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中文名称 英文名称 CAS号 化学式 结构式图片
—— 5-Hydroxy-5-trifluormethyl-5.6-dihydro-uracil 1481-04-5 C5H5F3N2O3
5-Hydroxy-5-trifluormethyl-5.6-dihydro-uracil
—— 1-[[2-chloro-4-[3-(3,5-dichlorophenyl)-3-(trifluoromethyl)pyrrolidin-1-yl]phenyl]methylideneamino]-3-(2,2-difluoroethyl)urea 1370263-06-1 C21H18Cl3F5N4O
1-[[2-chloro-4-[3-(3,5-dichlorophenyl)-3-(trifluoromethyl)pyrrolidin-1-yl]phenyl]methylideneamino]-3-(2,2-difluoroethyl)urea
—— N-[4-[4-(1,2, 3,4-Tetrahydro-6,7-dimethoxy-2-isoquinolinyl)butoxy]phenyl]-1-isoquinolinecarboxamide 159781-05-2 C31H33N3O4
N-[4-[4-(1,2, 3,4-Tetrahydro-6,7-dimethoxy-2-isoquinolinyl)butoxy]phenyl]-1-isoquinolinecarboxamide
—— 3-methylaminocarbonyloximino-4-methyl-1,2,3,4-tetrahydrocyclopent[b]indol-7-yl methylcarbamate 142284-20-6 C16H18N4O4
3-methylaminocarbonyloximino-4-methyl-1,2,3,4-tetrahydrocyclopent[b]indol-7-yl methylcarbamate
—— 6-chloro-3-((6,7-dimethoxyisoquinolin-4-yl)methyl)-4H-chromen-4-one 1605070-62-9 C21H16ClNO4
6-chloro-3-((6,7-dimethoxyisoquinolin-4-yl)methyl)-4H-chromen-4-one
—— 3'-fluoro-4'-[3-((R)-1-mercaptomethyl-3-methylbutylcarbamoyl)-5-propylpyrazol-1-ylmethyl]biphenyl-2-carboxylic acid 1260232-47-0 C27H32FN3O3S
3'-fluoro-4'-[3-((R)-1-mercaptomethyl-3-methylbutylcarbamoyl)-5-propylpyrazol-1-ylmethyl]biphenyl-2-carboxylic acid
—— N7-(2-mrpholinoethyl)-2-phenyl-5H-pyrido[3,2-b]indole-4,7-dicarboxamide 1235464-10-4 C25H25N5O3
N7-(2-mrpholinoethyl)-2-phenyl-5H-pyrido[3,2-b]indole-4,7-dicarboxamide
—— 4-{[(6-{2-chloro-4-[(E)-3-(4-{[2-(4-methoxyphenoxy)quinolin-6-yl]methyl}piperazin-1-yl)-3-oxoprop-1-en-1-yl]phenoxy}pyridin-3-yl)oxy]methyl}benzonitrile 1322779-14-5 C43H36ClN5O5
4-{[(6-{2-chloro-4-[(E)-3-(4-{[2-(4-methoxyphenoxy)quinolin-6-yl]methyl}piperazin-1-yl)-3-oxoprop-1-en-1-yl]phenoxy}pyridin-3-yl)oxy]methyl}benzonitrile
—— (8R)-8-(2-bromo-5-tert-butylphenyl)-2-[6-methoxy-5-(4-methylimidazol-1-yl)pyridin-2-yl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridine 1242311-26-7 C26H29BrN6O
(8R)-8-(2-bromo-5-tert-butylphenyl)-2-[6-methoxy-5-(4-methylimidazol-1-yl)pyridin-2-yl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridine
—— 9-ethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-6-(2-oxo-1,2-dihydro-1'H-spiro[indole-3,4'-piperidin]-1'-yl)-9H-purine-8-carboxamide 1365606-65-0 C24H25N9O3
9-ethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-6-(2-oxo-1,2-dihydro-1'H-spiro[indole-3,4'-piperidin]-1'-yl)-9H-purine-8-carboxamide
—— N-((4-chloro-6,6-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl)-N-ethylpropan-2-amine 1256956-35-0 C16H26ClN3
N-((4-chloro-6,6-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl)-N-ethylpropan-2-amine
