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苯并异恶唑

中文名称 英文名称 CAS号 化学式 结构式图片
—— (2R)-N-(3-amino-1,2-benzoxazol-6-yl)-2-[(2R)-4-[1-(3-fluoropyridin-4-yl)pyrazol-3-yl]-2-methyl-3-oxomorpholin-2-yl]-2-hydroxyacetamide —— C22H20FN7O5
(2R)-N-(3-amino-1,2-benzoxazol-6-yl)-2-[(2R)-4-[1-(3-fluoropyridin-4-yl)pyrazol-3-yl]-2-methyl-3-oxomorpholin-2-yl]-2-hydroxyacetamide
—— N-(3-amino-1,2-benzoxazol-6-yl)-2-[4-[4-chloro-1-(2-methoxypyridin-4-yl)pyrazol-3-yl]-3-oxomorpholin-2-yl]-2-hydroxypropanamide —— C23H22ClN7O6
N-(3-amino-1,2-benzoxazol-6-yl)-2-[4-[4-chloro-1-(2-methoxypyridin-4-yl)pyrazol-3-yl]-3-oxomorpholin-2-yl]-2-hydroxypropanamide
—— N-(3-amino-1,2-benzoxazol-6-yl)-2-hydroxy-2-[(2R,6S)-6-methyl-3-oxo-4-(1-pyridin-4-ylpyrazol-3-yl)morpholin-2-yl]acetamide —— C22H21N7O5
N-(3-amino-1,2-benzoxazol-6-yl)-2-hydroxy-2-[(2R,6S)-6-methyl-3-oxo-4-(1-pyridin-4-ylpyrazol-3-yl)morpholin-2-yl]acetamide
—— (2R)-N-(3-amino-1,2-benzoxazol-6-yl)-2-hydroxy-2-[(2R)-2-methyl-3-oxo-4-(4-pyridin-4-yl-1,3-thiazol-2-yl)morpholin-2-yl]acetamide —— C22H20N6O5S
(2R)-N-(3-amino-1,2-benzoxazol-6-yl)-2-hydroxy-2-[(2R)-2-methyl-3-oxo-4-(4-pyridin-4-yl-1,3-thiazol-2-yl)morpholin-2-yl]acetamide
—— (2R)-N-(3-amino-1,2-benzoxazol-6-yl)-2-hydroxy-2-[(2R)-2-methyl-4-[6-(oxan-4-yloxy)pyridin-2-yl]-3-oxomorpholin-2-yl]acetamide —— C24H27N5O7
(2R)-N-(3-amino-1,2-benzoxazol-6-yl)-2-hydroxy-2-[(2R)-2-methyl-4-[6-(oxan-4-yloxy)pyridin-2-yl]-3-oxomorpholin-2-yl]acetamide
—— N-(3-amino-1,2-benzoxazol-6-yl)-2-hydroxy-2-[4-[5-(2-methoxypyrimidin-4-yl)furan-2-yl]-3-oxomorpholin-2-yl]propanamide —— C23H22N6O7
N-(3-amino-1,2-benzoxazol-6-yl)-2-hydroxy-2-[4-[5-(2-methoxypyrimidin-4-yl)furan-2-yl]-3-oxomorpholin-2-yl]propanamide
—— N-(3-amino-1,2-benzoxazol-6-yl)-2-hydroxy-2-[2-methyl-4-[6-(1,2-oxazol-4-yl)pyridin-2-yl]-3-oxomorpholin-2-yl]acetamide —— C22H20N6O6
N-(3-amino-1,2-benzoxazol-6-yl)-2-hydroxy-2-[2-methyl-4-[6-(1,2-oxazol-4-yl)pyridin-2-yl]-3-oxomorpholin-2-yl]acetamide
—— N-(3-amino-1,2-benzoxazol-6-yl)-2-hydroxy-2-[2-methyl-4-[6-(3-methyl-1,2-oxazol-4-yl)pyridin-2-yl]-3-oxomorpholin-2-yl]acetamide —— C23H22N6O6
N-(3-amino-1,2-benzoxazol-6-yl)-2-hydroxy-2-[2-methyl-4-[6-(3-methyl-1,2-oxazol-4-yl)pyridin-2-yl]-3-oxomorpholin-2-yl]acetamide
—— N-(3-amino-1,2-benzoxazol-6-yl)-2-hydroxy-2-[2-methyl-3-oxo-4-(4-pyridin-4-yl-1,3-oxazol-2-yl)morpholin-2-yl]acetamide —— C22H20N6O6
N-(3-amino-1,2-benzoxazol-6-yl)-2-hydroxy-2-[2-methyl-3-oxo-4-(4-pyridin-4-yl-1,3-oxazol-2-yl)morpholin-2-yl]acetamide
—— (5R)-3-[5-(1,3-dioxolan-2-yl)-6-[ethyl-[(2S)-2-hydroxypropyl]amino]-7-fluoro-1,2-benzoxazol-3-yl]-5-methyl-1,3-oxazolidin-2-one —— C19H24FN3O6
