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中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-2-amino-N-[(1S,2S)-1-hydroxy-1-phenylpropan-2-yl]-N-methylpropanamide 185508-81-0 C13H20N2O2
(2R)-2-amino-N-[(1S,2S)-1-hydroxy-1-phenylpropan-2-yl]-N-methylpropanamide
—— 8-(methoxycarbonyl)octyl O-(benzyl 5-acetamido-4,7,8,9-tetra-O-acetyl-3,5-dideoxy-D-glycero-α-D-galacto-2-nonulopyranosylonate)-(2<*>3)-O-(2,4,6-tri-O-acetyl-β-D-galactopyranosyl)-(1<*>4)-6-O-acetyl-2-azido-2-deoxy-β-D-glucopyranoside 126168-68-1 C56H78N4O28
8-(methoxycarbonyl)octyl O-(benzyl 5-acetamido-4,7,8,9-tetra-O-acetyl-3,5-dideoxy-D-glycero-α-D-galacto-2-nonulopyranosylonate)-(2<*>3)-O-(2,4,6-tri-O-acetyl-β-D-galactopyranosyl)-(1<*>4)-6-O-acetyl-2-azido-2-deoxy-β-D-glucopyranoside
—— tert-Butyl (2S,4S)-2-(bromomethyl)-4-fluoropyrrolidine-1-carboxylate 2165773-57-7 C10H17BrFNO2
tert-Butyl (2S,4S)-2-(bromomethyl)-4-fluoropyrrolidine-1-carboxylate
—— Methyl 2-[[1-(4-chlorophenyl)-2-cyanoprop-2-enyl]amino]acetate 1141875-57-1 C13H13ClN2O2
Methyl 2-[[1-(4-chlorophenyl)-2-cyanoprop-2-enyl]amino]acetate
—— dimethyl (E)-2-acetylamino-2-p-tolylvinylphosphonate 1115365-46-2 C13H18NO4P
dimethyl (E)-2-acetylamino-2-p-tolylvinylphosphonate
—— 4-[p-(N,N'-dibutyl-N'-phenyl)phenylene-diamino]-phenyl-6-phenyl-2,2'-bipyridine 1142955-66-5 C42H42N4
4-[p-(N,N'-dibutyl-N'-phenyl)phenylene-diamino]-phenyl-6-phenyl-2,2'-bipyridine
—— 5-(3,5-bis(trifluoromethyl)phenyl)-3-((4'-fluoro-5'-isopropyl-2'-methoxy-4-fluorobiphenyl-2-yl)methyl)-4-methylthiazolidin-2-one 1370452-36-0 C29H25F8NO2S
5-(3,5-bis(trifluoromethyl)phenyl)-3-((4'-fluoro-5'-isopropyl-2'-methoxy-4-fluorobiphenyl-2-yl)methyl)-4-methylthiazolidin-2-one
—— (1R,2S)-N-(2,4-difluorophenyl)-2-(3-fluorophenyl)-2-{[(4-methoxymethyl-2-methylpyrimidin-5-yl)oxy]methyl}cyclopropanecarboxamide 1369765-03-6 C24H22F3N3O3
(1R,2S)-N-(2,4-difluorophenyl)-2-(3-fluorophenyl)-2-{[(4-methoxymethyl-2-methylpyrimidin-5-yl)oxy]methyl}cyclopropanecarboxamide
—— (E)-3-(4-((Z)-1-(1H-indazol-5-yl)-2-phenylbut-1-en-1-yl)-3-fluorophenyl)acrylic acid 1366770-76-4 C26H21FN2O2
(E)-3-(4-((Z)-1-(1H-indazol-5-yl)-2-phenylbut-1-en-1-yl)-3-fluorophenyl)acrylic acid
—— (3aR,4R,6S,7aR)-6-cyclohexyloxy-4-[(4R)-2,2-dimethyl-1,3-dioxolan-4-yl]-6-(4-methoxyphenyl)-2,2-dimethyl-3a,4,7,7a-tetrahydro-[1,3]dioxolo[4,5-c]pyran 1351958-30-9 C26H38O7
