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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-(4-(4-amino-1-((1r,4r)-4-(4-isopropylpiperazin-1-yl)cyclohexyl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)phenyl)-7-chlorobenzo[d]oxazol-2-amine 1253107-52-6 C31H36ClN9O
N-(4-(4-amino-1-((1r,4r)-4-(4-isopropylpiperazin-1-yl)cyclohexyl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)phenyl)-7-chlorobenzo[d]oxazol-2-amine
—— N-((1R,2S)-1-(1-(4-fluorophenyl)-1H-indazol-5-yloxy)-1-(6-methoxypyridin-3-yl)propan-2-yl)cyclopropanecarboxamide 1034148-16-7 C26H25FN4O3
N-((1R,2S)-1-(1-(4-fluorophenyl)-1H-indazol-5-yloxy)-1-(6-methoxypyridin-3-yl)propan-2-yl)cyclopropanecarboxamide
—— 1-Acetyl-3-m-nitrophenyl-5-methyl-1,2,4-triazol 61598-91-2 C11H10N4O3
1-Acetyl-3-m-nitrophenyl-5-methyl-1,2,4-triazol
—— N-(4-(4-amino-1-((1s,4s)-4-(4-isopropylpiperazin-1-yl)cyclohexyl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)phenyl)-7-chlorobenzo[d]oxazol-2-amine 1253107-53-7 C31H36ClN9O
N-(4-(4-amino-1-((1s,4s)-4-(4-isopropylpiperazin-1-yl)cyclohexyl)-1H-pyrazolo[3,4-d]pyrimidin-3-yl)phenyl)-7-chlorobenzo[d]oxazol-2-amine
—— 4-methyl-5-ethoxycarbonyloxyoxazole 19561-23-0 C7H9NO4
4-methyl-5-ethoxycarbonyloxyoxazole
—— 4-(3-hydroxy-5-phenyl-1H-pyrazol-1-yl)benzenesulfonamide 188817-18-7 C15H13N3O3S
4-(3-hydroxy-5-phenyl-1H-pyrazol-1-yl)benzenesulfonamide
—— [8-(4-bromo-2,6-dimethoxyphenyl)-2,7-dimethyl-pyrazolo[1,5-a][1,3,5]triazin-4-yl]bis(2-methoxyethyl)amine 1217490-78-2 C21H28BrN5O4
[8-(4-bromo-2,6-dimethoxyphenyl)-2,7-dimethyl-pyrazolo[1,5-a][1,3,5]triazin-4-yl]bis(2-methoxyethyl)amine
—— [8-(4-benzyloxy-2,6-dimethoxyphenyl)-2,7-dimethylpyrazolo[1,5-a][1,3,5]triazin-4-yl]bis(2-methoxyethyl)amine 1217490-66-8 C28H35N5O5
[8-(4-benzyloxy-2,6-dimethoxyphenyl)-2,7-dimethylpyrazolo[1,5-a][1,3,5]triazin-4-yl]bis(2-methoxyethyl)amine
—— 8-(4-benzyloxy-2,6-dimethoxyphenyl)-4-chloro-2,7-dimethylpyrazolo[1,5-a][1,3,5]triazine 1217490-63-5 C22H21ClN4O3
8-(4-benzyloxy-2,6-dimethoxyphenyl)-4-chloro-2,7-dimethylpyrazolo[1,5-a][1,3,5]triazine
—— (2-chloro-3-methyl-3H-imidazol-4-yl)-(4-isopropyl-piperazin-1-yl)-methanone 1160227-50-8 C12H19ClN4O
(2-chloro-3-methyl-3H-imidazol-4-yl)-(4-isopropyl-piperazin-1-yl)-methanone
—— 4-(4-benzyloxy-2,6-dimethoxyphenyl)-5-methyl-2H-pyrazol-3-ylamine 1217490-56-6 C19H21N3O3
