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中文名称 英文名称 CAS号 化学式 结构式图片
—— (R)-9-(4-(1-aminopropan-2-yl)phenyl)-8-methoxythieno[2,3-c]quinolin-4(5H)-one hydrochloride 1338544-93-6 C21H20N2O2S*ClH
(R)-9-(4-(1-aminopropan-2-yl)phenyl)-8-methoxythieno[2,3-c]quinolin-4(5H)-one hydrochloride
—— 1-[(4R)-2,2-diethyl-6-fluoro-3,4-dihydro-2H-chromen-4-yl]-3-(1-methyl-2-oxo-1,2-dihydroquinolin-5-yl)urea 1444789-64-3 C24H26FN3O3
1-[(4R)-2,2-diethyl-6-fluoro-3,4-dihydro-2H-chromen-4-yl]-3-(1-methyl-2-oxo-1,2-dihydroquinolin-5-yl)urea
—— (3S)-tert-butyl 3-((1-(2-chlorophenyl)-2-((3,3-difluorocyclobutyl)amino)-2-oxoethyl)(3-fluorophenyl)carbamoyl)-4-(4-cyanopyridin-2-yl)-5-oxopiperazine-1-carboxylate 1448346-61-9 C34H32ClF3N6O5
(3S)-tert-butyl 3-((1-(2-chlorophenyl)-2-((3,3-difluorocyclobutyl)amino)-2-oxoethyl)(3-fluorophenyl)carbamoyl)-4-(4-cyanopyridin-2-yl)-5-oxopiperazine-1-carboxylate
—— (S)-2-(4-(5-(3-chlorophenyl)-1H-pyrazol-3-yl)phenyl)morpholine hydrochloride 1447830-24-1 C19H18ClN3O*ClH
(S)-2-(4-(5-(3-chlorophenyl)-1H-pyrazol-3-yl)phenyl)morpholine hydrochloride
—— 1,1,1,2,2,3,3,4,4,5,5,6,6,7,7,8,8,9,9,10,10-Henicosafluoro-11-iodoundecane 1146953-90-3 C11H2F21I
1,1,1,2,2,3,3,4,4,5,5,6,6,7,7,8,8,9,9,10,10-Henicosafluoro-11-iodoundecane
—— Propyl 3-[2-[[4-[bis(3-methoxy-3-oxopropyl)amino]-2-hydroxyphenyl]diazenyl]-4-chloro-1,3-thiazol-5-yl]-2-cyanoprop-2-enoate 1114964-08-7 C24H26ClN5O7S
Propyl 3-[2-[[4-[bis(3-methoxy-3-oxopropyl)amino]-2-hydroxyphenyl]diazenyl]-4-chloro-1,3-thiazol-5-yl]-2-cyanoprop-2-enoate
—— N-[4-(2,4-difluorophenoxy)-3-(6-methyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-d]pyridazin-4-yl)phenyl]ethanesulfonamide 1446233-71-1 C21H18F2N4O4S
N-[4-(2,4-difluorophenoxy)-3-(6-methyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-d]pyridazin-4-yl)phenyl]ethanesulfonamide
—— 5-(8-hydroxy-1,4-dioxa-spiro[4.5]dec-8-yl)-1,3-dimethyl-1,3-dihydro-benzoimidazol-2-one 1252616-23-1 C17H22N2O4
5-(8-hydroxy-1,4-dioxa-spiro[4.5]dec-8-yl)-1,3-dimethyl-1,3-dihydro-benzoimidazol-2-one
—— 1-[4-(2-{(R)-2-[5-fluoro-7-(tetrahydro-pyran-4-ylamino)-1H-indol-2-yl]-4,5-dihydro-thiazol-4-yl}-ethyl)-piperazin-1-yl]-ethanone 1120344-27-5 C24H32FN5O2S
1-[4-(2-{(R)-2-[5-fluoro-7-(tetrahydro-pyran-4-ylamino)-1H-indol-2-yl]-4,5-dihydro-thiazol-4-yl}-ethyl)-piperazin-1-yl]-ethanone
—— 3-(5-methylpyridin-2-yl)-N-(2-phenylpropan-2-yl)-5-(2,2,2-trifluoro-1-hydroxyethyl)benzamide 1150249-75-4 C24H23F3N2O2
3-(5-methylpyridin-2-yl)-N-(2-phenylpropan-2-yl)-5-(2,2,2-trifluoro-1-hydroxyethyl)benzamide
—— 2-(5-morpholin-4-yl-pyridin-3-yl)-10-spirocyclopropyl-5,6,8,9,10,11-hexahydro-3,8,11-triaza-benzo[a]fluoren-7-one 1105661-74-2 C25H25N5O2
2-(5-morpholin-4-yl-pyridin-3-yl)-10-spirocyclopropyl-5,6,8,9,10,11-hexahydro-3,8,11-triaza-benzo[a]fluoren-7-one
