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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-3-(4-{[3-(2,6-dichlorophenyl)isoxazol-5-yl]methyl}piperazinyl)-1-[2-(4-chlorophenyl)benzoxazol-5-yloxy]propan-2-ol 1055973-52-8 C30H27Cl3N4O4
(2R)-3-(4-{[3-(2,6-dichlorophenyl)isoxazol-5-yl]methyl}piperazinyl)-1-[2-(4-chlorophenyl)benzoxazol-5-yloxy]propan-2-ol
—— 3,5-dibromo-4-methoxyphenyl 4-(3-butyl-2-oxoimidazolidin-1-yl)benzenesulfonate 1422528-07-1 C20H22Br2N2O5S
3,5-dibromo-4-methoxyphenyl 4-(3-butyl-2-oxoimidazolidin-1-yl)benzenesulfonate
—— (7R,8aS)-7-[(5-cyclopropylpyrazin-2-yl)oxy]-2-[(2,3-difluorophenyl)-sulfonyl]octahydropyrrolo[1,2-a]pyrazine 1429197-61-4 C20H22F2N4O3S
(7R,8aS)-7-[(5-cyclopropylpyrazin-2-yl)oxy]-2-[(2,3-difluorophenyl)-sulfonyl]octahydropyrrolo[1,2-a]pyrazine
—— (2S)-2-amino-3-{[(2-methoxy-5-sulfophenyl)carbamoyl]amino}propanoic acid 1333219-19-4 C11H15N3O7S
(2S)-2-amino-3-{[(2-methoxy-5-sulfophenyl)carbamoyl]amino}propanoic acid
—— 2-[(1S)-2-amino-1-(2-thienylmethyl)ethyl]-5-(4-chloro-1-methyl-1H-pyrazol-5-yl)isoindolin-1-one 1430057-08-1 C19H19ClN4OS
2-[(1S)-2-amino-1-(2-thienylmethyl)ethyl]-5-(4-chloro-1-methyl-1H-pyrazol-5-yl)isoindolin-1-one
—— 4-(3-(4-(adamantan-1-yl)phenoxy)propanoyl)-1,1-dimethylpiperazin-1-ium iodide 1429054-46-5 C25H37N2O2*I
4-(3-(4-(adamantan-1-yl)phenoxy)propanoyl)-1,1-dimethylpiperazin-1-ium iodide
—— 4-(3-chlorophenyl)-2-(piperidin-1-yl)-3-(1H-tetrazol-5-yl)-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridine 1569821-99-3 C22H25ClN6
4-(3-chlorophenyl)-2-(piperidin-1-yl)-3-(1H-tetrazol-5-yl)-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridine
—— 3-(N,N-dibutylamino)-4-phenoxy-5-ethylsulfonylbenzoic acid 1431501-04-0 C23H31NO5S
3-(N,N-dibutylamino)-4-phenoxy-5-ethylsulfonylbenzoic acid
—— (-)-(R)-3-isopropyl-N-(p-toluenesulfonyl)pyrrolidine 1417920-76-3 C14H21NO2S
(-)-(R)-3-isopropyl-N-(p-toluenesulfonyl)pyrrolidine
—— N-((S)-2-((3aS,6S,6aS)-6-chloro-3-oxodihydro-2H-furo[3,2-b]pyrrol-4(5H,6H,6aH)-yl)-1-cyclohexyl-2-oxoethyl)-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide 1187323-63-2 C23H25ClN4O6
N-((S)-2-((3aS,6S,6aS)-6-chloro-3-oxodihydro-2H-furo[3,2-b]pyrrol-4(5H,6H,6aH)-yl)-1-cyclohexyl-2-oxoethyl)-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
—— 3-(azulen-1-yl)-5-methylphenol 1189141-17-0 C17H14O
3-(azulen-1-yl)-5-methylphenol
—— 3-(2-chloro-benzoylamino)-N-(pyridine-2-ylmethyl)-benzamide 1185401-71-1 C20H16ClN3O2
3-(2-chloro-benzoylamino)-N-(pyridine-2-ylmethyl)-benzamide
