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—— 6-bromo-2-(4-fluorophenyl)-N-[[(2R)-oxolan-2-yl]methyl]imidazo[1,2-a]pyridin-3-amine —— C18H17BrFN3O
6-bromo-2-(4-fluorophenyl)-N-[[(2R)-oxolan-2-yl]methyl]imidazo[1,2-a]pyridin-3-amine
—— 6-Hydroxy-4-methyl-5-(morpholin-4-ylmethyl)-2-oxo-1-(2-phenylethyl)-1,2-dihydropyridine-3-carbonitrile —— C20H23N3O3
6-Hydroxy-4-methyl-5-(morpholin-4-ylmethyl)-2-oxo-1-(2-phenylethyl)-1,2-dihydropyridine-3-carbonitrile
—— 6-chloro-N-cyclohexyl-2-(4-methoxyphenyl)imidazo[1,2-a]pyridin-3-amine —— C20H22ClN3O
6-chloro-N-cyclohexyl-2-(4-methoxyphenyl)imidazo[1,2-a]pyridin-3-amine
—— 6-methyl-N-[[(2R)-oxolan-2-yl]methyl]-2-pyridin-4-ylimidazo[1,2-a]pyridin-3-amine —— C18H20N4O
6-methyl-N-[[(2R)-oxolan-2-yl]methyl]-2-pyridin-4-ylimidazo[1,2-a]pyridin-3-amine
—— 6-bromo-N-cyclopentyl-2-(4-methylphenyl)imidazo[1,2-a]pyridin-3-amine —— C19H20BrN3
6-bromo-N-cyclopentyl-2-(4-methylphenyl)imidazo[1,2-a]pyridin-3-amine
—— 6-bromo-N-cyclopentyl-2-(4-fluorophenyl)imidazo[1,2-a]pyridin-3-amine —— C18H17BrFN3
6-bromo-N-cyclopentyl-2-(4-fluorophenyl)imidazo[1,2-a]pyridin-3-amine
—— 6-bromo-2-(4-chlorophenyl)-N-cyclopentylimidazo[1,2-a]pyridin-3-amine —— C18H17BrClN3
6-bromo-2-(4-chlorophenyl)-N-cyclopentylimidazo[1,2-a]pyridin-3-amine
—— 6-[2-(4-Chloro-phenyl)-2-oxo-ethoxy]-8-ethyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile —— C21H21ClN2O3
6-[2-(4-Chloro-phenyl)-2-oxo-ethoxy]-8-ethyl-3,3-dimethyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— 6-[2-(4-Bromo-phenyl)-2-oxo-ethoxy]-3,3-dimethyl-8-phenyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile —— C25H21BrN2O3
6-[2-(4-Bromo-phenyl)-2-oxo-ethoxy]-3,3-dimethyl-8-phenyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— 6-[2-(4-Chloro-phenyl)-2-oxo-ethoxy]-3,3-dimethyl-8-propyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile —— C22H23ClN2O3
6-[2-(4-Chloro-phenyl)-2-oxo-ethoxy]-3,3-dimethyl-8-propyl-3,4-dihydro-1H-pyrano[3,4-c]pyridine-5-carbonitrile
—— 6,6-Dimethyl-2-[(2-oxo-2-phenylethyl)sulfanyl]-3,5,6,8-tetrahydro-4H-pyrano[4',3':4,5]thieno[2,3-D]pyrimidin-4-one —— C19H18N2O3S2
6,6-Dimethyl-2-[(2-oxo-2-phenylethyl)sulfanyl]-3,5,6,8-tetrahydro-4H-pyrano[4',3':4,5]thieno[2,3-D]pyrimidin-4-one
—— (6S)-N-(4-methylphenyl)-2-(4-methylphenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide —— C19H19N3O2S
(6S)-N-(4-methylphenyl)-2-(4-methylphenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide
—— (6R)-N-(4-fluorophenyl)-2-(4-methylphenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide —— C18H16FN3O2S
(6R)-N-(4-fluorophenyl)-2-(4-methylphenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide
—— (6S)-2-(2,5-dimethoxyphenyl)imino-N-(2-ethylphenyl)-4-oxo-1,3-thiazinane-6-carboxamide —— C21H23N3O4S
(6S)-2-(2,5-dimethoxyphenyl)imino-N-(2-ethylphenyl)-4-oxo-1,3-thiazinane-6-carboxamide
—— (6R)-2-(2,5-dimethoxyphenyl)imino-N-(4-fluorophenyl)-4-oxo-1,3-thiazinane-6-carboxamide —— C19H18FN3O4S
(6R)-2-(2,5-dimethoxyphenyl)imino-N-(4-fluorophenyl)-4-oxo-1,3-thiazinane-6-carboxamide
—— (6S)-2-(4-methylphenyl)imino-4-oxo-N-[3-(trifluoromethyl)phenyl]-1,3-thiazinane-6-carboxamide —— C19H16F3N3O2S
(6S)-2-(4-methylphenyl)imino-4-oxo-N-[3-(trifluoromethyl)phenyl]-1,3-thiazinane-6-carboxamide
—— (6R)-2-(4-methylphenyl)imino-N-naphthalen-1-yl-4-oxo-1,3-thiazinane-6-carboxamide —— C22H19N3O2S
(6R)-2-(4-methylphenyl)imino-N-naphthalen-1-yl-4-oxo-1,3-thiazinane-6-carboxamide
—— (6R)-2-(4-methylphenyl)imino-4-oxo-N-[3-(trifluoromethyl)phenyl]-1,3-thiazinane-6-carboxamide —— C19H16F3N3O2S
