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中文名称 英文名称 CAS号 化学式 结构式图片
—— pyrimid-2-yl-Pyr-N(Ph(3-F))Phg(2-Cl)-NHcHex 1448345-74-1 C29H29ClFN5O3
pyrimid-2-yl-Pyr-N(Ph(3-F))Phg(2-Cl)-NHcHex
—— 5-{4-[2-(4-fluoro-1H-indol-2-yl)-3-methybutan-2-yl]phenyl}pyrimidin-2-amine 1448608-82-9 C23H23FN4
5-{4-[2-(4-fluoro-1H-indol-2-yl)-3-methybutan-2-yl]phenyl}pyrimidin-2-amine
—— 4-ethyl-N-(4-methyl-2-phenylpentyl)-2-pyrimidin-2-yl-1,3-thiazole-5-carboxamide 1104272-73-2 C22H26N4OS
4-ethyl-N-(4-methyl-2-phenylpentyl)-2-pyrimidin-2-yl-1,3-thiazole-5-carboxamide
—— toluene-4-sulfonic acid 2-[1-(3-methoxy-propionyl)-piperidin-4-yl]-ethyl ester 1156468-27-7 C18H27NO5S
toluene-4-sulfonic acid 2-[1-(3-methoxy-propionyl)-piperidin-4-yl]-ethyl ester
—— 6-(5-hexyl-2-oxo-1,3-oxazolidin-3-yl)-3,4-dihydroisoquinolin-1(2H)-one 1174336-85-6 C18H24N2O3
6-(5-hexyl-2-oxo-1,3-oxazolidin-3-yl)-3,4-dihydroisoquinolin-1(2H)-one
—— 6-(benzothiazol-2-yloxy)-1H-indole-2-carbaldehyde 1256106-54-3 C16H10N2O2S
6-(benzothiazol-2-yloxy)-1H-indole-2-carbaldehyde
—— 1-(2-azatricyclo[3.3.1.1<sup>3</sup>'<sup>7</sup>]dec-2-yl)-3-(1,3-benzothiazol-2-yl)butan-1-one 1448697-55-9 C20H24N2OS
1-(2-azatricyclo[3.3.1.1<sup>3</sup>'<sup>7</sup>]dec-2-yl)-3-(1,3-benzothiazol-2-yl)butan-1-one
—— 2-({4-cyclopropyl-6-[4-(4-hydroxypiperidin-1-yl)phenyl]pyridin-2-yl}amino)pyridine-4-carbonitrile hydrochloride 1374140-49-4 C25H25N5O*ClH
2-({4-cyclopropyl-6-[4-(4-hydroxypiperidin-1-yl)phenyl]pyridin-2-yl}amino)pyridine-4-carbonitrile hydrochloride
—— 1-(1H-indol-5-yl)-6-[3-(4-methylpiperazin-1-ylmethyl)phenyl]-1,3-dihydroimidazo[4,5-b]pyrazin-2-one 1351477-08-1 C25H25N7O
1-(1H-indol-5-yl)-6-[3-(4-methylpiperazin-1-ylmethyl)phenyl]-1,3-dihydroimidazo[4,5-b]pyrazin-2-one
—— [2-(Hydroxymethyl)-4,5-bis(2-methoxyethoxy)phenyl]methanol 1107625-50-2 C14H22O6
[2-(Hydroxymethyl)-4,5-bis(2-methoxyethoxy)phenyl]methanol
—— 2-[4-[4-chloro-3-(6-chloro-1H-benzimidazol-2-yl)phenyl]piperazin-1-yl]-N-methylacetamide 1160832-86-9 C20H21Cl2N5O
2-[4-[4-chloro-3-(6-chloro-1H-benzimidazol-2-yl)phenyl]piperazin-1-yl]-N-methylacetamide
—— 1'-(4-tert-butyl-benzenesulfonyl)-2,3-dihydrospiro[(2-oxo)-indole-3,4'-piperidine]-1-yl-acetic acid methyl ester 1151786-50-3 C25H30N2O5S
