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苯二氮卓类

相关化合物

中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-[(4R)-6-(4-chlorophenyl)-1,8-dimethyl-4H-imidazo[1,2-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide —— C23H23ClN4O
2-[(4R)-6-(4-chlorophenyl)-1,8-dimethyl-4H-imidazo[1,2-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide
—— 2-[(4S)-8-[2-[2-[2-[2-[2-[2-[2-(2-aminoethoxy)ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-6-(4-chlorophenyl)-1-methyl-2,3,3a,4-tetrahydro-1H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide —— C37H57ClN6O9
2-[(4S)-8-[2-[2-[2-[2-[2-[2-[2-(2-aminoethoxy)ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]-6-(4-chlorophenyl)-1-methyl-2,3,3a,4-tetrahydro-1H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide
—— 5-(((4S)-6-(4-chlorophenyl)-4-(2-(ethylamino)-2-oxoethyl)-1-methyl-4H-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepin-8-yl)oxy)-N-phenylpentanamide —— C32H33ClN6O3
5-(((4S)-6-(4-chlorophenyl)-4-(2-(ethylamino)-2-oxoethyl)-1-methyl-4H-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepin-8-yl)oxy)-N-phenylpentanamide
—— 2-[(4S)-6-(4-chlorophenyl)-8-(4,5-dihydroxy-5-methylhexoxy)-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide —— C28H34ClN5O4
2-[(4S)-6-(4-chlorophenyl)-8-(4,5-dihydroxy-5-methylhexoxy)-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide
—— 2-[(4S)-6-(4-chlorophenyl)-1-methyl-8-(2-phenylethoxy)-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide —— C29H28ClN5O2
2-[(4S)-6-(4-chlorophenyl)-1-methyl-8-(2-phenylethoxy)-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide
—— 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-(2-naphthalen-2-ylethyl)acetamide —— C32H28ClN5O2
2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-(2-naphthalen-2-ylethyl)acetamide
—— N-(4-acetamidobutyl)-2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetamide —— C26H29ClN6O3
N-(4-acetamidobutyl)-2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetamide
—— N-[(4R)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-3-methylbutanamide —— C23H24ClN5O2
N-[(4R)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-3-methylbutanamide
—— 2-[(4S)-8-(aminomethoxy)-6-(4-chlorophenyl)-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide —— C22H23ClN6O2
2-[(4S)-8-(aminomethoxy)-6-(4-chlorophenyl)-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide
—— 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-(1-hydroxy-3H-2,1-benzoxaborol-5-yl)ethyl]acetamide —— C29H27BClN5O4
2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-(1-hydroxy-3H-2,1-benzoxaborol-5-yl)ethyl]acetamide
—— 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-(5,6-dihydroxy-1H-indol-2-yl)ethyl]acetamide —— C30H27ClN6O4
2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-(5,6-dihydroxy-1H-indol-2-yl)ethyl]acetamide
—— [4-[[[2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetyl]amino]methoxy]phenyl]boronic acid —— C27H25BClN5O5
[4-[[[2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetyl]amino]methoxy]phenyl]boronic acid
—— (3-((2-(2-(2-(2-(((4S)-6-(4-chlorophenyl)-4-(2-(ethylamino)-2-oxoethyl)-1-methyl-4H-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepin-8-yl)oxy)ethoxy)ethoxy)ethoxy)ethyl)carbamoyl)phenyl)boronic acid —— C36H42BClN6O8
