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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-{3-benzyl-2-[4-fluoro-2-(1-hydroxy-ethyl)-phenoxy]-quinolin-6-yl}-3-(4-chloro-benzyl)-thiourea 1173290-18-0 C32H27ClFN3O2S
1-{3-benzyl-2-[4-fluoro-2-(1-hydroxy-ethyl)-phenoxy]-quinolin-6-yl}-3-(4-chloro-benzyl)-thiourea
—— N-[N'-(2-tert-butylphenyl)-N-(2-oxo-3H-1,3-benzoxazol-6-yl)carbamimidoyl]-3-fluorobenzamide 1217242-20-0 C25H23FN4O3
N-[N'-(2-tert-butylphenyl)-N-(2-oxo-3H-1,3-benzoxazol-6-yl)carbamimidoyl]-3-fluorobenzamide
—— 4-(4'-methylbiphenyl-2-carboxamido)-N-methyl-N-[2-(5-carboxypentyl)phenyl]benzamide 183492-86-6 C34H34N2O4
4-(4'-methylbiphenyl-2-carboxamido)-N-methyl-N-[2-(5-carboxypentyl)phenyl]benzamide
—— 2-((3-oxo-3-(4-(5-phenyl-1,3,4-oxadiazol-2-yl)piperidin-1-yl)propyl)thio)quinazolin-4(3H)-one 1570178-10-7 C24H23N5O3S
2-((3-oxo-3-(4-(5-phenyl-1,3,4-oxadiazol-2-yl)piperidin-1-yl)propyl)thio)quinazolin-4(3H)-one
—— N,N-bis(methyl-d<sub>3</sub>)alanine methyl ester 1571901-51-3 C6H13NO2
N,N-bis(methyl-d<sub>3</sub>)alanine methyl ester
—— —— 1366019-32-0 C15H13N3O2S
—— N-[5-(2-amino-4-methyl-pyrimidin-5-yl)-2-chloro-phenyl]-benzenesulfonamide 1106312-90-6 C17H15ClN4O2S
N-[5-(2-amino-4-methyl-pyrimidin-5-yl)-2-chloro-phenyl]-benzenesulfonamide
—— Brutieridin 1162664-57-4 C34H42O19
Brutieridin
—— (2S,3S)-N-(4-(5-heptylpyridin-2-yl)phenyl)-3-hydroxypyrrolidine-2-carboxamide 1218816-86-4 C23H31N3O2
(2S,3S)-N-(4-(5-heptylpyridin-2-yl)phenyl)-3-hydroxypyrrolidine-2-carboxamide
—— 5-fluoro-2-(4-sulfamoylphenylamino)-1-(2-(trifluoromethyl)benzyl)-1H-benzo[d]imidazole-6-carboxamide 1175563-18-4 C22H17F4N5O3S
5-fluoro-2-(4-sulfamoylphenylamino)-1-(2-(trifluoromethyl)benzyl)-1H-benzo[d]imidazole-6-carboxamide
—— [(1R,2S)-1-[3,5-bis(trifluoromethyl)phenyl]-2-[[2-(4-fluoro-2-methoxy-5-propan-2-ylphenyl)-5-(trifluoromethyl)phenyl]methylamino]propyl] methyl carbonate 1220750-26-4 C31H29F10NO4
[(1R,2S)-1-[3,5-bis(trifluoromethyl)phenyl]-2-[[2-(4-fluoro-2-methoxy-5-propan-2-ylphenyl)-5-(trifluoromethyl)phenyl]methylamino]propyl] methyl carbonate
—— N,1-dimethyl-N-pyridazin-4-yl-5-(trifluoromethyl)pyrazole-4-carboxamide 1219837-96-3 C11H10F3N5O
N,1-dimethyl-N-pyridazin-4-yl-5-(trifluoromethyl)pyrazole-4-carboxamide
—— cyclopropyl(6-(3,5-dichloro-4-hydroxyphenyl)-4-(6-(pyrrolidin-3-ylamino)pyridin-3-ylamino)quinolin-3-yl)methanone 1356948-18-9 C28H25Cl2N5O2
cyclopropyl(6-(3,5-dichloro-4-hydroxyphenyl)-4-(6-(pyrrolidin-3-ylamino)pyridin-3-ylamino)quinolin-3-yl)methanone
—— 4-chloro-N-(3-methyl-4-(4-methyl-3-pyridinyl)phenyl)benzenesulfonamide 1357091-99-6 C19H17ClN2O2S
