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—— methyl (2Z,5S)-2-[[4-(dimethylamino)phenyl]methylidene]-5-(1,3-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H25N5O3S
methyl (2Z,5S)-2-[[4-(dimethylamino)phenyl]methylidene]-5-(1,3-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2Z,5S)-2-[[4-(difluoromethoxy)-3-methoxyphenyl]methylidene]-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H22F2N4O5S
methyl (2Z,5S)-2-[[4-(difluoromethoxy)-3-methoxyphenyl]methylidene]-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2Z,5S)-2-[(2,4-dimethoxyphenyl)methylidene]-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H24N4O5S
methyl (2Z,5S)-2-[(2,4-dimethoxyphenyl)methylidene]-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2Z,5S)-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-2-[[4-(trifluoromethyl)phenyl]methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C22H19F3N4O3S
methyl (2Z,5S)-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-2-[[4-(trifluoromethyl)phenyl]methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2Z,5R)-5-[4-(diethylamino)phenyl]-7-methyl-2-[(1-methylpyrazol-4-yl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H27N5O3S
methyl (2Z,5R)-5-[4-(diethylamino)phenyl]-7-methyl-2-[(1-methylpyrazol-4-yl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl N-[[5-chloro-2-(2-phenoxyethoxy)phenyl]methylideneamino]carbamate —— C17H17ClN2O4
methyl N-[[5-chloro-2-(2-phenoxyethoxy)phenyl]methylideneamino]carbamate
—— methyl (2Z,5S)-2-[(2,3-dimethoxyphenyl)methylidene]-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H24N4O5S
methyl (2Z,5S)-2-[(2,3-dimethoxyphenyl)methylidene]-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2Z,5S)-2-[(4-bromophenyl)methylidene]-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C21H19BrN4O3S
methyl (2Z,5S)-2-[(4-bromophenyl)methylidene]-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2Z,5R)-2-[(3-bromophenyl)methylidene]-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C21H19BrN4O3S
methyl (2Z,5R)-2-[(3-bromophenyl)methylidene]-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2Z,5R)-2-[(4-bromophenyl)methylidene]-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C21H19BrN4O3S
methyl (2Z,5R)-2-[(4-bromophenyl)methylidene]-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (1R,9R,13Z,16R)-13-[[3-[(2,3-dimethylphenoxy)methyl]-4-methoxyphenyl]methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C32H30N2O6S
methyl (1R,9R,13Z,16R)-13-[[3-[(2,3-dimethylphenoxy)methyl]-4-methoxyphenyl]methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— methyl (2Z,5R)-2-[(2-chloro-6-fluorophenyl)methylidene]-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C21H18ClFN4O3S
methyl (2Z,5R)-2-[(2-chloro-6-fluorophenyl)methylidene]-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Methyl 5-[[4-[1-(4-methoxyphenyl)cyclopropanecarbonyl]morpholin-2-yl]methoxy]pyridine-3-carboxylate —— C23H26N2O6
Methyl 5-[[4-[1-(4-methoxyphenyl)cyclopropanecarbonyl]morpholin-2-yl]methoxy]pyridine-3-carboxylate
—— methyl (2Z,5S)-2-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H26N4O4S
methyl (2Z,5S)-2-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2Z,5S)-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-2-[(4-methylphenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C22H22N4O3S
methyl (2Z,5S)-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-2-[(4-methylphenyl)methylidene]-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2Z,5R)-2-[(2,3-dimethoxyphenyl)methylidene]-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H24N4O5S
