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—— 9,9-dimethyl-N-[4-(1-methylpyrrol-3-yl)phenyl]-N-[4-(9-phenylcarbazol-3-yl)phenyl]fluoren-2-amine 1421752-91-1 C50H39N3
9,9-dimethyl-N-[4-(1-methylpyrrol-3-yl)phenyl]-N-[4-(9-phenylcarbazol-3-yl)phenyl]fluoren-2-amine
—— 4-Chloro-N-(imidazolidin-2-ylidene)-1H-pyrrolo[2,3-b]pyridin-5-amine 1421359-62-7 C10H10ClN5
4-Chloro-N-(imidazolidin-2-ylidene)-1H-pyrrolo[2,3-b]pyridin-5-amine
—— N-((4-chloro-2-methylphenyl)(phenyl)methyl)-2-(2-(1-(3-fluoropyridin-4-yl)-1-hydroxyethyl)benzofuran-5-yl)acetamide 1422168-30-6 C31H26ClFN2O3
N-((4-chloro-2-methylphenyl)(phenyl)methyl)-2-(2-(1-(3-fluoropyridin-4-yl)-1-hydroxyethyl)benzofuran-5-yl)acetamide
—— Ethyl 2-methyl-2-(2-methyl-5-nitrophenyl)sulfonylpropanoate 1335140-33-4 C13H17NO6S
Ethyl 2-methyl-2-(2-methyl-5-nitrophenyl)sulfonylpropanoate
—— (R)-6-(5-isopropyl-2-methylphenyl)-2-(3-methyl-1H-indol-4-yl)-4-(2-methylpiperidin-1-yl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine 1421249-61-7 C32H39N5
(R)-6-(5-isopropyl-2-methylphenyl)-2-(3-methyl-1H-indol-4-yl)-4-(2-methylpiperidin-1-yl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine
—— (R)-3-(5-cyano-3-fluoro-6-(5-fluoro-1H-pyrrolo[2,3-b]pyridin-3-yl)pyridin-2-ylamino)-4,4-dimethylpentanoic acid 1422051-36-2 C20H19F2N5O2
(R)-3-(5-cyano-3-fluoro-6-(5-fluoro-1H-pyrrolo[2,3-b]pyridin-3-yl)pyridin-2-ylamino)-4,4-dimethylpentanoic acid
—— 5-(2-cyano-4-(hydroxymethyl)phenoxy)picolinonitrile 1421434-89-0 C14H9N3O2
5-(2-cyano-4-(hydroxymethyl)phenoxy)picolinonitrile
—— 5-((3-(4-(1H-pyrrol-2-ylcarbonyl)piperazin-1-yl)azetidin-1-yl)carbonyl)-1-(6-trifluoromethylpyridin-3-yl)-1H-indole 1252765-45-9 C27H25F3N6O2
5-((3-(4-(1H-pyrrol-2-ylcarbonyl)piperazin-1-yl)azetidin-1-yl)carbonyl)-1-(6-trifluoromethylpyridin-3-yl)-1H-indole
—— N-(4-tert-butyl-2-(cyclohexylthio)benzyl)-2-(pyridin-2-yl)acetamide 1421473-89-3 C24H32N2OS
N-(4-tert-butyl-2-(cyclohexylthio)benzyl)-2-(pyridin-2-yl)acetamide
—— 2-[(dimethylamino)methyl]-N-[2-[4-(2-methylphenyl)piperazin-1-yl]-5-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyl]phenyl]-1,3-oxazole-4-carboxamide 1419869-74-1 C32H41N7O4
2-[(dimethylamino)methyl]-N-[2-[4-(2-methylphenyl)piperazin-1-yl]-5-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyl]phenyl]-1,3-oxazole-4-carboxamide
