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—— (S)-N-((S)-1-(2-chlorophenyl)-2-((3,3-difluorocyclobutyl)amino)-2-oxoethyl)-1-(4-cyanopyridin-2-yl)-N-(2,5-difluorophenyl)-5-oxopyrrolidine-2-carboxamide 1448347-70-3 C29H22ClF4N5O3
(S)-N-((S)-1-(2-chlorophenyl)-2-((3,3-difluorocyclobutyl)amino)-2-oxoethyl)-1-(4-cyanopyridin-2-yl)-N-(2,5-difluorophenyl)-5-oxopyrrolidine-2-carboxamide
—— N-{4-methoxy-3-[6-(pyridin-3-yl)-1H-imidazo[1,2-b]pyrazol-1-yl]phenyl}-3-(pentafluoro-λ<sup>6</sup>-sulphanyl)benzamide 1448316-06-0 C24H18F5N5O2S
N-{4-methoxy-3-[6-(pyridin-3-yl)-1H-imidazo[1,2-b]pyrazol-1-yl]phenyl}-3-(pentafluoro-λ<sup>6</sup>-sulphanyl)benzamide
—— 6-(3-fluorophenyl)-N-(1-pyrido[2,3-d]pyrimidin-2-ylpiperidin-4-yl)nicotinamide 1033839-37-0 C24H21FN6O
6-(3-fluorophenyl)-N-(1-pyrido[2,3-d]pyrimidin-2-ylpiperidin-4-yl)nicotinamide
—— 2-[4-({7-methoxy-3-[2-(methylamino)pyrimidin-4-yl]-1-naphthyl}amino)piperidin-1-yl]isonicotinonitrile 1313487-54-5 C27H27N7O
2-[4-({7-methoxy-3-[2-(methylamino)pyrimidin-4-yl]-1-naphthyl}amino)piperidin-1-yl]isonicotinonitrile
—— 2-(3-methylpiperidin-1-yl)-N-(6-(piperazin-1-yl)pyridin-3-yl)-4-(trifluoromethyl)oxazole-5-carboxamide 1228000-55-2 C20H25F3N6O2
2-(3-methylpiperidin-1-yl)-N-(6-(piperazin-1-yl)pyridin-3-yl)-4-(trifluoromethyl)oxazole-5-carboxamide
—— 6-[2-(2-Aminobenzimidazol-1-yl)ethylamino]-1-[[4-(difluoromethoxy)phenyl]methyl]-3-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1,3,5-triazine-2,4-dione 1148128-32-8 C29H27F2N7O4
6-[2-(2-Aminobenzimidazol-1-yl)ethylamino]-1-[[4-(difluoromethoxy)phenyl]methyl]-3-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1,3,5-triazine-2,4-dione
—— (2S,4S)-methyl 1-[4,4-bis(3-methyl-2-thienyl)-3-buten-1-yl]-4-fluoropyrrolidine-2-carboxylate 1157865-28-5 C20H24FNO2S2
(2S,4S)-methyl 1-[4,4-bis(3-methyl-2-thienyl)-3-buten-1-yl]-4-fluoropyrrolidine-2-carboxylate
—— 1-methyl-1H-indazole-3-carboxylic acid {(1R,3S,4S)-2-[2-dimethylamino-5-(3-fluoro-phenyl)-thiazole-4-carbonyl]-2-aza-bicyclo[2.2.1]hept-3-ylmethyl}-amide 1181571-85-6 C28H29FN6O2S
1-methyl-1H-indazole-3-carboxylic acid {(1R,3S,4S)-2-[2-dimethylamino-5-(3-fluoro-phenyl)-thiazole-4-carbonyl]-2-aza-bicyclo[2.2.1]hept-3-ylmethyl}-amide
—— (2S,4R)-2-(1-cyanocyclopropylcarbamoyl)-4-(2,6-dichlorobenzenesulfonyl)pyrrolidine-1-carboxylic acid tert-butyl ester 1252631-64-3 C20H23Cl2N3O5S