4-chloro-N-(3-methyl-4-(4-methyl-3-pyridinyl)phenyl)benzenesulfonamide
—— (2S,4R)-4-(2-chlorobenzenesulfonyl)-1-[1-(5-chloro-3-fluoropyridin-2-yl)cyclopropanecarbonyl]pyrrolidine-2-carboxylic acid (1-cyanocyclopropyl)amide 1569085-03-5 C24H21Cl2FN4O4S
(2S,4R)-4-(2-chlorobenzenesulfonyl)-1-[1-(5-chloro-3-fluoropyridin-2-yl)cyclopropanecarbonyl]pyrrolidine-2-carboxylic acid (1-cyanocyclopropyl)amide
—— 4-(2-cyclohexyl-6-methyl-3-(1H-tetrazol-5-yl)-5,6,7,8-tetrahydroquinolin-4-yl)-3,5-dimethylisoxazole 1569825-32-6 C22H28N6O
4-(2-cyclohexyl-6-methyl-3-(1H-tetrazol-5-yl)-5,6,7,8-tetrahydroquinolin-4-yl)-3,5-dimethylisoxazole
—— —— 1346981-28-9 C20H18ClN3O
—— 6-(4-hydroxy-phenyl)-1H-pyrazolo[3,4-b]pyridine-4-carboxylic acid methyl ester 1431977-97-7 C14H11N3O3
6-(4-hydroxy-phenyl)-1H-pyrazolo[3,4-b]pyridine-4-carboxylic acid methyl ester
—— ethyl 2-(3-nitro-2-pyridylhydrazono)phenylacetate 110606-60-5 C15H14N4O4
ethyl 2-(3-nitro-2-pyridylhydrazono)phenylacetate
—— (S)-1-(3,5-bis-(trifluoromethyl)phenyl)-3-((1-(piperidin-2-carbonyl)piperidin-4yl)methyl)urea 1274834-87-5 C21H26F6N4O2
(S)-1-(3,5-bis-(trifluoromethyl)phenyl)-3-((1-(piperidin-2-carbonyl)piperidin-4yl)methyl)urea
—— 3-[(4-Chloropyrimidin-2-yl)amino]benzenesulfonamide 1335140-75-4 C10H9ClN4O2S
3-[(4-Chloropyrimidin-2-yl)amino]benzenesulfonamide
—— 2-{4-[(1-tert-butyl-1H-tetrazol-5-yl)(4-chlorophenylamino)methyl]phenyl}-3-cyclohexylaminoimidazo[1,2-a]pyridine 1440522-60-0 C31H35ClN8
2-{4-[(1-tert-butyl-1H-tetrazol-5-yl)(4-chlorophenylamino)methyl]phenyl}-3-cyclohexylaminoimidazo[1,2-a]pyridine
—— 4-nitrobenzoic acid 2-[[(1-methylethyl)thio](methylthio)methylene]hydrazide 1366338-41-1 C12H15N3O3S2
4-nitrobenzoic acid 2-[[(1-methylethyl)thio](methylthio)methylene]hydrazide
—— 2-chloro-4-methyl-5-(trifluoromethyl)thiazole 141761-76-4 C5H3ClF3NS
2-chloro-4-methyl-5-(trifluoromethyl)thiazole
—— N-((2-(3-(3-fluorobenzyl)ureido)thiazol-4-yl)methyl)-N,3-dimethyl-5,6-dihydro-1,4-dioxine-2-carboxamide 1108709-34-7 C19H21FN4O4S
N-((2-(3-(3-fluorobenzyl)ureido)thiazol-4-yl)methyl)-N,3-dimethyl-5,6-dihydro-1,4-dioxine-2-carboxamide
—— 3-{3-[2-(3-methoxy-propyl)-pyridin-4-yl]-1H-indole-6-carbonyl}-benzenesulfonamide 1189544-90-8 C24H23N3O4S
3-{3-[2-(3-methoxy-propyl)-pyridin-4-yl]-1H-indole-6-carbonyl}-benzenesulfonamide
—— 6-(imidazo[1,2-a]pyrazin-3-yl)-N-[(2R,3S)-2-methylpiperidin-3-yl]pyrazin-2-amine 1207851-06-6 C16H19N7
6-(imidazo[1,2-a]pyrazin-3-yl)-N-[(2R,3S)-2-methylpiperidin-3-yl]pyrazin-2-amine