—— 3-[4-[[(4S)-2,2-dimethyl-1,3-dioxolan-4-yl]methoxy]-2-methylphenyl]-2-methylbenzaldehyde 1148022-42-7 C21H24O4
3-[4-[[(4S)-2,2-dimethyl-1,3-dioxolan-4-yl]methoxy]-2-methylphenyl]-2-methylbenzaldehyde
—— 7-methyl-N-(4-morpholin-4-ylbutyl)-1-(oxan-4-yl)-4-oxo-5H-pyrazolo[4,3-c]quinoline-8-carboxamide 1364614-72-1 C25H33N5O4
7-methyl-N-(4-morpholin-4-ylbutyl)-1-(oxan-4-yl)-4-oxo-5H-pyrazolo[4,3-c]quinoline-8-carboxamide
—— 2-fluoro-3-(indol-3-yl)propionic acid 131451-35-9 C11H10FNO2
2-fluoro-3-(indol-3-yl)propionic acid
—— (6-chloro-1H,3H-2,4,7a,8-tetraaza-cyclopenta[a]inden-2-yl)-[4-fluoro-2-(1,1,2,2-tetrafluoro-ethoxy)-phenyl]-methanone 1445803-35-9 C17H10ClF5N4O2
(6-chloro-1H,3H-2,4,7a,8-tetraaza-cyclopenta[a]inden-2-yl)-[4-fluoro-2-(1,1,2,2-tetrafluoro-ethoxy)-phenyl]-methanone
—— 3-fluoromethyl-2-methanesulfonyl-5-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)pyridine 1445651-55-7 C13H19BFNO4S
3-fluoromethyl-2-methanesulfonyl-5-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)pyridine
—— {(S)-3-[4-(6-methoxy-5-methyl-pyridin-3-yl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-yloxy]-pyrrolidin-1-yl}-(3-methyl-3h-imidazol-4-yl)-methanone 1446000-03-8 C24H27N5O4
{(S)-3-[4-(6-methoxy-5-methyl-pyridin-3-yl)-3,4-dihydro-2H-benzo[1,4]oxazin-6-yloxy]-pyrrolidin-1-yl}-(3-methyl-3h-imidazol-4-yl)-methanone
—— 9-hydroxymethyl-3-oxo-spiro[5.5]undecane 154464-91-2 C12H20O2
9-hydroxymethyl-3-oxo-spiro[5.5]undecane
—— (3-(5-chloro-2,4-dihydroxyphenyl)-1,4,6,7-tetrahydro-5H-pyrazolo[4,3-c]pyridin-5-yl)(4-((1,1-dioxidothiomorpholin-4-yl)methyl)phenyl)methanone 1228278-73-6 C24H25ClN4O5S
(3-(5-chloro-2,4-dihydroxyphenyl)-1,4,6,7-tetrahydro-5H-pyrazolo[4,3-c]pyridin-5-yl)(4-((1,1-dioxidothiomorpholin-4-yl)methyl)phenyl)methanone
—— N-{1-[3-(2-Methyl-3,3,3-trifluoropropoxycarbonylamino)benzyl]-indol-5-ylcarbonyl}-2-methylbenzene sulphonamide 141451-89-0 C28H26F3N3O5S
N-{1-[3-(2-Methyl-3,3,3-trifluoropropoxycarbonylamino)benzyl]-indol-5-ylcarbonyl}-2-methylbenzene sulphonamide
—— N,N-bis(4-aminobenzyl)isoxazol-3-amine 1252601-41-4 C17H18N4O
N,N-bis(4-aminobenzyl)isoxazol-3-amine
—— 4-(3-methoxy-pyridin-2-yloxy)-cyclohexanone 1252607-23-0 C12H15NO3
4-(3-methoxy-pyridin-2-yloxy)-cyclohexanone
—— N-{[6-chloro-4-(trifluoromethyl)pyridin-2-yl]carbamoyl}-5-(2-methoxyethyl)-4-methylthiophene-2-sulfonamide 1158787-70-2 C15H15ClF3N3O4S2
N-{[6-chloro-4-(trifluoromethyl)pyridin-2-yl]carbamoyl}-5-(2-methoxyethyl)-4-methylthiophene-2-sulfonamide
—— H-Cys-Leu-Pro-Thr-Arg-His-Met-Ala-Cys-OH 1160375-81-4 C41H70N14O11S3
H-Cys-Leu-Pro-Thr-Arg-His-Met-Ala-Cys-OH
—— 5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-yl)-N-cyclopentylpyridine-3-sulfonamide 1159823-92-3 C16H18N6O2S