(2S,4R)-2-(1-cyanocyclopropylcarbamoyl)-4-(2,6-dichlorobenzenesulfonyl)pyrrolidine-1-carboxylic acid tert-butyl ester
—— 2,2-dimethyl-propionic acid (R)-2-[7-amino-5-(2,2-dimethyl-propionyloxymethyl)-1H-indol-2-yl]-4,5-dihydro-thiazol-4-ylmethyl ester 1172997-16-8 C23H31N3O4S
2,2-dimethyl-propionic acid (R)-2-[7-amino-5-(2,2-dimethyl-propionyloxymethyl)-1H-indol-2-yl]-4,5-dihydro-thiazol-4-ylmethyl ester
—— [(R)-2-(7-cyclopentylamino-5-methoxy-1H-indol-2-yl)-4,5-dihydro-thiazol-4-yl]-acetic acid ethyl ester 1172996-59-6 C21H27N3O3S
[(R)-2-(7-cyclopentylamino-5-methoxy-1H-indol-2-yl)-4,5-dihydro-thiazol-4-yl]-acetic acid ethyl ester
—— N-[6-chloro-4-(ethylcarbamoyl)-1,3-benzodioxol-5-yl]-2-(3-chloropyridin-2-yl)-5-(trifluoromethyl)pyrazole-3-carboxamide 1103244-77-4 C20H14Cl2F3N5O4
N-[6-chloro-4-(ethylcarbamoyl)-1,3-benzodioxol-5-yl]-2-(3-chloropyridin-2-yl)-5-(trifluoromethyl)pyrazole-3-carboxamide
—— 2,N-dicyclohexyl-2-[5,6-difluoro-2-(4-methoxy-phenoxymethyl)-benzoimidazol-1-yl]-acetamide 1128218-66-5 C29H35F2N3O3
2,N-dicyclohexyl-2-[5,6-difluoro-2-(4-methoxy-phenoxymethyl)-benzoimidazol-1-yl]-acetamide
—— 11-(5-chloro-2-thienyl)-2-fluorodibenzo[b,f][1,4]thiazepine-8-carboxylic acid butyl amide 1019853-48-5 C22H18ClFN2OS2
11-(5-chloro-2-thienyl)-2-fluorodibenzo[b,f][1,4]thiazepine-8-carboxylic acid butyl amide
—— N-(3-(5-(2-((4-chlorophenyl)amino)pyrimidin-4-yl)imidazo[2,1-b][1,3]thiazol-6-yl)phenyl)benzamide 1159884-33-9 C28H19ClN6OS
N-(3-(5-(2-((4-chlorophenyl)amino)pyrimidin-4-yl)imidazo[2,1-b][1,3]thiazol-6-yl)phenyl)benzamide
—— 2-[2-(trifluoromethyl)benzyl]-N-[4-(trifluoromethyl)phenyl][1,3]thiazolo[5,4-d]pyrimidin-7-amine 1160607-20-4 C20H12F6N4S
2-[2-(trifluoromethyl)benzyl]-N-[4-(trifluoromethyl)phenyl][1,3]thiazolo[5,4-d]pyrimidin-7-amine
—— (R)-2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4H-chromen-3-yl 2-(tert-butoxycarbonylamino)-3-methylbutanoate 1158555-69-1 C25H27NO10
(R)-2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4H-chromen-3-yl 2-(tert-butoxycarbonylamino)-3-methylbutanoate
—— (4-butoxy-benzyl)-carbamic acid methyl ester 100618-96-0 C13H19NO3
(4-butoxy-benzyl)-carbamic acid methyl ester
—— 2-[3-(1-fluoropropyl)-5-(1H-pyrazolo[3,4-b]pyridin-4-yl)phenyl]-2-methylbutan-1-amine 1160500-24-2 C20H25FN4
2-[3-(1-fluoropropyl)-5-(1H-pyrazolo[3,4-b]pyridin-4-yl)phenyl]-2-methylbutan-1-amine
