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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-cyclobutyl-N-[[3-[6-(dimethylamino)pyridin-3-yl]-4-fluorophenyl]methyl]-1-methylimidazole-4-carboxamide 1366405-93-7 C23H26FN5O
N-cyclobutyl-N-[[3-[6-(dimethylamino)pyridin-3-yl]-4-fluorophenyl]methyl]-1-methylimidazole-4-carboxamide
—— (2S,4R)-4-hydroxy-1-(5-hydroxy-2-methylbenzoyl)-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide 1448186-98-8 C24H25N3O4S
(2S,4R)-4-hydroxy-1-(5-hydroxy-2-methylbenzoyl)-N-[[4-(4-methyl-1,3-thiazol-5-yl)phenyl]methyl]pyrrolidine-2-carboxamide
—— 2-ethylsulfanyl-N-[(3-fluorophenyl)-methyl]-6-[(3R)-3-(methoxymethyl)-morpholin-4-yl]-4-methyl-pyridine-3-carboxylic acid amide 1373487-54-7 C22H28FN3O3S
2-ethylsulfanyl-N-[(3-fluorophenyl)-methyl]-6-[(3R)-3-(methoxymethyl)-morpholin-4-yl]-4-methyl-pyridine-3-carboxylic acid amide
—— 1-(2'-(2-(diisopropylamino)ethoxy)-5'-(5-methyl-1,3,4-oxadiazol-2-yl)-4-(4(trifluoromethyl)thiazol-2-yl)-3,3'-bipyridin-6-yl)-3-ethylurea 1186109-13-6 C28H33F3N8O3S
1-(2'-(2-(diisopropylamino)ethoxy)-5'-(5-methyl-1,3,4-oxadiazol-2-yl)-4-(4(trifluoromethyl)thiazol-2-yl)-3,3'-bipyridin-6-yl)-3-ethylurea
—— sodium 6-chloro-7-(4-(6-(2,4-dichlorophenyl)pyridin-2-ylcarbamoyl)phenoxy)chroman-4-carboxylate 1233694-71-7 C28H18Cl3N2O5*Na
sodium 6-chloro-7-(4-(6-(2,4-dichlorophenyl)pyridin-2-ylcarbamoyl)phenoxy)chroman-4-carboxylate
—— 5-(piperidin-4-yl)-N-{5-[3-(trifluoromethyl)phenyl]-1H-benzimidazol-2-yl}imidazo[1,2-a]pyridine-2-carboxamide 1254170-09-6 C27H23F3N6O
5-(piperidin-4-yl)-N-{5-[3-(trifluoromethyl)phenyl]-1H-benzimidazol-2-yl}imidazo[1,2-a]pyridine-2-carboxamide
—— 5-[3-(2-bromo-5-fluorophenoxy)azetidin-1-yl]-N-(4-fluorophenyl)pyrazine-2-carboxamide 1222404-41-2 C20H15BrF2N4O2
5-[3-(2-bromo-5-fluorophenoxy)azetidin-1-yl]-N-(4-fluorophenyl)pyrazine-2-carboxamide
—— 2-morpholin-4-yl-N-6-pyridin-3-yl-[4,5']bipyrimidinyl-6,2'-diamine 1155305-48-8 C17H18N8O
2-morpholin-4-yl-N-6-pyridin-3-yl-[4,5']bipyrimidinyl-6,2'-diamine
—— 4-N-[1-[5-[[5-chloro-4-(trifluoromethyl)pyridin-2-yl]carbamoyl]-1,3-thiazol-2-yl]ethyl]-6-N-(2-hydroxyethyl)pyrimidine-4,6-dicarboxamide 1097249-27-8 C20H17ClF3N7O4S
4-N-[1-[5-[[5-chloro-4-(trifluoromethyl)pyridin-2-yl]carbamoyl]-1,3-thiazol-2-yl]ethyl]-6-N-(2-hydroxyethyl)pyrimidine-4,6-dicarboxamide
—— 5-chloro-N-(4-(octyloxy)-3-(trifluoromethyl)phenyl)-4-(pyrazin-2-yl)thiazol-2-amine 1088698-22-9 C22H24ClF3N4OS
5-chloro-N-(4-(octyloxy)-3-(trifluoromethyl)phenyl)-4-(pyrazin-2-yl)thiazol-2-amine
