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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-(3-(5-(2-(3-(2-(dimethylamino)ethyl)phenylamino)pyrimidin-4-yl)imidazo[2,1-b]thiazol-6-yl)phenyl)-2-phenylacetamide 1228004-70-3 C33H31N7OS
N-(3-(5-(2-(3-(2-(dimethylamino)ethyl)phenylamino)pyrimidin-4-yl)imidazo[2,1-b]thiazol-6-yl)phenyl)-2-phenylacetamide
—— N-(3-(5-(2-(4-(4-ethylpiperazin-1-yl)phenylamino)pyrimidin-4-yl)imidazo[2,1-b]thiazol-6-yl)phenyl)-2-phenylacetamide 1160061-35-7 C35H34N8OS
N-(3-(5-(2-(4-(4-ethylpiperazin-1-yl)phenylamino)pyrimidin-4-yl)imidazo[2,1-b]thiazol-6-yl)phenyl)-2-phenylacetamide
—— N6-[4-[2-[3,5-Di-tert-butylbenzamido]ethyl]benzyl]adenosine-5''-N-methylcarboxamide 1233488-03-3 C34H43N7O5
N6-[4-[2-[3,5-Di-tert-butylbenzamido]ethyl]benzyl]adenosine-5''-N-methylcarboxamide
—— N-[(2-chloro-4-fluorophenyl)methyl]-2-(3,5-dimethyl-2-phenylimidazol-4-yl)acetamide 1232975-52-8 C20H19ClFN3O
N-[(2-chloro-4-fluorophenyl)methyl]-2-(3,5-dimethyl-2-phenylimidazol-4-yl)acetamide
—— N-(7-benzyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c][2,7]naphthyridin-1-yl)isobutyramide 1228692-60-1 C25H32N6O
N-(7-benzyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c][2,7]naphthyridin-1-yl)isobutyramide
—— N-(4-chlorobenzyl)-8-(morpholin-4-ylmethyl)-6-oxo-2-(piperazin-1-ylmethyl)-6H-pyrrolo[3,2,1-ij]quinoline-5-carboxamide 1232152-27-0 C29H32ClN5O3
N-(4-chlorobenzyl)-8-(morpholin-4-ylmethyl)-6-oxo-2-(piperazin-1-ylmethyl)-6H-pyrrolo[3,2,1-ij]quinoline-5-carboxamide
—— N-(7-benzyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c][2,7]naphthyridin-1-yl)acetamide 1228692-58-7 C23H28N6O
N-(7-benzyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c][2,7]naphthyridin-1-yl)acetamide
—— N-ethyl-N'-[4-(1-ethyl-4-{2-[4-(1-pyrrolidinylmethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazol-3-yl)phenyl]urea 942918-25-4 C32H35N7O
N-ethyl-N'-[4-(1-ethyl-4-{2-[4-(1-pyrrolidinylmethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazol-3-yl)phenyl]urea
—— N-(3-bromophenyl)-6-(2-phenylethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine 1228352-51-9 C20H17BrN4
N-(3-bromophenyl)-6-(2-phenylethyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine
—— N-(7-benzyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c][2,7]naphthyridin-1-yl)propionamide 1228692-59-8 C24H30N6O
N-(7-benzyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c][2,7]naphthyridin-1-yl)propionamide
—— N-(7-benzyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c][2,7]naphthyridin-1-yl)cyclopentanecarboxamide 1348124-74-2 C27H34N6O
