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苯并恶嗪类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[2-[[(1S)-cyclohex-3-en-1-yl]methyl]pyrazol-3-yl]-7-(hydroxymethyl)-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide —— C21H26N4O3
N-[2-[[(1S)-cyclohex-3-en-1-yl]methyl]pyrazol-3-yl]-7-(hydroxymethyl)-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
—— N-[2-[[(1R)-cyclohex-3-en-1-yl]methyl]pyrazol-3-yl]-7-(hydroxymethyl)-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide —— C21H26N4O3
N-[2-[[(1R)-cyclohex-3-en-1-yl]methyl]pyrazol-3-yl]-7-(hydroxymethyl)-3,5-dihydro-2H-1,4-benzoxazepine-4-carboxamide
—— (2R)-4-methyl-N-[2-(4-sulfamoylphenyl)ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C18H21N3O4S
(2R)-4-methyl-N-[2-(4-sulfamoylphenyl)ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2S)-4-methyl-N-[2-(4-sulfamoylphenyl)ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C18H21N3O4S
(2S)-4-methyl-N-[2-(4-sulfamoylphenyl)ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2S)-N-[2-(1H-benzimidazol-2-yl)ethyl]-4-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C19H20N4O2
(2S)-N-[2-(1H-benzimidazol-2-yl)ethyl]-4-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— N-[2-(6-methoxy-2-phenyl-2,3-dihydro-4H-1,4-benzoxazin-4-yl)ethyl]benzamide —— C24H24N2O3
N-[2-(6-methoxy-2-phenyl-2,3-dihydro-4H-1,4-benzoxazin-4-yl)ethyl]benzamide
—— 2-ethoxy-3-[4-[2-(4-oxo-2H-1,3-benzoxazin-3-yl)ethoxy]phenyl]propanamide —— C21H24N2O5
2-ethoxy-3-[4-[2-(4-oxo-2H-1,3-benzoxazin-3-yl)ethoxy]phenyl]propanamide
—— (2R)-4-methyl-N-[(5-methylpyrazin-2-yl)methyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C16H18N4O2
(2R)-4-methyl-N-[(5-methylpyrazin-2-yl)methyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2R)-N-[2-(1H-benzimidazol-2-yl)ethyl]-4-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C19H20N4O2
(2R)-N-[2-(1H-benzimidazol-2-yl)ethyl]-4-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (7-oxophenoxazin-3-yl) [(E)-3-phenylprop-2-enyl] carbonate —— C22H15NO5
(7-oxophenoxazin-3-yl) [(E)-3-phenylprop-2-enyl] carbonate
—— (2S)-4-methyl-N-[(5-methylpyrazin-2-yl)methyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C16H18N4O2
(2S)-4-methyl-N-[(5-methylpyrazin-2-yl)methyl]-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— N-[2-(6-methoxy-3-phenyl-2,3-dihydro-4H-1,4-benzoxazin-4-yl)ethyl]butanamide —— C21H26N2O3
N-[2-(6-methoxy-3-phenyl-2,3-dihydro-4H-1,4-benzoxazin-4-yl)ethyl]butanamide
—— 3-Piperidin-1-ylpropyl 9-oxa-1,2-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraene-3-carboxylate —— C18H23N3O3
3-Piperidin-1-ylpropyl 9-oxa-1,2-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraene-3-carboxylate
—— 8-Azabicyclo[3.2.1]octan-3-yl 9-oxa-1,2-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraene-3-carboxylate —— C17H19N3O3