—— 1-(5-hydroxy-2-azatricyclo[3.3.1.1<sup>3,7</sup>]dec-2-yl)-3-(5-methoxy-4-methy-1H-indol-3-yl)butan-1-one 1448698-20-1 C23H30N2O3
1-(5-hydroxy-2-azatricyclo[3.3.1.1<sup>3,7</sup>]dec-2-yl)-3-(5-methoxy-4-methy-1H-indol-3-yl)butan-1-one
—— isopropyl (S)-2-(4-{[4-(1-(4-chlorophenyl)cyclopropylamino)-6-(2,2,2-trifluoroethoxy)-1,3,5-triazin-2-yl]amino}benzamido)-3-(2-(dimethylamino)-2-oxoacetamido)propanoate 1449396-96-6 C31H34ClF3N8O6
isopropyl (S)-2-(4-{[4-(1-(4-chlorophenyl)cyclopropylamino)-6-(2,2,2-trifluoroethoxy)-1,3,5-triazin-2-yl]amino}benzamido)-3-(2-(dimethylamino)-2-oxoacetamido)propanoate
—— N-{2,4-dimethyl-5-[6-(pyridin-3-yl)-1H-imidazo[1,2-b]pyrazol-1-yl]phenyl}-3-(1,1,1-trifluoro-2-methylpropan-2-yl)benzamide 1448316-72-0 C29H26F3N5O
N-{2,4-dimethyl-5-[6-(pyridin-3-yl)-1H-imidazo[1,2-b]pyrazol-1-yl]phenyl}-3-(1,1,1-trifluoro-2-methylpropan-2-yl)benzamide
—— 2-[4-[3-[1-(4-bromophenyl)-1-cyclopropylethyl]-1,2-oxazol-5-yl]pyrazol-1-yl]-N,N-dimethylethanamine 1448611-13-9 C21H25BrN4O
2-[4-[3-[1-(4-bromophenyl)-1-cyclopropylethyl]-1,2-oxazol-5-yl]pyrazol-1-yl]-N,N-dimethylethanamine
—— 8-(tert-butyldimethylsilyl)-2,3,6,7-tetrahydro-6-phenylfuro[2,3-f]isoindol-5-one 1411944-38-1 C22H27NO2Si
8-(tert-butyldimethylsilyl)-2,3,6,7-tetrahydro-6-phenylfuro[2,3-f]isoindol-5-one
—— 4-(4-hydroxy-pyridin-3-yl)-cyclohexanone 1252689-28-3 C11H13NO2
4-(4-hydroxy-pyridin-3-yl)-cyclohexanone
—— 5-(2,3-dihydrobenzofuran-5-yl)-3-(2-{4-[4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-2-propylphenyl]-1,4-diazepan-1-yl}-2-oxoethyl)-5-methylimidazolidine-2,4-dione 1254042-93-7 C31H34F6N4O5
5-(2,3-dihydrobenzofuran-5-yl)-3-(2-{4-[4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-2-propylphenyl]-1,4-diazepan-1-yl}-2-oxoethyl)-5-methylimidazolidine-2,4-dione
—— 2-{4-[2-(4-methyl-furazan-3-yl)-acetyl]-piperazin-1-yl}-N-pyridin-4-yl-benzamide 1253381-96-2 C21H22N6O3
2-{4-[2-(4-methyl-furazan-3-yl)-acetyl]-piperazin-1-yl}-N-pyridin-4-yl-benzamide
—— 3,4-dimethoxy-N-(2-oxo-2-{4-[2-(pyridin-3-ylcarbamoyl)-phenyl]-piperazin-1-yl}-ethyl)-benzamide 1253383-16-2 C27H29N5O5
3,4-dimethoxy-N-(2-oxo-2-{4-[2-(pyridin-3-ylcarbamoyl)-phenyl]-piperazin-1-yl}-ethyl)-benzamide
—— (4S,5R)-5-(2-hydroxy-2-methylpropyl)-4-methyloxazolidin-2-one 1453083-31-2 C8H15NO3
(4S,5R)-5-(2-hydroxy-2-methylpropyl)-4-methyloxazolidin-2-one
—— sodium 6-chloro-7-(4-(6'-methoxy-3,3'-bipyridin-6-ylcarbamoyl)phenoxy)chroman-4-carboxylate 1233694-44-4 C28H21ClN3O6*Na
sodium 6-chloro-7-(4-(6'-methoxy-3,3'-bipyridin-6-ylcarbamoyl)phenoxy)chroman-4-carboxylate
—— 5-methyl-imidazo[1,2-a]pyridine-2-carboxylic acid [5-(4-chloro-phenyl)-1H-benzoimidazol-2-yl]-amide 1254167-15-1 C22H16ClN5O
