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—— 2-[1-[(6-amino-5-bromopyrimidine-4-carbonyl)amino]ethyl]-N-[2-(2,2,2-trifluoroethoxy)-5-(trifluoromethyl)phenyl]-1,3-thiazole-5-carboxamide 1096709-42-0 C20H15BrF6N6O3S
2-[1-[(6-amino-5-bromopyrimidine-4-carbonyl)amino]ethyl]-N-[2-(2,2,2-trifluoroethoxy)-5-(trifluoromethyl)phenyl]-1,3-thiazole-5-carboxamide
—— 2-Methylmercapto-5-methoxy-4-methyl-pyrimidin 19175-01-0 C7H10N2OS
2-Methylmercapto-5-methoxy-4-methyl-pyrimidin
—— (3R)-3-{(1S,4S)-1,4-dimethyl-2-[(trimethylsilyl)oxy]-cyclohex-2-en-1-yl}butyl benzoate 1146476-04-1 C22H34O3Si
(3R)-3-{(1S,4S)-1,4-dimethyl-2-[(trimethylsilyl)oxy]-cyclohex-2-en-1-yl}butyl benzoate
—— {3-[7-(1-benzyl-1,2,3,6-tetrahydropyridin-4-yl)-4-morpholin-4-yl-5H-pyrrolo[3,2-d]pyrimidin-2-yl]phenyl}methanol 1155810-88-0 C29H31N5O2
{3-[7-(1-benzyl-1,2,3,6-tetrahydropyridin-4-yl)-4-morpholin-4-yl-5H-pyrrolo[3,2-d]pyrimidin-2-yl]phenyl}methanol
—— 2-amino-5-(1H-indol-3-yl)-5-(2-oxopropyl)-1H-imidazol-4(5H)-one 1146981-75-0 C14H14N4O2
2-amino-5-(1H-indol-3-yl)-5-(2-oxopropyl)-1H-imidazol-4(5H)-one
—— 2-methoxy-9-(2-methylphenyl)-7-(trifluoromethyl)imidazo[1,5-a]pyrido[3,2-e]pyrazin-6-amine 1156499-70-5 C18H14F3N5O
2-methoxy-9-(2-methylphenyl)-7-(trifluoromethyl)imidazo[1,5-a]pyrido[3,2-e]pyrazin-6-amine
—— [(R)-3-(6-fluoro-benzothiazol-2-ylamino)-pyrrolidin-1-yl]-(5-methyl-3-phenyl-isoxazol-4-yl)-methanone 1163122-14-2 C22H19FN4O2S
[(R)-3-(6-fluoro-benzothiazol-2-ylamino)-pyrrolidin-1-yl]-(5-methyl-3-phenyl-isoxazol-4-yl)-methanone
—— 2-[3-(cyclohexen-1-yl)-5-(1H-pyrazolo[3,4-b]pyridin-4-yl)phenyl]-2-methylpropan-1-amine 1160498-66-7 C22H26N4
2-[3-(cyclohexen-1-yl)-5-(1H-pyrazolo[3,4-b]pyridin-4-yl)phenyl]-2-methylpropan-1-amine
—— N'-[(2Z)-3-[4-(difluoromethoxy)phenyl]-5-methyl-1,3-thiazol-2(3H)-ylidene]-N,N-diethylurea 1163264-91-2 C16H19F2N3O2S
N'-[(2Z)-3-[4-(difluoromethoxy)phenyl]-5-methyl-1,3-thiazol-2(3H)-ylidene]-N,N-diethylurea
—— [1-(5-acetyl-furan-2-ylmethyl)-1H-pyrazol-4-yl]-carbamic acid 2-chloro-4-fluoro-benzyl ester 1163255-91-1 C18H15ClFN3O4
[1-(5-acetyl-furan-2-ylmethyl)-1H-pyrazol-4-yl]-carbamic acid 2-chloro-4-fluoro-benzyl ester
—— 5-bromo-2-(ethylaminomethyl)-3,4-dihydro-1H-naphthalen-2-amine 1221136-10-2 C13H19BrN2
5-bromo-2-(ethylaminomethyl)-3,4-dihydro-1H-naphthalen-2-amine