—— 2-(2,6-dichlorobenzyl)-N-[3-fluoro-4-(methylsulfonyl)phenyl][1,3]thiazolo[5,4-d]pyrimidin-7-amine 1160607-39-5 C19H13Cl2FN4O2S2
2-(2,6-dichlorobenzyl)-N-[3-fluoro-4-(methylsulfonyl)phenyl][1,3]thiazolo[5,4-d]pyrimidin-7-amine
—— tert-butyl (2S,3S,4S,5R)-5-acetoxy-3,4-bis(benzyloxy)-2-(benzyloxymethyl)piperidine-1-carboxylate 1161011-66-0 C34H41NO7
tert-butyl (2S,3S,4S,5R)-5-acetoxy-3,4-bis(benzyloxy)-2-(benzyloxymethyl)piperidine-1-carboxylate
—— (1R,2R,3R)-1-methoxycarbonyl-trans-2-furyl-cis-3-[(E)-2-(trimethylsilyl)vinyl]cyclopropane 1160615-49-5 C14H20O3Si
(1R,2R,3R)-1-methoxycarbonyl-trans-2-furyl-cis-3-[(E)-2-(trimethylsilyl)vinyl]cyclopropane
—— N-(2-chloro-6-(methyl-d3)phenyl)-2-(6-(4-(2,2-d2-2-hydroxyethyl)piperazin-1-yl)-2-methylpyrimidin-4-ylamino)thiazole-5-carboxamide 1160297-11-9 C22H26ClN7O2S
N-(2-chloro-6-(methyl-d3)phenyl)-2-(6-(4-(2,2-d2-2-hydroxyethyl)piperazin-1-yl)-2-methylpyrimidin-4-ylamino)thiazole-5-carboxamide
—— 9-(phenanthren-9-yl)-9H-carbazole-3-carbaldehyde 1097732-19-8 C27H17NO
9-(phenanthren-9-yl)-9H-carbazole-3-carbaldehyde
—— 3-chloro-4'-(1-imidazol-1-yl-propyl)-biphenyl-4-ol 1164120-71-1 C18H17ClN2O
3-chloro-4'-(1-imidazol-1-yl-propyl)-biphenyl-4-ol
—— 1-[4-(2-{(S)-1-[4-(2-aminopyrimidin-5-yl)phenyl]-1-cyclopropylethyl}oxazol-4-yl)pyrazol-1-yl]-2-methylpropan-2-ol 1448610-32-9 C25H28N6O2
1-[4-(2-{(S)-1-[4-(2-aminopyrimidin-5-yl)phenyl]-1-cyclopropylethyl}oxazol-4-yl)pyrazol-1-yl]-2-methylpropan-2-ol
—— (6-Ethylthieno[2,3-b]pyrrol-5-yl)-(1-propylpyrrolo[2,3-c]pyridin-3-yl)methanone 1328170-42-8 C19H19N3OS
(6-Ethylthieno[2,3-b]pyrrol-5-yl)-(1-propylpyrrolo[2,3-c]pyridin-3-yl)methanone
—— 1-[3-(trifluoromethoxy)phenyl]-1H-pyrazole-4-carbaldehyde 1366407-18-2 C11H7F3N2O2
1-[3-(trifluoromethoxy)phenyl]-1H-pyrazole-4-carbaldehyde
—— cyclohexyl(4-(2-(2,5-dichlorophenoxy)-5-nitrophenylsulfonyl)piperazin-1-yl)methanone 1253109-77-1 C23H25Cl2N3O6S
cyclohexyl(4-(2-(2,5-dichlorophenoxy)-5-nitrophenylsulfonyl)piperazin-1-yl)methanone
—— (S)-methyl 2-(2-azidoacetamido)-3-(3-(2-fluoroethoxy)benzylthio)propanoate 1071475-66-5 C15H19FN4O4S
(S)-methyl 2-(2-azidoacetamido)-3-(3-(2-fluoroethoxy)benzylthio)propanoate
—— 2-{4-[3-(4-acetylaminophenyl)ureido]phenyl}-5-ethoxy-6-morpholin-4-ylpyrimidine-4-carboxylic acid ethyl ester 1313718-18-1 C28H32N6O6
2-{4-[3-(4-acetylaminophenyl)ureido]phenyl}-5-ethoxy-6-morpholin-4-ylpyrimidine-4-carboxylic acid ethyl ester