(3-((2-(2-(2-(2-(((4S)-6-(4-chlorophenyl)-4-(2-(ethylamino)-2-oxoethyl)-1-methyl-4H-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepin-8-yl)oxy)ethoxy)ethoxy)ethoxy)ethyl)carbamoyl)phenyl)boronic acid
—— [4-[2-[[2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetyl]amino]ethoxy]phenyl]boronic acid —— C28H27BClN5O5
[4-[2-[[2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetyl]amino]ethoxy]phenyl]boronic acid
—— [4-[5-[[(4R)-6-(4-chlorophenyl)-1-methyl-4-(propanoylamino)-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-8-yl]oxy]pentanoylamino]phenyl]boronic acid —— C31H32BClN6O5
[4-[5-[[(4R)-6-(4-chlorophenyl)-1-methyl-4-(propanoylamino)-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-8-yl]oxy]pentanoylamino]phenyl]boronic acid
—— 5-[[[2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetyl]amino]methyl]-2-hydroxy-N-methoxybenzamide —— C29H27ClN6O5
5-[[[2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetyl]amino]methyl]-2-hydroxy-N-methoxybenzamide
—— 2-[(3S)-5-(4-chlorophenyl)-1-ethanimidoyl-2-imino-7-methoxy-3H-1,4-benzodiazepin-3-yl]-N-[2-[[hydroxy(dimethyl)silyl]methyl]phenyl]acetamide —— C29H32ClN5O3Si
2-[(3S)-5-(4-chlorophenyl)-1-ethanimidoyl-2-imino-7-methoxy-3H-1,4-benzodiazepin-3-yl]-N-[2-[[hydroxy(dimethyl)silyl]methyl]phenyl]acetamide
—— 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-[6-[hydroxy(dimethyl)silyl]quinolin-2-yl]ethyl]acetamide —— C33H33ClN6O3Si
2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-[6-[hydroxy(dimethyl)silyl]quinolin-2-yl]ethyl]acetamide
—— [3-[[[2-[(3S)-5-(4-chlorophenyl)-1-ethanimidoyl-2-imino-7-methoxy-3H-1,4-benzodiazepin-3-yl]acetyl]amino]methyl]phenyl]boronic acid —— C27H27BClN5O4
[3-[[[2-[(3S)-5-(4-chlorophenyl)-1-ethanimidoyl-2-imino-7-methoxy-3H-1,4-benzodiazepin-3-yl]acetyl]amino]methyl]phenyl]boronic acid
—— N-(2-acetamidoethyl)-2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetamide —— C24H25ClN6O3
N-(2-acetamidoethyl)-2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetamide
—— 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-[6-[hydroxy(dimethyl)silyl]quinolin-3-yl]ethyl]acetamide —— C33H33ClN6O3Si
2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-[6-[hydroxy(dimethyl)silyl]quinolin-3-yl]ethyl]acetamide
—— 2-[(4S)-6-(4-chlorophenyl)-8-(3-hydroxypropoxy)-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide —— C24H26ClN5O3
2-[(4S)-6-(4-chlorophenyl)-8-(3-hydroxypropoxy)-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide
—— N-(5-(2-((4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepin-4-yl)acetamido)pentyl)benzamide —— C32H33ClN6O3
N-(5-(2-((4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepin-4-yl)acetamido)pentyl)benzamide
—— 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-[6-[hydroxy(dimethyl)silyl]-1-benzothiophen-2-yl]ethyl]acetamide —— C32H32ClN5O3SSi
2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-[6-[hydroxy(dimethyl)silyl]-1-benzothiophen-2-yl]ethyl]acetamide
—— [6-[2-[[2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetyl]amino]ethyl]-1-benzothiophen-2-yl]boronic acid —— C30H27BClN5O4S
[6-[2-[[2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetyl]amino]ethyl]-1-benzothiophen-2-yl]boronic acid