5-methyl-imidazo[1,2-a]pyridine-2-carboxylic acid [5-(4-chloro-phenyl)-1H-benzoimidazol-2-yl]-amide
—— (R)-2-[2-[4-(3-methyl-1,2,4-oxadiazol-5-yl)-phenyl]-1,4-oxazepan-4-yl]-6-(3-fluoropyridin-4-yl)-3-methylpyrimidin-4(3H)-one 1246455-22-0 C24H23FN6O3
(R)-2-[2-[4-(3-methyl-1,2,4-oxadiazol-5-yl)-phenyl]-1,4-oxazepan-4-yl]-6-(3-fluoropyridin-4-yl)-3-methylpyrimidin-4(3H)-one
—— 6-methyl-imidazo[2,1-b]thiazole-5-carboxylic acid {(1R,3S,4S)-2-[5-(2-fluoro-phenyl)-thiazole-4-carbonyl]-2-aza-bicyclo[2.2.1]hept-3-ylmethyl}-amide 1181571-50-5 C24H22FN5O2S2
6-methyl-imidazo[2,1-b]thiazole-5-carboxylic acid {(1R,3S,4S)-2-[5-(2-fluoro-phenyl)-thiazole-4-carbonyl]-2-aza-bicyclo[2.2.1]hept-3-ylmethyl}-amide
—— 5-chloro-N-[6-chloro-2,2-difluoro-4-(propan-2-ylcarbamoyl)-1,3-benzodioxol-5-yl]-2-(3-chloropyridin-2-yl)pyrazole-3-carboxamide 1103245-15-3 C20H14Cl3F2N5O4
5-chloro-N-[6-chloro-2,2-difluoro-4-(propan-2-ylcarbamoyl)-1,3-benzodioxol-5-yl]-2-(3-chloropyridin-2-yl)pyrazole-3-carboxamide
—— 5-(4-amino-6-methyl-1,3,5-triazin-2-yl)-N-(2-methoxyethyl)-6-((6-methoxy-3-pyridinyl)amino)-pyridine-3-carboxamide 1253573-69-1 C19H22N8O3
5-(4-amino-6-methyl-1,3,5-triazin-2-yl)-N-(2-methoxyethyl)-6-((6-methoxy-3-pyridinyl)amino)-pyridine-3-carboxamide
—— 5-(5-(6-(benzo[d]thiazol-6-ylamino)-4-(isopropylamino)pyridin-3-yl)-1,3,4-oxadiazol-2-yl)-2-fluorobenzenesulfonamide 1447225-53-7 C23H20FN7O3S2
5-(5-(6-(benzo[d]thiazol-6-ylamino)-4-(isopropylamino)pyridin-3-yl)-1,3,4-oxadiazol-2-yl)-2-fluorobenzenesulfonamide
—— (RS)-N-(4-cyano-benzyl)-2-(3-fluoro-biphenyl-4-yl)-2-methoxy-acetamide 1055904-64-7 C23H19FN2O2
(RS)-N-(4-cyano-benzyl)-2-(3-fluoro-biphenyl-4-yl)-2-methoxy-acetamide
—— 2-bromo-5-[(3-chloro-4-fluoro-phenyl)-4-chloro-phenylamino]-1-isopropyl-1H-imidazole-4-carboxylic acid ethyl ester 1448869-96-2 C22H21BrCl2FN3O2
2-bromo-5-[(3-chloro-4-fluoro-phenyl)-4-chloro-phenylamino]-1-isopropyl-1H-imidazole-4-carboxylic acid ethyl ester
—— (S)-3-hydroxy-2-{4-[(1S,3S)-3-((R)-1-naphthalen-1-yl-ethylamino)-cyclohexyl]-benzoylamino}-propionic acid benzyl ester 1157579-57-1 C35H38N2O4
(S)-3-hydroxy-2-{4-[(1S,3S)-3-((R)-1-naphthalen-1-yl-ethylamino)-cyclohexyl]-benzoylamino}-propionic acid benzyl ester
—— 4-(pyrrolidin-1-yl)butyl 2-(4-((2-amino-4-(butylamino)-6-methylpyrimidin-5-yl)methyl)-3-hydroxyphenyl)acetate 1158803-46-3 C26H39N5O3
4-(pyrrolidin-1-yl)butyl 2-(4-((2-amino-4-(butylamino)-6-methylpyrimidin-5-yl)methyl)-3-hydroxyphenyl)acetate
—— 5-(4-methoxy-phenyl)-2-methyl-oxazole-4-carboxylic acid [1-(5-acetyl-furan-2-ylmethyl)-1H-pyrazol-4-yl]-amide 1163256-32-3 C22H20N4O5
