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中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-triisopropylsilanylsulfanyl-3,4,4a,9a-tetrahydro-1H-benzo[4,5]furo[2,3-c]pyridine-2-carboxylic acid tert-butyl ester 1357602-77-7 C25H41NO3SSi
7-triisopropylsilanylsulfanyl-3,4,4a,9a-tetrahydro-1H-benzo[4,5]furo[2,3-c]pyridine-2-carboxylic acid tert-butyl ester
—— 4-[3-[6-(5-benzylcarbamoyl-3'-fluoro-biphenyl-3-yloxy)-hexyl]-2-(2-carboxy-ethyl)-phenoxy]-butyric acid 1162259-74-6 C39H42FNO7
4-[3-[6-(5-benzylcarbamoyl-3'-fluoro-biphenyl-3-yloxy)-hexyl]-2-(2-carboxy-ethyl)-phenoxy]-butyric acid
—— methyl (7R)-7-[(tert-butoxycarbonyl)amino]-14-cyclohexyl-4-(piperidin-1-ylmethyl)-7,8-dihydro-6H-indolo[1,2-e][1,5]benzoxazocine-11-carboxylate 1104194-76-4 C36H47N3O5
methyl (7R)-7-[(tert-butoxycarbonyl)amino]-14-cyclohexyl-4-(piperidin-1-ylmethyl)-7,8-dihydro-6H-indolo[1,2-e][1,5]benzoxazocine-11-carboxylate
—— 4-[3-{6-[3-benzo[1,3]dioxol-5-yl-5-(2-difluoromethoxy-benzylcarbamoyl)-phenoxy]-hexyl}-2-(2-carboxy-ethyl)-phenoxy]-butyric acid 1162261-22-4 C41H43F2NO10
4-[3-{6-[3-benzo[1,3]dioxol-5-yl-5-(2-difluoromethoxy-benzylcarbamoyl)-phenoxy]-hexyl}-2-(2-carboxy-ethyl)-phenoxy]-butyric acid
—— (E)-N-(2-benzyloxy-phenyl)-3-(4-fluoro-3-acetoxy-phenyl)-acrylamide 1223569-81-0 C24H20FNO4
(E)-N-(2-benzyloxy-phenyl)-3-(4-fluoro-3-acetoxy-phenyl)-acrylamide
—— (R)-N-(4-cyanophenyl)-4-(4-(4-fluorophenyl)phthalazin-1-yl)-3-methylpiperazine-1-carboxamide 1228071-58-6 C27H23FN6O
(R)-N-(4-cyanophenyl)-4-(4-(4-fluorophenyl)phthalazin-1-yl)-3-methylpiperazine-1-carboxamide
—— 3-(6-aminopyridin-3-yl)-4-oxo-8-oxa-3,10-diazabicyclo[4.3.1]decane-10-carboxylic acid tert-butyl ester 1331847-87-0 C17H24N4O4
3-(6-aminopyridin-3-yl)-4-oxo-8-oxa-3,10-diazabicyclo[4.3.1]decane-10-carboxylic acid tert-butyl ester
—— 1-amino-N-[5-(4-{[2-ethyl-3-fluoro-4-(methylsulfonyl)-phenyl]carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)pyridin-2-yl]cyclopropane-carboxamide 1251161-39-3 C28H29FN4O5S
1-amino-N-[5-(4-{[2-ethyl-3-fluoro-4-(methylsulfonyl)-phenyl]carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)pyridin-2-yl]cyclopropane-carboxamide
—— 5-[3-(4-fluorophenyl)phenyl]-N-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-[1,2,4]triazolo[1,5-a]pyridin-2-amine 1142943-74-5 C30H28FN5O
5-[3-(4-fluorophenyl)phenyl]-N-[4-(2-pyrrolidin-1-ylethoxy)phenyl]-[1,2,4]triazolo[1,5-a]pyridin-2-amine
—— 4-{6-[2-fluoro-1-(fluoromethyl)ethoxy]-3-[3-methoxy-4-(pyrrolidin-3-yloxy)benzyl]-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl}piperidine-1-carbaldehyde 1162651-94-6 C29H34F2N4O6