—— N-{1-[3-(7-chloro-3-oxo-2,3-dihydro-benzo[1,4]thiazin-4-yl)-propyl]-piperidin-4-yl}-isobutyramide 1186229-74-2 C20H28ClN3O2S
N-{1-[3-(7-chloro-3-oxo-2,3-dihydro-benzo[1,4]thiazin-4-yl)-propyl]-piperidin-4-yl}-isobutyramide
—— (5R,7S,10S,12R)-N-{(1R,2S)-1-[(cyclopropylsulfonyl)carbamoyl]-2-ethenylcyclopropyl}-12-methyl-3,9-dioxo-10-(propan-2-yl)-6,7,9,10,11,12,13,14,15,16,17,18-dodecahydro-1H,5H-2,22:5,8-dimethano-4,2,8,11-benzoxatriazacycloicosine-7(3H)-carboxamide 1179843-08-3 C36H51N5O7S
(5R,7S,10S,12R)-N-{(1R,2S)-1-[(cyclopropylsulfonyl)carbamoyl]-2-ethenylcyclopropyl}-12-methyl-3,9-dioxo-10-(propan-2-yl)-6,7,9,10,11,12,13,14,15,16,17,18-dodecahydro-1H,5H-2,22:5,8-dimethano-4,2,8,11-benzoxatriazacycloicosine-7(3H)-carboxamide
—— (E)-N,N-Diethyl-4-[[3-dimethylamino-1-(3-hydroxyphenyl)]-1-propenyl]benzamide 189100-58-1 C22H28N2O2
(E)-N,N-Diethyl-4-[[3-dimethylamino-1-(3-hydroxyphenyl)]-1-propenyl]benzamide
—— (R)-3-(3-fluorophenyl)-N-(1-hydroxy-3-(1H-indol-3-yl)propan-2-yl)-7,8,9-trimethoxy-5,6-dihydropyrrolo[2,1-a]isoquinoline-2-carboxamide 1428796-27-3 C33H32FN3O5
(R)-3-(3-fluorophenyl)-N-(1-hydroxy-3-(1H-indol-3-yl)propan-2-yl)-7,8,9-trimethoxy-5,6-dihydropyrrolo[2,1-a]isoquinoline-2-carboxamide
—— 7-methoxy-2-methyl-4-[2-(1-methyl-4-thiazol-2-yl-1H-imidazol-2-yl)-ethyl]-quinazoline 1429781-47-4 C19H19N5OS
7-methoxy-2-methyl-4-[2-(1-methyl-4-thiazol-2-yl-1H-imidazol-2-yl)-ethyl]-quinazoline
—— N-[(S)-4-(8-chloro-1-methyl-2-oxo-1,2,3,4-tetrahydro-quinolin-6-yl)-5,6,7,8-tetrahydro-isoquinolin-8-yl]-propionamide 1428652-55-4 C22H24ClN3O2
N-[(S)-4-(8-chloro-1-methyl-2-oxo-1,2,3,4-tetrahydro-quinolin-6-yl)-5,6,7,8-tetrahydro-isoquinolin-8-yl]-propionamide
—— (5R)-5-benzyl-N-[1-(3-chlorophenyl)-2,2,2-trifluoroethyl]-3-[(1R)-1-(4-fluorophenyl)ethyl]-2,4-dioxo-1,3-oxazolidine-5-carboxamide 1430104-65-6 C27H21ClF4N2O4
(5R)-5-benzyl-N-[1-(3-chlorophenyl)-2,2,2-trifluoroethyl]-3-[(1R)-1-(4-fluorophenyl)ethyl]-2,4-dioxo-1,3-oxazolidine-5-carboxamide
—— N-[(1S)-1-cyclohexyl-2-(4-methylpiperazin-1-yl)ethyl]-2-[(4R)-7-(3-fluorophenyl)-1-oxo-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-4-yl]acetamide 1429925-10-9 C28H38FN5O2
N-[(1S)-1-cyclohexyl-2-(4-methylpiperazin-1-yl)ethyl]-2-[(4R)-7-(3-fluorophenyl)-1-oxo-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-4-yl]acetamide
—— 3-Nitro-4-pyridin-1-ium-1-ylbenzamide;chloride 1443647-42-4 C12H10N3O3*Cl
3-Nitro-4-pyridin-1-ium-1-ylbenzamide;chloride
—— Trimethyl-[2-(2,8,9-trioxa-5-aza-1-silabicyclo[3.3.3]undecan-1-ylmethylselanyl)ethynyl]silane 127072-75-7 C12H23NO3SeSi2
