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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-chloro-5-{5-[2-(methoxymethyl)-2'-methylbiphenyl-4-yl]-1,2,4-oxadiazol-3-yl}benzoic acid 1141472-80-1 C24H19ClN2O4
2-chloro-5-{5-[2-(methoxymethyl)-2'-methylbiphenyl-4-yl]-1,2,4-oxadiazol-3-yl}benzoic acid
—— 2-amino-N-(1-methyl-1-phenylethyl)-4-(4-methylpiperazin-1-yl)quinazoline-7-carboxamide 1246207-44-2 C23H28N6O
2-amino-N-(1-methyl-1-phenylethyl)-4-(4-methylpiperazin-1-yl)quinazoline-7-carboxamide
—— 9-{2-[((1R,2S)-1-{[(2S,4R)-4-(7-methoxy-2-phenyl-quinolin-4-yloxy)-pyrrolidine-2-carbonyl]-amino}-2-vinyl-cyclopropanecarbonyl)-sulfamoyl]-phenylcarbamoyl}-nonanoic acid 1051391-60-6 C43H49N5O9S
9-{2-[((1R,2S)-1-{[(2S,4R)-4-(7-methoxy-2-phenyl-quinolin-4-yloxy)-pyrrolidine-2-carbonyl]-amino}-2-vinyl-cyclopropanecarbonyl)-sulfamoyl]-phenylcarbamoyl}-nonanoic acid
—— N-[2-(5-Chloro-thiophen-3-yl)-2-oxo-ethyl]-4-fluoro-benzamide 113471-06-0 C13H9ClFNO2S
N-[2-(5-Chloro-thiophen-3-yl)-2-oxo-ethyl]-4-fluoro-benzamide
—— (1R,3S)-3-[(1R,2R)-2-tert-Butoxycarbonyl-1-((R)-methoxysulfinyl)-2-(2-methyl-propane-2-sulfonyl)-ethyl]-2,2-dimethyl-cyclopropanecarboxylic acid 3-phenoxy-benzyl ester 138383-26-3 C31H42O9S2
(1R,3S)-3-[(1R,2R)-2-tert-Butoxycarbonyl-1-((R)-methoxysulfinyl)-2-(2-methyl-propane-2-sulfonyl)-ethyl]-2,2-dimethyl-cyclopropanecarboxylic acid 3-phenoxy-benzyl ester
—— ethyl-6-(hydroxyimino)hexa-2,4-dienoate 1446478-86-9 C8H11NO3
ethyl-6-(hydroxyimino)hexa-2,4-dienoate
—— 3,6-dimethyl-7,8-diphenylimidazo[1,5-a]pyridine 1428368-03-9 C21H18N2
3,6-dimethyl-7,8-diphenylimidazo[1,5-a]pyridine
—— —— 1425946-53-7 C17H13IN2O
—— US9598416, Example 58 1443617-17-1 C24H28N6OS
US9598416, Example 58
—— 5-(3-tert-butyl-4-carbamoylphenyl)-1-(cyclohexylmethyl)-2-methyl-N-(oxan-4-yl)pyrrole-3-carboxamide 1442424-71-6 C29H41N3O3
5-(3-tert-butyl-4-carbamoylphenyl)-1-(cyclohexylmethyl)-2-methyl-N-(oxan-4-yl)pyrrole-3-carboxamide
—— 2,3-dihydro-5-(3-hydroxy-1-piperidinyl)-1-oxo-1H-indene-2-acetic acid 103422-79-3 C16H19NO4
2,3-dihydro-5-(3-hydroxy-1-piperidinyl)-1-oxo-1H-indene-2-acetic acid
—— 2,2,3-trimethyl-3-propylcyclopropane-1,1-dicarbonitrile 105695-02-1 C11H16N2
2,2,3-trimethyl-3-propylcyclopropane-1,1-dicarbonitrile
—— (S)-3-[6-(4-chloro-phenoxy)-pyridin-3-yl]-1-(4-methoxy-benzyl)-4-(3-trifluoromethyl-phenyl)-imidazolidin-2-one 1035487-71-8 C29H23ClF3N3O3
(S)-3-[6-(4-chloro-phenoxy)-pyridin-3-yl]-1-(4-methoxy-benzyl)-4-(3-trifluoromethyl-phenyl)-imidazolidin-2-one