—— [(2R,3aR,6aR)-2-{4-[3-(2-hydroxypropan-2-yl)phenyl]piperidin-1-yl}hexahydropentalen 3a(1H)-yl][3-(trifluoromethyl)-7,8-dihydro-1,6-naphthyridin-6(5H)-yl]methanone 1421062-98-7 C32H40F3N3O2
[(2R,3aR,6aR)-2-{4-[3-(2-hydroxypropan-2-yl)phenyl]piperidin-1-yl}hexahydropentalen 3a(1H)-yl][3-(trifluoromethyl)-7,8-dihydro-1,6-naphthyridin-6(5H)-yl]methanone
—— (S)-3-(4-(1-(5-fluoropyridin-2-yl)ethylamino)-5-methylpyrimidin-2-ylamino)pyridin-2(1H)-one 1421757-87-0 C17H17FN6O
(S)-3-(4-(1-(5-fluoropyridin-2-yl)ethylamino)-5-methylpyrimidin-2-ylamino)pyridin-2(1H)-one
—— 8-chloro-2-phenyl-3-[(1S)-1-(pyrido[3,4-d]pyrimidin-4-ylamino)ethyl]isoquinolin-1-one 1420622-94-1 C24H18ClN5O
8-chloro-2-phenyl-3-[(1S)-1-(pyrido[3,4-d]pyrimidin-4-ylamino)ethyl]isoquinolin-1-one
—— 2-(4,4-difluorocyclohexylamino)-4-((1R,2R)-2-hydroxycyclopentylamino)-pyrimidine-5-carboxamide 1403855-36-6 C16H23F2N5O2
2-(4,4-difluorocyclohexylamino)-4-((1R,2R)-2-hydroxycyclopentylamino)-pyrimidine-5-carboxamide
—— N-[5-[2-[(4-hydroxy-1,1-dioxothiolan-3-yl)amino]ethylcarbamoyl]-2-[4-(2-methylphenyl)piperazin-1-yl]phenyl]furan-2-carboxamide 1419869-26-3 C29H35N5O6S
N-[5-[2-[(4-hydroxy-1,1-dioxothiolan-3-yl)amino]ethylcarbamoyl]-2-[4-(2-methylphenyl)piperazin-1-yl]phenyl]furan-2-carboxamide
—— 2-[(4-[2-(2-(dimethylamino)ethoxy)-4-fluorophenyl]piperazin-1-yl)methyl]pyrrolo[1,2-a]quinazolin-5(4H)-one 1417562-83-4 C26H30FN5O2
2-[(4-[2-(2-(dimethylamino)ethoxy)-4-fluorophenyl]piperazin-1-yl)methyl]pyrrolo[1,2-a]quinazolin-5(4H)-one
—— (S)-1-(6-(5-(1-methyl-1H-pyrazole-4-yl)-1H-pyrazolo[3,4-c]pyridine-3-yl)pyridin-2-yl)piperidin-3-amine 1422438-84-3 C20H22N8
(S)-1-(6-(5-(1-methyl-1H-pyrazole-4-yl)-1H-pyrazolo[3,4-c]pyridine-3-yl)pyridin-2-yl)piperidin-3-amine
—— N-{1-(3-ethoxypropyl)-2-[(5-methylthiophen-2-ylcarbamoyl)amino]-1H-benzimidazol-5-yl}-2-ethyl-N-methylbutanamide 1424296-85-4 C25H35N5O3S
N-{1-(3-ethoxypropyl)-2-[(5-methylthiophen-2-ylcarbamoyl)amino]-1H-benzimidazol-5-yl}-2-ethyl-N-methylbutanamide
—— 4-chloro-5-(3-chloro-2-fluorophenyl)isothiazole-3-carboxylic acid 1422386-98-8 C10H4Cl2FNO2S
4-chloro-5-(3-chloro-2-fluorophenyl)isothiazole-3-carboxylic acid
—— 1-[(1R)-1-cyclohexylethyl]-3-[7-[1-(3-morpholin-4-ylpropyl)pyrazol-4-yl]-1,5-naphthyridin-2-yl]urea 1422125-21-0 C27H37N7O2
1-[(1R)-1-cyclohexylethyl]-3-[7-[1-(3-morpholin-4-ylpropyl)pyrazol-4-yl]-1,5-naphthyridin-2-yl]urea