Trimethyl-[2-(2,8,9-trioxa-5-aza-1-silabicyclo[3.3.3]undecan-1-ylmethylselanyl)ethynyl]silane
—— (2S)-2-[4-[4-(2-fluoroethyl)phenyl]-2-methylquinolin-3-yl]-2-[(2-methylpropan-2-yl)oxy]acetic acid 1155270-98-6 C24H26FNO3
(2S)-2-[4-[4-(2-fluoroethyl)phenyl]-2-methylquinolin-3-yl]-2-[(2-methylpropan-2-yl)oxy]acetic acid
—— 4-(2-cyclopropylmethoxy-5-fluoro-phenyl)-5H-pyrrolo[3,2-d]pyrimidine-7-carboxylic acid [1-(2-methoxy-acetyl)-piperidin-4-yl]-amide 1185839-39-7 C25H28FN5O4
4-(2-cyclopropylmethoxy-5-fluoro-phenyl)-5H-pyrrolo[3,2-d]pyrimidine-7-carboxylic acid [1-(2-methoxy-acetyl)-piperidin-4-yl]-amide
—— 1-(4-hydroxy-4-methylpentyl)-2,7-dimethoxynaphthalene 1140910-75-3 C18H24O3
1-(4-hydroxy-4-methylpentyl)-2,7-dimethoxynaphthalene
—— (1S,3S)-3-benzyl-4-oxo-1-phenylbutyl nitrate 1092798-43-0 C17H17NO4
(1S,3S)-3-benzyl-4-oxo-1-phenylbutyl nitrate
—— (E)-3-(Furo<3,4-b>furan-4-yl)-2-propennitril 113893-50-8 C9H5NO2
(E)-3-(Furo<3,4-b>furan-4-yl)-2-propennitril
—— (1Z,6Z)-2,7,12,21-tetraphenyl-13-oxa-16,25,27,28-tetrazaheptacyclo[13.9.2.13,6.18,11.012,17.016,20.022,25]octacosa-1,3(28),4,6,8,10,15(26),17,19,21,23-undecaene 131074-83-4 C47H32N4O
(1Z,6Z)-2,7,12,21-tetraphenyl-13-oxa-16,25,27,28-tetrazaheptacyclo[13.9.2.13,6.18,11.012,17.016,20.022,25]octacosa-1,3(28),4,6,8,10,15(26),17,19,21,23-undecaene
—— 2-(2-methyl-2-decyl)-2-imidazoline 117818-10-7 C14H28N2
2-(2-methyl-2-decyl)-2-imidazoline
—— (S)-2-mesitylpropanenitrile 1421692-24-1 C12H15N
(S)-2-mesitylpropanenitrile
—— N-benzyl-1-(5-(4-nitrophenyl)furan-2-yl)methanimine 1392096-61-5 C18H14N2O3
N-benzyl-1-(5-(4-nitrophenyl)furan-2-yl)methanimine
—— 2,3,5,6-tetrafluoro-4-[(1S,9R)-4-(2,3,4,5,6-pentafluorophenyl)-8-oxa-2,4,5-triazatetracyclo[7.7.0.02,6.011,16]hexadeca-5,11,13,15-tetraen-3-ylidene]cyclohexa-2,5-dien-1-one 1449013-58-4 C24H10F9N3O2
2,3,5,6-tetrafluoro-4-[(1S,9R)-4-(2,3,4,5,6-pentafluorophenyl)-8-oxa-2,4,5-triazatetracyclo[7.7.0.02,6.011,16]hexadeca-5,11,13,15-tetraen-3-ylidene]cyclohexa-2,5-dien-1-one
—— methyl 2-[2-[(2S)-3-bromo-2-(phenylmethoxycarbonylamino)propoxy]phenyl]-3-cyclohexyl-1H-indole-6-carboxylate 1325208-63-6 C33H35BrN2O5
methyl 2-[2-[(2S)-3-bromo-2-(phenylmethoxycarbonylamino)propoxy]phenyl]-3-cyclohexyl-1H-indole-6-carboxylate
—— (2S)-2-(dimethylamino)-2-methyl-1,1,3-triphenylpropan-1-ol 1030884-68-4 C24H27NO
(2S)-2-(dimethylamino)-2-methyl-1,1,3-triphenylpropan-1-ol
—— (2R)-2-amino-2-ethyl-4-[5-(5-phenylpentanoyl)thiophen-2-yl]butan-1-ol 1171214-89-3 C21H29NO2S