—— (8S)-8-amino-3-[2,6-difluoro-4-[(5R)-2-oxo-5-(triazol-1-ylmethyl)-1,3-oxazolidin-3-yl]phenyl]-1,2,4,5,8,9-hexahydropyridazino[1,2-a][1,2,5]triazepine-7,10-dione 1138149-46-8 C20H22F2N8O4
(8S)-8-amino-3-[2,6-difluoro-4-[(5R)-2-oxo-5-(triazol-1-ylmethyl)-1,3-oxazolidin-3-yl]phenyl]-1,2,4,5,8,9-hexahydropyridazino[1,2-a][1,2,5]triazepine-7,10-dione
—— 4,4,6,6-tetramethyl-2-[(2,2,3,3-tetramethyl-cyclopropanecarbonyl)-amino]-4,6-dihydrothieno[2,3-c]furan-3-carboxylic acid 1010798-51-2 C19H27NO4S
4,4,6,6-tetramethyl-2-[(2,2,3,3-tetramethyl-cyclopropanecarbonyl)-amino]-4,6-dihydrothieno[2,3-c]furan-3-carboxylic acid
—— 1-[4-(5-ethyl-[1,2,4]oxadiazol-3-yl)-benzoyl]-40phenyl-piperidine-4-carboxylic acid ((S)-1-phenyl-ethyl)-amide 1246386-56-0 C31H32N4O3
1-[4-(5-ethyl-[1,2,4]oxadiazol-3-yl)-benzoyl]-40phenyl-piperidine-4-carboxylic acid ((S)-1-phenyl-ethyl)-amide
—— (R)-4-hydroxy-7-(1-hydroxy-2-(9-(4-(2-methylfuran-3-carbonyl)-l-oxa-4,9-diazaspiro[5.5]undecan-9-yl)nonylamino)ethyl)benzo[d]thiazol-2(3H)-one 1179334-95-2 C32H46N4O6S
(R)-4-hydroxy-7-(1-hydroxy-2-(9-(4-(2-methylfuran-3-carbonyl)-l-oxa-4,9-diazaspiro[5.5]undecan-9-yl)nonylamino)ethyl)benzo[d]thiazol-2(3H)-one
—— N-(5-tert-butyl-4-methyl-thiazol-2-yl)-2-{4-[2-(3,5-dimethyl-pyrazol-1-yl)-acetyl]-piperazin-1-yl}-benzamide 1253381-81-5 C26H34N6O2S
N-(5-tert-butyl-4-methyl-thiazol-2-yl)-2-{4-[2-(3,5-dimethyl-pyrazol-1-yl)-acetyl]-piperazin-1-yl}-benzamide
—— N-[3-methoxy-4-(2-methyl-4-pyridinyl)phenyl]-1-(1-methylethyl)-5-[3-(4-morpholinyl)phenoxy]-1H-1,2,4-triazol-3-amine 1314874-70-8 C28H32N6O3
N-[3-methoxy-4-(2-methyl-4-pyridinyl)phenyl]-1-(1-methylethyl)-5-[3-(4-morpholinyl)phenoxy]-1H-1,2,4-triazol-3-amine
—— {[3'-({4-[(3,5-dioxo-1,2,4-oxadiazolidine-2-yl)methyl]phenoxy}methyl)-2,2',6-trimethylbiphenyl-4-yl]oxy} acetic acid 1148023-54-4 C27H26N2O7
{[3'-({4-[(3,5-dioxo-1,2,4-oxadiazolidine-2-yl)methyl]phenoxy}methyl)-2,2',6-trimethylbiphenyl-4-yl]oxy} acetic acid
—— N-((2R,6S,13aS,14aR,16aS,Z)-2-(3-ethyl-7-fluoroquinoxalin-2-yloxy)-14a-(cyclopropylsulfonylcarbamoyl)-5,16-dioxo-1,2,3,5,6,7,8,9,10,11,13a,14,14a,15,16,16a-hexadecahydrocyclopropa[e]pyrrolo[1,2-a][1,4]diazacyclopentadecin-6-yl)-3-methylisoxazole-5-carboxamide 1352301-95-1 C36H42FN7O8S