—— N-[(4,6-dimethyl-2-oxo-1,2-dihydro-3-pyridinyl)methyl]-3-methyl-1-(1-methylethyl)-6-(4-morpholinyl)-1H-indole-4-carboxamide 1346574-99-9 C25H32N4O3
N-[(4,6-dimethyl-2-oxo-1,2-dihydro-3-pyridinyl)methyl]-3-methyl-1-(1-methylethyl)-6-(4-morpholinyl)-1H-indole-4-carboxamide
—— 1-(2-phenylpropan-2-yl)-1H-pyrazol-4-amine 1422982-51-1 C12H15N3
1-(2-phenylpropan-2-yl)-1H-pyrazol-4-amine
—— (R,E)-1-(3-(4-amino-3-(3-methoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)pyrrolidin-1-yl)-4-(cyclobutyl(methyl)amino)but-2-en-1-one 1422827-12-0 C25H31N7O2
(R,E)-1-(3-(4-amino-3-(3-methoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)pyrrolidin-1-yl)-4-(cyclobutyl(methyl)amino)but-2-en-1-one
—— 3-(6-(piperazin-1-yl)pyridin-2-yl)-5-(tetrahydrofuran-3-yl)-1H-pyrazolo[3,4-c]pyridine 1422439-23-3 C19H22N6O
3-(6-(piperazin-1-yl)pyridin-2-yl)-5-(tetrahydrofuran-3-yl)-1H-pyrazolo[3,4-c]pyridine
—— N-[1-(3-hydroxypropyl)-2-{[(3-methylthiophen-2-yl)carbamoyl]amino}-1H-benzimidazol-5-yl]-N-methylbenzamide 1424297-45-9 C24H25N5O3S
N-[1-(3-hydroxypropyl)-2-{[(3-methylthiophen-2-yl)carbamoyl]amino}-1H-benzimidazol-5-yl]-N-methylbenzamide
—— N-[1-(3-amino-3-oxopropyl)-2-{[(4-cyanophenyl)carbamoyl]amino}-1H-benzimidazol-5-yl]-N-methylcyclohexanecarboxamide 1424296-41-2 C26H29N7O3
N-[1-(3-amino-3-oxopropyl)-2-{[(4-cyanophenyl)carbamoyl]amino}-1H-benzimidazol-5-yl]-N-methylcyclohexanecarboxamide
—— N-(4-fluorophenyl)-N-{[6-(4-phenylpiperazin-1-yl)pyridin-3-yl]methyl}pyridazine-4-carboxamide 1033832-77-7 C27H25FN6O
N-(4-fluorophenyl)-N-{[6-(4-phenylpiperazin-1-yl)pyridin-3-yl]methyl}pyridazine-4-carboxamide
—— 1-chloro-5,6,7,8-tetrahydrocarbazole-3-carboxylic acid 1007568-15-1 C13H12ClNO2
1-chloro-5,6,7,8-tetrahydrocarbazole-3-carboxylic acid
—— N-(4-fluorophenyl)-N-{[6-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}pyrimidine-4-carboxamide 1033832-60-8 C22H23FN6O
N-(4-fluorophenyl)-N-{[6-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}pyrimidine-4-carboxamide
—— N-(4-methylphenyl)-N-[(2-pyrrolidin-1-yl-1,3-thiazol-5-yl)methyl]-1-benzothiophene-2-carboxamide 1033832-92-6 C24H23N3OS2
N-(4-methylphenyl)-N-[(2-pyrrolidin-1-yl-1,3-thiazol-5-yl)methyl]-1-benzothiophene-2-carboxamide
—— (R)-1-(3-(2-(5-methyl-2-(4-trifluoromethylphenyl)oxazol-4-yl)ethoxy)benzyl)piperidine-2-carboxylic acid methyl ester 1065334-58-8 C27H29F3N2O4