8-Azabicyclo[3.2.1]octan-3-yl 9-oxa-1,2-diazatricyclo[6.3.1.04,12]dodeca-2,4(12),5,7-tetraene-3-carboxylate
—— (2S)-N-[[3-(methoxymethyl)-1H-pyrazol-5-yl]methyl]-N,4-dimethyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C17H22N4O3
(2S)-N-[[3-(methoxymethyl)-1H-pyrazol-5-yl]methyl]-N,4-dimethyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2R)-N-[[3-(methoxymethyl)-1H-pyrazol-5-yl]methyl]-N,4-dimethyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C17H22N4O3
(2R)-N-[[3-(methoxymethyl)-1H-pyrazol-5-yl]methyl]-N,4-dimethyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— 2-methyl-6,7,8,9,10,11-hexahydro-4H-cycloocta[g][1,4]benzoxazine-3-thione —— C15H19NOS
2-methyl-6,7,8,9,10,11-hexahydro-4H-cycloocta[g][1,4]benzoxazine-3-thione
—— (5R)-5-(azidomethyl)-3-(4-methyl-2,3-dihydro-1,4-benzoxazin-7-yl)-1,3-oxazolidin-2-one —— C13H15N5O3
(5R)-5-(azidomethyl)-3-(4-methyl-2,3-dihydro-1,4-benzoxazin-7-yl)-1,3-oxazolidin-2-one
—— [2-oxo-2-(3-oxo-4H-1,4-benzoxazin-6-yl)ethyl] (Z)-3-quinolin-2-ylprop-2-enoate —— C22H16N2O5
[2-oxo-2-(3-oxo-4H-1,4-benzoxazin-6-yl)ethyl] (Z)-3-quinolin-2-ylprop-2-enoate
—— [2-oxo-2-(3-oxo-4H-1,4-benzoxazin-6-yl)ethyl] (Z)-3-(1,3-benzothiazol-2-yl)prop-2-enoate —— C20H14N2O5S
[2-oxo-2-(3-oxo-4H-1,4-benzoxazin-6-yl)ethyl] (Z)-3-(1,3-benzothiazol-2-yl)prop-2-enoate
—— 2,12,14-Trioxa-7-azatetracyclo[7.7.0.03,7.011,15]hexadeca-1(16),9,11(15)-triene-6,8-dione —— C12H9NO5
2,12,14-Trioxa-7-azatetracyclo[7.7.0.03,7.011,15]hexadeca-1(16),9,11(15)-triene-6,8-dione
—— [4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methanone —— C21H25N3O3
[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-[(2S)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methanone
—— 3-hydroxy-6-methyl-6H-benzo[b][4,1]benzoxazepin-8-one —— C14H11NO3
3-hydroxy-6-methyl-6H-benzo[b][4,1]benzoxazepin-8-one
—— [4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-[(2R)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methanone —— C21H25N3O3
[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-[(2R)-4-methyl-2,3-dihydro-1,4-benzoxazin-2-yl]methanone
—— 1-Ethynyl-5,6-difluoro-4-propan-2-yl-4-(trifluoromethyl)-3,1-benzoxazin-2-one —— C14H10F5NO2
1-Ethynyl-5,6-difluoro-4-propan-2-yl-4-(trifluoromethyl)-3,1-benzoxazin-2-one
—— 4-(8-fluoro-4,4-dimethyl-2-oxo-1H-3,1-benzoxazin-6-yl)thiophene-2-carbonitrile —— C15H11FN2O2S
4-(8-fluoro-4,4-dimethyl-2-oxo-1H-3,1-benzoxazin-6-yl)thiophene-2-carbonitrile
—— 1-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-3-(8-fluoro-3-oxo-4H-1,4-benzoxazin-6-yl)urea —— C16H19FN4O3
1-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-3-(8-fluoro-3-oxo-4H-1,4-benzoxazin-6-yl)urea
—— 1-[(3S)-1-azabicyclo[2.2.2]octan-3-yl]-3-(8-fluoro-3-oxo-4H-1,4-benzoxazin-6-yl)urea —— C16H19FN4O3
