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中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-methyl-3-(3-methyl-1-(6-methylaminopyrimidin-4-yl)-1H-pyrazol-5-ylamino)-N-(3-methyl-5-trifluoromethylphenyl)-benzamide 1018471-09-4 C25H24F3N7O
4-methyl-3-(3-methyl-1-(6-methylaminopyrimidin-4-yl)-1H-pyrazol-5-ylamino)-N-(3-methyl-5-trifluoromethylphenyl)-benzamide
—— (4S,5S,6R)-4-((tert-butyldimethylsilyl)oxy)-10-((tert-butyldiphenylsilyl)oxy)-1-((4-methoxybenzyl)oxy)-5-methyl-6-((triethylsilyl)oxy)decan-2-one 1196801-46-3 C47H76O6Si3
(4S,5S,6R)-4-((tert-butyldimethylsilyl)oxy)-10-((tert-butyldiphenylsilyl)oxy)-1-((4-methoxybenzyl)oxy)-5-methyl-6-((triethylsilyl)oxy)decan-2-one
—— 1-ethyl-1,4-dihydro-7-methyl-N'-(1-((4-methylpiperazin-1-yl)methyl)-2-oxoindolin-3-ylidene)-4-oxo-1,8-naphthyridine-3-carbohydrazide 1253047-40-3 C26H29N7O3
1-ethyl-1,4-dihydro-7-methyl-N'-(1-((4-methylpiperazin-1-yl)methyl)-2-oxoindolin-3-ylidene)-4-oxo-1,8-naphthyridine-3-carbohydrazide
—— N-(benzylideneamino)-5-(4-fluorophenyl)-2-oxo-N-phenyl-1,3,4-oxadiazole-3-carboxamide 121649-31-8 C22H15FN4O3
N-(benzylideneamino)-5-(4-fluorophenyl)-2-oxo-N-phenyl-1,3,4-oxadiazole-3-carboxamide
—— (2,2-dimethyl-2H-thiochromen-4-yl)-(4-methoxyphenyl)methanol 1072932-99-0 C19H20O2S
(2,2-dimethyl-2H-thiochromen-4-yl)-(4-methoxyphenyl)methanol
—— ethyl (E)-4-hydroxy-4-(2-thiophen-2-yl-benzoxazol-6-yl)-but-2-enoate 1346701-90-3 C17H15NO4S
ethyl (E)-4-hydroxy-4-(2-thiophen-2-yl-benzoxazol-6-yl)-but-2-enoate
—— (S)-2-azido-1-iodo-3-methylbutane 1067878-89-0 C5H10IN3
(S)-2-azido-1-iodo-3-methylbutane
—— N-[2-oxo-2-(1'H,3H-spiro[2-benzofuran-1,4'-piperidin]-1'-yl)ethyl]-9H-fluoren-9-amine 1039165-07-5 C27H26N2O2
N-[2-oxo-2-(1'H,3H-spiro[2-benzofuran-1,4'-piperidin]-1'-yl)ethyl]-9H-fluoren-9-amine
—— Propyl 3-[(5-amino-3,4-dimethylthieno[2,3-c]pyridazine-6-carbonyl)amino]pyrrolidine-1-carboxylate 1451995-35-9 C17H23N5O3S
Propyl 3-[(5-amino-3,4-dimethylthieno[2,3-c]pyridazine-6-carbonyl)amino]pyrrolidine-1-carboxylate
—— tert-butyl N-methyl-N-[1-[[5-(7-fluoro-2-methylimidazo[1,2-a]pyridin-3-yl)-6-[2-tri(propan-2-yl)silylethynyl]pyridin-2-yl]amino]-1-oxopropan-2-yl]carbamate 1452573-45-3 C33H46FN5O3Si
tert-butyl N-methyl-N-[1-[[5-(7-fluoro-2-methylimidazo[1,2-a]pyridin-3-yl)-6-[2-tri(propan-2-yl)silylethynyl]pyridin-2-yl]amino]-1-oxopropan-2-yl]carbamate
—— (8-chloro-[1,2,4]triazolo[1,5-a]pyrazin-2-yl)-(3-methyl-3H-benzotriazol-5-yl)amine 1451388-98-9 C12H9ClN8
(8-chloro-[1,2,4]triazolo[1,5-a]pyrazin-2-yl)-(3-methyl-3H-benzotriazol-5-yl)amine
—— 1,4-dimethyl-5-(6-(trifluoromethyl)-1H-indazol-4-yl)pyridin-2(1H)-one 1454298-98-6 C15H12F3N3O
1,4-dimethyl-5-(6-(trifluoromethyl)-1H-indazol-4-yl)pyridin-2(1H)-one
—— 4-(3-cyano-4-methylphenyl)-N-(thiazol-2-yl)-3,4-dihydro-2H-benzo[b][1,4]oxazine-7-sulfonamide 1450921-28-4 C19H16N4O3S2