(5R)-3-[5-(1,3-dioxolan-2-yl)-6-[ethyl-[(2S)-2-hydroxypropyl]amino]-7-fluoro-1,2-benzoxazol-3-yl]-5-methyl-1,3-oxazolidin-2-one
—— 6,7-Difluoro-3-(2-oxo-1,3-oxazolidin-3-yl)-1,2-benzoxazole-5-carbaldehyde —— C11H6F2N2O4
6,7-Difluoro-3-(2-oxo-1,3-oxazolidin-3-yl)-1,2-benzoxazole-5-carbaldehyde
—— 7-fluoro-3-[(4R,5R)-4-(fluoromethyl)-5-methyl-2-oxo-1,3-oxazolidin-3-yl]-6-[(2R)-2-methylmorpholin-4-yl]-1,2-benzoxazole-5-carbaldehyde —— C18H19F2N3O5
7-fluoro-3-[(4R,5R)-4-(fluoromethyl)-5-methyl-2-oxo-1,3-oxazolidin-3-yl]-6-[(2R)-2-methylmorpholin-4-yl]-1,2-benzoxazole-5-carbaldehyde
—— 2-(4-Aminobenzo[d]isoxazol-3-yl)propan-2-ol —— C10H12N2O2
2-(4-Aminobenzo[d]isoxazol-3-yl)propan-2-ol
—— 3-Chloro-6-(2,6-dimethylmorpholin-4-yl)-7-fluoro-1,2-benzoxazole-5-carbaldehyde —— C14H14ClFN2O3
3-Chloro-6-(2,6-dimethylmorpholin-4-yl)-7-fluoro-1,2-benzoxazole-5-carbaldehyde
—— 1-(1,2-Benzoxazol-3-yl)-2-(3-methoxyanilino)-2-phenylethanone —— C22H18N2O3
1-(1,2-Benzoxazol-3-yl)-2-(3-methoxyanilino)-2-phenylethanone
—— (5R)-3-[6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-5-(1,3-dioxolan-2-yl)-7-fluoro-1,2-benzoxazol-3-yl]-5-methanimidoyl-1,3-oxazolidin-2-one —— C20H23FN4O6
(5R)-3-[6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-5-(1,3-dioxolan-2-yl)-7-fluoro-1,2-benzoxazol-3-yl]-5-methanimidoyl-1,3-oxazolidin-2-one
—— 6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-7-fluoro-3-[4-(oxan-4-yl)-2-oxo-1,3-oxazolidin-3-yl]-1,2-benzoxazole-5-carbaldehyde —— C22H26FN3O6
6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-7-fluoro-3-[4-(oxan-4-yl)-2-oxo-1,3-oxazolidin-3-yl]-1,2-benzoxazole-5-carbaldehyde
—— (5S)-3-[6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-5-(1,3-dioxolan-2-yl)-7-fluoro-1,2-benzoxazol-3-yl]-5-ethyl-1,3-oxazolidin-2-one —— C21H26FN3O6
(5S)-3-[6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-5-(1,3-dioxolan-2-yl)-7-fluoro-1,2-benzoxazol-3-yl]-5-ethyl-1,3-oxazolidin-2-one
—— 3-[(4S)-4-[3-[tert-butyl(diphenyl)silyl]oxypropyl]-2-oxo-1,3-oxazolidin-3-yl]-6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-7-fluoro-1,2-benzoxazole-5-carbaldehyde —— C36H42FN3O6Si
3-[(4S)-4-[3-[tert-butyl(diphenyl)silyl]oxypropyl]-2-oxo-1,3-oxazolidin-3-yl]-6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-7-fluoro-1,2-benzoxazole-5-carbaldehyde
—— 3-[5-(1,3-Dioxolan-2-yl)-6,7-difluoro-1,2-benzoxazol-3-yl]-4-ethynyl-1,3-oxazolidin-2-one —— C15H10F2N2O5
3-[5-(1,3-Dioxolan-2-yl)-6,7-difluoro-1,2-benzoxazol-3-yl]-4-ethynyl-1,3-oxazolidin-2-one
—— (4S)-((S)-4-allyl-2-oxooxazolidin-3-yl)-6-((2R,6R)-2,6-dimethylmorpholino)-7-fluorobenzo[d]isoxazole-5-carbaldehyde —— C20H22FN3O5