4-(4-benzyloxy-2,6-dimethoxyphenyl)-5-methyl-2H-pyrazol-3-ylamine
—— [8-(3-bromo-2,6-dimethoxyphenyl)-2,7-dimethyl-pyrazolo[1,5-a][1,3,5]triazin-4-yl]bis(2-methoxyethyl)amine 1217490-84-0 C21H28BrN5O4
[8-(3-bromo-2,6-dimethoxyphenyl)-2,7-dimethyl-pyrazolo[1,5-a][1,3,5]triazin-4-yl]bis(2-methoxyethyl)amine
—— trifluoromethanesulfonic acid 4-{4-[bis(2-methoxyethyl)amino]-2,7-dimethylpyrazolo[1,5-a][1,3,5]triazin-8-yl}-3,5-dimethoxyphenyl ester 1217490-72-6 C22H28F3N5O7S
trifluoromethanesulfonic acid 4-{4-[bis(2-methoxyethyl)amino]-2,7-dimethylpyrazolo[1,5-a][1,3,5]triazin-8-yl}-3,5-dimethoxyphenyl ester
—— [8-(2,6-dimethoxyphenyl)-2,7-dimethyl-pyrazolo[1,5-a][1,3,5]triazin-4-yl]bis(2-methoxyethyl)amine 1217490-81-7 C21H29N5O4
[8-(2,6-dimethoxyphenyl)-2,7-dimethyl-pyrazolo[1,5-a][1,3,5]triazin-4-yl]bis(2-methoxyethyl)amine
—— N-(2-diethylaminoethyl)-1-phenyl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide hydrochloride 60656-35-1 C23H26N4O*ClH
N-(2-diethylaminoethyl)-1-phenyl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide hydrochloride
—— 4-{[bis(2-methoxyethyl)amino]-2,7-dimethyl-pyrazolo[1,5-a][1,3,5]triazin-8-yl}-3,5-dimethoxyphenol 1217490-69-1 C21H29N5O5
4-{[bis(2-methoxyethyl)amino]-2,7-dimethyl-pyrazolo[1,5-a][1,3,5]triazin-8-yl}-3,5-dimethoxyphenol
—— 1-(4-chlorophenyl)-4-formyl-5-hydroxy-1H-pyrazole-3-carboxamide 61378-76-5 C11H8ClN3O3
1-(4-chlorophenyl)-4-formyl-5-hydroxy-1H-pyrazole-3-carboxamide
—— 1-(4-nitrophenyl)-5-phenyl-1H-1,2,3-triazole-4-carboxylic acid 1236-33-5 C15H10N4O4
1-(4-nitrophenyl)-5-phenyl-1H-1,2,3-triazole-4-carboxylic acid
—— 5-amino-3-(4-methoxyphenyl)-1-methyl-1H-pyrazole-4-carbonitrile 58791-91-6 C12H12N4O
5-amino-3-(4-methoxyphenyl)-1-methyl-1H-pyrazole-4-carbonitrile
—— 3,5-Dimethyl-1-(3-trifluoromethyl-phenyl)-1H-pyrazole-4-carboxylic acid 956950-77-9 C13H11F3N2O2
3,5-Dimethyl-1-(3-trifluoromethyl-phenyl)-1H-pyrazole-4-carboxylic acid
—— [3,5-dimethyl-1-(3-trifluoromethyl-phenyl)-1H-pyrazol-4-yl]-(4-isopropyl-piperazin-1-yl)-methanone 1107656-98-3 C20H25F3N4O
[3,5-dimethyl-1-(3-trifluoromethyl-phenyl)-1H-pyrazol-4-yl]-(4-isopropyl-piperazin-1-yl)-methanone
—— 4-(3,5-diisopropyl-pyrazol-1-yl)-cyclohexanone 946859-70-7 C15H24N2O
4-(3,5-diisopropyl-pyrazol-1-yl)-cyclohexanone
