-7 C19H22N2O2
2-[(benzyloxyimino)]-N-(4-tert-butylphenyl)acetamide
—— (CO)4Cr(4,4'-dimethyl-2,2'-bipyridine) 15740-68-8 C16H12CrN2O4
(CO)4Cr(4,4'-dimethyl-2,2'-bipyridine)
—— 2,3-epoxy-2,3,5,6-tetrachloro-2,3-dihydro-1.4-dioxin 133349-07-2 C4Cl4O3
2,3-epoxy-2,3,5,6-tetrachloro-2,3-dihydro-1.4-dioxin
—— 1-[4,4-bis(4-hydroxy-3,5-dimethoxyphenyl)piperidin-1-yl]ethan-1-one 134594-67-5 C23H29NO7
1-[4,4-bis(4-hydroxy-3,5-dimethoxyphenyl)piperidin-1-yl]ethan-1-one
—— —— 138612-73-4 C44H27ClN4Ni
—— (E)-2-(2-(4-(trifluoromethyl)phenyl)ethenyl)benzaldehyde 1220094-34-7 C16H11F3O
(E)-2-(2-(4-(trifluoromethyl)phenyl)ethenyl)benzaldehyde
—— (1E,4E)-2,3,4-trimethyl-1,5-diphenylpenta-1,4-dien-3-ol 1415893-77-4 C20H22O
(1E,4E)-2,3,4-trimethyl-1,5-diphenylpenta-1,4-dien-3-ol
—— 1-(6-iodo-2H-pyrazolo[4,3-b]pyridin-2-yl)propan-2-one 1227628-25-2 C9H8IN3O
1-(6-iodo-2H-pyrazolo[4,3-b]pyridin-2-yl)propan-2-one
—— —— 1099062-76-6 C19H23ClFN5O
—— —— 1099060-77-1 C19H26ClFN6O
—— 2-(3-aminosulfonylphenyl)amino-4-[(S)-2-(hydroxymethyl)pyrrolidin-1-yl]-7H-pyrrolo[2,3-d]pyrimidine 1070164-73-6 C17H20N6O3S
2-(3-aminosulfonylphenyl)amino-4-[(S)-2-(hydroxymethyl)pyrrolidin-1-yl]-7H-pyrrolo[2,3-d]pyrimidine
—— 5-(3-Dimethylamino-butyl)-10,11-dihydro-5H-dibenzo[b,f]azepine-3-sulfonic acid dimethylamide 10302-10-0 C22H31N3O2S
5-(3-Dimethylamino-butyl)-10,11-dihydro-5H-dibenzo[b,f]azepine-3-sulfonic acid dimethylamide
—— 4-[[5-methyl-3-[3-[4-(trifluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]pyrazol-1-yl]methyl]-N-[2-(oxan-2-yl)ethyl]pyridin-2-amine 1227147-57-0 C26H27F3N6O3
4-[[5-methyl-3-[3-[4-(trifluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]pyrazol-1-yl]methyl]-N-[2-(oxan-2-yl)ethyl]pyridin-2-amine
—— 4-[4-((5R,8S,11R,13S,14S,17S)-5,17-dihydroxy-5',5',13-trimethyl-17-pentafluoroethyl-2,3,4,5,6,7,8,11,12,13,14,15,16,17-tetradecahydro-1H-spiro[cyclopenta[a]phenanthrene-3,2'-[1,3]dioxane]-11-yl)phenylethynyl]benzoic acid 1262017-29-7 C40H43F5O6
4-[4-((5R,8S,11R,13S,14S,17S)-5,17-dihydroxy-5',5',13-trimethyl-17-pentafluoroethyl-2,3,4,5,6,7,8,11,12,13,14,15,16,17-tetradecahydro-1H-spiro[cyclopenta[a]phenanthrene-3,2'-[1,3]dioxane]-11-yl)phenylethynyl]benzoic acid
—— {(3S,4R)-4-(4-chloro-phenyl)-1-[1-(1-methyl-cyclopropanecarbonyl)-piperidine-4-carbonyl]-pyrrolidin-3-yl}-methyl-carbamic acid 1-cyclopropyl-ethyl ester 1310820-01-9 C28H38ClN3O4
{(3S,4R)-4-(4-chloro-phenyl)-1-[1-(1-methyl-cyclopropanecarbonyl)-piperidine-4-carbonyl]-pyrrolidin-3-yl}-methyl-carbamic acid 1-cyclopropyl-ethyl ester