(3aR,4R,6S,7aR)-6-cyclohexyloxy-4-[(4R)-2,2-dimethyl-1,3-dioxolan-4-yl]-6-(4-methoxyphenyl)-2,2-dimethyl-3a,4,7,7a-tetrahydro-[1,3]dioxolo[4,5-c]pyran
—— 2-[3-(3-chlorophenyl)-1-{4-[2-(morpholin-4-yl)ethyl]phenyl}-5-oxo-1,5-dihydro-4H-1,2,4-triazol-4-yl]-N-(1,1,1-trifluoropropan-2-yl)acetamide 1370446-04-0 C25H27ClF3N5O3
2-[3-(3-chlorophenyl)-1-{4-[2-(morpholin-4-yl)ethyl]phenyl}-5-oxo-1,5-dihydro-4H-1,2,4-triazol-4-yl]-N-(1,1,1-trifluoropropan-2-yl)acetamide
—— (5S,5'S,8S,8'S,10aR,10a'R)-3,3'-adipoylbis(N-benzhydryl-5-((S)-2-(methylamino)propanamido)-6-oxodecahydropyrrolo-[1,2-a][1,5]diazocine-8-carboxamide) 1352130-33-6 C60H76N10O8
(5S,5'S,8S,8'S,10aR,10a'R)-3,3'-adipoylbis(N-benzhydryl-5-((S)-2-(methylamino)propanamido)-6-oxodecahydropyrrolo-[1,2-a][1,5]diazocine-8-carboxamide)
—— N-[[5-[4-(benzotriazol-1-ylmethoxy)phenyl]-1,3,4-oxadiazol-2-yl]methyl]-2-oxo-8-phenyloctanamide 1369795-81-2 C30H30N6O4
N-[[5-[4-(benzotriazol-1-ylmethoxy)phenyl]-1,3,4-oxadiazol-2-yl]methyl]-2-oxo-8-phenyloctanamide
—— 1-(4-(4-(4-(4-(aminomethyl)piperidin-1-yl)furo[3,2-d]pyrimidin-2-ylamino)phenyl)piperazin-1-yl)ethanone 1372531-28-6 C24H31N7O2
1-(4-(4-(4-(4-(aminomethyl)piperidin-1-yl)furo[3,2-d]pyrimidin-2-ylamino)phenyl)piperazin-1-yl)ethanone
—— (S)-3-(2,6-difluoro-4-(methylsulfonyl)phenylamino)-1'-(5-(1,1-difluoroethyl)-1,2,4-oxadiazol-3-yl)-1,4'-bipiperidin-2-one 1365998-25-9 C21H25F4N5O4S
(S)-3-(2,6-difluoro-4-(methylsulfonyl)phenylamino)-1'-(5-(1,1-difluoroethyl)-1,2,4-oxadiazol-3-yl)-1,4'-bipiperidin-2-one
—— 3-[[4-(4-fluorophenoxy)phenyl]methoxymethyl]piperidine 876148-18-4 C19H22FNO2
3-[[4-(4-fluorophenoxy)phenyl]methoxymethyl]piperidine
—— Ethyl 5-(furan-2-carbonylamino)-1-(4-methoxyphenyl)pyrazolo[3,4-d][1,3]thiazole-3-carboxylate 866838-26-8 C19H16N4O5S
Ethyl 5-(furan-2-carbonylamino)-1-(4-methoxyphenyl)pyrazolo[3,4-d][1,3]thiazole-3-carboxylate
—— 5-(6-methyl-2-pyridinyl)-2-thiophenesulfonyl chloride 874959-49-6 C10H8ClNO2S2
5-(6-methyl-2-pyridinyl)-2-thiophenesulfonyl chloride
—— Mes-D-Abu(4-piperidyl)-Hyp(piperidine-1-carbonyl)-Phe(3-amidino)-benzoxazol-2-yl 959424-90-9 C38H50N8O8S
Mes-D-Abu(4-piperidyl)-Hyp(piperidine-1-carbonyl)-Phe(3-amidino)-benzoxazol-2-yl
—— 1-(1-Adamantyloxy)ethyl 4-[[5-[1-(1-adamantyloxy)ethoxy]-2-cyano-5-oxopentan-2-yl]diazenyl]-4-cyanopentanoate 957580-99-3 C36H52N4O6