—— (R)-3-amino-4-(4-(6-aminopyridin-3-yl)phenyl)-1-((R)-3-(1-(3-methoxypropyl)-5-methyl-3-(trifluoromethyl)-1H-pyrrol-2-yl)piperidin-1-yl)butan-1-one 1246359-90-9 C30H38F3N5O2
(R)-3-amino-4-(4-(6-aminopyridin-3-yl)phenyl)-1-((R)-3-(1-(3-methoxypropyl)-5-methyl-3-(trifluoromethyl)-1H-pyrrol-2-yl)piperidin-1-yl)butan-1-one
—— 3-Chloro-2,5-dimethoxy-bicyclo[4.2.0]octa-1,3,5-triene-7-carboxylic acid methyl ester 110137-91-2 C12H13ClO4
3-Chloro-2,5-dimethoxy-bicyclo[4.2.0]octa-1,3,5-triene-7-carboxylic acid methyl ester
—— (9R,9aS,12aR,13S)9,13-diphenyl-11-(2-(pyridin-3-yloxy)phenyl)-12a,13-dihydro-9H-9,13-methanophenanthro[9,10-f]isoindole-10,12,14(9aH,11H)-trione 1438384-23-6 C44H28N2O4
(9R,9aS,12aR,13S)9,13-diphenyl-11-(2-(pyridin-3-yloxy)phenyl)-12a,13-dihydro-9H-9,13-methanophenanthro[9,10-f]isoindole-10,12,14(9aH,11H)-trione
—— ethyl (6-((6-methoxy-2-methylpyridin-3-yl)methoxy)-1-benzothiophen-3-yl)acetate 1452475-34-1 C20H21NO4S
ethyl (6-((6-methoxy-2-methylpyridin-3-yl)methoxy)-1-benzothiophen-3-yl)acetate
—— (S)-3-amino-1-(6-((2-propylpentyl)oxy)pyridin-2-yl)propan-1-ol 1448434-88-5 C16H28N2O2
(S)-3-amino-1-(6-((2-propylpentyl)oxy)pyridin-2-yl)propan-1-ol
—— ((4R,5S)-5-((1R,2R)-1-(benzyloxycarbonylamino)-2-hydroxypent-4-enyl)-2,2-dimethyl-1,3-dioxolan-4-yl)methyl benzoate 1148122-93-3 C26H31NO7
((4R,5S)-5-((1R,2R)-1-(benzyloxycarbonylamino)-2-hydroxypent-4-enyl)-2,2-dimethyl-1,3-dioxolan-4-yl)methyl benzoate
—— (2E)-N-[(1S)-1-benzyl-2-methoxyethyl]-3-(1H-pyrrolo[2,3-b]pyridin-3-yl)acrylamide 1160981-55-4 C20H21N3O2
(2E)-N-[(1S)-1-benzyl-2-methoxyethyl]-3-(1H-pyrrolo[2,3-b]pyridin-3-yl)acrylamide
—— 4-(2-{[6-((S)-3-methoxypyrrolidin-1-yl)-2-phenylpyrimidine-4-carbonyl]amino}-2-phosphonoacetyl)piperazine-1-carboxylic acid butyl ester 1159500-89-6 C27H37N6O8P
4-(2-{[6-((S)-3-methoxypyrrolidin-1-yl)-2-phenylpyrimidine-4-carbonyl]amino}-2-phosphonoacetyl)piperazine-1-carboxylic acid butyl ester
—— (2,6-dimethoxy-phenyl)-[(R)-3-(6-fluoro-quinoxalin-2-ylamino)-pyrrolidin-1-yl]-methanone 1163122-08-4 C21H21FN4O3
(2,6-dimethoxy-phenyl)-[(R)-3-(6-fluoro-quinoxalin-2-ylamino)-pyrrolidin-1-yl]-methanone
—— 7-methoxy-3,4-dimethyl-1-propyl-imidazo[1,5-a]quinoxaline 1159794-12-3 C16H19N3O
7-methoxy-3,4-dimethyl-1-propyl-imidazo[1,5-a]quinoxaline
—— 5-[5-(Quinolin-3-ylamino)-3,4-dihydro-1H-[2,6]naphthyridine-2-sulfonyl]-furan-2-carboxylic acid methyl ester 1104023-05-3 C23H20N4O5S