—— 1-(4-(2-(2-p-tolyloxazol-4-yl)ethoxy)benzyl)piperidine-2-carboxylic acid 1065335-79-6 C25H28N2O4
1-(4-(2-(2-p-tolyloxazol-4-yl)ethoxy)benzyl)piperidine-2-carboxylic acid
—— 9-p-Chlorobenzyl-6-(7-chloroquinolin-2-ylmethoxy)-1,2,3,4-tetrahydrocarbazol-1-ylacetic acid 141179-76-2 C31H26Cl2N2O3
9-p-Chlorobenzyl-6-(7-chloroquinolin-2-ylmethoxy)-1,2,3,4-tetrahydrocarbazol-1-ylacetic acid
—— (4-{[5-hydroxy-6-(3-methoxycyclohexyl)-pyridin-2-yl]methyl}-2,3,5-trimethylphenoxy)acetic acid 1253211-53-8 C24H31NO5
(4-{[5-hydroxy-6-(3-methoxycyclohexyl)-pyridin-2-yl]methyl}-2,3,5-trimethylphenoxy)acetic acid
—— (S)-α-[(S)-2-[(t-butylsulphonyl)methyl]-4-phenylbutyramido]-N-[(1S,2R,3S)-1-(cyclohexylmethyl)-3-cyclopropyl-2,3-dihydroxypropyl]imidazole-4-propionamide 126222-44-4 C34H52N4O6S
(S)-α-[(S)-2-[(t-butylsulphonyl)methyl]-4-phenylbutyramido]-N-[(1S,2R,3S)-1-(cyclohexylmethyl)-3-cyclopropyl-2,3-dihydroxypropyl]imidazole-4-propionamide
—— 3-[4-[5-Bromo-1-ethyl-3-(1H-tetrazol-5-yl)-2-pyrrolyl]benzyl]-7-methyl-2-propyl-3H-imidazo[4,5-b]pyridine 142014-63-9 C24H25BrN8
3-[4-[5-Bromo-1-ethyl-3-(1H-tetrazol-5-yl)-2-pyrrolyl]benzyl]-7-methyl-2-propyl-3H-imidazo[4,5-b]pyridine
—— 4-(4-Hexanoylamino-indol-1-ylmethyl)-3-methoxy-benzoic acid methyl ester 104436-19-3 C24H28N2O4
4-(4-Hexanoylamino-indol-1-ylmethyl)-3-methoxy-benzoic acid methyl ester
—— 4-[(2-mercaptomethyl-3-phenylpropionyl)amino]-2-hydroxybenzoic acid 123986-45-8 C17H17NO4S
4-[(2-mercaptomethyl-3-phenylpropionyl)amino]-2-hydroxybenzoic acid
—— US9499502, 9cy-a 1403464-23-2 C23H23FN6O4S
US9499502, 9cy-a
—— (S)-4-oxo-2-[7-oxo-4-(4-trifluoromethoxy-phenyl)-[1,4]diazepan-1-yl]-butyric acid methyl ester 1206599-92-9 C17H19F3N2O5
(S)-4-oxo-2-[7-oxo-4-(4-trifluoromethoxy-phenyl)-[1,4]diazepan-1-yl]-butyric acid methyl ester
—— 5-chloro-6-(3-methoxyphenyl)-2-methyl-8-morpholinoimidazo[1,2-a]pyrazine 1252594-97-0 C18H19ClN4O2
5-chloro-6-(3-methoxyphenyl)-2-methyl-8-morpholinoimidazo[1,2-a]pyrazine
—— 4-chloro-N-[3-methoxy-5-(trifluoromethyl)phenyl]phthalazin-1-amine 1365802-97-6 C16H11ClF3N3O
4-chloro-N-[3-methoxy-5-(trifluoromethyl)phenyl]phthalazin-1-amine
—— 4-(benzo[d]oxazol-2-ylamino)-N-(thiazol-2-yl)benzenesulfonamide 1104804-94-5 C16H12N4O3S2
4-(benzo[d]oxazol-2-ylamino)-N-(thiazol-2-yl)benzenesulfonamide
—— (3R,5S,8S,13R,15E)-8-cyclohexyl-N-((1R,2S)-1-{[(cyclopropylsulfonyl)amino]carbonyl}-2-vinylcyclopropyl)-22-ethoxy-18-methoxy-13-methyl-7,10-dioxo-2,11-dioxa-6,9,21-triazatetracyclo[15.6.2.1(3,6).0(20,24)]hexacosa-1(23),15,17,19,21,24-hexaene-5-carboxamide 1021437-12-6 C41H53N5O10S