(4S)-((S)-4-allyl-2-oxooxazolidin-3-yl)-6-((2R,6R)-2,6-dimethylmorpholino)-7-fluorobenzo[d]isoxazole-5-carbaldehyde
—— 6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-7-fluoro-3-(5-methyl-2-oxo-1,3-oxazolidin-3-yl)-1,2-benzoxazole-5-carbaldehyde —— C18H20FN3O5
6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-7-fluoro-3-(5-methyl-2-oxo-1,3-oxazolidin-3-yl)-1,2-benzoxazole-5-carbaldehyde
—— 3-[6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-5-(1,3-dioxolan-2-yl)-7-fluoro-1,2-benzoxazol-3-yl]-5-(hydroxymethyl)-1,3-oxazolidin-2-one —— C20H24FN3O7
3-[6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-5-(1,3-dioxolan-2-yl)-7-fluoro-1,2-benzoxazol-3-yl]-5-(hydroxymethyl)-1,3-oxazolidin-2-one
—— 2-[[5-(1,3-Dioxolan-2-yl)-6,7-difluoro-1,2-benzoxazol-3-yl]amino]but-3-yn-1-ol —— C14H12F2N2O4
2-[[5-(1,3-Dioxolan-2-yl)-6,7-difluoro-1,2-benzoxazol-3-yl]amino]but-3-yn-1-ol
—— 6-((2R,6R)-2,6-dimethylmorpholino)-3-((4S)-4-ethynyl-2-oxooxazolidin-3-yl)-7-fluorobenzo[d]isoxazole-5-carbaldehyde —— C19H18FN3O5
6-((2R,6R)-2,6-dimethylmorpholino)-3-((4S)-4-ethynyl-2-oxooxazolidin-3-yl)-7-fluorobenzo[d]isoxazole-5-carbaldehyde
—— 6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-7-fluoro-3-[4-[(1S)-1-methoxyethyl]-2-oxo-1,3-oxazolidin-3-yl]-1,2-benzoxazole-5-carbaldehyde —— C20H24FN3O6
6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-7-fluoro-3-[4-[(1S)-1-methoxyethyl]-2-oxo-1,3-oxazolidin-3-yl]-1,2-benzoxazole-5-carbaldehyde
—— 6,7-difluoro-3-((4S,5R)-4-(methoxymethyl)-5-methyl-2-oxooxazolidin-3-yl)benzo[d]isoxazole-5-carbaldehyde —— C14H12F2N2O5
6,7-difluoro-3-((4S,5R)-4-(methoxymethyl)-5-methyl-2-oxooxazolidin-3-yl)benzo[d]isoxazole-5-carbaldehyde
—— (4S)-3-(7-chloro-6-((2R,6R)-2,6-dimethylmorpholino)-5-(1,3-dioxolan-2-yl)benzo[d]isoxazol-3-yl)-4-(3-fluoropropyl)oxazolidin-2-one —— C22H27ClFN3O6
(4S)-3-(7-chloro-6-((2R,6R)-2,6-dimethylmorpholino)-5-(1,3-dioxolan-2-yl)benzo[d]isoxazol-3-yl)-4-(3-fluoropropyl)oxazolidin-2-one
—— 6-((2R,6R)-2,6-dimethylmorpholino)-7-fluoro-3-(2-oxo-4-(pyridin-4-yl)oxazolidin-3-yl)benzo[d]isoxazole-5-carbaldehyde —— C22H21FN4O5
6-((2R,6R)-2,6-dimethylmorpholino)-7-fluoro-3-(2-oxo-4-(pyridin-4-yl)oxazolidin-3-yl)benzo[d]isoxazole-5-carbaldehyde
—— 3-[7-chloro-6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-5-(1,3-dioxolan-2-yl)-1,2-benzoxazol-3-yl]-5-(methoxymethyl)-1,3-oxazolidin-2-one —— C21H26ClN3O7
3-[7-chloro-6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-5-(1,3-dioxolan-2-yl)-1,2-benzoxazol-3-yl]-5-(methoxymethyl)-1,3-oxazolidin-2-one
—— 2-((5-(1,3-dioxolan-2-yl)-6,7-difluorobenzo[d]isoxazol-3-yl)amino)-2-(pyridin-2-yl)ethanol —— C17H15F2N3O4