5-(2-amino-[1,2,4]triazolo[1,5-a]pyridin-yl)-N-cyclopentylpyridine-3-sulfonamide
—— 2-[6-chloro-5-fluoro-2-(4-fluoro-phenylsulfanylmethyl)-benzoimidazol-1-yl]-2,N-dicyclohexyl-acetamide 1128219-15-7 C28H32ClF2N3OS
2-[6-chloro-5-fluoro-2-(4-fluoro-phenylsulfanylmethyl)-benzoimidazol-1-yl]-2,N-dicyclohexyl-acetamide
—— 2-{4-[4-(2,6-di-tert-butyl-pyrimidin-4-yl)-piperazin-1-yl]-butyl}-2H-[1,2,4]triazine-3,5-dione 1147785-32-7 C23H37N7O2
2-{4-[4-(2,6-di-tert-butyl-pyrimidin-4-yl)-piperazin-1-yl]-butyl}-2H-[1,2,4]triazine-3,5-dione
—— methyl-[2-(4-methyl-dibenzo[b,f]oxepin-10-yl)-ethyl]-carbamic acid tert-butyl ester 1184947-40-7 C23H27NO3
methyl-[2-(4-methyl-dibenzo[b,f]oxepin-10-yl)-ethyl]-carbamic acid tert-butyl ester
—— N-(2-chloro-pyridin-4-yl)-2-{4-[2-(3,5-dimethyl-pyrazol-1-yl)-acetyl]-piperazin-1-yl}-benzamide 1253382-74-9 C23H25ClN6O2
N-(2-chloro-pyridin-4-yl)-2-{4-[2-(3,5-dimethyl-pyrazol-1-yl)-acetyl]-piperazin-1-yl}-benzamide
—— Tert-butyl 4-[3-[3-[[3-(3,5-difluorophenyl)-6-oxopyridazin-1-yl]methyl]phenyl]-1,2,4-oxadiazol-5-yl]piperazine-1-carboxylate 1007099-07-1 C28H28F2N6O4
Tert-butyl 4-[3-[3-[[3-(3,5-difluorophenyl)-6-oxopyridazin-1-yl]methyl]phenyl]-1,2,4-oxadiazol-5-yl]piperazine-1-carboxylate
—— 3-(4,4-difluoropiperidin-1-yl)-N-{2,4-dimethyl-5-[6-(pyridin-3-yl)-1H-imidazo[1,2-b]pyrazol-1-yl]phenyl}benzamide 1448316-71-9 C30H28F2N6O
3-(4,4-difluoropiperidin-1-yl)-N-{2,4-dimethyl-5-[6-(pyridin-3-yl)-1H-imidazo[1,2-b]pyrazol-1-yl]phenyl}benzamide
—— N<sup>2</sup>-(1-methylcyclopropyl)-6-phenyl-N<sup>4</sup>-(pyridin-4-yl)-1,3,5-triazine-2,4-diamine 1446503-11-2 C18H18N6
N<sup>2</sup>-(1-methylcyclopropyl)-6-phenyl-N<sup>4</sup>-(pyridin-4-yl)-1,3,5-triazine-2,4-diamine
—— Tert-butyl 3-[4-(1-acetamidoethyl)phenyl]azetidine-1-carboxylate 1446021-07-3 C18H26N2O3
Tert-butyl 3-[4-(1-acetamidoethyl)phenyl]azetidine-1-carboxylate
—— tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(1-methylindazol-6-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate 1428666-52-7 C29H33N5O3
tert-butyl (1R,3S,4S)-3-[[(1S)-1-cyano-2-[4-(1-methylindazol-6-yl)phenyl]ethyl]carbamoyl]-2-azabicyclo[2.2.1]heptane-2-carboxylate
—— 7-methyl-1-(oxan-4-yl)-8-[4-(oxan-4-yl)piperazine-1-carbonyl]-5H-pyrazolo[4,3-c]quinolin-4-one 1364607-15-7 C26H33N5O4
7-methyl-1-(oxan-4-yl)-8-[4-(oxan-4-yl)piperazine-1-carbonyl]-5H-pyrazolo[4,3-c]quinolin-4-one
—— 5-cyclopropyl-4-[2-(N-methyl-N-methylsulphonyl)amino-benzoyl]isoxazole 158579-54-5 C15H16N2O4S
5-cyclopropyl-4-[2-(N-methyl-N-methylsulphonyl)amino-benzoyl]isoxazole
—— N-({1-[4-(4-methylsulfanyl-phenyl)-cyclohex-3-enyl]-azetidin-3-ylcarbamoyl}-methyl)-3-trifluoromethyl-benzamide 1252615-95-4 C26H28F3N3O2S
N-({1-[4-(4-methylsulfanyl-phenyl)-cyclohex-3-enyl]-azetidin-3-ylcarbamoyl}-methyl)-3-trifluoromethyl-benzamide