N-(7-benzyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c][2,7]naphthyridin-1-yl)cyclopentanecarboxamide
—— N-[2-(3,5-ditert-butyl-4-hydroxyphenyl)ethyl]-N'-[4-[[[9-[(2R,3R,4S,5S)-3,4-dihydroxy-5-(methylcarbamoyl)oxolan-2-yl]purin-6-yl]amino]methyl]phenyl]butanediamide 1233488-14-6 C38H50N8O7
N-[2-(3,5-ditert-butyl-4-hydroxyphenyl)ethyl]-N'-[4-[[[9-[(2R,3R,4S,5S)-3,4-dihydroxy-5-(methylcarbamoyl)oxolan-2-yl]purin-6-yl]amino]methyl]phenyl]butanediamide
—— N1-((1S,2S)-1-((R)-4-(3-chlorophenylsulfonyl)piperazin-2-yl)-3-(3,5-difluorophenyl)-1-hydroxypropan-2-yl)-5-methyl-N3,N3-dipropylisophthalamide 1230559-08-6 C34H41ClF2N4O5S
N1-((1S,2S)-1-((R)-4-(3-chlorophenylsulfonyl)piperazin-2-yl)-3-(3,5-difluorophenyl)-1-hydroxypropan-2-yl)-5-methyl-N3,N3-dipropylisophthalamide
—— N-(3-{4-[1-ethyl-3-(4-{[(phenylamino)carbonyl]amino}phenyl)-1H-pyrazol-4-yl]-1H-pyrrolo[2,3-b]pyridin-2-yl}phenyl)acetamide 942918-14-1 C33H29N7O2
N-(3-{4-[1-ethyl-3-(4-{[(phenylamino)carbonyl]amino}phenyl)-1H-pyrazol-4-yl]-1H-pyrrolo[2,3-b]pyridin-2-yl}phenyl)acetamide
—— N-phenyl-N'-{4-[4-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrazol-3-yl]phenyl}urea 942919-20-2 C23H18N6O
N-phenyl-N'-{4-[4-(1H-pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrazol-3-yl]phenyl}urea
—— N1-((1S,2S)-1-((R)-4-(2-chlorophenylsulfonyl)piperazin-2-yl)-3-(3,5-difluorophenyl)-1-hydroxypropan-2-yl)-5-methyl-N3,N3-dipropylisophthalamide 1230559-06-4 C34H41ClF2N4O5S
N1-((1S,2S)-1-((R)-4-(2-chlorophenylsulfonyl)piperazin-2-yl)-3-(3,5-difluorophenyl)-1-hydroxypropan-2-yl)-5-methyl-N3,N3-dipropylisophthalamide
—— N1-((1S,2S)-3-(3,5-difluorophenyl)-1-((R)-4-(3,5-dimethylisoxazol-4-ylsulfonyl)piperazin-2-yl)-1-hydroxypropan-2-yl)-5-methyl-N3,N3-dipropylisophthalamide 1230559-28-0 C33H43F2N5O6S
N1-((1S,2S)-3-(3,5-difluorophenyl)-1-((R)-4-(3,5-dimethylisoxazol-4-ylsulfonyl)piperazin-2-yl)-1-hydroxypropan-2-yl)-5-methyl-N3,N3-dipropylisophthalamide
—— N-(7-benzyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c][2,7]naphthyridin-1-yl)pivalamide 1228692-61-2 C26H34N6O
N-(7-benzyl-5-(piperidin-1-yl)-6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c][2,7]naphthyridin-1-yl)pivalamide
—— N-(1,3-Benzothiazol-2-ylmethyl)-N-(5,6,7,8-tetrahydroquinolin-8-yl)butane-1,4-diamine 794499-02-8 C21H26N4S
N-(1,3-Benzothiazol-2-ylmethyl)-N-(5,6,7,8-tetrahydroquinolin-8-yl)butane-1,4-diamine
—— N-(3-(2-(4-(2-oxo-1,2,3,4-tetrahydroquinolin-7-yloxy)piperidin-1-yl)ethoxy)phenyl)methanesulfonamide 1227498-06-7 C23H29N3O5S