—— 2-(4-(benzyloxy)-1-ethyl-6-fluoro-1H-indol-3-yl)-N-phenethylethanamine 1265217-33-1 C27H29FN2O
2-(4-(benzyloxy)-1-ethyl-6-fluoro-1H-indol-3-yl)-N-phenethylethanamine
—— 6-(2-ethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(2R,3S)-2-methylpiperidin-3-yl]pyrazin-2-amine 1207851-09-9 C17H22N6S
6-(2-ethylimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(2R,3S)-2-methylpiperidin-3-yl]pyrazin-2-amine
—— 2-N-(8-cyclopentyl-4,6,8,11-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6,10,12-hexaen-5-yl)-5-N-methyl-5-N-piperidin-3-ylpyridine-2,5-diamine 1169692-74-3 C25H30N8
2-N-(8-cyclopentyl-4,6,8,11-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6,10,12-hexaen-5-yl)-5-N-methyl-5-N-piperidin-3-ylpyridine-2,5-diamine
—— 1-cyclopentyl-1H-pyrazole-3-carboxylic acid 1006348-93-1 C9H12N2O2
1-cyclopentyl-1H-pyrazole-3-carboxylic acid
—— 4-(4-Fluorophenyl)-1-methylsulfonyl-5-phenyl-2,3,6,7-tetrahydroazepine 1342798-58-6 C19H20FNO2S
4-(4-Fluorophenyl)-1-methylsulfonyl-5-phenyl-2,3,6,7-tetrahydroazepine
—— 3-[(6-Bromoquinazolin-2-yl)amino]-5-morpholin-4-ylbenzamide 1036744-81-6 C19H18BrN5O2
3-[(6-Bromoquinazolin-2-yl)amino]-5-morpholin-4-ylbenzamide
—— (4R,5R,8R,11S,14R,17S)-4,5-dihydroxy-3,6,9,12,15-pentaoxo-14-(2-phenylethyl)-11-[(4-phenylphenyl)methyl]-8-(thiophen-2-ylmethyl)-2,7,10,13,16-pentazabicyclo[17.2.2]tricosa-1(21),19,22-triene-17-carboxylic acid 1211439-69-8 C45H45N5O9S
(4R,5R,8R,11S,14R,17S)-4,5-dihydroxy-3,6,9,12,15-pentaoxo-14-(2-phenylethyl)-11-[(4-phenylphenyl)methyl]-8-(thiophen-2-ylmethyl)-2,7,10,13,16-pentazabicyclo[17.2.2]tricosa-1(21),19,22-triene-17-carboxylic acid
—— isopropyl 4-(4-(4-(oxazol-5-yl)phenylamino)-6H-pyrimido[5,4-b][1,4]oxazin-8(7H)-yl)piperidine-1-carboxylate 1079053-51-2 C24H28N6O4
isopropyl 4-(4-(4-(oxazol-5-yl)phenylamino)-6H-pyrimido[5,4-b][1,4]oxazin-8(7H)-yl)piperidine-1-carboxylate
—— 2-methyl-2-[methyl(oxan-4-ylmethyl)amino]-N-[3-[1-(oxan-2-yloxymethyl)cyclopentyl]-1,2-oxazol-5-yl]propanamide 1259021-40-3 C25H41N3O5
2-methyl-2-[methyl(oxan-4-ylmethyl)amino]-N-[3-[1-(oxan-2-yloxymethyl)cyclopentyl]-1,2-oxazol-5-yl]propanamide
—— [(3S,4R)-4-(4-chloro-phenyl)-1-(1,1-dioxo-hexahydro-1λ<sup>6</sup>-thiopyran-4-carbonyl)-pyrrolidin-3-yl]-methyl-carbamic acid 4-fluoro-phenyl ester 1310819-22-7 C24H26ClFN2O5S
[(3S,4R)-4-(4-chloro-phenyl)-1-(1,1-dioxo-hexahydro-1λ<sup>6</sup>-thiopyran-4-carbonyl)-pyrrolidin-3-yl]-methyl-carbamic acid 4-fluoro-phenyl ester
—— 8-cyclopentyl-N-[5-[4-(propan-2-ylamino)piperidin-1-yl]pyridin-2-yl]-4,6,8,11-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6,10,12-hexaen-5-amine 1169698-33-2 C27H34N8