1'-(4-tert-butyl-benzenesulfonyl)-2,3-dihydrospiro[(2-oxo)-indole-3,4'-piperidine]-1-yl-acetic acid methyl ester
—— 1-(2-{4-[4-fluoro-2-(2-methoxypyrimidin-5-yl)phenyl]piperazin-1-yl}-2-oxoethyl)-1,3-dihydro-2H-benzimidazol-2-one 1253938-23-6 C24H23FN6O3
1-(2-{4-[4-fluoro-2-(2-methoxypyrimidin-5-yl)phenyl]piperazin-1-yl}-2-oxoethyl)-1,3-dihydro-2H-benzimidazol-2-one
—— 2-(3,5-dimethyl-pyrazol-1-yl)-1-(4-{2-[(1S,4S)-2-(2-oxa-5-aza-bicyclo[2.2.1]hept-5-yl)pyrimidin-5-yl]phenyl}piperazin-1-yl)ethanone 1253937-82-4 C26H31N7O2
2-(3,5-dimethyl-pyrazol-1-yl)-1-(4-{2-[(1S,4S)-2-(2-oxa-5-aza-bicyclo[2.2.1]hept-5-yl)pyrimidin-5-yl]phenyl}piperazin-1-yl)ethanone
—— 2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(4-fluoro-2-{2-[4-(methylsulfonyl)piperidin-1-yl]pyrimidin-5-yl}phenyl)piperazin-1-yl]ethanone 1253938-13-4 C27H34FN7O3S
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(4-fluoro-2-{2-[4-(methylsulfonyl)piperidin-1-yl]pyrimidin-5-yl}phenyl)piperazin-1-yl]ethanone
—— 1-[4-(4-Aminopiperidin-1-yl)-2-methoxyphenyl]-9-(6-methoxypyridin-3-yl)benzo[h][1,6]naphthyridin-2-one 1222998-88-0 C30H29N5O3
1-[4-(4-Aminopiperidin-1-yl)-2-methoxyphenyl]-9-(6-methoxypyridin-3-yl)benzo[h][1,6]naphthyridin-2-one
—— 5-[7-[(5R)-5-[(S)-hydroxy(phenyl)methyl]-5-methyl-4H-1,2-oxazol-3-yl]-4-oxo-3-phenylquinazolin-2-yl]pentanoic acid 1373277-60-1 C30H29N3O5
5-[7-[(5R)-5-[(S)-hydroxy(phenyl)methyl]-5-methyl-4H-1,2-oxazol-3-yl]-4-oxo-3-phenylquinazolin-2-yl]pentanoic acid
—— (4-Methylpiperazin-1-yl)-[3-[[2-methyl-4-[3-[4-(trifluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]pyrrol-1-yl]methyl]phenyl]methanone 1225380-02-8 C27H26F3N5O3
(4-Methylpiperazin-1-yl)-[3-[[2-methyl-4-[3-[4-(trifluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl]pyrrol-1-yl]methyl]phenyl]methanone
—— N-tert-butyl-2-{[1-(5'-chloro-3-methyl-2,4'-bipyridin-2'-yl)piperidin-4-yl]oxy}acetamide 1373614-54-0 C22H29ClN4O2
N-tert-butyl-2-{[1-(5'-chloro-3-methyl-2,4'-bipyridin-2'-yl)piperidin-4-yl]oxy}acetamide
—— 1-(5-hydroxy-2-azatricyclo[3.3.1.1<sup>3</sup>'<sup>7</sup>]dec-2-yl)-3-(5-methoxy-1H-indol-3-yl)butan-1-one 1448697-59-3 C22H28N2O3
1-(5-hydroxy-2-azatricyclo[3.3.1.1<sup>3</sup>'<sup>7</sup>]dec-2-yl)-3-(5-methoxy-1H-indol-3-yl)butan-1-one