N-(3-(2-(4-(2-oxo-1,2,3,4-tetrahydroquinolin-7-yloxy)piperidin-1-yl)ethoxy)phenyl)methanesulfonamide
—— N-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)benzamide 1233719-56-6 C16H11ClN2O2
N-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)benzamide
—— N-(3-(2-(8-((2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)methyl)-3-azabicyclo[3.2.1]octan-3-yl)ethoxy)phenyl)methanesulfonamide 1227498-10-3 C26H33N3O4S
N-(3-(2-(8-((2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)methyl)-3-azabicyclo[3.2.1]octan-3-yl)ethoxy)phenyl)methanesulfonamide
—— N1-((1S,2S)-3-(3,5-difluorophenyl)-1-hydroxy-1-((R)-4-(pyridin-4-ylsulfonyl)piperazin-2-yl)propan-2-yl)-5-methyl-N3,N3-dipropylisophthalamide 1230559-20-2 C33H41F2N5O5S
N1-((1S,2S)-3-(3,5-difluorophenyl)-1-hydroxy-1-((R)-4-(pyridin-4-ylsulfonyl)piperazin-2-yl)propan-2-yl)-5-methyl-N3,N3-dipropylisophthalamide
—— N1-((1S,2S)-3-(3,5-difluorophenyl)-1-hydroxy-1-((R)-4-(1-methyl-1H-imidazol-4-ylsulfonyl)piperazin-2-yl)propan-2-yl)-5-methyl-N3,N3-dipropylisophthalamide 1230559-19-9 C32H42F2N6O5S
N1-((1S,2S)-3-(3,5-difluorophenyl)-1-hydroxy-1-((R)-4-(1-methyl-1H-imidazol-4-ylsulfonyl)piperazin-2-yl)propan-2-yl)-5-methyl-N3,N3-dipropylisophthalamide
—— N-(2-fluoro-5-(2-(4-(2-oxo-1,2,3,4-tetrahydroquinolin-7-yloxy)piperidin-1-yl)ethoxy)phenyl)methanesulfonamide 1227498-07-8 C23H28FN3O5S
N-(2-fluoro-5-(2-(4-(2-oxo-1,2,3,4-tetrahydroquinolin-7-yloxy)piperidin-1-yl)ethoxy)phenyl)methanesulfonamide
—— N-[[(6aR,7R,10aS)-1,4-difluoro-10a-[4-(trifluoromethyl)phenyl]sulfonyl-6,6a,7,8,9,10-hexahydrobenzo[c]chromen-7-yl]methyl]-N-ethylmethanesulfonamide 1237802-35-5 C24H26F5NO5S2
N-[[(6aR,7R,10aS)-1,4-difluoro-10a-[4-(trifluoromethyl)phenyl]sulfonyl-6,6a,7,8,9,10-hexahydrobenzo[c]chromen-7-yl]methyl]-N-ethylmethanesulfonamide
—— N-ethyl-5-(4-phenyl-2-pyridin-3-yl-1,3-thiazol-5-yl)-1H-pyrazole-3-carboxamide 1232031-33-2 C20H17N5OS
N-ethyl-5-(4-phenyl-2-pyridin-3-yl-1,3-thiazol-5-yl)-1H-pyrazole-3-carboxamide
—— N-(2-morpholinoethyl)-3-(3-phenylureido)benzamide 1229653-33-1 C20H24N4O3
N-(2-morpholinoethyl)-3-(3-phenylureido)benzamide
—— N1-((1S,2S)-3-(3,5-difluorophenyl)-1-((R)-4-(2,4-dimethylthiazol-5-ylsulfonyl)piperazin-2-yl)-1-hydroxypropan-2-yl)-5-methyl-N3,N3-dipropylisophthalamide 1230559-23-5 C33H43F2N5O5S2
N1-((1S,2S)-3-(3,5-difluorophenyl)-1-((R)-4-(2,4-dimethylthiazol-5-ylsulfonyl)piperazin-2-yl)-1-hydroxypropan-2-yl)-5-methyl-N3,N3-dipropylisophthalamide