—— [2-Amino-6-[2-[3-(dimethylamino)propoxy]phenyl]quinazolin-4-yl]-(1,3-dihydroisoindol-2-yl)methanone 1349794-53-1 C28H29N5O2
[2-Amino-6-[2-[3-(dimethylamino)propoxy]phenyl]quinazolin-4-yl]-(1,3-dihydroisoindol-2-yl)methanone
—— Pyrimidine-5-carboxylic acid-N-(1-((5-(2-(trifluoromethyl)phenylamino)pyridin-2-yl)methylcarbamoyl)cyclopropyl)amide 1242452-08-9 C22H19F3N6O2
Pyrimidine-5-carboxylic acid-N-(1-((5-(2-(trifluoromethyl)phenylamino)pyridin-2-yl)methylcarbamoyl)cyclopropyl)amide
—— 7-(3-thienylsulfonyl)-6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c][2,7]naphthyridine 1234374-27-6 C13H12N4O2S2
7-(3-thienylsulfonyl)-6,7,8,9-tetrahydro-3H-pyrazolo[3,4-c][2,7]naphthyridine
—— 4-(2-methoxyethoxy)-8-[(R)-(tetrahydrofuran-3-yl)oxy]quinoline-2-carboxylic acid isopropyl-(R)-piperidin-3-ylamide 1443458-09-0 C25H35N3O5
4-(2-methoxyethoxy)-8-[(R)-(tetrahydrofuran-3-yl)oxy]quinoline-2-carboxylic acid isopropyl-(R)-piperidin-3-ylamide
—— 3-{[tert-butyl(diphenyl)silyl]oxy}-2-(4-fluorophenyl)-N-[4-(2-{[2-methoxy-4-(methylsulfonyl)phenyl]amino}[1,2,4]triazolo[1,5-a]pyridin-6-yl)phenyl]propanamide 1443764-22-4 C45H44FN5O5SSi
3-{[tert-butyl(diphenyl)silyl]oxy}-2-(4-fluorophenyl)-N-[4-(2-{[2-methoxy-4-(methylsulfonyl)phenyl]amino}[1,2,4]triazolo[1,5-a]pyridin-6-yl)phenyl]propanamide
—— ethyl 1-[4-(aminosulfonyl)phenyl]-5-cyclopentyl-1H-1,2,4-triazole-3-carboxylate 1006904-93-3 C16H20N4O4S
ethyl 1-[4-(aminosulfonyl)phenyl]-5-cyclopentyl-1H-1,2,4-triazole-3-carboxylate
—— 1-(4-tert-butyl-benzoyl)amino-5-morpholino-2,4-dinitro-benzene 1072919-53-9 C21H24N4O6
1-(4-tert-butyl-benzoyl)amino-5-morpholino-2,4-dinitro-benzene
—— 2-(2-chloro-5-(((tert-butylcarbonyl)amino)methyl)phenylamino)-6-(2,2-difluoroethoxy)-1-methyl-1H-benzo[d]imidazole-5-carboxylic acid 1242269-89-1 C23H25ClF2N4O4
2-(2-chloro-5-(((tert-butylcarbonyl)amino)methyl)phenylamino)-6-(2,2-difluoroethoxy)-1-methyl-1H-benzo[d]imidazole-5-carboxylic acid
—— 2-[3-(5,6-Dimethylpyridin-2-yl)-5-phenylpyrazol-1-yl]-1-(2-methyl-4,6-dihydropyrrolo[3,4-d][1,3]thiazol-5-yl)ethanone 1440953-27-4 C24H23N5OS
2-[3-(5,6-Dimethylpyridin-2-yl)-5-phenylpyrazol-1-yl]-1-(2-methyl-4,6-dihydropyrrolo[3,4-d][1,3]thiazol-5-yl)ethanone
—— [4-(1,3,3a,4,6,6a-hexahydrofuro[3,4-c]pyrrol-5-yl)piperidin-1-yl]-[5-methyl-6-[[(1S,3R)-3-phenylcyclohexyl]methylamino]pyrimidin-4-yl]methanone 1416329-41-3 C30H41N5O2
[4-(1,3,3a,4,6,6a-hexahydrofuro[3,4-c]pyrrol-5-yl)piperidin-1-yl]-[5-methyl-6-[[(1S,3R)-3-phenylcyclohexyl]methylamino]pyrimidin-4-yl]methanone