—— (E)-6-amino-9-((1-(4-(dimethylamino)but-2-enoyl)piperidin-4-yl)methyl)-7-(4-phenoxyphenyl)-7H-purin-8(9H)-one 1448445-07-5 C29H33N7O3
(E)-6-amino-9-((1-(4-(dimethylamino)but-2-enoyl)piperidin-4-yl)methyl)-7-(4-phenoxyphenyl)-7H-purin-8(9H)-one
—— 2-[(3-Aminopyrazol-1-yl)methyl]pyridin-3-ol 1372892-00-6 C9H10N4O
2-[(3-Aminopyrazol-1-yl)methyl]pyridin-3-ol
—— 2-[1-(2,2-dimethylpropyl)-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-4-(hexahydro-4H-furo[3,2-b]pyrrol-4-ylmethyl)benzonitrile 1352423-36-9 C26H31N5O2
2-[1-(2,2-dimethylpropyl)-3-methyl-2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-5-yl]-4-(hexahydro-4H-furo[3,2-b]pyrrol-4-ylmethyl)benzonitrile
—— 3-({6-[(2-hydroxy-3-methylbenzyl)amino]-9-(benzyl)-9H-purin-2-yl}amino)-2-methyl-pentan-2-ol 1257695-51-4 C26H32N6O2
3-({6-[(2-hydroxy-3-methylbenzyl)amino]-9-(benzyl)-9H-purin-2-yl}amino)-2-methyl-pentan-2-ol
—— (2S)-N-[(1S)-1-(2-chlorophenyl)-2-[(3,3-difluorocyclobutyl)amino]-2-oxoethyl]-N-(3-fluorophenyl)-5-oxo-1-(1,3-thiazol-2-yl)pyrrolidine-2-carboxamide 1448345-83-2 C26H22ClF3N4O3S
(2S)-N-[(1S)-1-(2-chlorophenyl)-2-[(3,3-difluorocyclobutyl)amino]-2-oxoethyl]-N-(3-fluorophenyl)-5-oxo-1-(1,3-thiazol-2-yl)pyrrolidine-2-carboxamide
—— 1-[2-[2-[2-[Bis(2-hydroxydodecyl)amino]ethoxy]ethoxy]ethylamino]dodecan-2-ol 1220890-35-6 C42H88N2O5
1-[2-[2-[2-[Bis(2-hydroxydodecyl)amino]ethoxy]ethoxy]ethylamino]dodecan-2-ol
—— 1-(4-(3-ethyl-4-(methyl(1-methyl-1H-imidazo[4,5-c]pyridin-6-yl)amino)phenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl)cyclopropanecarbonitrile 1449668-16-9 C26H28N6O
1-(4-(3-ethyl-4-(methyl(1-methyl-1H-imidazo[4,5-c]pyridin-6-yl)amino)phenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl)cyclopropanecarbonitrile
—— (R)-N-{1-[6-(thiazolo[4,5-b]pyridin-2-yloxy)-benzofuran-3-ylmethyl]-pyrrolidin-3-yl}-acetamide 1256105-32-4 C21H20N4O3S
(R)-N-{1-[6-(thiazolo[4,5-b]pyridin-2-yloxy)-benzofuran-3-ylmethyl]-pyrrolidin-3-yl}-acetamide
—— 5-[2-(3-fluorophenyl)-1-methyl-1H-benzimidazol-5-yl]-3-isopropyl-6-methyl-3,6-dihydro-2H-1,3,4-thiadiazin-2-one 1151821-34-9 C21H21FN4OS
5-[2-(3-fluorophenyl)-1-methyl-1H-benzimidazol-5-yl]-3-isopropyl-6-methyl-3,6-dihydro-2H-1,3,4-thiadiazin-2-one