2-((5-(1,3-dioxolan-2-yl)-6,7-difluorobenzo[d]isoxazol-3-yl)amino)-2-(pyridin-2-yl)ethanol
—— 6,7-difluoro-3-[4-[(1R)-1-hydroxyethyl]-2-oxo-1,3-oxazolidin-3-yl]-1,2-benzoxazole-5-carbaldehyde —— C13H10F2N2O5
6,7-difluoro-3-[4-[(1R)-1-hydroxyethyl]-2-oxo-1,3-oxazolidin-3-yl]-1,2-benzoxazole-5-carbaldehyde
—— (R)-2-(5-(1,3-dioxolan-2-yl)-6,7-difluorobenzo[d]isoxazol-3-ylamino)-2-(1-methyl-1H-1,2,4-triazol-5-yl)ethanol —— C15H15F2N5O4
(R)-2-(5-(1,3-dioxolan-2-yl)-6,7-difluorobenzo[d]isoxazol-3-ylamino)-2-(1-methyl-1H-1,2,4-triazol-5-yl)ethanol
—— (5S)-3-(6-((2R,6R)-2,6-Dimethylmorpholino)-5-(1,3-dioxolan-2-yl)-7-fluorobenzo[d]isoxazol-3-yl)-5-(hydroxymethyl)oxazolidin-2-one —— C20H24FN3O7
(5S)-3-(6-((2R,6R)-2,6-Dimethylmorpholino)-5-(1,3-dioxolan-2-yl)-7-fluorobenzo[d]isoxazol-3-yl)-5-(hydroxymethyl)oxazolidin-2-one
—— 6,7-Difluoro-3-[4-(2-hydroxyethyl)-2-oxo-1,3-oxazolidin-3-yl]-1,2-benzoxazole-5-carbaldehyde —— C13H10F2N2O5
6,7-Difluoro-3-[4-(2-hydroxyethyl)-2-oxo-1,3-oxazolidin-3-yl]-1,2-benzoxazole-5-carbaldehyde
—— 6,7-difluoro-3-[4-[(1R)-1-methoxyethyl]-2-oxo-1,3-oxazolidin-3-yl]-1,2-benzoxazole-5-carbaldehyde —— C14H12F2N2O5
6,7-difluoro-3-[4-[(1R)-1-methoxyethyl]-2-oxo-1,3-oxazolidin-3-yl]-1,2-benzoxazole-5-carbaldehyde
—— (5R)-3-[6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-5-(1,3-dioxolan-2-yl)-7-fluoro-1,2-benzoxazol-3-yl]-5-[(E)-methoxyiminomethyl]-1,3-oxazolidin-2-one —— C21H25FN4O7
(5R)-3-[6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-5-(1,3-dioxolan-2-yl)-7-fluoro-1,2-benzoxazol-3-yl]-5-[(E)-methoxyiminomethyl]-1,3-oxazolidin-2-one
—— (4S)-4-(3-(tert-butyldiphenylsilyloxy)propyl)-3-(6-((2R,6R)-2,6-dimethylmorpholino)-5-(1,3-dioxolan-2-yl)-7-fluorobenzo[d]isoxazol-3-yl)oxazolidin-2-one —— C38H46FN3O7Si
(4S)-4-(3-(tert-butyldiphenylsilyloxy)propyl)-3-(6-((2R,6R)-2,6-dimethylmorpholino)-5-(1,3-dioxolan-2-yl)-7-fluorobenzo[d]isoxazol-3-yl)oxazolidin-2-one
—— 6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-7-fluoro-3-[4-[(1R)-1-hydroxyethyl]-2-oxo-1,3-oxazolidin-3-yl]-1,2-benzoxazole-5-carbaldehyde —— C19H22FN3O6
6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-7-fluoro-3-[4-[(1R)-1-hydroxyethyl]-2-oxo-1,3-oxazolidin-3-yl]-1,2-benzoxazole-5-carbaldehyde
—— 3-[5-(1,3-dioxolan-2-yl)-6,7-difluoro-1,2-benzoxazol-3-yl]-4-[(1S)-1-methoxyethyl]-1,3-oxazolidin-2-one —— C16H16F2N2O6
3-[5-(1,3-dioxolan-2-yl)-6,7-difluoro-1,2-benzoxazol-3-yl]-4-[(1S)-1-methoxyethyl]-1,3-oxazolidin-2-one
—— 2-[[5-(1,3-Dioxolan-2-yl)-6,7-difluoro-1,2-benzoxazol-3-yl]amino]-2-(2-methyl-1,2,4-triazol-3-yl)ethanol —— C15H15F2N5O4