(R)-1-(3-(2-(5-methyl-2-(4-trifluoromethylphenyl)oxazol-4-yl)ethoxy)benzyl)piperidine-2-carboxylic acid methyl ester
—— N-(4-fluorophenyl)-N-{[6-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}pyridine-2-carboxamide 1033832-57-3 C23H24FN5O
N-(4-fluorophenyl)-N-{[6-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}pyridine-2-carboxamide
—— N-[5-[4-(4-cyanophenyl)piperidine-1-carbonyl]-2-methyl-phenyl]-6-(methyl-propan-2-yl-amino)pyridine-3-carboxamide 1027354-01-3 C30H33N5O2
N-[5-[4-(4-cyanophenyl)piperidine-1-carbonyl]-2-methyl-phenyl]-6-(methyl-propan-2-yl-amino)pyridine-3-carboxamide
—— N-[5-[4-(4-cyanophenyl)piperidine-1-carbonyl]-2-methyl-phenyl]-6-methyl-pyridine-3-carboxamide 1027353-12-3 C27H26N4O2
N-[5-[4-(4-cyanophenyl)piperidine-1-carbonyl]-2-methyl-phenyl]-6-methyl-pyridine-3-carboxamide
—— [6-bromo-2-(2,4-dichloro-benzyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-carbamic acid tert-butyl ester 1067912-43-9 C20H17BrCl2N2O4
[6-bromo-2-(2,4-dichloro-benzyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-carbamic acid tert-butyl ester
—— 6-(dimethylcarbamoyl)-5-[2-(7-methoxy-2,3-dihydro-1H-inden-1-ylidene)ethyl]-1,2-dimethyl-1H-benzimidazol-4-yl pivalate 1034023-39-6 C29H35N3O4
6-(dimethylcarbamoyl)-5-[2-(7-methoxy-2,3-dihydro-1H-inden-1-ylidene)ethyl]-1,2-dimethyl-1H-benzimidazol-4-yl pivalate
—— ethyl 2-(7-methoxy-4-oxo-3,4-dihydro-2H-3-chromenyl)-2-oxoacetate 1015695-22-3 C14H14O6
ethyl 2-(7-methoxy-4-oxo-3,4-dihydro-2H-3-chromenyl)-2-oxoacetate
—— 7-(3-chlorophenyl)-1-(2,4-dichlorophenyl)-4,4-dimethyl-1,4-dihydrochromeno[4,3-c]pyrazole-3-carboxylic acid 1015695-45-0 C25H17Cl3N2O3
7-(3-chlorophenyl)-1-(2,4-dichlorophenyl)-4,4-dimethyl-1,4-dihydrochromeno[4,3-c]pyrazole-3-carboxylic acid
—— N-(3-{[2-(1,1-dioxido-2,3-dihydro-1,4-benzothiazepin-4(5H)-yl)-6-methylquinolin-4-yl]amino}propyl)acetamide 1422500-76-2 C24H28N4O3S
N-(3-{[2-(1,1-dioxido-2,3-dihydro-1,4-benzothiazepin-4(5H)-yl)-6-methylquinolin-4-yl]amino}propyl)acetamide
—— N-[2-amino-1-(2,2,2-trifluoroethyl)-1H-benzimidazol-5-yl]-N-methylcyclohexanecarboxamide 1424299-03-5 C17H21F3N4O
N-[2-amino-1-(2,2,2-trifluoroethyl)-1H-benzimidazol-5-yl]-N-methylcyclohexanecarboxamide
—— N-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]-4-methylspiro[7H-thieno[3,2-d]pyrimidine-6,1'-cyclobutane]-2-amine 1422354-24-2 C21H23N5OS
N-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]-4-methylspiro[7H-thieno[3,2-d]pyrimidine-6,1'-cyclobutane]-2-amine