5-[5-(Quinolin-3-ylamino)-3,4-dihydro-1H-[2,6]naphthyridine-2-sulfonyl]-furan-2-carboxylic acid methyl ester
—— 7-[(2,6-dimethylbenzyl)oxy]-4-[4-(methylsulfonyl)phenyl]-2-naphthoic acid 1160271-18-0 C27H24O5S
7-[(2,6-dimethylbenzyl)oxy]-4-[4-(methylsulfonyl)phenyl]-2-naphthoic acid
—— 1-(1-benzyl-3-oxo-2,3-dihydro-1H-indazol-5-yl)-3-(2-methoxy-phenyl)-urea 1160165-48-9 C22H20N4O3
1-(1-benzyl-3-oxo-2,3-dihydro-1H-indazol-5-yl)-3-(2-methoxy-phenyl)-urea
—— N-cyclohexyl-5-methyl-4-(1H-pyrazol-4-yl)thiazol-2-amine 1105039-04-0 C13H18N4S
N-cyclohexyl-5-methyl-4-(1H-pyrazol-4-yl)thiazol-2-amine
—— 3-{(Z)-1-[4-((imidazol-4-yl)methyl)anilino]-1-phenylmethylidene}-2-indolinone 1139221-00-3 C25H20N4O
3-{(Z)-1-[4-((imidazol-4-yl)methyl)anilino]-1-phenylmethylidene}-2-indolinone
—— 8-(2-chloro-6-fluorophenyl)-5,6,7,8-tetrahydro-N-[4-(2-methyl-4-pyridinyl)phenyl]-[1,2,4]triazolo[1,5-a]pyridin-2-amine 1314787-50-2 C24H21ClFN5
8-(2-chloro-6-fluorophenyl)-5,6,7,8-tetrahydro-N-[4-(2-methyl-4-pyridinyl)phenyl]-[1,2,4]triazolo[1,5-a]pyridin-2-amine
—— (3-{7-[(diethylamino)methyl]-4-morpholin-4-yl-5H-pyrrolo[3,2-d]pyrimidin-2-yl}phenyl)methanol 1155810-70-0 C22H29N5O2
(3-{7-[(diethylamino)methyl]-4-morpholin-4-yl-5H-pyrrolo[3,2-d]pyrimidin-2-yl}phenyl)methanol
—— N-((1S,2R)-2-hydroxy-cyclopentyl)-6-(5-methyl-3-phenyl-isoxazol-4-ylmethoxy)-nicotinamide 1159601-59-8 C22H23N3O4
N-((1S,2R)-2-hydroxy-cyclopentyl)-6-(5-methyl-3-phenyl-isoxazol-4-ylmethoxy)-nicotinamide
—— 4-[6-(1H-pyrazolo[3,4-b]pyridin-4-yl)pyridin-2-yl]piperidine-4-carbonitrile 1160498-01-0 C17H16N6
4-[6-(1H-pyrazolo[3,4-b]pyridin-4-yl)pyridin-2-yl]piperidine-4-carbonitrile
—— 6-methyl-8-(4-nitrobenzyl)-3-phenylpyrimido[5,4-e][1,2,4]triazine-5,7(6H,8H)-dione 1207377-93-2 C19H14N6O4
6-methyl-8-(4-nitrobenzyl)-3-phenylpyrimido[5,4-e][1,2,4]triazine-5,7(6H,8H)-dione
—— (1,5-naphthyridin-2-yl)methanamine 1060816-75-2 C9H9N3
(1,5-naphthyridin-2-yl)methanamine
—— 1-methylethyl 2-(4-{[3-({[4-(1-methylethyl)phenyl]methyl}oxy)phenyl]methyl}-1-piperazinyl)-3-pyridinecarboxylate 1315558-58-7 C30H37N3O3
1-methylethyl 2-(4-{[3-({[4-(1-methylethyl)phenyl]methyl}oxy)phenyl]methyl}-1-piperazinyl)-3-pyridinecarboxylate
—— (1-methyl-3-sulfamoyl-1H-indol-7-yloxy)-acetic acid ethyl ester 1158210-83-3 C13H16N2O5S
(1-methyl-3-sulfamoyl-1H-indol-7-yloxy)-acetic acid ethyl ester
—— (2S)-2-((2-((5-cyclopropyl-1H-pyrazol-3-yl)amino)pyrrolo[2,1-f][1,2,4]triazin-4-yl)amino)-3-methyl-1-butanol 1026146-36-0 C17H23N7O