4-{6-[2-fluoro-1-(fluoromethyl)ethoxy]-3-[3-methoxy-4-(pyrrolidin-3-yloxy)benzyl]-2,4-dioxo-3,4-dihydroquinazolin-1(2H)-yl}piperidine-1-carbaldehyde
—— 2-(3H-1-(4-chloro-benzenesulfonylamino)-5',7'-dimethoxy-spiro[cyclohexane-4,3'-indene]-1'-yl)-propionic acid ethyl ester 1151766-44-7 C27H32ClNO6S
2-(3H-1-(4-chloro-benzenesulfonylamino)-5',7'-dimethoxy-spiro[cyclohexane-4,3'-indene]-1'-yl)-propionic acid ethyl ester
—— 5-[[4-(cyclopropylamino)-3-methylsulfonyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl]amino]-1,3-dihydrobenzimidazole-2-thione 1037474-90-0 C16H16N8O2S2
5-[[4-(cyclopropylamino)-3-methylsulfonyl-2H-pyrazolo[3,4-d]pyrimidin-6-yl]amino]-1,3-dihydrobenzimidazole-2-thione
—— Methyl 5-(methanesulfonamido)-2-[2-[2-methoxy-5-(2-methoxypyridin-3-yl)-3-(1-methylcyclopropyl)phenyl]ethynyl]benzoate 1256489-14-1 C28H28N2O6S
Methyl 5-(methanesulfonamido)-2-[2-[2-methoxy-5-(2-methoxypyridin-3-yl)-3-(1-methylcyclopropyl)phenyl]ethynyl]benzoate
—— 7-(1H-indol-3-yl)-3-oxo-5-thioxo-2,3,5,6-tetrahydro[1,2,4]triazolo[4,3-c]pyrimidine-8-carbonitrile 1558023-19-0 C14H8N6OS
7-(1H-indol-3-yl)-3-oxo-5-thioxo-2,3,5,6-tetrahydro[1,2,4]triazolo[4,3-c]pyrimidine-8-carbonitrile
—— (S)-N-(2-hydroxy-3-methoxybenzylidene)-1-phenylethylamine 1204611-64-2 C16H17NO2
(S)-N-(2-hydroxy-3-methoxybenzylidene)-1-phenylethylamine
—— ethyl 5-((3,4-difluorobenzyl)oxy)-2-(p-tolyl)benzofuran-3-carboxylate 1390638-47-7 C25H20F2O4
ethyl 5-((3,4-difluorobenzyl)oxy)-2-(p-tolyl)benzofuran-3-carboxylate
—— —— 1421519-63-2 C34H47N6O20S*Na
—— 4-tert-butylcyclohexyl 4-methylbenzoate 1036648-28-8 C18H26O2
4-tert-butylcyclohexyl 4-methylbenzoate
—— (-)-2-phenylthiocyclopent-2-ene-1-ol 157239-36-6 C11H12OS
(-)-2-phenylthiocyclopent-2-ene-1-ol
—— 1-m-tolyl-1,2-dihydro-benzo[d][1,3]thiazin-4-one 16075-11-9 C15H13NOS
1-m-tolyl-1,2-dihydro-benzo[d][1,3]thiazin-4-one
—— 4,5-dihydro-2-(4-iodophenyl)-3-(3,4-dimethoxyphenyl)-2H-benzo[g]indazole 1432465-04-7 C25H21IN2O2
4,5-dihydro-2-(4-iodophenyl)-3-(3,4-dimethoxyphenyl)-2H-benzo[g]indazole
—— N-(3-carbamoyl-5-ethyl-1-(2-morpholinoethyl)-1H-pyrazol-4-yl)-2-ethoxy-5-((4-ethylpiperazin-1-yl)sulfonyl)nicotinamide 1356129-73-1 C26H40N8O6S
N-(3-carbamoyl-5-ethyl-1-(2-morpholinoethyl)-1H-pyrazol-4-yl)-2-ethoxy-5-((4-ethylpiperazin-1-yl)sulfonyl)nicotinamide
—— —— 174903-12-9 C24H18EuF3O2
—— —— 180260-23-5 C19H17BrFeO2
—— 2-(3-nitrophenyl)-4-p-tolyloxazole 1418206-06-0 C16H12N2O3
2-(3-nitrophenyl)-4-p-tolyloxazole
—— 8-(3,5-dimethyl-isoxazole-4-sulfonyl)-2-[4-(2-methoxy-1,1-dimethylethyl)-phenyl]-2,8-diaza-spiro[4.5]decan-1-one 1255712-53-8 C24H33N3O5S