—— 4-((2-(2-(2-(2-(((4S)-6-(4-chlorophenyl)-4-(2-(ethylamino)-2-oxoethyl)-1-methyl-4H-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepin-8-yl)oxy)ethoxy)ethoxy)ethoxy)ethyl)carbamoyl)phenylboronic acid —— C36H42BClN6O8
4-((2-(2-(2-(2-(((4S)-6-(4-chlorophenyl)-4-(2-(ethylamino)-2-oxoethyl)-1-methyl-4H-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepin-8-yl)oxy)ethoxy)ethoxy)ethoxy)ethyl)carbamoyl)phenylboronic acid
—— 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-[5-[hydroxy(dimethyl)silyl]-1-benzothiophen-2-yl]ethyl]acetamide —— C32H32ClN5O3SSi
2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-[5-[hydroxy(dimethyl)silyl]-1-benzothiophen-2-yl]ethyl]acetamide
—— 3-[3-[[[2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetyl]amino]methyl]phenoxy]-2-cyclopentyl-2-hydroxypropanoic acid —— C35H36ClN5O6
3-[3-[[[2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetyl]amino]methyl]phenoxy]-2-cyclopentyl-2-hydroxypropanoic acid
—— 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-(2,3-dihydroxy-3-methylbutyl)acetamide —— C25H28ClN5O4
2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-(2,3-dihydroxy-3-methylbutyl)acetamide
—— 2-[(3S)-5-(4-chlorophenyl)-1-ethanimidoyl-2-imino-7-methoxy-3H-1,4-benzodiazepin-3-yl]-N-[(1-hydroxy-3H-2,1-benzoxaborol-4-yl)methyl]acetamide —— C28H27BClN5O4
2-[(3S)-5-(4-chlorophenyl)-1-ethanimidoyl-2-imino-7-methoxy-3H-1,4-benzodiazepin-3-yl]-N-[(1-hydroxy-3H-2,1-benzoxaborol-4-yl)methyl]acetamide
—— 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-[3-[hydroxy(dimethyl)silyl]quinolin-7-yl]ethyl]acetamide —— C33H33ClN6O3Si
2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-[3-[hydroxy(dimethyl)silyl]quinolin-7-yl]ethyl]acetamide
—— 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[[4-hydroxy-3-(hydroxymethyl)phenyl]methyl]acetamide —— C28H26ClN5O4
2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[[4-hydroxy-3-(hydroxymethyl)phenyl]methyl]acetamide
—— 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-[3-[hydroxy(dimethyl)silyl]-1-benzothiophen-5-yl]ethyl]acetamide —— C32H32ClN5O3SSi
2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-[3-[hydroxy(dimethyl)silyl]-1-benzothiophen-5-yl]ethyl]acetamide
—— 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-[3-[hydroxy(dimethyl)silyl]-1-benzothiophen-6-yl]ethyl]acetamide —— C32H32ClN5O3SSi
2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-[3-[hydroxy(dimethyl)silyl]-1-benzothiophen-6-yl]ethyl]acetamide
—— 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[4-[[hydroxy(dimethyl)silyl]methyl]phenyl]acetamide —— C29H30ClN5O3Si
2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[4-[[hydroxy(dimethyl)silyl]methyl]phenyl]acetamide
—— [2-[[[2-[(3S)-5-(4-chlorophenyl)-1-ethanimidoyl-2-imino-7-methoxy-3H-1,4-benzodiazepin-3-yl]acetyl]amino]methyl]phenyl]boronic acid —— C27H27BClN5O4
[2-[[[2-[(3S)-5-(4-chlorophenyl)-1-ethanimidoyl-2-imino-7-methoxy-3H-1,4-benzodiazepin-3-yl]acetyl]amino]methyl]phenyl]boronic acid
—— [6-[2-[[2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetyl]amino]ethyl]-1H-indol-3-yl]boronic acid —— C30H28BClN6O4
[6-[2-[[2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetyl]amino]ethyl]-1H-indol-3-yl]boronic acid
—— 2-[(4S)-6-(4-chlorophenyl)-8-(3,4-dihydroxy-4-methylpentoxy)-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide —— C27H32ClN5O4