(2S)-2-((2-((5-cyclopropyl-1H-pyrazol-3-yl)amino)pyrrolo[2,1-f][1,2,4]triazin-4-yl)amino)-3-methyl-1-butanol
—— 5-nitro-6-(2,4,5-trichlorophenylamino)pyridin-2-ol 1217350-22-5 C11H6Cl3N3O3
5-nitro-6-(2,4,5-trichlorophenylamino)pyridin-2-ol
—— 4-(6-methoxy-4-piperazin-1-yl-2-naphthyl)-N-(3-methoxypropyl)pyrimidin-2-amine 1313486-97-3 C23H29N5O2
4-(6-methoxy-4-piperazin-1-yl-2-naphthyl)-N-(3-methoxypropyl)pyrimidin-2-amine
—— N-(4-bromophenyl)-8-hydroxy-N-methylquinoline-7-carboxamide 1313602-03-7 C17H13BrN2O2
N-(4-bromophenyl)-8-hydroxy-N-methylquinoline-7-carboxamide
—— N-[(2R,3S)-2-(4-bromophenyl)tetrahydro-2H-pyran-3-yl]propane-2-sulfonamide 1219633-46-1 C14H20BrNO3S
N-[(2R,3S)-2-(4-bromophenyl)tetrahydro-2H-pyran-3-yl]propane-2-sulfonamide
—— benzyl 2-cycloheptyl-4,4-dimethyl-3-oxo-1,2-diazetidine-1-carboxylate 1224513-44-3 C19H26N2O3
benzyl 2-cycloheptyl-4,4-dimethyl-3-oxo-1,2-diazetidine-1-carboxylate
—— —— 1383275-18-0 C18H21NO2S2
—— ethyl 6-bromo-3-(3-(naphthalen-1-yloxy)propyl)-1H-indole-2-carboxylate 1079251-83-4 C24H22BrNO3
ethyl 6-bromo-3-(3-(naphthalen-1-yloxy)propyl)-1H-indole-2-carboxylate
—— N-acetyl-N-(4-trifluoromethylphenyl)-4-acetoxy-5-chloro-1,2-dihydro-1-methyl-2-oxoquinoline-3-carboxamide 1373261-06-3 C22H16ClF3N2O5
N-acetyl-N-(4-trifluoromethylphenyl)-4-acetoxy-5-chloro-1,2-dihydro-1-methyl-2-oxoquinoline-3-carboxamide
—— —— 1234581-31-7 C26H23NO3
—— 9,10-diiodo-6-oxaspiro[4.5]dec-9-ene 1352458-97-9 C9H12I2O
9,10-diiodo-6-oxaspiro[4.5]dec-9-ene
—— N-(2-hydroxyethyl)-3-[2-(4-iodophenyl)-3-methylbutan-2-yl]-N-methyl-1H-indole-6-carboxamide 1448611-23-1 C23H27IN2O2
N-(2-hydroxyethyl)-3-[2-(4-iodophenyl)-3-methylbutan-2-yl]-N-methyl-1H-indole-6-carboxamide
—— (1S<sup>*</sup>,6S<sup>*</sup>)-6-(1-benzyloxypentyl)-3,4,5,6-tetrahydropyran-2,4-dione 141554-39-4 C17H22O4
(1S<sup>*</sup>,6S<sup>*</sup>)-6-(1-benzyloxypentyl)-3,4,5,6-tetrahydropyran-2,4-dione
—— ethyl 5-phenylimidazo<1,2-a>quinoline-2-carboxylate 113508-57-9 C20H16N2O2
ethyl 5-phenylimidazo<1,2-a>quinoline-2-carboxylate
—— 2-diazo-1-(1,1-dioxido-4-thiomorpholinyl)ethanone 1342316-11-3 C6H9N3O3S
2-diazo-1-(1,1-dioxido-4-thiomorpholinyl)ethanone
—— 3-[4-(2-iodobenzyloxy)phenyl]isoxazole-5-carboxylic acid amide 1613165-83-5 C17H13IN2O3
3-[4-(2-iodobenzyloxy)phenyl]isoxazole-5-carboxylic acid amide