(2R)-2-amino-2-ethyl-4-[5-(5-phenylpentanoyl)thiophen-2-yl]butan-1-ol
—— 6-Methoxy-2,2,5,7-tetramethylchromene 1352188-71-6 C14H18O2
6-Methoxy-2,2,5,7-tetramethylchromene
—— 2,3,5-trimethyl-4-(chloromethyl)selenophene 126458-41-1 C8H11ClSe
2,3,5-trimethyl-4-(chloromethyl)selenophene
—— 3,9,15,35-tetratert-butyl-39,40-dihydroxy-19,30-dioxahexacyclo[15.14.7.17,11.133,37.05,31.013,18]tetraconta-1,3,5(31),7,9,11(40),13(18),14,16,33,35,37(39)-dodecaene-20,29-dione 128217-32-3 C54H70O6
3,9,15,35-tetratert-butyl-39,40-dihydroxy-19,30-dioxahexacyclo[15.14.7.17,11.133,37.05,31.013,18]tetraconta-1,3,5(31),7,9,11(40),13(18),14,16,33,35,37(39)-dodecaene-20,29-dione
—— US8653087, III-313 1213246-01-5 C21H18F3N9O2S
US8653087, III-313
—— 5-(5,6-dimethoxypyridin-3-yl)-2-(5-ethyl-1H-1,2,4-triazol-3-yl)-3H-isoindol-1-one 1315535-04-6 C19H19N5O3
5-(5,6-dimethoxypyridin-3-yl)-2-(5-ethyl-1H-1,2,4-triazol-3-yl)-3H-isoindol-1-one
—— US8653087, III-342 1213246-29-7 C21H19F3N10OS
US8653087, III-342
—— 2,8-dibromo-5H-benzo[b][1,4]benzoxazepin-6-one 1246661-76-6 C13H7Br2NO2
2,8-dibromo-5H-benzo[b][1,4]benzoxazepin-6-one
—— 2-[N-(3-Acetylaminobenzoyl)amino]-4-[(2-diisopropylaminoethyl)aminocarbonyl]-1,3-thiazole 185105-77-5 C21H29N5O3S
2-[N-(3-Acetylaminobenzoyl)amino]-4-[(2-diisopropylaminoethyl)aminocarbonyl]-1,3-thiazole
—— pregna-Δ<sup>4,17(20)</sup>-dien-3-one 1667-83-0 C21H30O
pregna-Δ<sup>4,17(20)</sup>-dien-3-one
—— 3-(cyano-dimethyl-methyl)-N-(6-methyl-5-{4-[5-(4-methyl-piperazin-1-yl)-pyridine-3-yl]-1,2,3-triazol-1-yl}-pyridin-3-yl)-benzamide 1219947-68-8 C29H31N9O
3-(cyano-dimethyl-methyl)-N-(6-methyl-5-{4-[5-(4-methyl-piperazin-1-yl)-pyridine-3-yl]-1,2,3-triazol-1-yl}-pyridin-3-yl)-benzamide
—— 1-(4-Isopropylphenyl)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]urea 1227091-12-4 C20H26N4O
1-(4-Isopropylphenyl)-3-[2-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)ethyl]urea
—— 2-[4-[2-(5-methoxypyridin-3-yl)-4-methyl-5-oxo-7H-pyrrolo[3,4-b]pyridin-6-yl]pyrazol-1-yl]acetonitrile 1315536-60-7 C19H16N6O2
2-[4-[2-(5-methoxypyridin-3-yl)-4-methyl-5-oxo-7H-pyrrolo[3,4-b]pyridin-6-yl]pyrazol-1-yl]acetonitrile
—— 2-[benzyl(hydroxy)amino]-2-cyclohexylacetonitrile 1373354-78-9 C15H20N2O
2-[benzyl(hydroxy)amino]-2-cyclohexylacetonitrile
—— 2,3,4,6-tetrabromo-5-methoxytoluene 136401-01-9 C8H6Br4O
2,3,4,6-tetrabromo-5-methoxytoluene
—— 2-(3-amino-5-(trifluoromethyl)phenyl)isoindoline-1,3-dione 1610038-13-5 C15H9F3N2O2
2-(3-amino-5-(trifluoromethyl)phenyl)isoindoline-1,3-dione