(6R)-2-(4-methylphenyl)imino-4-oxo-N-[3-(trifluoromethyl)phenyl]-1,3-thiazinane-6-carboxamide
—— (6S)-N-(4-fluorophenyl)-2-(4-methylphenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide —— C18H16FN3O2S
(6S)-N-(4-fluorophenyl)-2-(4-methylphenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide
—— (6R)-N-(4-methylphenyl)-2-(4-methylphenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide —— C19H19N3O2S
(6R)-N-(4-methylphenyl)-2-(4-methylphenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide
—— 6-(4-bromophenyl)-7-hydroxy-1,3-dimethyl-5H-pyrrolo[3,2-d]pyrimidine-2,4-dione —— C14H12BrN3O3
6-(4-bromophenyl)-7-hydroxy-1,3-dimethyl-5H-pyrrolo[3,2-d]pyrimidine-2,4-dione
—— (6R)-2-(4-methylphenyl)imino-4-oxo-N-[2-(trifluoromethyl)phenyl]-1,3-thiazinane-6-carboxamide —— C19H16F3N3O2S
(6R)-2-(4-methylphenyl)imino-4-oxo-N-[2-(trifluoromethyl)phenyl]-1,3-thiazinane-6-carboxamide
—— (6S)-2-(2,5-dimethoxyphenyl)imino-N-(4-fluorophenyl)-4-oxo-1,3-thiazinane-6-carboxamide —— C19H18FN3O4S
(6S)-2-(2,5-dimethoxyphenyl)imino-N-(4-fluorophenyl)-4-oxo-1,3-thiazinane-6-carboxamide
—— (6R)-N-(2,4-difluorophenyl)-2-(4-methylphenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide —— C18H15F2N3O2S
(6R)-N-(2,4-difluorophenyl)-2-(4-methylphenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide
—— (6S)-N-(2,4-difluorophenyl)-2-(4-methylphenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide —— C18H15F2N3O2S
(6S)-N-(2,4-difluorophenyl)-2-(4-methylphenyl)imino-4-oxo-1,3-thiazinane-6-carboxamide
—— 6-ethyl-2-(3-phenylprop-2-enoylcarbamothioylamino)-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxamide —— C20H22N4O2S2
6-ethyl-2-(3-phenylprop-2-enoylcarbamothioylamino)-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxamide
—— (6R)-6-(2-hydroxy-5-methoxyphenyl)-9,9-dimethyl-6,8,10,11-tetrahydro-5H-benzo[b][1,4]benzodiazepin-7-one —— C22H24N2O3
(6R)-6-(2-hydroxy-5-methoxyphenyl)-9,9-dimethyl-6,8,10,11-tetrahydro-5H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-6-(2-hydroxy-5-methoxyphenyl)-9,9-dimethyl-6,8,10,11-tetrahydro-5H-benzo[b][1,4]benzodiazepin-7-one —— C22H24N2O3
(6S)-6-(2-hydroxy-5-methoxyphenyl)-9,9-dimethyl-6,8,10,11-tetrahydro-5H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-6-(5-chloro-2-hydroxyphenyl)-9,9-dimethyl-6,8,10,11-tetrahydro-5H-benzo[b][1,4]benzodiazepin-7-one —— C21H21ClN2O2
(6S)-6-(5-chloro-2-hydroxyphenyl)-9,9-dimethyl-6,8,10,11-tetrahydro-5H-benzo[b][1,4]benzodiazepin-7-one
—— (6R)-6-(5-chloro-2-hydroxyphenyl)-9,9-dimethyl-6,8,10,11-tetrahydro-5H-benzo[b][1,4]benzodiazepin-7-one —— C21H21ClN2O2
(6R)-6-(5-chloro-2-hydroxyphenyl)-9,9-dimethyl-6,8,10,11-tetrahydro-5H-benzo[b][1,4]benzodiazepin-7-one
—— 6,7-dimethyl-3-[(R)-(4-methylpiperidin-1-yl)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C24H32N6O2
6,7-dimethyl-3-[(R)-(4-methylpiperidin-1-yl)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6,7-dimethyl-3-[(S)-morpholin-4-yl-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C22H28N6O3
6,7-dimethyl-3-[(S)-morpholin-4-yl-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6,7-dimethyl-3-[(R)-(4-methylpiperazin-1-yl)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C23H31N7O2
6,7-dimethyl-3-[(R)-(4-methylpiperazin-1-yl)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6,7-dimethyl-3-[(R)-morpholin-4-yl-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C22H28N6O3
6,7-dimethyl-3-[(R)-morpholin-4-yl-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— (6S,9S)-9-phenyl-6-thiophen-2-yl-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C25H19F3N2O2S