(3R,5S,8S,13R,15E)-8-cyclohexyl-N-((1R,2S)-1-{[(cyclopropylsulfonyl)amino]carbonyl}-2-vinylcyclopropyl)-22-ethoxy-18-methoxy-13-methyl-7,10-dioxo-2,11-dioxa-6,9,21-triazatetracyclo[15.6.2.1(3,6).0(20,24)]hexacosa-1(23),15,17,19,21,24-hexaene-5-carboxamide
—— 2-(4-fluorophenethylamino)benzo[d]thiazole-6-carbonitrile 1409949-05-8 C16H12FN3S
2-(4-fluorophenethylamino)benzo[d]thiazole-6-carbonitrile
—— 9-[4'-(β-Methylaminocarbonyloxyethyl)anilino]-2,7-dimethoxyacridine 135753-82-1 C25H25N3O4
9-[4'-(β-Methylaminocarbonyloxyethyl)anilino]-2,7-dimethoxyacridine
—— 1-(3-(4-(5-(3,5-dichloro-4-fluorophenyl)-5-(trifluoromethyl)-4,5-dihydroisoxazol-3-yl)phenyl)-3-fluoroazetidin-1-yl)-2-methyl-1-oxopropane-2-sulfonamide 1357612-14-6 C23H20Cl2F5N3O4S
1-(3-(4-(5-(3,5-dichloro-4-fluorophenyl)-5-(trifluoromethyl)-4,5-dihydroisoxazol-3-yl)phenyl)-3-fluoroazetidin-1-yl)-2-methyl-1-oxopropane-2-sulfonamide
—— 4-(1-(4-chlorobenzyl)-1H-pyrazol-3-ylamino)-N-(thiazol-2-yl)-2-(trifluoromethyl)benzenesulfonamide 1104806-01-0 C20H15ClF3N5O2S2
4-(1-(4-chlorobenzyl)-1H-pyrazol-3-ylamino)-N-(thiazol-2-yl)-2-(trifluoromethyl)benzenesulfonamide
—— (E)-5-(((2-hydroxyphenyl)imino)methyl)-2-methoxyphenol 1415567-41-7 C14H13NO3
(E)-5-(((2-hydroxyphenyl)imino)methyl)-2-methoxyphenol
—— N-[(2R,3S)-2-(2'-ethoxybiphenyl-4-yl)-6-oxopiperidin-3-yl]propane-2-sulfonamide 1219634-08-8 C22H28N2O4S
N-[(2R,3S)-2-(2'-ethoxybiphenyl-4-yl)-6-oxopiperidin-3-yl]propane-2-sulfonamide
—— 3-(3-Chlorophenyl)sulfonyl-5,7-dimethyl-2-methylsulfinylpyrazolo[1,5-a]pyrimidine 1220641-62-2 C15H14ClN3O3S2
3-(3-Chlorophenyl)sulfonyl-5,7-dimethyl-2-methylsulfinylpyrazolo[1,5-a]pyrimidine
—— 6-acetamido-N-phenyl-2,3-dihydropyrido[3,2-b][1,4]oxazine-4-carboxamide 1214929-07-3 C16H16N4O3
6-acetamido-N-phenyl-2,3-dihydropyrido[3,2-b][1,4]oxazine-4-carboxamide
—— N-[(1R)-5-[5-(3-cyano-4-propan-2-yloxyphenyl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydronaphthalen-1-yl]morpholine-4-carboxamide 1307230-63-2 C27H29N5O4
N-[(1R)-5-[5-(3-cyano-4-propan-2-yloxyphenyl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydronaphthalen-1-yl]morpholine-4-carboxamide
—— N1-(2-Benzylaminocarbonyl-3-methylbutanoyl)-N4-(benzyl-oxycarbonyl)-2,2-difluoro-3-hydroxy-6-methyl-1,4-heptanediamine 119844-25-6 C29H39F2N3O5
N1-(2-Benzylaminocarbonyl-3-methylbutanoyl)-N4-(benzyl-oxycarbonyl)-2,2-difluoro-3-hydroxy-6-methyl-1,4-heptanediamine
—— 1-[[4-(hexahydro-1H-azepin-1-yl)-phenyl]-sulphonyl]-4-hydroxy-pyrrolidinon 143136-22-5 C16H22N2O4S
1-[[4-(hexahydro-1H-azepin-1-yl)-phenyl]-sulphonyl]-4-hydroxy-pyrrolidinon
—— 2-Methyl-2-acetylaminomethyl-6-chlorochroman-4-ol 144312-63-0 C13H16ClNO3
2-Methyl-2-acetylaminomethyl-6-chlorochroman-4-ol
—— methyl 4-(6-hexanamido-2,3,5-trimethylindol-1-ylmethyl)-3-methoxybenzoate 104446-89-1 C27H34N2O4