—— 4-Chloro-1,3-dihydrothieno[3,4-c]pyridine-7-carbonitrile 1357188-61-4 C8H5ClN2S
4-Chloro-1,3-dihydrothieno[3,4-c]pyridine-7-carbonitrile
—— 1-Ethyl-3-[4-hydroxy-3-(1-propylpyrazol-4-yl)phenyl]-5-phenyl-7-(trifluoromethyl)-1,5-benzodiazepine-2,4-dione 1329989-27-6 C30H27F3N4O3
1-Ethyl-3-[4-hydroxy-3-(1-propylpyrazol-4-yl)phenyl]-5-phenyl-7-(trifluoromethyl)-1,5-benzodiazepine-2,4-dione
—— (R)-((3S,7S)-7-((2R,5R)-2-methyl-5-(2-(triethylsilyloxy)propan-2-yl)tetrahydrofuran-2-yl)-1-((5R,6R,8R)-8-((S)-2-methyl-5-oxotetrahydrofuran-2-yl)-2-oxo-1,3,7-trioxaspiro[4.5]decan-6-yl)-4-methylene-7-(triethylsilyloxy)heptan-3-yl)-2-methoxy-2-phenylethanoate 1312080-64-0 C49H80O12Si2
(R)-((3S,7S)-7-((2R,5R)-2-methyl-5-(2-(triethylsilyloxy)propan-2-yl)tetrahydrofuran-2-yl)-1-((5R,6R,8R)-8-((S)-2-methyl-5-oxotetrahydrofuran-2-yl)-2-oxo-1,3,7-trioxaspiro[4.5]decan-6-yl)-4-methylene-7-(triethylsilyloxy)heptan-3-yl)-2-methoxy-2-phenylethanoate
—— (E)-N-((E)-4-phenylbut-3-en-2-ylidene)butan-1-amine 1217341-41-7 C14H19N
(E)-N-((E)-4-phenylbut-3-en-2-ylidene)butan-1-amine
—— 10-Oxo-bicyclo<4.3.1>decan-1-carbonsaeure 13348-05-5 C11H16O3
10-Oxo-bicyclo<4.3.1>decan-1-carbonsaeure
—— 4-(4-tert-butylphenyl)nonan-5-one 1268834-08-7 C19H30O
4-(4-tert-butylphenyl)nonan-5-one
—— —— 1446556-62-2 C26H26N8O2
—— [(E)-3-(Diphenyl-phosphinoyl)-3-methoxy-2-methyl-allyl]-trimethyl-silane 107832-79-1 C20H27O2PSi
[(E)-3-(Diphenyl-phosphinoyl)-3-methoxy-2-methyl-allyl]-trimethyl-silane
—— 2-<(2-Acetylphenyl)(4-methoxyphenyl)amino>benzoesaeure-methylester 104033-88-7 C23H21NO4
2-<(2-Acetylphenyl)(4-methoxyphenyl)amino>benzoesaeure-methylester
—— N-[(Z)-1-benzamidohept-5-enyl]benzamide 102853-11-2 C21H24N2O2
N-[(Z)-1-benzamidohept-5-enyl]benzamide
—— 3-(4-Hydroxy-2,2,6,6-tetramethylpiperidin-1-yl)oxypropanoic acid 1001081-24-8 C12H23NO4
3-(4-Hydroxy-2,2,6,6-tetramethylpiperidin-1-yl)oxypropanoic acid
—— 2-(4-chlorophenyl)-N-[3-[(2-chlorophenyl)sulfamoyl]-4-morpholin-4-ylphenyl]acetamide 1033344-53-4 C24H23Cl2N3O4S
2-(4-chlorophenyl)-N-[3-[(2-chlorophenyl)sulfamoyl]-4-morpholin-4-ylphenyl]acetamide
—— 4-(3-methyl-4,5,6,7-tetrahydro-1H-indazol-1-yl)benzenesulfonamide 1006907-52-3 C14H17N3O2S
4-(3-methyl-4,5,6,7-tetrahydro-1H-indazol-1-yl)benzenesulfonamide
—— 2-Piperazinemethanol, 6-methyl-1-[2-(1-methylethyl)phenyl]- 1784882-83-2 C15H24N2O
2-Piperazinemethanol, 6-methyl-1-[2-(1-methylethyl)phenyl]-
—— 7-[(2R,5S)-2,5-dimethylpiperazin-1-yl]-3-(8-methylimidazo[1,2-a]pyridin-2-yl)-2H-chromen-2-one 1446329-02-7 C23H24N4O2