1-[(3S)-1-azabicyclo[2.2.2]octan-3-yl]-3-(8-fluoro-3-oxo-4H-1,4-benzoxazin-6-yl)urea
—— 2-[4-[2-[(3-Amino-1,2-benzothiazol-5-yl)-benzylamino]-3-cyclohexylpropanoyl]-2,3-dihydro-1,4-benzoxazin-7-yl]benzenesulfonamide —— C37H39N5O4S2
2-[4-[2-[(3-Amino-1,2-benzothiazol-5-yl)-benzylamino]-3-cyclohexylpropanoyl]-2,3-dihydro-1,4-benzoxazin-7-yl]benzenesulfonamide
—— methyl 3-[3-(6-chloro-2-oxospiro[1H-3,1-benzoxazine-4,4'-piperidine]-1'-yl)propylcarbamoyl]-4-(3,4-difluorophenyl)-6-(methoxymethyl)-2-oxo-1,4-dihydropyrimidine-5-carboxylate —— C30H32ClF2N5O7
methyl 3-[3-(6-chloro-2-oxospiro[1H-3,1-benzoxazine-4,4'-piperidine]-1'-yl)propylcarbamoyl]-4-(3,4-difluorophenyl)-6-(methoxymethyl)-2-oxo-1,4-dihydropyrimidine-5-carboxylate
—— (2S)-2-amino-5-(diaminomethylideneamino)pentanoic acid;(2R)-2-ethoxy-3-[4-(2-phenoxazin-10-ylethoxy)phenyl]propanoic acid —— C31H39N5O7
(2S)-2-amino-5-(diaminomethylideneamino)pentanoic acid;(2R)-2-ethoxy-3-[4-(2-phenoxazin-10-ylethoxy)phenyl]propanoic acid
—— Tert-butyl 5-(aminomethyl)-11-fluoro-10-[3-[(2-methylpropan-2-yl)oxycarbonylamino]pyrrolidin-1-yl]-14-oxo-8-oxa-1-azatetracyclo[7.7.1.02,7.013,17]heptadeca-2(7),3,5,9(17),10,12,15-heptaene-15-carboxylate —— C30H35FN4O6
Tert-butyl 5-(aminomethyl)-11-fluoro-10-[3-[(2-methylpropan-2-yl)oxycarbonylamino]pyrrolidin-1-yl]-14-oxo-8-oxa-1-azatetracyclo[7.7.1.02,7.013,17]heptadeca-2(7),3,5,9(17),10,12,15-heptaene-15-carboxylate
—— 18-(3-Aminopyrrolidin-1-yl)-19-fluoro-22-oxo-16-oxa-1-azahexacyclo[15.7.1.02,15.04,13.07,12.021,25]pentacosa-2(15),3,7,9,11,13,17(25),18,20,23-decaene-23-carboxylic acid —— C28H22FN3O4
18-(3-Aminopyrrolidin-1-yl)-19-fluoro-22-oxo-16-oxa-1-azahexacyclo[15.7.1.02,15.04,13.07,12.021,25]pentacosa-2(15),3,7,9,11,13,17(25),18,20,23-decaene-23-carboxylic acid
—— 4-(2-Methoxyethylamino)-3-[3-oxo-3-[7-(2-sulfamoylphenyl)-2,3-dihydro-1,4-benzoxazin-4-yl]propyl]benzenecarboximidamide —— C27H31N5O5S
4-(2-Methoxyethylamino)-3-[3-oxo-3-[7-(2-sulfamoylphenyl)-2,3-dihydro-1,4-benzoxazin-4-yl]propyl]benzenecarboximidamide
—— 6-[[[3-[[(3-chlorophenyl)methylamino]methyl]phenyl]methylamino]methyl]-2-methyl-2H-1,4-benzoxazin-3-amine;trihydrochloride —— C25H30Cl4N4O
6-[[[3-[[(3-chlorophenyl)methylamino]methyl]phenyl]methylamino]methyl]-2-methyl-2H-1,4-benzoxazin-3-amine;trihydrochloride
—— N-[2-(6-methyl-2-oxospiro[1H-3,1-benzoxazine-4,4'-piperidine]-1'-yl)ethyl]-3-(4-methylphenyl)-8,9-dihydro-7H-benzo[7]annulene-6-carboxamide —— C34H37N3O3
N-[2-(6-methyl-2-oxospiro[1H-3,1-benzoxazine-4,4'-piperidine]-1'-yl)ethyl]-3-(4-methylphenyl)-8,9-dihydro-7H-benzo[7]annulene-6-carboxamide
—— 4-[[3-[(4-chlorophenyl)methyl]imidazol-4-yl]methyl]-N-[2-(2-methoxyphenyl)ethyl]-2,3-dihydro-1,4-benzoxazine-8-carboxamide —— C29H29ClN4O3