—— 2,2-dimethyl-5-morpholin-4-yl-N-(2-morpholin-4-ylethyl)-N-(pyridin-3-ylmethyl)-1,4-dihydro-2H-pyrano[4'',3'':4',5']pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-8-amine 1247025-90-6 C30H37N7O3S
2,2-dimethyl-5-morpholin-4-yl-N-(2-morpholin-4-ylethyl)-N-(pyridin-3-ylmethyl)-1,4-dihydro-2H-pyrano[4'',3'':4',5']pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-8-amine
—— 3-((3,3-diphenylpropyloxy)methyl)-7-methoxybenzofuran 181053-15-6 C25H24O3
3-((3,3-diphenylpropyloxy)methyl)-7-methoxybenzofuran
—— N-(5-(3-(1H-benzo[d]imidazol-2-yl)-1H-indazol-5-yl)pyridin-3-yl)-3-methylbutanamide 1616951-63-3 C24H22N6O
N-(5-(3-(1H-benzo[d]imidazol-2-yl)-1H-indazol-5-yl)pyridin-3-yl)-3-methylbutanamide
—— 6-(4-hydroxy-2-methoxyphenyl)-3-methyl-1H-pyrazolo[3,4-b]pyridine-4-carboxylic acid 1429171-44-7 C15H13N3O4
6-(4-hydroxy-2-methoxyphenyl)-3-methyl-1H-pyrazolo[3,4-b]pyridine-4-carboxylic acid
—— 5'-fluoro-4'-(2-hydroxyethoxy)-2,2'-dimethylbiphenyl-3-carbaldehyde 1147857-54-2 C17H17FO3
5'-fluoro-4'-(2-hydroxyethoxy)-2,2'-dimethylbiphenyl-3-carbaldehyde
—— 1-{1-[4-(3-pyrrolidin-1-ylpropoxy)phenyl]-1H-pyrazol-4-yl}pyrrolidine-2-one 1152748-34-9 C20H26N4O2
1-{1-[4-(3-pyrrolidin-1-ylpropoxy)phenyl]-1H-pyrazol-4-yl}pyrrolidine-2-one
—— tert-butyl {1-(2,3-dichlorophenyl)-2-[(ethylsulphonyl)amino]ethyl}carbamate 1245622-40-5 C15H22Cl2N2O4S
tert-butyl {1-(2,3-dichlorophenyl)-2-[(ethylsulphonyl)amino]ethyl}carbamate
—— N-[2-methoxy-4-[1-(2-methoxyethyl)-2-oxo-benzofuro[3,2-d]pyrimidin-4-yl]phenyl]-2-pyrrolidin-1-yl-acetamide 1251585-55-3 C26H28N4O5
N-[2-methoxy-4-[1-(2-methoxyethyl)-2-oxo-benzofuro[3,2-d]pyrimidin-4-yl]phenyl]-2-pyrrolidin-1-yl-acetamide
—— 2-(4-{[2-(2-fluorophenyl)-1-methylethyl]amino}-2-oxo-1,2-dihydropyridin-3-yl)-6-(3-pyrrolidin-1-ylpropyl)-6,7-dihydroimidazo[4,5-f]isoindol-5(3H)-one 1188411-02-0 C30H33FN6O2
2-(4-{[2-(2-fluorophenyl)-1-methylethyl]amino}-2-oxo-1,2-dihydropyridin-3-yl)-6-(3-pyrrolidin-1-ylpropyl)-6,7-dihydroimidazo[4,5-f]isoindol-5(3H)-one
—— 7-methyl-N-[3-[methyl-(1-methylpiperidin-4-yl)amino]-3-oxopropyl]-1-(oxan-4-yl)-4-oxo-5H-pyrazolo[4,3-c]quinoline-8-carboxamide 1364936-45-7 C27H36N6O4
7-methyl-N-[3-[methyl-(1-methylpiperidin-4-yl)amino]-3-oxopropyl]-1-(oxan-4-yl)-4-oxo-5H-pyrazolo[4,3-c]quinoline-8-carboxamide
—— 1-cyclopentyl-7-methyl-N-(oxan-4-ylmethyl)-4-oxo-5H-pyrazolo[4,3-c]quinoline-8-carboxamide 1364617-53-7 C23H28N4O3
1-cyclopentyl-7-methyl-N-(oxan-4-ylmethyl)-4-oxo-5H-pyrazolo[4,3-c]quinoline-8-carboxamide
—— 2-[[(2S)-pyrrolidine-2-carbonyl]amino]butanoic acid 1493764-39-8 C9H16N2O3
2-[[(2S)-pyrrolidine-2-carbonyl]amino]butanoic acid
—— 3-[(2,2-Dimethylpropyl)amino]propanenitrile 100551-78-8 C8H16N2
3-[(2,2-Dimethylpropyl)amino]propanenitrile