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—— 5-chloro-N<sup>2</sup>-((prop-2-yloxy)-5-methyl-4-(piperidin-4-yl)phenyl)-N<sup>4</sup>-(2-(isopropylsulfonyl)phenyl)pyrimidine-2,4-diamine —— C28H36ClN5O3S
5-chloro-N<sup>2</sup>-((prop-2-yloxy)-5-methyl-4-(piperidin-4-yl)phenyl)-N<sup>4</sup>-(2-(isopropylsulfonyl)phenyl)pyrimidine-2,4-diamine
—— 6-chloro-N<sup>3</sup>-[5-(dimethylphosphoryl)-2-methoxyphenyl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine —— C21H25ClN5O4PS
6-chloro-N<sup>3</sup>-[5-(dimethylphosphoryl)-2-methoxyphenyl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine
—— 3-amino-N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)propanamide —— C22H25ClN6O3S
3-amino-N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)propanamide
—— N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)-2-(hexahydropyrrolo[3,4-b]pyrrol-1(2H)-yl)acetamide —— C27H32ClN7O3S
N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)-2-(hexahydropyrrolo[3,4-b]pyrrol-1(2H)-yl)acetamide
—— (E)-N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)-amino)pyrimidin-2-yl)amino)phenyl)-2-(4-(4-(dimethylamino)but-2-enoyl)piperazin-1-yl)acetamide —— C31H39ClN8O4S
(E)-N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)-amino)pyrimidin-2-yl)amino)phenyl)-2-(4-(4-(dimethylamino)but-2-enoyl)piperazin-1-yl)acetamide
—— N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)-2-morpholinoacetamide —— C25H29ClN6O4S
N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)-2-morpholinoacetamide
—— ethyl (2S,3aS,6S)-6-(2-methyl-2-propenyl)-2,3,3a,4,5,6-hexahydro-1H-indolo<3,2,1-de><1,5>naphthyridine-2-carboxylate —— C21H26N2O2
ethyl (2S,3aS,6S)-6-(2-methyl-2-propenyl)-2,3,3a,4,5,6-hexahydro-1H-indolo<3,2,1-de><1,5>naphthyridine-2-carboxylate
—— N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)-2-(1H-indol-2-yl)acetamide —— C29H27ClN6O3S
N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)-2-(1H-indol-2-yl)acetamide
—— N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)-2-(hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl)acetamide —— C27H32ClN7O3S
N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)-2-(hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl)acetamide
—— (E)-5-chloro-2-(2-(2,4-difluorobenzylidene)hydrazinyl)-N-(2-(isopropylsulfonyl)phenyl)pyrimidin-4-amine —— C20H18ClF2N5O2S
(E)-5-chloro-2-(2-(2,4-difluorobenzylidene)hydrazinyl)-N-(2-(isopropylsulfonyl)phenyl)pyrimidin-4-amine
—— N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)-2-(4-(2-hydroxyacetyl)piperazin-1-yl)acetamide —— C27H32ClN7O5S
N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)-2-(4-(2-hydroxyacetyl)piperazin-1-yl)acetamide
—— 6-chloro-N<sup>3</sup>-[4-(1-ethyl-4-oxido-1,4-azaphosphinan-4-yl)-2-methoxyphenyl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine —— C25H32ClN6O4PS
6-chloro-N<sup>3</sup>-[4-(1-ethyl-4-oxido-1,4-azaphosphinan-4-yl)-2-methoxyphenyl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine
—— N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)-amino)pyrimidin-2-yl)amino)phenyl)-1-(4-(dimethylamino)butanoyl)azetidine-3-carboxamide —— C29H36ClN7O4S
N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)-amino)pyrimidin-2-yl)amino)phenyl)-1-(4-(dimethylamino)butanoyl)azetidine-3-carboxamide
—— 2-(2,5-diazabicyclo[2.2.1]heptan-2-yl)-N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)acetamide —— C26H30ClN7O3S
2-(2,5-diazabicyclo[2.2.1]heptan-2-yl)-N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)acetamide
—— (E)-5-chloro-2-(2-(1-(4-fluorophenyl)ethylidene)hydrazinyl)-N-(2-(isopropylsulfonyl)phenyl)pyrimidin-4-amine —— C21H21ClFN5O2S
(E)-5-chloro-2-(2-(1-(4-fluorophenyl)ethylidene)hydrazinyl)-N-(2-(isopropylsulfonyl)phenyl)pyrimidin-4-amine
—— N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)-2-(piperazin-1-yl)acetamide —— C25H30ClN7O3S
N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)-2-(piperazin-1-yl)acetamide
—— N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)-2-(3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl)acetamide —— C27H31ClN6O4S
N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)-2-(3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl)acetamide
—— 1-amino-N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)cyclopropanecarboxamide —— C23H25ClN6O3S
1-amino-N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)cyclopropanecarboxamide
—— nickel-tin —— NiSn
nickel-tin
—— 5-chloro-N<sup>2</sup>-(2-(2-d-prop-2-yloxyl)-5-methyl-4-(2,2,6,6-tetrafluoropiperidin-4-yl)phenyl)-N<sup>4</sup>-(2-(isopropylsulfonyl)phenyl)pyrimidine-2,4-diamine —— C28H36ClN5O3S
5-chloro-N<sup>2</sup>-(2-(2-d-prop-2-yloxyl)-5-methyl-4-(2,2,6,6-tetrafluoropiperidin-4-yl)phenyl)-N<sup>4</sup>-(2-(isopropylsulfonyl)phenyl)pyrimidine-2,4-diamine
—— 2-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)acetamide —— C27H31ClN6O4S
2-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)acetamide
—— N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)-2-(4-methylpiperazin-1-yl)acetamide —— C26H32ClN7O3S
N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)-2-(4-methylpiperazin-1-yl)acetamide
—— 5-chloro-N<sup>2</sup>-(2-(d<sub>7</sub>-isopropoxy)-5-methyl-4-(piperidin-4-yl)phenyl)-N<sup>4</sup>-(2-(isopropylsulfonyl)phenyl)pyrimidine-2,4-diamine —— C28H36ClN5O3S
5-chloro-N<sup>2</sup>-(2-(d<sub>7</sub>-isopropoxy)-5-methyl-4-(piperidin-4-yl)phenyl)-N<sup>4</sup>-(2-(isopropylsulfonyl)phenyl)pyrimidine-2,4-diamine
—— (E)-5-chloro-N-(2-(isopropylsulfonyl)phenyl)-2-(2-(1-(4-methoxyphenyl)ethylidene)hydrazinyl)pyrimidin-4-amine —— C22H24ClN5O3S
(E)-5-chloro-N-(2-(isopropylsulfonyl)phenyl)-2-(2-(1-(4-methoxyphenyl)ethylidene)hydrazinyl)pyrimidin-4-amine
—— (S)-2-amino-N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)-3-(1H-imidazol-4-yl)propanamide —— C25H27ClN8O3S