8-(3,5-dimethyl-isoxazole-4-sulfonyl)-2-[4-(2-methoxy-1,1-dimethylethyl)-phenyl]-2,8-diaza-spiro[4.5]decan-1-one
—— 1-(ethylpropyl)-6-prop-1-ynylimidazo[4,5-b]pyridin-2-ol 1064782-76-8 C14H17N3O
1-(ethylpropyl)-6-prop-1-ynylimidazo[4,5-b]pyridin-2-ol
—— N-[5-[1-(2-methylpropyl)pyrazol-4-yl]-[1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide 1142938-05-3 C17H20N6O
N-[5-[1-(2-methylpropyl)pyrazol-4-yl]-[1,2,4]triazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide
—— 4-((1S,3R)-1-biphenyl-4-ylmethyl-3-ethoxycarbonyl-butylcarbamoyl)-pyridine-2-carboxylicacid 1257265-68-1 C27H28N2O5
4-((1S,3R)-1-biphenyl-4-ylmethyl-3-ethoxycarbonyl-butylcarbamoyl)-pyridine-2-carboxylicacid
—— methyl 4-[[(2R)-4-ethoxy-4-oxo-1-[4-[3-(trifluoromethyl)phenyl]phenyl]butan-2-yl]amino]-4-oxobutanoate 1257443-54-1 C24H26F3NO5
methyl 4-[[(2R)-4-ethoxy-4-oxo-1-[4-[3-(trifluoromethyl)phenyl]phenyl]butan-2-yl]amino]-4-oxobutanoate
—— 4-{[2-ethyl-3-fluoro-4-(methylsulfonyl)phenyl]carbonyl}-7-(4-morpholin-4-ylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine 1251161-96-2 C29H31FN2O5S
4-{[2-ethyl-3-fluoro-4-(methylsulfonyl)phenyl]carbonyl}-7-(4-morpholin-4-ylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
—— N-(4-chloro-3-methylphenyl)-4-(6-pyridin-3-ylpyrazolo[1,5-a]pyrimidin-3-yl)thiophene-2-carboxamide 1109282-63-4 C23H16ClN5OS
N-(4-chloro-3-methylphenyl)-4-(6-pyridin-3-ylpyrazolo[1,5-a]pyrimidin-3-yl)thiophene-2-carboxamide
—— Ethyl 5-(5-formyl-6-hydroxy-2-naphthalenyl)-2-thiophenecarboxylate 1093119-41-5 C18H14O4S
Ethyl 5-(5-formyl-6-hydroxy-2-naphthalenyl)-2-thiophenecarboxylate
—— (±)-3,4-dihydro-7-hydroxy-8-methyl-2H-1-benzopyran 1154741-15-7 C10H12O2
(±)-3,4-dihydro-7-hydroxy-8-methyl-2H-1-benzopyran
—— 4-amino-N-(benzo[d][1,3]dioxol-5-yl)thieno[3,2-d]pyrimidine-7-carboxamide 1318129-57-5 C14H10N4O3S
4-amino-N-(benzo[d][1,3]dioxol-5-yl)thieno[3,2-d]pyrimidine-7-carboxamide
—— (RS)-1-({2-[(S)-2-oxo-3-(3-oxo-3,4-dihydro-2H-benzo[1,4]oxazin-6-yl)-oxazolidin-5-yl]-ethylamino}-methyl)-1,2-dihydro-pyrrolo[3,2,1-ij]quinolin-4-one 1220976-76-0 C25H24N4O5
(RS)-1-({2-[(S)-2-oxo-3-(3-oxo-3,4-dihydro-2H-benzo[1,4]oxazin-6-yl)-oxazolidin-5-yl]-ethylamino}-methyl)-1,2-dihydro-pyrrolo[3,2,1-ij]quinolin-4-one
—— 1-pyridin-3-yl-5-[(3-pyridin-3-ylpyrrolidin-1-yl)carbonyl]-2-[3-(trifluoromethoxy)phenyl]-1H-benzimidazole 1225213-39-7 C29H22F3N5O2
1-pyridin-3-yl-5-[(3-pyridin-3-ylpyrrolidin-1-yl)carbonyl]-2-[3-(trifluoromethoxy)phenyl]-1H-benzimidazole
—— 3-(4-fluorophenyl)-2-oxo-2H-1,2'-bipyridine-5-carboxylic acid 1225462-76-9 C17H11FN2O3
3-(4-fluorophenyl)-2-oxo-2H-1,2'-bipyridine-5-carboxylic acid