methyl (2Z,5R)-2-[(2,3-dimethoxyphenyl)methylidene]-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2Z,5S)-5-(1,3-dimethylpyrazol-4-yl)-7-methyl-3-oxo-2-[(3-phenoxyphenyl)methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H24N4O4S
methyl (2Z,5S)-5-(1,3-dimethylpyrazol-4-yl)-7-methyl-3-oxo-2-[(3-phenoxyphenyl)methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (6S)-2-[[6-bromo-2-(4-butylphenyl)quinoline-4-carbonyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C31H31BrN2O3S
methyl (6S)-2-[[6-bromo-2-(4-butylphenyl)quinoline-4-carbonyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— methyl (1R,9R,13Z,16R)-13-[[5-[(3-chloro-4-fluorophenoxy)methyl]furan-2-yl]methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate —— C27H20ClFN2O6S
methyl (1R,9R,13Z,16R)-13-[[5-[(3-chloro-4-fluorophenoxy)methyl]furan-2-yl]methylidene]-9-methyl-14-oxo-8-oxa-12-thia-10,15-diazatetracyclo[7.6.1.02,7.011,15]hexadeca-2,4,6,10-tetraene-16-carboxylate
—— methyl 2-[[2-[(4Z)-4-[(1-methylpyrazol-4-yl)methylidene]-5-oxo-1-phenylimidazol-2-yl]sulfanylacetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C26H25N5O4S2
methyl 2-[[2-[(4Z)-4-[(1-methylpyrazol-4-yl)methylidene]-5-oxo-1-phenylimidazol-2-yl]sulfanylacetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— methyl (2Z,5R)-2-[(3,4-dimethoxyphenyl)methylidene]-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H24N4O5S
methyl (2Z,5R)-2-[(3,4-dimethoxyphenyl)methylidene]-5-(1,5-dimethylpyrazol-4-yl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (6R)-6-(2-methylbutan-2-yl)-2-[[6-methyl-2-(4-propan-2-ylphenyl)quinoline-4-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C35H40N2O3S
methyl (6R)-6-(2-methylbutan-2-yl)-2-[[6-methyl-2-(4-propan-2-ylphenyl)quinoline-4-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— Methyl 2-(4-ethoxyanilino)-3-[hydroxy-(4-methylphenyl)methylidene]-4,5-dioxo-1-phenylpyrrolidine-2-carboxylate —— C28H26N2O6
Methyl 2-(4-ethoxyanilino)-3-[hydroxy-(4-methylphenyl)methylidene]-4,5-dioxo-1-phenylpyrrolidine-2-carboxylate
—— Methyl 4-[[4-(4-methoxyphenyl)-3-methylpiperazine-1-carbothioyl]amino]benzoate —— C21H25N3O3S
Methyl 4-[[4-(4-methoxyphenyl)-3-methylpiperazine-1-carbothioyl]amino]benzoate
—— Methyl 2-[4-(hexanoylamino)phenoxy]benzenecarboxylate —— C20H23NO4
Methyl 2-[4-(hexanoylamino)phenoxy]benzenecarboxylate
—— methyl (2Z,5R)-2-[[4-methoxy-3-[(2-methylphenoxy)methyl]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H30N2O6S
methyl (2Z,5R)-2-[[4-methoxy-3-[(2-methylphenoxy)methyl]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2Z,5R)-2-(furan-3-ylmethylidene)-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C21H18N2O5S
methyl (2Z,5R)-2-(furan-3-ylmethylidene)-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Methyl 4-(4-carbamoyl-5-methyl-1-propan-2-yl-2-propylpyrrol-3-yl)benzoate —— C20H26N2O3
Methyl 4-(4-carbamoyl-5-methyl-1-propan-2-yl-2-propylpyrrol-3-yl)benzoate
—— Methyl 3-methyl-2-[[4-(2-phenylethenyl)piperazine-1-carbonyl]amino]pentanoate —— C20H29N3O3
Methyl 3-methyl-2-[[4-(2-phenylethenyl)piperazine-1-carbonyl]amino]pentanoate
—— methyl 4-[hydroxy-[1-(3-morpholin-4-ylpropyl)-4,5-dioxo-2-phenylpyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate —— C26H31N3O6
methyl 4-[hydroxy-[1-(3-morpholin-4-ylpropyl)-4,5-dioxo-2-phenylpyrrolidin-3-ylidene]methyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
—— Methyl 3-[4-carbamoyl-1-[2-(3,4-dimethoxyphenyl)ethyl]-5-methyl-3-(4-pyrrolidin-1-ylphenyl)pyrrol-2-yl]propanoate —— C30H37N3O5
Methyl 3-[4-carbamoyl-1-[2-(3,4-dimethoxyphenyl)ethyl]-5-methyl-3-(4-pyrrolidin-1-ylphenyl)pyrrol-2-yl]propanoate
—— Methyl 4-(1-benzyl-4-carbamoyl-5-methyl-2-propylpyrrol-3-yl)benzoate —— C24H26N2O3
Methyl 4-(1-benzyl-4-carbamoyl-5-methyl-2-propylpyrrol-3-yl)benzoate
—— Methyl 6-[[4-(dimethylamino)phenyl]carbamoyl]pyridine-3-carboxylate —— C16H17N3O3