—— N-(2-fluoro-5-(2-(8-((2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)methyl)-3-azabicyclo[3.2.1]octan-3-yl)ethoxy)phenyl)methanesulfonamide 1227498-11-4 C26H32FN3O4S
N-(2-fluoro-5-(2-(8-((2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)methyl)-3-azabicyclo[3.2.1]octan-3-yl)ethoxy)phenyl)methanesulfonamide
—— N-[3-(1,4-dihydroimidazo[4,5-c]pyrazol-5-yl)-4-methylphenyl]-3-morpholin-4-yl-5-(trifluoromethyl)benzamide 1236202-62-2 C23H21F3N6O2
N-[3-(1,4-dihydroimidazo[4,5-c]pyrazol-5-yl)-4-methylphenyl]-3-morpholin-4-yl-5-(trifluoromethyl)benzamide
—— N1-((1S,2S)-3-(3,5-difluorophenyl)-1-hydroxy-1-((R)-4-(1,3,5-trimethyl-1H-pyrazol-4-ylsulfonyl)piperazin-2-yl)propan-2-yl)-5-methyl-N3,N3-dipropylisophthalamide 1230559-27-9 C34H46F2N6O5S
N1-((1S,2S)-3-(3,5-difluorophenyl)-1-hydroxy-1-((R)-4-(1,3,5-trimethyl-1H-pyrazol-4-ylsulfonyl)piperazin-2-yl)propan-2-yl)-5-methyl-N3,N3-dipropylisophthalamide
—— N-(1-oxo-1,2-dihydroisoquinolin-6-yl)-1-phenylmethanesulfonamide 1233719-55-5 C16H14N2O3S
N-(1-oxo-1,2-dihydroisoquinolin-6-yl)-1-phenylmethanesulfonamide
—— N1-((1S,2S)-3-(3,5-difluorophenyl)-1-hydroxy-1-((R)-4-(3-methoxyphenylsulfonyl)piperazin-2-yl)propan-2-yl)-5-methyl-N3,N3-dipropylisophthalamide 1230559-12-2 C35H44F2N4O6S
N1-((1S,2S)-3-(3,5-difluorophenyl)-1-hydroxy-1-((R)-4-(3-methoxyphenylsulfonyl)piperazin-2-yl)propan-2-yl)-5-methyl-N3,N3-dipropylisophthalamide
—— N-[[(6aR,7R,10aS)-1,4-difluoro-10a-[4-(trifluoromethyl)phenyl]sulfonyl-6,6a,7,8,9,10-hexahydrobenzo[c]chromen-7-yl]methyl]-N-ethyl-1,1,1-trifluoromethanesulfonamide 1237802-37-7 C24H23F8NO5S2
N-[[(6aR,7R,10aS)-1,4-difluoro-10a-[4-(trifluoromethyl)phenyl]sulfonyl-6,6a,7,8,9,10-hexahydrobenzo[c]chromen-7-yl]methyl]-N-ethyl-1,1,1-trifluoromethanesulfonamide
—— N-(3-(2-(4-((2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)methyl)piperidin-1-yl)ethoxy)phenyl)methanesulfonamide 1227498-03-4 C24H31N3O4S
N-(3-(2-(4-((2-oxo-1,2,3,4-tetrahydroquinolin-7-yl)methyl)piperidin-1-yl)ethoxy)phenyl)methanesulfonamide
—— N-(3-imidazol-1-ylpropyl)-1-(4-methoxynaphthalen-1-yl)sulfonyl-2,3-dihydroindole-3-carboxamide 583813-42-7 C26H26N4O4S
N-(3-imidazol-1-ylpropyl)-1-(4-methoxynaphthalen-1-yl)sulfonyl-2,3-dihydroindole-3-carboxamide
—— N-Ethyl-5-[4-methyl-2-(3-pyridinyl)-5-thiazolyl]-1H-pyrazole-3-carboxamide 1232031-31-0 C15H15N5OS
N-Ethyl-5-[4-methyl-2-(3-pyridinyl)-5-thiazolyl]-1H-pyrazole-3-carboxamide
—— N-[2-(diethylamino)ethyl]-1-(4-methoxynaphthalen-1-yl)sulfonyl-2,3-dihydroindole-3-carboxamide 583813-40-5 C26H31N3O4S