—— [(S)-2-((S)-2-carbamoylpyrrolidin-1-yl)-1-(2-fluoro-4-{(R)-3-[1-(3-isopropyl-[1,2,4]oxadiazol-5-yl)piperidin-4-yl]butoxy}phenyl)-2-oxoethyl]carbamic acid tert-butyl ester 1131872-31-5 C32H47FN6O6
[(S)-2-((S)-2-carbamoylpyrrolidin-1-yl)-1-(2-fluoro-4-{(R)-3-[1-(3-isopropyl-[1,2,4]oxadiazol-5-yl)piperidin-4-yl]butoxy}phenyl)-2-oxoethyl]carbamic acid tert-butyl ester
—— 5-[2-(benzyloxy)ethoxy]pyrazin-2-amine 1174229-70-9 C13H15N3O2
5-[2-(benzyloxy)ethoxy]pyrazin-2-amine
—— 4-[3-(1H-benzimidazol-2-yl)-4-chlorophenyl]-N-phenylpiperazine-1-carboxamide 1160832-76-7 C24H22ClN5O
4-[3-(1H-benzimidazol-2-yl)-4-chlorophenyl]-N-phenylpiperazine-1-carboxamide
—— 2-(3-methoxyphenyl)-4-(4-methoxyphenyl)-1H-imidazole-5-carboxamide 1082440-05-8 C18H17N3O3
2-(3-methoxyphenyl)-4-(4-methoxyphenyl)-1H-imidazole-5-carboxamide
—— N-(4-fluorobenzyl)-4-ethyl-2-pyrimidin-2-yl-1,3-thiazole-5-carboxamide 1104272-55-0 C17H15FN4OS
N-(4-fluorobenzyl)-4-ethyl-2-pyrimidin-2-yl-1,3-thiazole-5-carboxamide
—— N-(2,4-difluorobenzyl)-4-ethyl-2-pyrimidin-2-yl-1,3-thiazole-5-carboxamide 1104271-80-8 C17H14F2N4OS
N-(2,4-difluorobenzyl)-4-ethyl-2-pyrimidin-2-yl-1,3-thiazole-5-carboxamide
—— {1-[6-(thiazolo[4,5-b]pyridin-2-yloxy)-benzofuran-3-ylmethyl]-piperidin-4-yl}-carbamic acid tert-butyl ester 1256103-88-4 C25H28N4O4S
{1-[6-(thiazolo[4,5-b]pyridin-2-yloxy)-benzofuran-3-ylmethyl]-piperidin-4-yl}-carbamic acid tert-butyl ester
—— 4-{4-[(2-tert-butylphenoxy)methyl]piperidin-1-yl}-4-oxobutanoic acid 1146958-07-7 C20H29NO4
4-{4-[(2-tert-butylphenoxy)methyl]piperidin-1-yl}-4-oxobutanoic acid
—— 1-(2,4-dichloro-phenyl)-4-fluoromethyl-5-(4-fluoro-phenyl)-4,5-dihydro-1H-pyrazole-3-carboxylic acid piperidin-1-ylamide 1026860-19-4 C22H22Cl2F2N4O
1-(2,4-dichloro-phenyl)-4-fluoromethyl-5-(4-fluoro-phenyl)-4,5-dihydro-1H-pyrazole-3-carboxylic acid piperidin-1-ylamide
—— N-[4-(2,3-dihydro-1,4-benzodioxin-2-yl)benzyl]-2-methyl-1-(pyrrolidin-1-yl)propan-2-amine 1400794-21-9 C23H30N2O2
N-[4-(2,3-dihydro-1,4-benzodioxin-2-yl)benzyl]-2-methyl-1-(pyrrolidin-1-yl)propan-2-amine
—— 1-amino-7-(3-fluorophenyl)-N-[(3-methoxyphenyl)methyl]isoquinoline-4-carboxamide 1449277-64-8 C24H20FN3O2