—— methyl ((S)-1-(((1R,2S)-2-(5-(4-(2-((S)-1-((S)-2-(methoxycarbonyl)amino-3-methylbutanoyl)pyrrolidin-2-yl)-1,4,5,6-tetrahydrobenzo[3,4]cyclohepta[1,2-d]imidazol-8-yl)phenyl)-1H-imidazol-2-yl)cyclopentyl)amino)-3-methyl-1-oxobutan-2-yl)carbamate 1422428-12-3 C44H56N8O6
methyl ((S)-1-(((1R,2S)-2-(5-(4-(2-((S)-1-((S)-2-(methoxycarbonyl)amino-3-methylbutanoyl)pyrrolidin-2-yl)-1,4,5,6-tetrahydrobenzo[3,4]cyclohepta[1,2-d]imidazol-8-yl)phenyl)-1H-imidazol-2-yl)cyclopentyl)amino)-3-methyl-1-oxobutan-2-yl)carbamate
—— 2-[1-tert-butyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-4-[2-oxo-2-(2-phenylpyrrolidin-1-yl)ethyl]-1,3-thiazole 1421847-90-6 C28H29FN4OS
2-[1-tert-butyl-5-(4-fluorophenyl)-1H-pyrazol-4-yl]-4-[2-oxo-2-(2-phenylpyrrolidin-1-yl)ethyl]-1,3-thiazole
—— N-[2-amino-1-(3-ethoxypropyl)-1H-benzimidazol-5-yl]-4-fluoro-N-methylbenzamide 1424298-63-4 C20H23FN4O2
N-[2-amino-1-(3-ethoxypropyl)-1H-benzimidazol-5-yl]-4-fluoro-N-methylbenzamide
—— 3-(6-fluoropyridin-2-yl)-1-(tetrahydro-2H-pyran-2-yl)-5-(tetrahydro-2H-pyran-3-yl)-1H-pyrazolo[3,4-c]pyridine 1422443-03-5 C21H23FN4O2
3-(6-fluoropyridin-2-yl)-1-(tetrahydro-2H-pyran-2-yl)-5-(tetrahydro-2H-pyran-3-yl)-1H-pyrazolo[3,4-c]pyridine
—— 1-((R)-(3,5-dimethylisoxazol-4-yl)(5-(2-(((S)-(2,4-dimethylphenyl)(phenyl)methyl)amino)-2-oxoethyl)benzofuran-2-yl)methoxy)cyclopropanecarboxylic acid 1422167-87-0 C35H34N2O6
1-((R)-(3,5-dimethylisoxazol-4-yl)(5-(2-(((S)-(2,4-dimethylphenyl)(phenyl)methyl)amino)-2-oxoethyl)benzofuran-2-yl)methoxy)cyclopropanecarboxylic acid
—— [4-(3,5-dimethylpyridin-2-yl)piperazin-1-yl] (2-fluoro-4-iodophenyl)methanone 1346123-96-3 C18H19FIN3O
[4-(3,5-dimethylpyridin-2-yl)piperazin-1-yl] (2-fluoro-4-iodophenyl)methanone
—— 3-(3-chloro-4-(trifluoromethyl)phenyl)-1-methyl-N-(1,2,4-thiadiazol-5-yl)-1H-indole-6-sulfonamide 1423161-20-9 C18H12ClF3N4O2S2
3-(3-chloro-4-(trifluoromethyl)phenyl)-1-methyl-N-(1,2,4-thiadiazol-5-yl)-1H-indole-6-sulfonamide
—— (S)-1-(4-chloro-3-methoxyphenyl)-1-(1-prop-2-ene-1-ylpiperidine-2-yl)methanamine 1007109-45-6 C16H23ClN2O
(S)-1-(4-chloro-3-methoxyphenyl)-1-(1-prop-2-ene-1-ylpiperidine-2-yl)methanamine
—— N-(5-(ethylthio)-4-(morpholinomethyl)pyridin-2-yl)-2,2-dimethylbutanamide 1029127-18-1 C18H29N3O2S
N-(5-(ethylthio)-4-(morpholinomethyl)pyridin-2-yl)-2,2-dimethylbutanamide