—— (RS)-4-(2'-fluoro-3'-methoxy-biphenyl-3-yl)-4-(4-methoxy-phenyl)-4,5-dihydro-oxazol-2-yl-amine formate 1180017-34-8 CH2O2*C23H21FN2O3
(RS)-4-(2'-fluoro-3'-methoxy-biphenyl-3-yl)-4-(4-methoxy-phenyl)-4,5-dihydro-oxazol-2-yl-amine formate
—— N-methyl-6-methylsulfanyl-N-pyridin-3-ylpyridine-3-carboxamide 1246663-27-3 C13H13N3OS
N-methyl-6-methylsulfanyl-N-pyridin-3-ylpyridine-3-carboxamide
—— (R)-4-(4-bromophenyl)-3-tert-butoxycarbonylaminobutyric acid butyl ester 1257446-41-5 C19H28BrNO4
(R)-4-(4-bromophenyl)-3-tert-butoxycarbonylaminobutyric acid butyl ester
—— (2R,4S)-5-biphenyl-4-yl-2-methyl-4-(2-1H-tetrazol-5-yl-acetylamido)-pentanoic acid 1257264-54-2 C21H23N5O3
(2R,4S)-5-biphenyl-4-yl-2-methyl-4-(2-1H-tetrazol-5-yl-acetylamido)-pentanoic acid
—— 3-(cyclopentanecarbonylamino)-N,4-dimethyl-N-pyridin-3-ylbenzamide 1246665-30-4 C20H23N3O2
3-(cyclopentanecarbonylamino)-N,4-dimethyl-N-pyridin-3-ylbenzamide
—— 8-N-[(2-amino-1,3-benzothiazol-6-yl)methyl]-3-N-(3-methylbutyl)-2-thiophen-3-ylimidazo[1,2-a]pyridine-3,8-dicarboxamide 1038692-63-5 C26H26N6O2S2
8-N-[(2-amino-1,3-benzothiazol-6-yl)methyl]-3-N-(3-methylbutyl)-2-thiophen-3-ylimidazo[1,2-a]pyridine-3,8-dicarboxamide
—— 3-[3-(2-tert-butylphenoxy)azetidin-1-yl]-3-oxopropylprop-2-enoate 1146960-71-5 C19H25NO4
3-[3-(2-tert-butylphenoxy)azetidin-1-yl]-3-oxopropylprop-2-enoate
—— 2-ethyl-3-N-[(2S)-1-hydroxy-4-methylpentan-2-yl]-8-N-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]imidazo[1,2-a]pyridine-3,8-dicarboxamide 1038390-66-7 C28H35N5O4
2-ethyl-3-N-[(2S)-1-hydroxy-4-methylpentan-2-yl]-8-N-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]imidazo[1,2-a]pyridine-3,8-dicarboxamide
—— 1-{1-[(benzyloxy)acetyl]piperidin-3-yl}-3-(3,4-dimethoxybenzyl)-6-[2-fluoro-1-(fluoromethyl)ethoxy]quinazoline-2,4(1H,3H)-dione 1140590-28-8 C34H37F2N3O7
1-{1-[(benzyloxy)acetyl]piperidin-3-yl}-3-(3,4-dimethoxybenzyl)-6-[2-fluoro-1-(fluoromethyl)ethoxy]quinazoline-2,4(1H,3H)-dione
—— 4-{[6-amino-9-(2-{1-[(2S)-2-hydroxypropanoyl]piperidin-4-yl}ethyl)-9H-purin-8-yl]thio}-5-bromobenzene-1,2-diol 1156467-67-2 C21H25BrN6O4S
4-{[6-amino-9-(2-{1-[(2S)-2-hydroxypropanoyl]piperidin-4-yl}ethyl)-9H-purin-8-yl]thio}-5-bromobenzene-1,2-diol
—— methyl 4-{4-[(2,6-di-tert-butyl-4-fluorophenoxy)methyl]piperidin-1-yl}-4-oxobutanoate 1146959-62-7 C25H38FNO4
methyl 4-{4-[(2,6-di-tert-butyl-4-fluorophenoxy)methyl]piperidin-1-yl}-4-oxobutanoate
—— 3-N-[(2S)-1-hydroxybutan-2-yl]-8-N-[(4-morpholin-4-ylphenyl)methyl]-2-thiophen-3-ylimidazo[1,2-a]pyridine-3,8-dicarboxamide 1038388-24-7 C28H31N5O4S
3-N-[(2S)-1-hydroxybutan-2-yl]-8-N-[(4-morpholin-4-ylphenyl)methyl]-2-thiophen-3-ylimidazo[1,2-a]pyridine-3,8-dicarboxamide