—— ethyl 2-(chloromethyl)-1,3-oxazole-4-carboxylate 68683-09-0 C7H8ClNO3
ethyl 2-(chloromethyl)-1,3-oxazole-4-carboxylate
—— 5-Morpholino-2-n-propyloxazol-4-carbonitril 60791-65-3 C11H15N3O2
5-Morpholino-2-n-propyloxazol-4-carbonitril
—— ethyl 5-oxo-4,5-dihydro-1,2,4-oxadiazole-3-carboxylate 42526-30-7 C5H6N2O4
ethyl 5-oxo-4,5-dihydro-1,2,4-oxadiazole-3-carboxylate
—— 2-<<2-hydroxy-1-(hydroxymethyl)ethoxy>methyl>thiazole-4-carboxamide 112475-07-7 C8H12N2O4S
2-<<2-hydroxy-1-(hydroxymethyl)ethoxy>methyl>thiazole-4-carboxamide
—— 2-phenyl-[1,2,4]triazolo[5,1-<i>a</i>]isoindol-5-one 57387-99-2 C15H9N3O
2-phenyl-[1,2,4]triazolo[5,1-<i>a</i>]isoindol-5-one
—— 5-chloro-3-(3-(trifluoromethoxy)phenyl)pyrazolo[1,5-a]pyrimidin-7-amine 1418143-31-3 C13H8ClF3N4O
5-chloro-3-(3-(trifluoromethoxy)phenyl)pyrazolo[1,5-a]pyrimidin-7-amine
—— N-(tetrahydro-2H-pyran-4-yl)-3-(3-(trifluoromethoxy)phenyl)pyrazolo[1,5-a]pyrimidin-5-amine 1361951-32-7 C18H17F3N4O2
N-(tetrahydro-2H-pyran-4-yl)-3-(3-(trifluoromethoxy)phenyl)pyrazolo[1,5-a]pyrimidin-5-amine
—— 2,4,N,N'-tetraethyl-[1,2,4]thiadiazolidine-3,5-diylidenediamine 61449-29-4 C10H20N4S
2,4,N,N'-tetraethyl-[1,2,4]thiadiazolidine-3,5-diylidenediamine
—— Ethyl 5-(isoxazol-3-yl)-1,2,4-oxadiazole-3-carboxylate 1343187-68-7 C8H7N3O4
Ethyl 5-(isoxazol-3-yl)-1,2,4-oxadiazole-3-carboxylate
—— ethyl 5-(thiophen-3-ylmethyl)-1,2,4-oxadiazole-3-carboxylate 1258503-91-1 C10H10N2O3S
ethyl 5-(thiophen-3-ylmethyl)-1,2,4-oxadiazole-3-carboxylate
—— 5-(2,4-Difluorophenyl)-1-(4-methylsulfonylphenyl)imidazole(77 % yield) 265113-49-3 C16H12F2N2O2S
5-(2,4-Difluorophenyl)-1-(4-methylsulfonylphenyl)imidazole(77 % yield)
—— 5-(3-fluoro-4-methanesulfonyl-phenyl)-[1,2,4]oxadiazole-3-carboxylic acid ethyl ester 1557037-69-0 C12H11FN2O5S
5-(3-fluoro-4-methanesulfonyl-phenyl)-[1,2,4]oxadiazole-3-carboxylic acid ethyl ester
—— 5-(4-cyano-3-fluoro-phenyl)-[1,2,4]oxadiazole-3-carboxylic acid ethyl ester 1557037-63-4 C12H8FN3O3
5-(4-cyano-3-fluoro-phenyl)-[1,2,4]oxadiazole-3-carboxylic acid ethyl ester
—— 5-(4-cyano-2-fluoro-phenyl)-[1,2,4]oxadiazole-3-carboxylic acid ethyl ester 1415836-66-6 C12H8FN3O3
5-(4-cyano-2-fluoro-phenyl)-[1,2,4]oxadiazole-3-carboxylic acid ethyl ester
—— (E)-N'-(2,4-difluorobenzylidene)-2-(2-methyl-5-nitro-1H-imidazol-1-yl)acetohydrazide 1436413-94-3 C13H11F2N5O3