5-(4-methoxy-phenyl)-2-methyl-oxazole-4-carboxylic acid [1-(5-acetyl-furan-2-ylmethyl)-1H-pyrazol-4-yl]-amide
—— [6-(Pentane-2-sulfonyl)-5,6,7,8-tetrahydro-[2,6]naphthyridin-1-yl]-quinolin-3-yl-amine 1104023-34-8 C22H26N4O2S
[6-(Pentane-2-sulfonyl)-5,6,7,8-tetrahydro-[2,6]naphthyridin-1-yl]-quinolin-3-yl-amine
—— (R)-5-(1-(tert-butyldimethylsilanyloxy)-2-(3-(3-(4-(2-methylthiazol-4-yl-carbonyl)-1-oxa-4,9-diazaspiro[5.5]undec-9-yl)propoxy)benzylamino)ethyl)-8-hydroxyquinoline-2(1H)-one 1179338-77-2 C40H55N5O6SSi
(R)-5-(1-(tert-butyldimethylsilanyloxy)-2-(3-(3-(4-(2-methylthiazol-4-yl-carbonyl)-1-oxa-4,9-diazaspiro[5.5]undec-9-yl)propoxy)benzylamino)ethyl)-8-hydroxyquinoline-2(1H)-one
—— 2-(4-{3-[4-(2-dimethylaminoethylcarbamoyl)phenyl]ureido}phenyl)-5-ethoxy-6-morpholin-4-ylpyrimidine-4-carboxylic acid ethyl ester 1313717-93-9 C31H39N7O6
2-(4-{3-[4-(2-dimethylaminoethylcarbamoyl)phenyl]ureido}phenyl)-5-ethoxy-6-morpholin-4-ylpyrimidine-4-carboxylic acid ethyl ester
—— N-[(4-chlorophenyl)-methyl]-2-ethoxy-4-methyl-6-[(3R)-3-methyl-morpholin-4-yl]-pyridine-3-carboxylic acid amide 1373488-47-1 C21H26ClN3O3
N-[(4-chlorophenyl)-methyl]-2-ethoxy-4-methyl-6-[(3R)-3-methyl-morpholin-4-yl]-pyridine-3-carboxylic acid amide
—— (3S)-N-(1-{[5-chloro-3-(trifluoromethyl)-1-benzothiophen-2-yl]carbonyl}azetidin-3-yl)-1-(1,3-thiazol-4-ylcarbonyl)pyrrolidin-3-amine 1373524-44-7 C21H18ClF3N4O2S2
(3S)-N-(1-{[5-chloro-3-(trifluoromethyl)-1-benzothiophen-2-yl]carbonyl}azetidin-3-yl)-1-(1,3-thiazol-4-ylcarbonyl)pyrrolidin-3-amine
—— 3-[4-(2-ethoxy-ethylsulfanyl)-1H-pyrazol-3-yl]-pyridine 1073552-12-1 C12H15N3OS
3-[4-(2-ethoxy-ethylsulfanyl)-1H-pyrazol-3-yl]-pyridine
—— N-(4,4-dimethyl-pentyl)-2-(3-methoxy-propyl)-4-methyl-6-morpholin-4-yl-pyridine-3-carboxylic acid amide 1373489-27-0 C22H37N3O3
N-(4,4-dimethyl-pentyl)-2-(3-methoxy-propyl)-4-methyl-6-morpholin-4-yl-pyridine-3-carboxylic acid amide
—— (S)-2-(2-methoxymethyl-pyrrolidin-1-yl)-N-{4-[4-(5-methyl-1H-pyrazol-3-ylamino)-pyrrolo[2,1-f][1,2,4]triazin-2-ylsulfanyl]-phenyl}-acetamide 1315585-73-9 C24H28N8O2S
(S)-2-(2-methoxymethyl-pyrrolidin-1-yl)-N-{4-[4-(5-methyl-1H-pyrazol-3-ylamino)-pyrrolo[2,1-f][1,2,4]triazin-2-ylsulfanyl]-phenyl}-acetamide
—— 2-methyl-7-(((R)-3-phenylpyrrolidin-1-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one 1246082-68-7 C20H22N2O2
2-methyl-7-(((R)-3-phenylpyrrolidin-1-yl)methyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
—— 3-(2-(3-(3-(dimethylamino)propoxy)benzyl)-4-methyl-1-oxo-1,2-dihydroisoquinolin-6-yl)-4-methylbenzoic acid methyl ester 1070295-07-6 C31H34N2O4