1-amino-7-(3-fluorophenyl)-N-[(3-methoxyphenyl)methyl]isoquinoline-4-carboxamide
—— 5-[3-(4-fluorophenyl)-7-[5-[(R)-methoxy(phenyl)methyl]-1,2-oxazol-3-yl]-4-oxoquinazolin-2-yl]hexanoic acid 1373275-84-3 C31H28FN3O5
5-[3-(4-fluorophenyl)-7-[5-[(R)-methoxy(phenyl)methyl]-1,2-oxazol-3-yl]-4-oxoquinazolin-2-yl]hexanoic acid
—— 2-[1-{4-[2-(4-cyanopiperidin-1-yl)ethyl]phenyl}-3-(4-fluoro-3-methoxyphenyl)-5-oxo-1,5-dihydro-4H-1,2,4-triazol-4-yl]-N-(propan-2-yl)acetamide 1370446-62-0 C28H33FN6O3
2-[1-{4-[2-(4-cyanopiperidin-1-yl)ethyl]phenyl}-3-(4-fluoro-3-methoxyphenyl)-5-oxo-1,5-dihydro-4H-1,2,4-triazol-4-yl]-N-(propan-2-yl)acetamide
—— N-(5-tert-butyl-1,2-oxazol-3-yl)-3-[4-[5-[4-(dimethylamino)piperidin-1-yl]pyridin-3-yl]triazol-1-yl]-4-methylbenzamide 1334683-86-1 C29H36N8O2
N-(5-tert-butyl-1,2-oxazol-3-yl)-3-[4-[5-[4-(dimethylamino)piperidin-1-yl]pyridin-3-yl]triazol-1-yl]-4-methylbenzamide
—— 2-[4-(1-tert-butoxycarbonylamino-cyclobutyl)-phenyl]-8-methyl-3-phenyl-imidazo[1,2-a]pyridine-6-carboxylic acid methyl ester 1356001-69-8 C31H33N3O4
2-[4-(1-tert-butoxycarbonylamino-cyclobutyl)-phenyl]-8-methyl-3-phenyl-imidazo[1,2-a]pyridine-6-carboxylic acid methyl ester
—— 5-[(2,4-dichlorophenoxy)methyl]-3-phenyl-1,3-oxazolidin-2-one 1174337-75-7 C16H13Cl2NO3
5-[(2,4-dichlorophenoxy)methyl]-3-phenyl-1,3-oxazolidin-2-one
—— t-butyl dicyclohexylphosphinyl acetate 1186034-91-2 C18H33O3P
t-butyl dicyclohexylphosphinyl acetate
—— 2-[2-chloro-5-[4-(1-pyridin-4-ylethyl)piperazin-1-yl]phenyl]-1H-benzimidazole 1160830-05-6 C24H24ClN5
2-[2-chloro-5-[4-(1-pyridin-4-ylethyl)piperazin-1-yl]phenyl]-1H-benzimidazole
—— 2-(4,4-difluorocyclohexyl)ethyl 4-methylbenzenesulfonate 1156468-41-5 C15H20F2O3S
2-(4,4-difluorocyclohexyl)ethyl 4-methylbenzenesulfonate
—— 1-oxo-2-(4-trifluoromethoxy-phenyl)-2,8-diaza-spiro[4.5]decane-8-carboxylic acid isobutyl-methyl-amide 1255714-85-2 C21H28F3N3O3
1-oxo-2-(4-trifluoromethoxy-phenyl)-2,8-diaza-spiro[4.5]decane-8-carboxylic acid isobutyl-methyl-amide
—— 4-methyl-N-{4-methyl-2-[4-(trifluoromethyl)phenyl]pentyl}-2-pyrimidin-2-yl-1,3-thiazole-5-carboxamide 1104273-69-9 C22H23F3N4OS
4-methyl-N-{4-methyl-2-[4-(trifluoromethyl)phenyl]pentyl}-2-pyrimidin-2-yl-1,3-thiazole-5-carboxamide