(E)-N'-(2,4-difluorobenzylidene)-2-(2-methyl-5-nitro-1H-imidazol-1-yl)acetohydrazide
—— 4-amino-5-(4-isopropyl-1,3-thiazol-2-yl)-4H-1,2,4-triazole-3-thiol 1198603-98-3 C8H11N5S2
4-amino-5-(4-isopropyl-1,3-thiazol-2-yl)-4H-1,2,4-triazole-3-thiol
—— 2,6-Bis[1-(4-carboxyphenyl)-4,5,6,7-tetrahydrobenzopyrazol-3-yl]pyridine diethyl ester 154420-40-3 C37H37N5O4
2,6-Bis[1-(4-carboxyphenyl)-4,5,6,7-tetrahydrobenzopyrazol-3-yl]pyridine diethyl ester
—— 4-(((3-(3-(trifluoromethoxy)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)amino)methyl)tetrahydro-2H-thiopyran 1,1-dioxide 1361951-33-8 C19H19F3N4O3S
4-(((3-(3-(trifluoromethoxy)phenyl)pyrazolo[1,5-a]pyrimidin-5-yl)amino)methyl)tetrahydro-2H-thiopyran 1,1-dioxide
—— 4-(3-(trifluoromethoxy)phenyl)-1H-pyrazol-5-amine 1361951-73-6 C10H8F3N3O
4-(3-(trifluoromethoxy)phenyl)-1H-pyrazol-5-amine
—— 5,7-dichloro-3-(3-(trifluoromethoxy)phenyl)pyrazolo[1,5-a]pyrimidine 1418143-30-2 C13H6Cl2F3N3O
5,7-dichloro-3-(3-(trifluoromethoxy)phenyl)pyrazolo[1,5-a]pyrimidine
—— 5-(2,4-difluorophenyl)-3-(trifluoromethyl)-1H-pyrazole —— C10H5F5N2
5-(2,4-difluorophenyl)-3-(trifluoromethyl)-1H-pyrazole
—— 5-chloro-3-(3-(trifluoromethoxy)phenyl)pyrazolo[1,5-a]pyrimidine 1361951-79-2 C13H7ClF3N3O
5-chloro-3-(3-(trifluoromethoxy)phenyl)pyrazolo[1,5-a]pyrimidine
—— N-((1-methylpiperidin-4-yl)methyl)-3-(3-(trifluoromethoxy)phenyl)pyrazolo[1,5-a]pyrimidin-5-amine 1361951-49-6 C20H22F3N5O
N-((1-methylpiperidin-4-yl)methyl)-3-(3-(trifluoromethoxy)phenyl)pyrazolo[1,5-a]pyrimidin-5-amine
—— N-(1-(1H-imidazole-1-carbonyl)piperidin-4-yl)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide 1443990-84-8 C26H23Cl3N6O2
N-(1-(1H-imidazole-1-carbonyl)piperidin-4-yl)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide
—— 3,5-bis(3-(trifluoromethyl)phenyl)-4H-1,2,4-triazole 58884-90-5 C16H9F6N3
3,5-bis(3-(trifluoromethyl)phenyl)-4H-1,2,4-triazole
—— 3-bromo-5-(2-chloro-4-fluorophenyl)-α-(2,4-difluorophenyl)-1-methyl-1H-pyrazole-4-methanol 1361019-54-6 C17H11BrClF3N2O
3-bromo-5-(2-chloro-4-fluorophenyl)-α-(2,4-difluorophenyl)-1-methyl-1H-pyrazole-4-methanol
—— 2-Isopropyl-5-phenyl-thiazol 19968-75-3 C12H13NS
2-Isopropyl-5-phenyl-thiazol
—— 4-(thiazol-2-yl)thiazol-2-amine 7520-81-2 C6H5N3S2
4-(thiazol-2-yl)thiazol-2-amine