1-(1-Adamantyloxy)ethyl 4-[[5-[1-(1-adamantyloxy)ethoxy]-2-cyano-5-oxopentan-2-yl]diazenyl]-4-cyanopentanoate
—— 14-Methoxy-2-oxo-1,3,10-trioxa-2lambda4-thiacycloheptadecan-9-one 1122438-72-5 C14H26O6S
14-Methoxy-2-oxo-1,3,10-trioxa-2lambda4-thiacycloheptadecan-9-one
—— 4-[(3R)-3-[methyl(methylsulfamoyl)amino]pyrrolidin-1-yl]-7H-pyrrolo[2,3-d]pyrimidine 1360092-28-9 C12H18N6O2S
4-[(3R)-3-[methyl(methylsulfamoyl)amino]pyrrolidin-1-yl]-7H-pyrrolo[2,3-d]pyrimidine
—— (1R,2S)-N-(3,4-difluorophenyl)-2-(3-fluoro-5-methoxyphenyl)-2-{[(4-methoxymethyl-2-methylpyrimidin-5-yl)oxy]methyl}cyclopropanecarboxamide 1369765-40-1 C25H24F3N3O4
(1R,2S)-N-(3,4-difluorophenyl)-2-(3-fluoro-5-methoxyphenyl)-2-{[(4-methoxymethyl-2-methylpyrimidin-5-yl)oxy]methyl}cyclopropanecarboxamide
—— 1-[2-[5-amino-1-(cyclopropylmethyl)-8-(2-furyl)-2-oxo-[1,2,4]triazolo[5,1-f]purin-3-yI]ethyl]pyrazoIe-4-carboxyIic acid 1367365-99-8 C20H19N9O4
1-[2-[5-amino-1-(cyclopropylmethyl)-8-(2-furyl)-2-oxo-[1,2,4]triazolo[5,1-f]purin-3-yI]ethyl]pyrazoIe-4-carboxyIic acid
—— 5-[(2,5-dimethyl-4-thiazolyl)acetyl]-4,5,6,7-tetrahydro-3-(4-pyridinyl)-1H-pyrazolo[4,3-c]pyridine 1366050-82-9 C18H19N5OS
5-[(2,5-dimethyl-4-thiazolyl)acetyl]-4,5,6,7-tetrahydro-3-(4-pyridinyl)-1H-pyrazolo[4,3-c]pyridine
—— [(1S,11S,13R,16S)-16-[tert-butyl(dimethyl)silyl]oxy-11-(2-hydroxyethyl)-9-oxo-10,17-dioxatricyclo[11.3.1.03,8]heptadeca-3(8),4,6-trien-7-yl] acetate 1350978-98-1 C25H38O7Si
[(1S,11S,13R,16S)-16-[tert-butyl(dimethyl)silyl]oxy-11-(2-hydroxyethyl)-9-oxo-10,17-dioxatricyclo[11.3.1.03,8]heptadeca-3(8),4,6-trien-7-yl] acetate
—— 2-({4-[({2-[ethyl(methylsulfonyl)amino]pyridin-3-yl}amino)methyl]-7H-pyrrolo[2,3-d]pyrimidin-2-yl}amino)-N-methylbenzamide 1372263-51-8 C23H26N8O3S
2-({4-[({2-[ethyl(methylsulfonyl)amino]pyridin-3-yl}amino)methyl]-7H-pyrrolo[2,3-d]pyrimidin-2-yl}amino)-N-methylbenzamide
—— sodium 3-(phenylacetamido)but-1-enesulfonate 134077-06-8 C12H14NO4S*Na
sodium 3-(phenylacetamido)but-1-enesulfonate
—— N-[4-(6,7-dimethoxyquinolin-4-yloxy)-2-fluorophenyl]-3-methylbenzenesulfonamide 1192298-28-4 C24H21FN2O5S
N-[4-(6,7-dimethoxyquinolin-4-yloxy)-2-fluorophenyl]-3-methylbenzenesulfonamide
—— (4-bromophenyl)(4-(4-(pyridin-4-yl)piperazine-1-carbonyl)piperazin-1-yl)methanone 875545-73-6 C21H24BrN5O2
(4-bromophenyl)(4-(4-(pyridin-4-yl)piperazine-1-carbonyl)piperazin-1-yl)methanone