Methyl 6-[[4-(dimethylamino)phenyl]carbamoyl]pyridine-3-carboxylate
—— Methyl 3-[1-[2-(diethylcarbamoyl)-3,6-difluorobenzoyl]piperidin-4-yl]-2-oxo-1,3-oxazolidine-4-carboxylate —— C22H27F2N3O6
Methyl 3-[1-[2-(diethylcarbamoyl)-3,6-difluorobenzoyl]piperidin-4-yl]-2-oxo-1,3-oxazolidine-4-carboxylate
—— methyl (2Z,5S)-2-[[4-methoxy-3-[(2-methylphenoxy)methyl]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H30N2O6S
methyl (2Z,5S)-2-[[4-methoxy-3-[(2-methylphenoxy)methyl]phenyl]methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Methyl 2-cyano-3-[(2,4-dichlorophenyl)amino]prop-2-enoate —— C11H8Cl2N2O2
Methyl 2-cyano-3-[(2,4-dichlorophenyl)amino]prop-2-enoate
—— methyl (2Z,5S)-5-(1,5-dimethylpyrazol-4-yl)-2-(furan-3-ylmethylidene)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C19H18N4O4S
methyl (2Z,5S)-5-(1,5-dimethylpyrazol-4-yl)-2-(furan-3-ylmethylidene)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Methyl 2-acetamido-4-[8-(2,6-difluoro-3-methylbenzoyl)-2,8-diazaspiro[4.5]decan-2-yl]-4-oxobutanoate —— C23H29F2N3O5
Methyl 2-acetamido-4-[8-(2,6-difluoro-3-methylbenzoyl)-2,8-diazaspiro[4.5]decan-2-yl]-4-oxobutanoate
—— methyl 2-(3-amino-3-oxopropyl)-4,6-dioxo-3-[4-(trifluoromethoxy)phenyl]-3a,6a-dihydro-3H-pyrrolo[3,4-d][1,2]oxazole-5-carboxylate —— C17H16F3N3O7
methyl 2-(3-amino-3-oxopropyl)-4,6-dioxo-3-[4-(trifluoromethoxy)phenyl]-3a,6a-dihydro-3H-pyrrolo[3,4-d][1,2]oxazole-5-carboxylate
—— methyl (2Z,5R)-2-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H26N4O4S
methyl (2Z,5R)-2-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2Z,5R)-2-[(1,5-dimethylpyrazol-4-yl)methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C22H22N4O4S
methyl (2Z,5R)-2-[(1,5-dimethylpyrazol-4-yl)methylidene]-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl (2Z,5S)-2-(furan-3-ylmethylidene)-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C21H18N2O5S
methyl (2Z,5S)-2-(furan-3-ylmethylidene)-5-(4-methoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Methyl 3,6-dioxospiro[11,13,15-trioxatetracyclo[8.6.0.02,7.012,16]hexadec-9-ene-14,1'-cyclohexane]-7-carboxylate —— C20H24O7
Methyl 3,6-dioxospiro[11,13,15-trioxatetracyclo[8.6.0.02,7.012,16]hexadec-9-ene-14,1'-cyclohexane]-7-carboxylate
—— Methyl 2-[(2-fluorophenyl)carbamoylamino]-3-methylbutanoate —— C13H17FN2O3
Methyl 2-[(2-fluorophenyl)carbamoylamino]-3-methylbutanoate
—— Methyl 6,18-dimethoxy-17-(3-oxobutanoyloxy)-1,3,11,12,14,15,16,17,18,19,20,21-dodecahydroyohimban-19-carboxylate —— C27H34N2O7
Methyl 6,18-dimethoxy-17-(3-oxobutanoyloxy)-1,3,11,12,14,15,16,17,18,19,20,21-dodecahydroyohimban-19-carboxylate
—— methyl 2-[[5-[(Z)-2-cyano-3-methoxy-3-oxoprop-1-enyl]-2-methoxyphenyl]methoxy]benzoate —— C21H19NO6
methyl 2-[[5-[(Z)-2-cyano-3-methoxy-3-oxoprop-1-enyl]-2-methoxyphenyl]methoxy]benzoate
—— methyl (Z)-2-cyano-3-[4-methoxy-3-[(3-nitro-1,2,4-triazol-1-yl)methyl]phenyl]prop-2-enoate —— C15H13N5O5
methyl (Z)-2-cyano-3-[4-methoxy-3-[(3-nitro-1,2,4-triazol-1-yl)methyl]phenyl]prop-2-enoate
—— methyl (2Z,5R)-2-[(3,4-dimethoxyphenyl)methylidene]-7-methyl-5-(3-nitrophenyl)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H21N3O7S
methyl (2Z,5R)-2-[(3,4-dimethoxyphenyl)methylidene]-7-methyl-5-(3-nitrophenyl)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— methyl N-[3-(4-methoxyphenyl)-5-phenyl-3,4-dihydropyrazole-2-carbothioyl]carbamate —— C19H19N3O3S
methyl N-[3-(4-methoxyphenyl)-5-phenyl-3,4-dihydropyrazole-2-carbothioyl]carbamate
—— Methyl 2-[[2-(1-amino-3-methylbutyl)-1,3-thiazole-4-carbonyl]amino]-3-benzylsulfanylpropanoate —— C20H27N3O3S2
Methyl 2-[[2-(1-amino-3-methylbutyl)-1,3-thiazole-4-carbonyl]amino]-3-benzylsulfanylpropanoate