N-[2-(diethylamino)ethyl]-1-(4-methoxynaphthalen-1-yl)sulfonyl-2,3-dihydroindole-3-carboxamide
—— N-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-3-phenylpropanamide 1233719-57-7 C18H15ClN2O2
N-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-3-phenylpropanamide
—— N-(cyclopropylmethyl)-4-((4-methoxy-N-(pyridin-3-ylmethyl)phenylsulfonamido)methyl)benzamide 1234457-66-9 C25H27N3O4S
N-(cyclopropylmethyl)-4-((4-methoxy-N-(pyridin-3-ylmethyl)phenylsulfonamido)methyl)benzamide
—— N-methyl-N-(1-methylpiperidin-4-yl)-1-[4-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydroindole-3-carboxamide 583813-78-9 C23H26F3N3O3S
N-methyl-N-(1-methylpiperidin-4-yl)-1-[4-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydroindole-3-carboxamide
—— N-(4-oxo-3,4-dihydroquinazolin-8-yl)-2-phenylacetamide 1233719-48-6 C16H13N3O2
N-(4-oxo-3,4-dihydroquinazolin-8-yl)-2-phenylacetamide
—— N-[[(6aR,7R,10aS)-1,4-difluoro-10a-[4-(trifluoromethyl)phenyl]sulfonyl-6,6a,7,8,9,10-hexahydrobenzo[c]chromen-7-yl]methyl]-N-cyclopropyl-1,1,1-trifluoromethanesulfonamide 1237802-43-5 C25H23F8NO5S2
N-[[(6aR,7R,10aS)-1,4-difluoro-10a-[4-(trifluoromethyl)phenyl]sulfonyl-6,6a,7,8,9,10-hexahydrobenzo[c]chromen-7-yl]methyl]-N-cyclopropyl-1,1,1-trifluoromethanesulfonamide
—— N-(1-oxo-1,2-dihydroisoquinolin-6-yl)-2-phenylacetamide 1233719-45-3 C17H14N2O2
N-(1-oxo-1,2-dihydroisoquinolin-6-yl)-2-phenylacetamide
—— N-(4-oxo-3,4-dihydroquinazolin-7-yl)-2-phenylacetamide 1233719-44-2 C16H13N3O2
N-(4-oxo-3,4-dihydroquinazolin-7-yl)-2-phenylacetamide
—— N-[[(6aR,7R,10aS)-1,4-difluoro-10a-[4-(trifluoromethyl)phenyl]sulfonyl-6,6a,7,8,9,10-hexahydrobenzo[c]chromen-7-yl]methyl]-N-cyclopropylethanesulfonamide 1237802-42-4 C26H28F5NO5S2
N-[[(6aR,7R,10aS)-1,4-difluoro-10a-[4-(trifluoromethyl)phenyl]sulfonyl-6,6a,7,8,9,10-hexahydrobenzo[c]chromen-7-yl]methyl]-N-cyclopropylethanesulfonamide
—— N-methyl-N-(1-methylpiperidin-4-yl)-1-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydroindole-3-carboxamide 583813-56-3 C23H26F3N3O3S
N-methyl-N-(1-methylpiperidin-4-yl)-1-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydroindole-3-carboxamide
—— N-(2-(4-sulfamoylphenylamino)-5,6-dihydrobenzo[h]quinazolin-8-yl)furan-2-carboxamide 1239413-42-3 C23H19N5O4S
N-(2-(4-sulfamoylphenylamino)-5,6-dihydrobenzo[h]quinazolin-8-yl)furan-2-carboxamide
—— N-(2-(4-sulfamoylphenylamino)-5,6-dihydrobenzo[h]quinazolin-8-yl)isobutyramide 1239413-40-1 C22H23N5O3S
N-(2-(4-sulfamoylphenylamino)-5,6-dihydrobenzo[h]quinazolin-8-yl)isobutyramide