2-[(4S)-6-(4-chlorophenyl)-8-(3,4-dihydroxy-4-methylpentoxy)-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide
—— 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-[2-[hydroxy(dimethyl)silyl]-1-benzothiophen-5-yl]ethyl]acetamide —— C32H32ClN5O3SSi
2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-[2-[hydroxy(dimethyl)silyl]-1-benzothiophen-5-yl]ethyl]acetamide
—— 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[3-[[hydroxy(dimethyl)silyl]methyl]phenyl]acetamide —— C29H30ClN5O3Si
2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[3-[[hydroxy(dimethyl)silyl]methyl]phenyl]acetamide
—— 2-[(3S)-5-(4-chlorophenyl)-1-ethanimidoyl-2-imino-7-methoxy-3H-1,4-benzodiazepin-3-yl]-N-[(1-hydroxy-3H-2,1-benzoxaborol-7-yl)methyl]acetamide —— C28H27BClN5O4
2-[(3S)-5-(4-chlorophenyl)-1-ethanimidoyl-2-imino-7-methoxy-3H-1,4-benzodiazepin-3-yl]-N-[(1-hydroxy-3H-2,1-benzoxaborol-7-yl)methyl]acetamide
—— 4-[2-[[2-[(3S)-5-(4-chlorophenyl)-1-ethanimidoyl-2-imino-7-methoxy-3H-1,4-benzodiazepin-3-yl]acetyl]amino]ethoxy]-N-[[hydroxy(dimethyl)silyl]methyl]benzamide —— C32H37ClN6O5Si
4-[2-[[2-[(3S)-5-(4-chlorophenyl)-1-ethanimidoyl-2-imino-7-methoxy-3H-1,4-benzodiazepin-3-yl]acetyl]amino]ethoxy]-N-[[hydroxy(dimethyl)silyl]methyl]benzamide
—— 2-[(3S)-5-(4-chlorophenyl)-1-ethanimidoyl-2-imino-7-methoxy-3H-1,4-benzodiazepin-3-yl]-N-[[3-hydroxy-4-(hydroxymethyl)phenyl]methyl]acetamide —— C28H28ClN5O4
2-[(3S)-5-(4-chlorophenyl)-1-ethanimidoyl-2-imino-7-methoxy-3H-1,4-benzodiazepin-3-yl]-N-[[3-hydroxy-4-(hydroxymethyl)phenyl]methyl]acetamide
—— 2-[6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-[2-[[2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetyl]amino]ethylcarbamoylamino]ethyl]acetamide —— C45H44Cl2N12O5
2-[6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[2-[2-[[2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetyl]amino]ethylcarbamoylamino]ethyl]acetamide
—— N-[2-(6-bromo-1-benzofuran-2-yl)ethyl]-2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetamide —— C30H25BrClN5O3
N-[2-(6-bromo-1-benzofuran-2-yl)ethyl]-2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetamide
—— N-[(4R)-8-methoxy-1-methyl-6-(4-methylphenyl)-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-2-methylpropanamide —— C23H25N5O2
N-[(4R)-8-methoxy-1-methyl-6-(4-methylphenyl)-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-2-methylpropanamide
—— 2-[(4S)-6-[4-[2-[2-(2-aminoethoxy)ethoxy]ethylsulfanyl]phenyl]-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide —— C28H36N6O4S
2-[(4S)-6-[4-[2-[2-(2-aminoethoxy)ethoxy]ethylsulfanyl]phenyl]-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide
—— 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[(3,4-dihydroxyphenoxy)methyl]acetamide —— C27H24ClN5O5
2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-[(3,4-dihydroxyphenoxy)methyl]acetamide
—— N-[2-(7-bromo-1-benzothiophen-3-yl)ethyl]-2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetamide —— C30H25BrClN5O2S
N-[2-(7-bromo-1-benzothiophen-3-yl)ethyl]-2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]acetamide
—— 3-[3-[[(4R)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]carbamoyl]phenoxy]-2-cyclopentyl-2-hydroxypropanoic acid —— C33H32ClN5O6
3-[3-[[(4R)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]carbamoyl]phenoxy]-2-cyclopentyl-2-hydroxypropanoic acid