4-(3-cyano-4-methylphenyl)-N-(thiazol-2-yl)-3,4-dihydro-2H-benzo[b][1,4]oxazine-7-sulfonamide
—— 1-{[4-(2-tert-butylphenoxy)piperidin-1-yl]carbonyl}cyclopropanecarboxylic acid 1146957-63-2 C20H27NO4
1-{[4-(2-tert-butylphenoxy)piperidin-1-yl]carbonyl}cyclopropanecarboxylic acid
—— 2-[4-(2-methoxy-ethyl)-phenyl]-8-(2-trifluoromethoxy-benzenesulfonyl)-2,8-diaza-spiro[4.5]decan-1-one 1255712-46-9 C24H27F3N2O5S
2-[4-(2-methoxy-ethyl)-phenyl]-8-(2-trifluoromethoxy-benzenesulfonyl)-2,8-diaza-spiro[4.5]decan-1-one
—— 1-(1-acetylpiperidin-3-yl)-3-(3,4-dimethoxybenzyl)-2,4-dioxo-1,2,3,4-tetrahydroquinazoline-6-carbonitrile 1140590-14-2 C25H26N4O5
1-(1-acetylpiperidin-3-yl)-3-(3,4-dimethoxybenzyl)-2,4-dioxo-1,2,3,4-tetrahydroquinazoline-6-carbonitrile
—— 3-methyl-N-{4-methyl-2-[4-(trifluoromethyl)phenyl]pentyl}-1-pyrazin-2-yl-1H-pyrazole-4-carboxamide 1104270-51-0 C22H24F3N5O
3-methyl-N-{4-methyl-2-[4-(trifluoromethyl)phenyl]pentyl}-1-pyrazin-2-yl-1H-pyrazole-4-carboxamide
—— triethylammonium dichloro(2-[(diethylamino)methyl]-4-methylphenolato)zincate(II) 189204-51-1 C6H16N*C12H18Cl2NOZn
triethylammonium dichloro(2-[(diethylamino)methyl]-4-methylphenolato)zincate(II)
—— 2-(1-methyl-1H-indol-3-yl)-3-[(trimethylsilyl)ethynyl]benzo[g]quinoxaline 1533429-29-6 C26H23N3Si
2-(1-methyl-1H-indol-3-yl)-3-[(trimethylsilyl)ethynyl]benzo[g]quinoxaline
—— (2S,3S)-3-methyl-2-[[methyl(pyridin-3-ylmethyl)carbamoyl]amino]pentanoic acid 1260720-71-5 C14H21N3O3
(2S,3S)-3-methyl-2-[[methyl(pyridin-3-ylmethyl)carbamoyl]amino]pentanoic acid
—— 1-(3-aminopyrazin-2-yl)-3-methyl-N-({1-[4-(trifluoromethyl)phenyl]cyclohexyl}methyl)-1H-pyrazole-4-carboxamide 1104270-67-8 C23H25F3N6O
1-(3-aminopyrazin-2-yl)-3-methyl-N-({1-[4-(trifluoromethyl)phenyl]cyclohexyl}methyl)-1H-pyrazole-4-carboxamide
—— 7-(2-methyl-1H-benzimidazol-6-yl)-4-{6-methyl-5-[(3-methylphenyl)methyl]pyrimidin-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepine 1256946-05-0 C30H29N5O
7-(2-methyl-1H-benzimidazol-6-yl)-4-{6-methyl-5-[(3-methylphenyl)methyl]pyrimidin-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
—— (S)-2-hydroxyethyl 1-(1-(tert-butyldimethylsilyloxy)-3,3-dimethylbutan-2-yl)-6-(6-(3-ethylureido)-4-(4-(trifluoromethyl)thiazol-2-yl)pyridin-3-yl)-4-oxo-1,4-dihydroquinoline-3-carboxylate 1258213-35-2 C36H46F3N5O6SSi
(S)-2-hydroxyethyl 1-(1-(tert-butyldimethylsilyloxy)-3,3-dimethylbutan-2-yl)-6-(6-(3-ethylureido)-4-(4-(trifluoromethyl)thiazol-2-yl)pyridin-3-yl)-4-oxo-1,4-dihydroquinoline-3-carboxylate
—— 1-methyl-1H-imidazole-4-carboxylic acid {4-[2-(4-cyclohexylamino-1H-pyrazolo[4,3-c]pyridin-3-yl)-ethyl]-phenyl}-amide 1246348-63-9 C25H29N7O
1-methyl-1H-imidazole-4-carboxylic acid {4-[2-(4-cyclohexylamino-1H-pyrazolo[4,3-c]pyridin-3-yl)-ethyl]-phenyl}-amide