2-[[5-(1,3-Dioxolan-2-yl)-6,7-difluoro-1,2-benzoxazol-3-yl]amino]-2-(2-methyl-1,2,4-triazol-3-yl)ethanol
—— 3-[6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-5-(1,3-dioxolan-2-yl)-7-fluoro-1,2-benzoxazol-3-yl]-5-(fluoromethyl)-1,3-oxazolidin-2-one —— C20H23F2N3O6
3-[6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-5-(1,3-dioxolan-2-yl)-7-fluoro-1,2-benzoxazol-3-yl]-5-(fluoromethyl)-1,3-oxazolidin-2-one
—— (5S)-5-((tert-butyldiphenylsilyloxy)methyl)-3-(7-chloro-6-((2R,6R)-2,6-dimethylmorpholino)-5-(1,3-dioxolan-2-yl)benzo[d]isoxazol-3-yl)oxazolidin-2-one —— C36H42ClN3O7Si
(5S)-5-((tert-butyldiphenylsilyloxy)methyl)-3-(7-chloro-6-((2R,6R)-2,6-dimethylmorpholino)-5-(1,3-dioxolan-2-yl)benzo[d]isoxazol-3-yl)oxazolidin-2-one
—— (4R)-3-(5-(1,3-dioxolan-2-yl)-6,7-difluorobenzo[d]isoxazol-3-yl)-4-((S)-1-methoxyethyl)oxazolidin-2-one —— C16H16F2N2O6
(4R)-3-(5-(1,3-dioxolan-2-yl)-6,7-difluorobenzo[d]isoxazol-3-yl)-4-((S)-1-methoxyethyl)oxazolidin-2-one
—— 4-[3-[tert-butyl(diphenyl)silyl]oxypropyl]-3-[6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-5-(1,3-dioxolan-2-yl)-7-fluoro-1,2-benzoxazol-3-yl]-1,3-oxazolidin-2-one —— C38H46FN3O7Si
4-[3-[tert-butyl(diphenyl)silyl]oxypropyl]-3-[6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-5-(1,3-dioxolan-2-yl)-7-fluoro-1,2-benzoxazol-3-yl]-1,3-oxazolidin-2-one
—— 6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-7-fluoro-3-[4-(2-hydroxyethyl)-2-oxo-1,3-oxazolidin-3-yl]-1,2-benzoxazole-5-carbaldehyde —— C19H22FN3O6
6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-7-fluoro-3-[4-(2-hydroxyethyl)-2-oxo-1,3-oxazolidin-3-yl]-1,2-benzoxazole-5-carbaldehyde
—— 6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-7-fluoro-3-[4-[(1S)-1-hydroxyethyl]-2-oxo-1,3-oxazolidin-3-yl]-1,2-benzoxazole-5-carbaldehyde —— C19H22FN3O6
6-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-7-fluoro-3-[4-[(1S)-1-hydroxyethyl]-2-oxo-1,3-oxazolidin-3-yl]-1,2-benzoxazole-5-carbaldehyde
—— 2-(5-(1,3-dioxolan-2-yl)-6,7-difluorobenzo[d]isoxazol-3-ylamino)-2-(tetrahydro-2H-pyran-4-yl)ethanol —— C17H20F2N2O5
2-(5-(1,3-dioxolan-2-yl)-6,7-difluorobenzo[d]isoxazol-3-ylamino)-2-(tetrahydro-2H-pyran-4-yl)ethanol
—— (S)-6,7-difluoro-3-(4-(1-methyl-1H-1,2,4-triazol-5-yl)-2-oxooxazolidin-3-yl)benzo[d]isoxazole-5-carbaldehyde —— C14H9F2N5O4
(S)-6,7-difluoro-3-(4-(1-methyl-1H-1,2,4-triazol-5-yl)-2-oxooxazolidin-3-yl)benzo[d]isoxazole-5-carbaldehyde
—— (S)-2-(5-(1,3-dioxolan-2-yl)-6,7-difluorobenzo[d]isoxazol-3-ylamino)-2-(1-methyl-1H-1,2,4-triazol-5-yl)ethanol —— C15H15F2N5O4
(S)-2-(5-(1,3-dioxolan-2-yl)-6,7-difluorobenzo[d]isoxazol-3-ylamino)-2-(1-methyl-1H-1,2,4-triazol-5-yl)ethanol