7-[(2R,5S)-2,5-dimethylpiperazin-1-yl]-3-(8-methylimidazo[1,2-a]pyridin-2-yl)-2H-chromen-2-one
—— 4-[2-(2-fluoro-5-methylphenoxy)-5-(methylsulfonyl)phenyl]-6-methyl-1,6-dihydro-7H-pyrrolo[2,3-c]pyridin-7-one 1446234-08-7 C22H19FN2O4S
4-[2-(2-fluoro-5-methylphenoxy)-5-(methylsulfonyl)phenyl]-6-methyl-1,6-dihydro-7H-pyrrolo[2,3-c]pyridin-7-one
—— 1-(5-(7-((4-methoxybenzyl)(methyl)amino)-1-ethyl-2-oxo-1,2-dihydro-1,6-naphthyridin-3-yl)-2,4-difluorophenyl)-3-(3-chlorophenyl)urea 1442471-80-8 C32H28ClF2N5O3
1-(5-(7-((4-methoxybenzyl)(methyl)amino)-1-ethyl-2-oxo-1,2-dihydro-1,6-naphthyridin-3-yl)-2,4-difluorophenyl)-3-(3-chlorophenyl)urea
—— N-cyclopropyl-N-[(3R,4S)-3-fluoro-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl]-5-(3-methyl-1H-1,2,4-triazol-1-yl)pyrazine-2-carboxamide 1415836-06-4 C22H22F4N8O
N-cyclopropyl-N-[(3R,4S)-3-fluoro-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl]-5-(3-methyl-1H-1,2,4-triazol-1-yl)pyrazine-2-carboxamide
—— EWLCNPMDI 1445949-97-2 C49H73N11O15S2
EWLCNPMDI
—— (S)-2-(benzo[d]thiazol-2-ylthio)-N-(3-hydroxy-1-oxo-1-(2-(2-oxoindolin-3-ylidene)hydrazineyl)propan-2-yl)acetamide 1311513-68-4 C20H17N5O4S2
(S)-2-(benzo[d]thiazol-2-ylthio)-N-(3-hydroxy-1-oxo-1-(2-(2-oxoindolin-3-ylidene)hydrazineyl)propan-2-yl)acetamide
—— —— 1393680-58-4 C19H14N6O2
—— 3,6-diiodo-9-(4-methylpentyl)-9H-carbazole 1564289-02-6 C18H19I2N
3,6-diiodo-9-(4-methylpentyl)-9H-carbazole
—— N-[1-[1-[6-[[(2R,6S)-6-(4-chlorophenyl)oxan-2-yl]methylamino]-5-methoxypyrimidine-4-carbonyl]piperidin-4-yl]piperidin-4-yl]-N-methylmethanesulfonamide 1312589-74-4 C30H43ClN6O5S
N-[1-[1-[6-[[(2R,6S)-6-(4-chlorophenyl)oxan-2-yl]methylamino]-5-methoxypyrimidine-4-carbonyl]piperidin-4-yl]piperidin-4-yl]-N-methylmethanesulfonamide
—— 4-amino-3-(2,4-difluorophenylazo)naphthalene-1-sulfonic acid sodium salt 1357165-12-8 C16H10F2N3O3S*Na
4-amino-3-(2,4-difluorophenylazo)naphthalene-1-sulfonic acid sodium salt
—— 5-(6-chloro-1-oxo-3,4-dihydro-1H-isoindolin-2-yl)-N-methylnicotinamide 1440514-39-5 C16H14ClN3O2
5-(6-chloro-1-oxo-3,4-dihydro-1H-isoindolin-2-yl)-N-methylnicotinamide
—— sodium 4-(2-chlorobenzyloxy)-2-(3-fluorophenyl)-1,3-thiazole-5-carboxylate 1445752-86-2 C17H10ClFNO3S*Na
sodium 4-(2-chlorobenzyloxy)-2-(3-fluorophenyl)-1,3-thiazole-5-carboxylate
—— 6-(3-Methylanilino)-4-azatricyclo[6.2.1.02,7]undeca-2(7),5-dien-3-one 1357188-83-0 C17H18N2O
6-(3-Methylanilino)-4-azatricyclo[6.2.1.02,7]undeca-2(7),5-dien-3-one