—— ethyl hydrogen [3-methoxy-4-({4-[(2-methyl-3-oxo-2,3-dihydro-1H-isoindol-4-yl)amino]-5-(trifluoromethyl)pyrimidin-2-yl}amino)benzyl]phosphonate 1257994-37-8 C24H25F3N5O5P
ethyl hydrogen [3-methoxy-4-({4-[(2-methyl-3-oxo-2,3-dihydro-1H-isoindol-4-yl)amino]-5-(trifluoromethyl)pyrimidin-2-yl}amino)benzyl]phosphonate
—— cyclohexyl-{5-[6-(2-morpholin-4-ylethylamino)pyridin-3-yl]imidazo[2,1-b][1,3,4]thiadiazol-2-yl}amine 1206204-38-7 C21H29N7OS
cyclohexyl-{5-[6-(2-morpholin-4-ylethylamino)pyridin-3-yl]imidazo[2,1-b][1,3,4]thiadiazol-2-yl}amine
—— N-(5-(cyclopropylcarbamoyl)-2-methylphenyl)-1H-indazole-6-carboxamide 1026767-37-2 C19H18N4O2
N-(5-(cyclopropylcarbamoyl)-2-methylphenyl)-1H-indazole-6-carboxamide
—— 5-amino-2-(4-benzylpiperidin-1-yl)-4-dimethylamino-6-thiomorpholinopyrimidine 1190065-97-4 C22H32N6S
5-amino-2-(4-benzylpiperidin-1-yl)-4-dimethylamino-6-thiomorpholinopyrimidine
—— 5-chloro-3-(2,4-dioxo-1H-quinazolin-3-yl)-1-[(3-hydroxyphenyl)methyl]indole-2-carboxylic acid 1154598-51-2 C24H16ClN3O5
5-chloro-3-(2,4-dioxo-1H-quinazolin-3-yl)-1-[(3-hydroxyphenyl)methyl]indole-2-carboxylic acid
—— N-[4-cyano-3-(trifluoromethyl)phenyl]-3-(ethanesulfonyl)-2-[4-(trifluoromethyl)phenyl]-2-hydroxypropanamide 1355935-63-5 C20H16F6N2O4S
N-[4-cyano-3-(trifluoromethyl)phenyl]-3-(ethanesulfonyl)-2-[4-(trifluoromethyl)phenyl]-2-hydroxypropanamide
—— 1-(2-([6-({5-[{2-[({[(2S)-1'-{2-[(5R)-3-[3,5-bis(trifluoromethyl)benzoyl]-5-(4-fluorophenyl)-1,3-oxazolidin-5-yl]ethyl}-2,3-dihydrospiro[indene-1,4'-piperidin]-2-yl]oxy}acetyl)(methyl)amino]ethyl}(methyl)carbamoyl]-4-methyl-2-thienyl}amino)hexanoyl](methyl)amino)ethyl)piperidin-4-yl biphenyl-2-ylcarbamate 1246245-83-9 C72H83F7N8O8S
1-(2-([6-({5-[{2-[({[(2S)-1'-{2-[(5R)-3-[3,5-bis(trifluoromethyl)benzoyl]-5-(4-fluorophenyl)-1,3-oxazolidin-5-yl]ethyl}-2,3-dihydrospiro[indene-1,4'-piperidin]-2-yl]oxy}acetyl)(methyl)amino]ethyl}(methyl)carbamoyl]-4-methyl-2-thienyl}amino)hexanoyl](methyl)amino)ethyl)piperidin-4-yl biphenyl-2-ylcarbamate
—— 1-isoquinolin-5-ylmethyl-piperazine-2-carboxylic acid (2-dimethylaminoethyl)amide 1021484-02-5 C19H27N5O
1-isoquinolin-5-ylmethyl-piperazine-2-carboxylic acid (2-dimethylaminoethyl)amide
—— —— 1021311-18-1 C27H33N3O2S
—— 17β-Hydroxy-17α-vinyl-4-androsten<3,2-c>pyrazol 100323-04-4 C22H30N2O
17β-Hydroxy-17α-vinyl-4-androsten<3,2-c>pyrazol
—— —— 1075185-52-2 C19H16FN5O
—— tert-butyl N-[(4-methoxypyridin-3-yl)methyl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate 1214728-83-2 C17H26N2O5
tert-butyl N-[(4-methoxypyridin-3-yl)methyl]-N-[(2-methylpropan-2-yl)oxycarbonyl]carbamate