8-cyclopentyl-N-[5-[4-(propan-2-ylamino)piperidin-1-yl]pyridin-2-yl]-4,6,8,11-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6,10,12-hexaen-5-amine
—— N-[5-[(3S)-3-methylpiperazin-1-yl]pyridin-2-yl]-8-[(3R)-pyrrolidin-3-yl]-4,6,8,11-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6,10,12-hexaen-5-amine 1169696-98-3 C23H27N9
N-[5-[(3S)-3-methylpiperazin-1-yl]pyridin-2-yl]-8-[(3R)-pyrrolidin-3-yl]-4,6,8,11-tetrazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6,10,12-hexaen-5-amine
—— [(8S)-4-[(3S,4R)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidine-3-carbonyl]-8-(4-chlorophenyl)-1,4-diazocan-1-yl]-cyclopentylmethanone 1207511-23-6 C33H42ClF2N3O2
[(8S)-4-[(3S,4R)-1-tert-butyl-4-(2,4-difluorophenyl)pyrrolidine-3-carbonyl]-8-(4-chlorophenyl)-1,4-diazocan-1-yl]-cyclopentylmethanone
—— 4-methyl-thiophene-2-carboxylic acid thiazol-2-ylamide 1185852-99-6 C9H8N2OS2
4-methyl-thiophene-2-carboxylic acid thiazol-2-ylamide
—— 7-amino-1-ethoxy-3-methoxy-10-methyl-6-[4-(2-pyridynyl)-1-piperazinyl]-9(10H)-acridinone 1152309-01-7 C26H29N5O3
7-amino-1-ethoxy-3-methoxy-10-methyl-6-[4-(2-pyridynyl)-1-piperazinyl]-9(10H)-acridinone
—— (2-methoxy-ethyl)-(3-quinolin-6-ylmethyl-imidazo[1,2-b]pyridazin-6-yl)-amine 1185764-62-8 C19H19N5O
(2-methoxy-ethyl)-(3-quinolin-6-ylmethyl-imidazo[1,2-b]pyridazin-6-yl)-amine
—— 6-O-(4-methylbenzoyl)galanthamine 1190931-54-4 C25H27NO4
6-O-(4-methylbenzoyl)galanthamine
—— benzyl 3-((7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-3-yl)ethynyl)phenylcarbamate 1181621-16-8 C24H19N3O3
benzyl 3-((7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-3-yl)ethynyl)phenylcarbamate
—— 1-[1-(3,3-dimethylbut-1-yn-1-yl)cyclohexyl]piperidine 1404592-47-7 C17H29N
1-[1-(3,3-dimethylbut-1-yn-1-yl)cyclohexyl]piperidine
—— diethyl 2-[(2-chlorophenoxy)methyl]-2-ethylpropanedioate 110449-99-5 C16H21ClO5
diethyl 2-[(2-chlorophenoxy)methyl]-2-ethylpropanedioate
—— (2S,3R,4R)-1-(N-methyl-N-((R)-1-phenylethyl)amino)-3-(benzyloxy)-4-methylhex-5-en-2-yl acetate 1338481-40-5 C25H33NO3
(2S,3R,4R)-1-(N-methyl-N-((R)-1-phenylethyl)amino)-3-(benzyloxy)-4-methylhex-5-en-2-yl acetate
—— 4-(3-fluoro-4-quinolin-6-ylphenyl)-N-hydroxy-2-methyl-2-(methylsulfonyl)butanamide 1289623-81-9 C21H21FN2O4S
4-(3-fluoro-4-quinolin-6-ylphenyl)-N-hydroxy-2-methyl-2-(methylsulfonyl)butanamide
—— 2,3,4,5-Tetrafluoro-6-[[6-[2-(2-methoxyethoxy)ethoxy]-1-oxidopyridin-1-ium-3-yl]carbamoyl]benzoic acid 1269512-66-4 C18H16F4N2O7
2,3,4,5-Tetrafluoro-6-[[6-[2-(2-methoxyethoxy)ethoxy]-1-oxidopyridin-1-ium-3-yl]carbamoyl]benzoic acid