(6S,9S)-9-phenyl-6-thiophen-2-yl-5-(2,2,2-trifluoroacetyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6,7-dimethyl-3-[(S)-(4-methylpiperidin-1-yl)-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C24H32N6O2
6,7-dimethyl-3-[(S)-(4-methylpiperidin-1-yl)-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6,7-dimethyl-3-[(R)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]-(4-phenylpiperazin-1-yl)methyl]-1H-quinolin-2-one —— C28H33N7O2
6,7-dimethyl-3-[(R)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]-(4-phenylpiperazin-1-yl)methyl]-1H-quinolin-2-one
—— 6,7-dimethyl-3-[(R)-morpholin-4-yl-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C22H28N6O3
6,7-dimethyl-3-[(R)-morpholin-4-yl-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6,7-dimethyl-3-[(R)-(4-methylpiperidin-1-yl)-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C24H32N6O2
6,7-dimethyl-3-[(R)-(4-methylpiperidin-1-yl)-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— (6S,9R)-5-acetyl-9-(4-chlorophenyl)-6-(3-methoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C28H25ClN2O3
(6S,9R)-5-acetyl-9-(4-chlorophenyl)-6-(3-methoxyphenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6,7-dimethyl-3-[(R)-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]-piperidin-1-ylmethyl]-1H-quinolin-2-one —— C23H30N6O2
6,7-dimethyl-3-[(R)-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]-piperidin-1-ylmethyl]-1H-quinolin-2-one
—— 6,7-dimethyl-3-[(R)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]-piperidin-1-ylmethyl]-1H-quinolin-2-one —— C23H30N6O2
6,7-dimethyl-3-[(R)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]-piperidin-1-ylmethyl]-1H-quinolin-2-one
—— 6,7-dimethyl-3-[(S)-(4-methylpiperazin-1-yl)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C23H31N7O2
6,7-dimethyl-3-[(S)-(4-methylpiperazin-1-yl)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6,7-dimethyl-3-[(S)-(4-methylpiperidin-1-yl)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C24H32N6O2
6,7-dimethyl-3-[(S)-(4-methylpiperidin-1-yl)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— (6S,9S)-5-(cyclopropanecarbonyl)-6-(3-methoxyphenyl)-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C30H28N2O3
(6S,9S)-5-(cyclopropanecarbonyl)-6-(3-methoxyphenyl)-9-phenyl-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— 6,7-dimethyl-3-[(S)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]-(4-phenylpiperazin-1-yl)methyl]-1H-quinolin-2-one —— C28H33N7O2
6,7-dimethyl-3-[(S)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]-(4-phenylpiperazin-1-yl)methyl]-1H-quinolin-2-one
—— 6-ethyl-3-[(R)-(4-methylpiperidin-1-yl)-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C24H32N6O2
6-ethyl-3-[(R)-(4-methylpiperidin-1-yl)-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6-ethyl-3-[(S)-[4-(furan-2-carbonyl)piperazin-1-yl]-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C27H31N7O4
6-ethyl-3-[(S)-[4-(furan-2-carbonyl)piperazin-1-yl]-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6,7-dimethoxy-2-[(6-oxo-4-phenyl-1H-pyrimidin-2-yl)sulfanylmethyl]-3H-quinazolin-4-one —— C21H18N4O4S
6,7-dimethoxy-2-[(6-oxo-4-phenyl-1H-pyrimidin-2-yl)sulfanylmethyl]-3H-quinazolin-4-one
—— 6,7-dimethyl-3-[(S)-[(3R)-3-methylpiperidin-1-yl]-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C24H32N6O2
6,7-dimethyl-3-[(S)-[(3R)-3-methylpiperidin-1-yl]-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one