methyl 4-(6-hexanamido-2,3,5-trimethylindol-1-ylmethyl)-3-methoxybenzoate
—— 1-methoxy-4-[2-[2-(4-methoxyphenyl)sulfanylphenyl]sulfanylphenyl]sulfanylbenzene 131376-22-2 C26H22O2S3
1-methoxy-4-[2-[2-(4-methoxyphenyl)sulfanylphenyl]sulfanylphenyl]sulfanylbenzene
—— (E)-6-(2-Methoxy-phenyl)-hex-5-enoic acid 128577-54-8 C13H16O3
(E)-6-(2-Methoxy-phenyl)-hex-5-enoic acid
—— 4-(2-methyl-1,3-dioxolan-2-yl)-2-methylthiocycloheptimidazole 129242-40-6 C13H14N2O2S
4-(2-methyl-1,3-dioxolan-2-yl)-2-methylthiocycloheptimidazole
—— 6-chloro-2-methylaminomethylbenzo-1,4-dioxane 142032-48-2 C10H12ClNO2
6-chloro-2-methylaminomethylbenzo-1,4-dioxane
—— 9-[3'-(Methylaminocarbonyloxymethyl)anilino]-3,6-dimethoxyacridine 135786-47-9 C24H23N3O4
9-[3'-(Methylaminocarbonyloxymethyl)anilino]-3,6-dimethoxyacridine
—— 6-[3-cyano-1-cyclobutyl-6-(trifluoromethoxy)-1H-indol-2-yl]-N-[(2R)-1,1,1-trifluoropropan-2-yl]pyridine-3-sulfonamide 1248575-61-2 C22H18F6N4O3S
6-[3-cyano-1-cyclobutyl-6-(trifluoromethoxy)-1H-indol-2-yl]-N-[(2R)-1,1,1-trifluoropropan-2-yl]pyridine-3-sulfonamide
—— 3-[(2R,6S)-10-hydroxy-6,11,11-trimethyl-1,2,5,6-tetrahydro-4H-2,6-methanobenzo[d]azocine-3-carbonyl]benzoic acid methyl ester 1155851-25-4 C24H27NO4
3-[(2R,6S)-10-hydroxy-6,11,11-trimethyl-1,2,5,6-tetrahydro-4H-2,6-methanobenzo[d]azocine-3-carbonyl]benzoic acid methyl ester
—— 5-((S)-1-ethyl-piperidin-3-yloxy)-9H-dipyrido[2,3-b;4',3'-d]pyrrole-6-carbonitrile 1312754-80-5 C18H19N5O
5-((S)-1-ethyl-piperidin-3-yloxy)-9H-dipyrido[2,3-b;4',3'-d]pyrrole-6-carbonitrile
—— (S)-3-chloro-4-(3-hydroxypiperidin-1-yl)-9H-dipyrido[2,3-b;4',3'-d]pyrrole-6-carbonitrile 1312754-11-2 C16H14ClN5O
(S)-3-chloro-4-(3-hydroxypiperidin-1-yl)-9H-dipyrido[2,3-b;4',3'-d]pyrrole-6-carbonitrile
—— (S)-(3,5-dinitrophenyl)(3-(4-methoxyphenoxy)pyrrolidin-1-yl)methanone 1204418-82-5 C18H17N3O7
(S)-(3,5-dinitrophenyl)(3-(4-methoxyphenoxy)pyrrolidin-1-yl)methanone
—— (2Z,5Z)-ethyl 2-{4-[5-{(2-cyclopropylcarbonylamino)(1,3-thiazol-5-yl)methylene}-4-oxo(1,3-thiazolidin-2-ylidene)azamethyl]-3-methylphenoxy}acetate 1253209-84-5 C22H22N4O5S2
(2Z,5Z)-ethyl 2-{4-[5-{(2-cyclopropylcarbonylamino)(1,3-thiazol-5-yl)methylene}-4-oxo(1,3-thiazolidin-2-ylidene)azamethyl]-3-methylphenoxy}acetate
—— 4-{[5-(ethylthio)-3-(trifluoromethyl)-1H-1,2,4-triazol-1-yl]methyl}-2-methylaniline 1207089-86-8 C13H15F3N4S
4-{[5-(ethylthio)-3-(trifluoromethyl)-1H-1,2,4-triazol-1-yl]methyl}-2-methylaniline
—— N,N-diethyl-4-[4-(1-isopropyl-1H-pyrrolo[2,3-c]pyridin-3-yl)-pyrimidin-2-ylamino]-3-methoxy-benzamide 1221153-10-1 C26H30N6O2
N,N-diethyl-4-[4-(1-isopropyl-1H-pyrrolo[2,3-c]pyridin-3-yl)-pyrimidin-2-ylamino]-3-methoxy-benzamide