3-(2-(3-(3-(dimethylamino)propoxy)benzyl)-4-methyl-1-oxo-1,2-dihydroisoquinolin-6-yl)-4-methylbenzoic acid methyl ester
—— 6-{(S)-1-[(3R,4S)-4-(3,4-difluorophenyl)-1-(6-methylpyridazine-4-carbonyl)pyrrolidin-3-yl]ethoxy}nicotinonitrile 1115961-41-5 C24H21F2N5O2
6-{(S)-1-[(3R,4S)-4-(3,4-difluorophenyl)-1-(6-methylpyridazine-4-carbonyl)pyrrolidin-3-yl]ethoxy}nicotinonitrile
—— 2-morpholinoethyl (S)-2-(4-{[4-(1-(4-chlorophenyl)cyclopropylamino)-6-(2,2,2-trifluoroethoxy)-1,3,5-triazin-2-yl]amino}benzamido)-3-(2-(dimethylamino)-2-oxoacetamido)propanoate 1449396-97-7 C34H39ClF3N9O7
2-morpholinoethyl (S)-2-(4-{[4-(1-(4-chlorophenyl)cyclopropylamino)-6-(2,2,2-trifluoroethoxy)-1,3,5-triazin-2-yl]amino}benzamido)-3-(2-(dimethylamino)-2-oxoacetamido)propanoate
—— (4-{6-amino-5-[1-(5-fluoro-2-methoxyphenyl)ethoxy]pyridin-3-yl}-1,3-thiazol-5-yl)methanol 1346814-67-2 C18H18FN3O3S
(4-{6-amino-5-[1-(5-fluoro-2-methoxyphenyl)ethoxy]pyridin-3-yl}-1,3-thiazol-5-yl)methanol
—— 2-cyclopropyl-1-{[3-(methoxycarbonyl)phenyl]sulfonyl}-1,2,2',3',5',6'-hexahydrospiro[indole-3,4'-thiopyran]-5-carboxylic acid 1',1'-dioxide 1448039-37-9 C24H25NO8S2
2-cyclopropyl-1-{[3-(methoxycarbonyl)phenyl]sulfonyl}-1,2,2',3',5',6'-hexahydrospiro[indole-3,4'-thiopyran]-5-carboxylic acid 1',1'-dioxide
—— 6-(2,6-difluoro-phenyl)-N-(5-fluoro-pyridin-3-yl)-N'-isopropyl-[1,3,5]triazine-2,4-diamine 1446504-57-9 C17H15F3N6
6-(2,6-difluoro-phenyl)-N-(5-fluoro-pyridin-3-yl)-N'-isopropyl-[1,3,5]triazine-2,4-diamine
—— 2-chloro-3-(4-methoxyphenyl)-5-methyl-5-(m-tolyl)-7H-thieno[2,3-b]pyridine-4,6-dione 1313503-46-6 C22H18ClNO3S
2-chloro-3-(4-methoxyphenyl)-5-methyl-5-(m-tolyl)-7H-thieno[2,3-b]pyridine-4,6-dione
—— (2R,6S,13aS,14aR,16aS,Z)-2-(8-fluoro-3-methylquinoxalin-2-yloxy)-6-(1-methyl-1H-pyrazole-3-carboxamido)-N-(1-methylcyclopropylsulfonyl)-5,16-dioxo-1,2,3,5,6,7,8,9,10,11,13a,14,14a,15,16,16a-hexadecahydrocyclopropa[e]pyrrolo[1,2-a][1,4]diazacyclopentadecine-14a-carboxamide 1352301-28-0 C36H43FN8O7S
(2R,6S,13aS,14aR,16aS,Z)-2-(8-fluoro-3-methylquinoxalin-2-yloxy)-6-(1-methyl-1H-pyrazole-3-carboxamido)-N-(1-methylcyclopropylsulfonyl)-5,16-dioxo-1,2,3,5,6,7,8,9,10,11,13a,14,14a,15,16,16a-hexadecahydrocyclopropa[e]pyrrolo[1,2-a][1,4]diazacyclopentadecine-14a-carboxamide
—— 2-[4-ethoxy-2-methyl-5-(1-methylethyl)phenyl]-N-[3-methoxy-4-(3-methyl-1H-1,2,4-triazol-1-yl)phenyl]-3-methyl-2H-indazol-7-amine 1259032-43-3 C30H34N6O2
2-[4-ethoxy-2-methyl-5-(1-methylethyl)phenyl]-N-[3-methoxy-4-(3-methyl-1H-1,2,4-triazol-1-yl)phenyl]-3-methyl-2H-indazol-7-amine