4-[[3-[(4-chlorophenyl)methyl]imidazol-4-yl]methyl]-N-[2-(2-methoxyphenyl)ethyl]-2,3-dihydro-1,4-benzoxazine-8-carboxamide
—— [(3S,5S)-7-chloro-5-(2,3-dimethoxyphenyl)-1-(2,2-dimethylpropyl)-2-oxo-5H-4,1-benzoxazepin-3-yl]methanesulfonic acid —— C23H28ClNO7S
[(3S,5S)-7-chloro-5-(2,3-dimethoxyphenyl)-1-(2,2-dimethylpropyl)-2-oxo-5H-4,1-benzoxazepin-3-yl]methanesulfonic acid
—— (6R)-6-hydroxy-N-(5,7,8-trimethyl-3-oxo-4H-1,4-benzoxazin-6-yl)-1,4-oxazepane-4-carboxamide —— C17H23N3O5
(6R)-6-hydroxy-N-(5,7,8-trimethyl-3-oxo-4H-1,4-benzoxazin-6-yl)-1,4-oxazepane-4-carboxamide
—— 6-[(6S)-6-hydroxy-1,4-diazepane-1-carbonyl]-4-methyl-1,4-benzoxazin-3-one —— C15H19N3O4
6-[(6S)-6-hydroxy-1,4-diazepane-1-carbonyl]-4-methyl-1,4-benzoxazin-3-one
—— 6-[(6R)-6-hydroxy-1,4-diazepane-1-carbonyl]-4-methyl-1,4-benzoxazin-3-one —— C15H19N3O4
6-[(6R)-6-hydroxy-1,4-diazepane-1-carbonyl]-4-methyl-1,4-benzoxazin-3-one
—— (2R)-N-(3-oxo-4H-1,4-benzoxazin-7-yl)-2-(pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide —— C18H21N5O4
(2R)-N-(3-oxo-4H-1,4-benzoxazin-7-yl)-2-(pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide
—— (2S)-N-(3-oxo-4H-1,4-benzoxazin-7-yl)-2-(pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide —— C18H21N5O4
(2S)-N-(3-oxo-4H-1,4-benzoxazin-7-yl)-2-(pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide
—— (6S)-6-hydroxy-N-(5,7,8-trimethyl-3-oxo-4H-1,4-benzoxazin-6-yl)-1,4-oxazepane-4-carboxamide —— C17H23N3O5
(6S)-6-hydroxy-N-(5,7,8-trimethyl-3-oxo-4H-1,4-benzoxazin-6-yl)-1,4-oxazepane-4-carboxamide
—— 2-Naphthalenecarboximidamide, 7-[[2,3-dihydro-7-[[1-(1-iminoethyl)-4-piperidinyl]oxy]-3-oxo-4H-1,4-benzoxazin-4-yl]methyl]- —— C27H29N5O3
2-Naphthalenecarboximidamide, 7-[[2,3-dihydro-7-[[1-(1-iminoethyl)-4-piperidinyl]oxy]-3-oxo-4H-1,4-benzoxazin-4-yl]methyl]-
—— 6-[[[5-(aminomethyl)cyclohexen-1-yl]methylamino]methyl]-2-methyl-2H-1,4-benzoxazin-3-amine —— C18H26N4O
6-[[[5-(aminomethyl)cyclohexen-1-yl]methylamino]methyl]-2-methyl-2H-1,4-benzoxazin-3-amine
—— 2a-[4-(1,2,3,4,4a,5-Hexahydropyrazino[2,1-c]-1,4-benzoxazin-3-yl)-butyl]-2a,3,4,5-tetrahydro-1H-benz[cd]indol-2-one 230300-90-0 C26H31N3O2
2a-[4-(1,2,3,4,4a,5-Hexahydropyrazino[2,1-c]-1,4-benzoxazin-3-yl)-butyl]-2a,3,4,5-tetrahydro-1H-benz[cd]indol-2-one
—— (2S)-N-(cyclohexen-1-ylmethyl)-4-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C17H22N2O2
(2S)-N-(cyclohexen-1-ylmethyl)-4-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— (2R)-N-(cyclohexen-1-ylmethyl)-4-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide —— C17H22N2O2
(2R)-N-(cyclohexen-1-ylmethyl)-4-methyl-2,3-dihydro-1,4-benzoxazine-2-carboxamide
—— 1-[[(5S)-3-ethyl-4,5-dihydro-1,2-oxazol-5-yl]methyl]-3-(3-oxo-4H-1,4-benzoxazin-7-yl)urea —— C15H18N4O4
1-[[(5S)-3-ethyl-4,5-dihydro-1,2-oxazol-5-yl]methyl]-3-(3-oxo-4H-1,4-benzoxazin-7-yl)urea