—— (E)-2-(butylselanyliodomethylene)tetrahydroselenophene 1414874-94-4 C9H15ISe2
(E)-2-(butylselanyliodomethylene)tetrahydroselenophene
—— N-[[1-[(4-amino-2-methylpyrimidin-5-yl)methyl]-5-iodotriazol-4-yl]methyl]benzamide 1428141-01-8 C16H16IN7O
N-[[1-[(4-amino-2-methylpyrimidin-5-yl)methyl]-5-iodotriazol-4-yl]methyl]benzamide
—— 3-phenyl-N-(3-(piperidin-1-yl)propyl)-3H-spiro[isobenzofuran-1,4'-piperidine]-1'-carboxamide 875546-95-5 C27H35N3O2
3-phenyl-N-(3-(piperidin-1-yl)propyl)-3H-spiro[isobenzofuran-1,4'-piperidine]-1'-carboxamide
—— (1R,2S)-2-ammo-1-{[(2-{4-[(3-chlorobenzyl)oxy]phenyl}ethyl)amino]methyl}-3-(3,5-difluorophenyl)propyl 3-[(dipropylamino)carbonyl]-5-methylbenzoate 674316-11-1 C40H46ClF2N3O4
(1R,2S)-2-ammo-1-{[(2-{4-[(3-chlorobenzyl)oxy]phenyl}ethyl)amino]methyl}-3-(3,5-difluorophenyl)propyl 3-[(dipropylamino)carbonyl]-5-methylbenzoate
—— (R)-1-(tert-butoxycarbonyl)-3-[[2-(4-chlorophenyl)-4-methylthiazol-5-yl]methoxy]piperidine 876148-42-4 C21H27ClN2O3S
(R)-1-(tert-butoxycarbonyl)-3-[[2-(4-chlorophenyl)-4-methylthiazol-5-yl]methoxy]piperidine
—— 5-bromo-2-[3-(5-bromo-1,3-dihydro-1,3,3-trimethyl-2H-indol-2-yliden)-1-propen-1-yl]-1,3,3-trimethyl-3H-indolium iodide 1254943-06-0 C25H27Br2N2*I
5-bromo-2-[3-(5-bromo-1,3-dihydro-1,3,3-trimethyl-2H-indol-2-yliden)-1-propen-1-yl]-1,3,3-trimethyl-3H-indolium iodide
—— methyl 2-[[(1R,2S)-2-[[2-[[(1R,2S)-2-[[2-[[(1R,2S)-2-[[2-[[(1R,2S)-2-(phenylmethoxycarbonylamino)cyclobutanecarbonyl]amino]acetyl]amino]cyclobutanecarbonyl]amino]acetyl]amino]cyclobutanecarbonyl]amino]acetyl]amino]cyclobutanecarbonyl]amino]acetate 1353742-66-1 C37H50N8O11
methyl 2-[[(1R,2S)-2-[[2-[[(1R,2S)-2-[[2-[[(1R,2S)-2-[[2-[[(1R,2S)-2-(phenylmethoxycarbonylamino)cyclobutanecarbonyl]amino]acetyl]amino]cyclobutanecarbonyl]amino]acetyl]amino]cyclobutanecarbonyl]amino]acetyl]amino]cyclobutanecarbonyl]amino]acetate
—— 1-(4-(2-amino-9-benzyl-8-(4-fluorophenyl)-9H-purin-6-yl)piperazin-1-yl)-2-(4-chlorophenoxy)ethanone 1245321-14-5 C30H27ClFN7O2
1-(4-(2-amino-9-benzyl-8-(4-fluorophenyl)-9H-purin-6-yl)piperazin-1-yl)-2-(4-chlorophenoxy)ethanone
—— 4-(4-(4-fluorophenoxy)phenyl)-2-(4-methylpiperazin-1-yl)quinazoline 1371596-00-7 C25H23FN4O
4-(4-(4-fluorophenoxy)phenyl)-2-(4-methylpiperazin-1-yl)quinazoline
—— N-[[5-(4-methylphenyl)-1,3,4-oxadiazol-2-yl]methyl]-2-oxo-7-(4-phenylphenyl)heptanamide 1369795-16-3 C29H29N3O3