N-((2R,6S,13aS,14aR,16aS,Z)-2-(3-ethyl-7-fluoroquinoxalin-2-yloxy)-14a-(cyclopropylsulfonylcarbamoyl)-5,16-dioxo-1,2,3,5,6,7,8,9,10,11,13a,14,14a,15,16,16a-hexadecahydrocyclopropa[e]pyrrolo[1,2-a][1,4]diazacyclopentadecin-6-yl)-3-methylisoxazole-5-carboxamide
—— 6-(2,3-dihydro-1H-indol-1-yl)-2-ethylsulfanyl-N-[(3-fluorophenyl)-methyl]-4-methyl-pyridine-3-carboxylic acid amide 1373488-78-8 C24H24FN3OS
6-(2,3-dihydro-1H-indol-1-yl)-2-ethylsulfanyl-N-[(3-fluorophenyl)-methyl]-4-methyl-pyridine-3-carboxylic acid amide
—— 3-chloro-6-(4-chloro-2-fluoro-3-methoxy-phenyl)-4-[(2,4-dimethoxyphenyl-methyl)-amino]-pyridine-2-carboxylic acid methyl ester 1259329-76-4 C23H21Cl2FN2O5
3-chloro-6-(4-chloro-2-fluoro-3-methoxy-phenyl)-4-[(2,4-dimethoxyphenyl-methyl)-amino]-pyridine-2-carboxylic acid methyl ester
—— 9-methylheptadeca-1,16-diene-7,11-dione 1149661-58-4 C18H30O2
9-methylheptadeca-1,16-diene-7,11-dione
—— 1-(4-{2-[(R)-2-(5-chloro-7-cyclopentylamino-1H-indol-2-yl)-4,5-dihydro-thiazol-4-yl]-ethyl}-piperazin-1-yl)-ethanone 1120344-01-5 C24H32ClN5OS
1-(4-{2-[(R)-2-(5-chloro-7-cyclopentylamino-1H-indol-2-yl)-4,5-dihydro-thiazol-4-yl]-ethyl}-piperazin-1-yl)-ethanone
—— N-(benzyloxy)-5-{[5,6-dihydro-4H-pyrrolo[3,2,1-ij]quinolin-1-yl(oxo)acetyl]amino}pentanamide 1122597-55-0 C25H27N3O4
N-(benzyloxy)-5-{[5,6-dihydro-4H-pyrrolo[3,2,1-ij]quinolin-1-yl(oxo)acetyl]amino}pentanamide
—— DHK19 1071471-49-2 C16H13N5O2S3
DHK19
—— 4-(5-methyl-pyridin-2-yloxy)-cyclohexanone 1252607-19-4 C12H15NO2
4-(5-methyl-pyridin-2-yloxy)-cyclohexanone
—— (2S)-methyl 2-(2-azidoacetamido)-3-(3-(2-fluoroethoxy)benzylsulfinyl)propanoate 1071475-67-6 C15H19FN4O5S
(2S)-methyl 2-(2-azidoacetamido)-3-(3-(2-fluoroethoxy)benzylsulfinyl)propanoate
—— phenyl 1-(4-(trifluoromethyl)phenyl)-3,4-dihydroisoquinoline-2(1H)-carboxylate 1159996-17-4 C23H18F3NO2
phenyl 1-(4-(trifluoromethyl)phenyl)-3,4-dihydroisoquinoline-2(1H)-carboxylate
—— N-[(1R,2R)-1-hydroxy-1-[4-(5-methylhexoxy)phenyl]-3-pyrrolidin-1-ylpropan-2-yl]-6-(4-methoxyphenyl)-6-oxohexanamide 1092470-00-2 C33H48N2O5
N-[(1R,2R)-1-hydroxy-1-[4-(5-methylhexoxy)phenyl]-3-pyrrolidin-1-ylpropan-2-yl]-6-(4-methoxyphenyl)-6-oxohexanamide
—— N-[4-bromo-2-methyl-6-(methylcarbamoyl)phenyl]-2-(3-chloropyridin-2-yl)-5-[[5-(difluoromethyl)tetrazol-2-yl]methyl]pyrazole-3-carboxamide 1229657-50-4 C21H17BrClF2N9O2
N-[4-bromo-2-methyl-6-(methylcarbamoyl)phenyl]-2-(3-chloropyridin-2-yl)-5-[[5-(difluoromethyl)tetrazol-2-yl]methyl]pyrazole-3-carboxamide