(S)-2-amino-N-(3-((5-chloro-4-((2-(isopropylsulfonyl)phenyl)amino)pyrimidin-2-yl)amino)phenyl)-3-(1H-imidazol-4-yl)propanamide
—— 6-chloro-N<sup>3</sup>-[4-(diethylphosphoryl)-2-methoxyphenyl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine —— C23H29ClN5O4PS
6-chloro-N<sup>3</sup>-[4-(diethylphosphoryl)-2-methoxyphenyl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine
—— 6-chloro-N<sup>3</sup>-[4-(dimethylphosphoryl)-2-ethylphenyl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine —— C22H27ClN5O3PS
6-chloro-N<sup>3</sup>-[4-(dimethylphosphoryl)-2-ethylphenyl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine
—— 6-chloro-N<sup>3</sup>-[4-(dimethylphosphoryl)-2-(trifluoromethoxy)phenyl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine —— C21H22ClF3N5O4PS
6-chloro-N<sup>3</sup>-[4-(dimethylphosphoryl)-2-(trifluoromethoxy)phenyl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine
—— 6-chloro-N<sup>3</sup>-[6-(dimethylphosphoryl)-2-methoxypyridin-3-yl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine —— C20H24ClN6O4PS
6-chloro-N<sup>3</sup>-[6-(dimethylphosphoryl)-2-methoxypyridin-3-yl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine
—— 6-chloro-N<sup>3</sup>-[4-(dimethylphosphoryl)-2-fluorophenyl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine —— C20H22ClFN5O3PS
6-chloro-N<sup>3</sup>-[4-(dimethylphosphoryl)-2-fluorophenyl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine
—— 2-benzyloxetan-3-one —— C10H10O2
2-benzyloxetan-3-one
—— 6-chloro-N<sup>3</sup>-{2-methoxy-4-[4-(4-methyl-4-oxido-1,4-azaphosphinan-1-yl)piperidin-1-yl]phenyl}-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine —— C29H39ClN7O4PS
6-chloro-N<sup>3</sup>-{2-methoxy-4-[4-(4-methyl-4-oxido-1,4-azaphosphinan-1-yl)piperidin-1-yl]phenyl}-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine
—— 6-chloro-N<sup>3</sup>-[2-methoxy-4-(4-methyl-4-oxido-1,4-azaphosphinan-1-yl)phenyl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine —— C24H30ClN6O4PS
6-chloro-N<sup>3</sup>-[2-methoxy-4-(4-methyl-4-oxido-1,4-azaphosphinan-1-yl)phenyl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine
—— (2S,3S,3'S)-ethyl-2-benzyl-2',3',4',9'-tetrahydrospiro[oxetane-3,1'-pyrido[3,4-b]indole]-3'-carboxylate —— C23H24N2O3
(2S,3S,3'S)-ethyl-2-benzyl-2',3',4',9'-tetrahydrospiro[oxetane-3,1'-pyrido[3,4-b]indole]-3'-carboxylate
—— (2S,3aS,8aS)-ethyl 3a-(3-((S)-2-amino-3-ethoxy-3-oxopropyl)-1H-indol-6-yl)-1,2,3,3a,8,8a-hexahydropyrrolo[2, 3-b]indole-2-carboxylate —— C26H30N4O4
(2S,3aS,8aS)-ethyl 3a-(3-((S)-2-amino-3-ethoxy-3-oxopropyl)-1H-indol-6-yl)-1,2,3,3a,8,8a-hexahydropyrrolo[2, 3-b]indole-2-carboxylate
—— 6-chloro-N<sup>3</sup>-[4-(dimethylphosphoryl)-2-methylphenyl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine —— C21H25ClN5O3PS
6-chloro-N<sup>3</sup>-[4-(dimethylphosphoryl)-2-methylphenyl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine
—— 6-chloro-N<sup>3</sup>-[2-chloro-4-(dimethylphosphoryl)phenyl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine —— C20H22Cl2N5O3PS
6-chloro-N<sup>3</sup>-[2-chloro-4-(dimethylphosphoryl)phenyl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine
—— (2S,2'S,3aR,3'aR,8aS,8'aS)-diethyl 2,2',3,3',8,8a,8',8'a-octahydro-1H,1'H-[3a,3'a-bipyrrolo[2, 3-b]indole]-2,2'-dicarboxylate —— C26H30N4O4
(2S,2'S,3aR,3'aR,8aS,8'aS)-diethyl 2,2',3,3',8,8a,8',8'a-octahydro-1H,1'H-[3a,3'a-bipyrrolo[2, 3-b]indole]-2,2'-dicarboxylate
—— (2R,3R,3'S)-ethyl-2-benzyl-2',3',4',9'-tetrahydrospiro[oxetane-3,1'-pyrido[3,4-b]-indole]-3'-carboxylate —— C23H24N2O3
(2R,3R,3'S)-ethyl-2-benzyl-2',3',4',9'-tetrahydrospiro[oxetane-3,1'-pyrido[3,4-b]-indole]-3'-carboxylate
—— (2S,2'S,3aS,3'aS,8aR,8'aR)-diethyl 2,2',3,3',8,8a,8',8'a-octahydro-1H,1'H-[3a, 3'a-bipyrrolo[2,3-b]indole]-2,2'-dicarboxylate —— C26H30N4O4
(2S,2'S,3aS,3'aS,8aR,8'aR)-diethyl 2,2',3,3',8,8a,8',8'a-octahydro-1H,1'H-[3a, 3'a-bipyrrolo[2,3-b]indole]-2,2'-dicarboxylate
—— 6-chloro-N<sup>3</sup>-[5-(dimethylphosphoryl)-3-methoxypyrazin-2-yl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine —— C19H23ClN7O4PS
6-chloro-N<sup>3</sup>-[5-(dimethylphosphoryl)-3-methoxypyrazin-2-yl]-N<sup>5</sup>-[2-(propan-2-ylsulfonyl)phenyl]-1,2,4-triazine-3,5-diamine
—— (2S,3aR,8aR)-ethyl 3a-(3-((S)-2-amino-3-ethoxy-3-oxopropyl)-1H-indol-6-yl)-1,2,3,3a,8,8a-hexahydropyrrolo[2,3-b]indole-2-carboxylate —— C26H30N4O4
(2S,3aR,8aR)-ethyl 3a-(3-((S)-2-amino-3-ethoxy-3-oxopropyl)-1H-indol-6-yl)-1,2,3,3a,8,8a-hexahydropyrrolo[2,3-b]indole-2-carboxylate
—— 7-amino-5-bromo-3-chloro-1H-indole —— C8H6BrClN2
7-amino-5-bromo-3-chloro-1H-indole
—— (1S,2S,3S)-ethyl 2-phenethyl-2',3',4',9'-tetrahydrospiro[oxetane-3,1'-pyrido[3,4-b]indole]-3'-carboxylate —— C24H26N2O3
(1S,2S,3S)-ethyl 2-phenethyl-2',3',4',9'-tetrahydrospiro[oxetane-3,1'-pyrido[3,4-b]indole]-3'-carboxylate
—— 5-Bromo-3-chloro-7-nitro-1H-indole —— C8H4BrClN2O2
5-Bromo-3-chloro-7-nitro-1H-indole
—— 5-chloro-N2-(2-isopropoxy-5-methyl-4-(1-(1-methylpiperidin-4-yl)piperidin-4-yl)phenyl )-N4-(2-(isopropylsulfonyl)phenyl)pyrimidine-2,4-diamine hydrochloride —— C34H47ClN6O3S*(x)ClH
5-chloro-N2-(2-isopropoxy-5-methyl-4-(1-(1-methylpiperidin-4-yl)piperidin-4-yl)phenyl )-N4-(2-(isopropylsulfonyl)phenyl)pyrimidine-2,4-diamine hydrochloride
—— (S)-ethyl 2-((S)-2-(((benzyloxy)carbonyl)(methyl)amino)propanamido)-3-(1H-indol-3-yl)propanoate —— C25H29N3O5
(S)-ethyl 2-((S)-2-(((benzyloxy)carbonyl)(methyl)amino)propanamido)-3-(1H-indol-3-yl)propanoate
—— (1R,2R,3S)-ethyl 2-phenethyl-2',3',4',9'-tetrahydrospiro[oxetane-3,1'-pyrido[3,4-b]indole]-3'-carboxylate —— C24H26N2O3
(1R,2R,3S)-ethyl 2-phenethyl-2',3',4',9'-tetrahydrospiro[oxetane-3,1'-pyrido[3,4-b]indole]-3'-carboxylate
—— <i>N</i>,<i>N</i>-diethyl-DL-aspartic acid —— C8H15NO4
<i>N</i>,<i>N</i>-diethyl-DL-aspartic acid
—— Gold--lambda~2~-stannane (5/1) 12006-74-5 Au5Sn
Gold--lambda~2~-stannane (5/1)