N-[[5-(4-methylphenyl)-1,3,4-oxadiazol-2-yl]methyl]-2-oxo-7-(4-phenylphenyl)heptanamide
—— 6-chloro-3-(1-(N-(4-chIorobenzyl)acetamido)-2-(cyclohexylamino)-2-oxoethyl)-1H-indole-2-carboxylic acid 1364488-78-7 C26H27Cl2N3O4
6-chloro-3-(1-(N-(4-chIorobenzyl)acetamido)-2-(cyclohexylamino)-2-oxoethyl)-1H-indole-2-carboxylic acid
—— 2-[5-hydroxy-2-(4-hydroxy-phenyl)-7-methyl-benzofuran-3-yl]-thiophene-3-carbonitrile 1191045-72-3 C20H13NO3S
2-[5-hydroxy-2-(4-hydroxy-phenyl)-7-methyl-benzofuran-3-yl]-thiophene-3-carbonitrile
—— 4-bromo-5-(3,4-dihydro-1H-isoquinolin-2-yl)-benzofuran-2-carboxylic acid 1192171-62-2 C18H14BrNO3
4-bromo-5-(3,4-dihydro-1H-isoquinolin-2-yl)-benzofuran-2-carboxylic acid
—— N-(5-{[(2-chloro-5-fluorophenyl)oxy]methyl}-1,3,4-thiadiazol-2-yl)-1,2,3,4-tetrahydro-6-isoquinolinecarboxamide hydrochloride 1052693-10-3 C19H16ClFN4O2S*ClH
N-(5-{[(2-chloro-5-fluorophenyl)oxy]methyl}-1,3,4-thiadiazol-2-yl)-1,2,3,4-tetrahydro-6-isoquinolinecarboxamide hydrochloride
—— 2-(5-piperidin-4-yl-2H-[1,2,4]triazol-3-yl)-6-trifluoromethyl-pyridine hydrochloride 1240108-71-7 C13H14F3N5*ClH
2-(5-piperidin-4-yl-2H-[1,2,4]triazol-3-yl)-6-trifluoromethyl-pyridine hydrochloride
—— methyl 2-[4-(pyridin-3-ylethynyl)phenyl]pyridine-4-carboxylate 1244017-04-6 C20H14N2O2
methyl 2-[4-(pyridin-3-ylethynyl)phenyl]pyridine-4-carboxylate
—— 1-phenyl-3-{1-[1-(t-butyloxycarbonyl)-1H-pyrrolo[2,3-b]pyridin-3-ylmethyl]-1H-indol-4-yl}urea 1268390-83-5 C28H27N5O3
1-phenyl-3-{1-[1-(t-butyloxycarbonyl)-1H-pyrrolo[2,3-b]pyridin-3-ylmethyl]-1H-indol-4-yl}urea
—— N-1-aza-bicyclo[2.2.2]oct-3R-yl-4-fluoro-N-[2-fluoro-5-(2-oxo-2,3-dihydro-benzooxazol-6-yl)-benzyl]-benzamide hydrochloride 906002-59-3 C28H25F2N3O3*ClH
N-1-aza-bicyclo[2.2.2]oct-3R-yl-4-fluoro-N-[2-fluoro-5-(2-oxo-2,3-dihydro-benzooxazol-6-yl)-benzyl]-benzamide hydrochloride
—— N-(3-tert-butylpyrazolo[1,5-a]pyrimidin-2-yl)-3-cyclohexylpropanamide 1375087-48-1 C19H28N4O
N-(3-tert-butylpyrazolo[1,5-a]pyrimidin-2-yl)-3-cyclohexylpropanamide
—— 5-(4-bromophenyl)-3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-(2,4-dichlorophenyl)-N-(pyridin-2-yl)-1H-pyrazole-4-carboxamide 1161827-58-2 C27H21BrCl2N6OS
5-(4-bromophenyl)-3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-(2,4-dichlorophenyl)-N-(pyridin-2-yl)-1H-pyrazole-4-carboxamide