—— (2R,4S)-5-biphenyl-4-yl-2-methyl-4-[(1H-pyrazole-4-carbonyl)-amino]-pentanoic acid 1257263-97-0 C22H23N3O3
(2R,4S)-5-biphenyl-4-yl-2-methyl-4-[(1H-pyrazole-4-carbonyl)-amino]-pentanoic acid
—— Methyl 4-[[[2-chloro-5-[(3-fluorophenyl)methoxy]benzoyl]amino]methyl]benzoate 1148147-01-6 C23H19ClFNO4
Methyl 4-[[[2-chloro-5-[(3-fluorophenyl)methoxy]benzoyl]amino]methyl]benzoate
—— <i>N</i>-[3-(5-oxo-3-phenyl-isoxazol-4-ylidene)-propenyl]-acetanilide 110441-23-1 C20H16N2O3
<i>N</i>-[3-(5-oxo-3-phenyl-isoxazol-4-ylidene)-propenyl]-acetanilide
—— N3,N3,N7,N7,4,8-hexamethyl-1,5-diphenyl-2l3,6l3,9-trioxa-4,8-diaza-1l4,5l4-diborabicyclo[3.3.1]nona-2,6-diene-3,7-diamine 124357-29-5 C20H28B2N4O3
N3,N3,N7,N7,4,8-hexamethyl-1,5-diphenyl-2l3,6l3,9-trioxa-4,8-diaza-1l4,5l4-diborabicyclo[3.3.1]nona-2,6-diene-3,7-diamine
—— N-methyl-N-[3-({[2-{[1-(methylsulfonyl)piperidin-4-yl]amino}-5-(trifluoromethyl)pyrimidin-4-yl]amino}methyl)pyridin-2-yl]methanesulfonamide 1073155-14-2 C19H26F3N7O4S2
N-methyl-N-[3-({[2-{[1-(methylsulfonyl)piperidin-4-yl]amino}-5-(trifluoromethyl)pyrimidin-4-yl]amino}methyl)pyridin-2-yl]methanesulfonamide
—— 3-(3-iodo-5-methoxyphenyl)thiophene 1123157-86-7 C11H9IOS
3-(3-iodo-5-methoxyphenyl)thiophene
—— 2,6-dichloro-N-(2-(6-hydroxypyridin-2-ylamino)pyridin-4-yl)benzamide 1258293-23-0 C17H12Cl2N4O2
2,6-dichloro-N-(2-(6-hydroxypyridin-2-ylamino)pyridin-4-yl)benzamide
—— cyclopropanecarboxylic acid (3-(5-(3-(6-amino-5-trifluoromethylpyridin-3-yl)imidazo[1,2-b]pyridazin-6-yl)pyridin-2-yloxy)propyl)amide 1084952-90-8 C24H22F3N7O2
cyclopropanecarboxylic acid (3-(5-(3-(6-amino-5-trifluoromethylpyridin-3-yl)imidazo[1,2-b]pyridazin-6-yl)pyridin-2-yloxy)propyl)amide
—— N-(6-(6-chloro-5-((3-thiophenylsulfonyl)amino)-3-pyridinyl)-1,3-benzothiazol-2-yl)acetamide 1112981-13-1 C18H13ClN4O3S3
N-(6-(6-chloro-5-((3-thiophenylsulfonyl)amino)-3-pyridinyl)-1,3-benzothiazol-2-yl)acetamide
—— 7-ethylamino-N-(1H-indazol-6-yl)-8-methylquinazoline-2-amine 1169790-56-0 C18H18N6
7-ethylamino-N-(1H-indazol-6-yl)-8-methylquinazoline-2-amine
—— N-[4-(4-{[2-ethyl-3-fluoro-4-(methylsulfonyl)-phenyl]carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-2-(methyloxy)phenyl]-acetamide 1251163-04-8 C28H29FN2O6S
N-[4-(4-{[2-ethyl-3-fluoro-4-(methylsulfonyl)-phenyl]carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-2-(methyloxy)phenyl]-acetamide
—— N-{(1S)-1-[6-[(4-tert-butylphenyl)sulfonyl]-2-(trifluoromethyl)-6,11-dihydro-5H-pyrido[2,3-b][1,5]benzodiazepin-8-yl]ethyl}acetamide 1034046-01-9 C27H29F3N4O3S
N-{(1S)-1-[6-[(4-tert-butylphenyl)sulfonyl]-2-(trifluoromethyl)-6,11-dihydro-5H-pyrido[2,3-b][1,5]benzodiazepin-8-yl]ethyl}acetamide
—— 1-[6-(4-imidazol-1-yl-3-oxo-1H-pyrazol-2-yl)pyrimidin-4-yl]-N-methylpiperidine-3-carboxamide 1154030-01-9 C17H20N8O2
1-[6-(4-imidazol-1-yl-3-oxo-1H-pyrazol-2-yl)pyrimidin-4-yl]-N-methylpiperidine-3-carboxamide
—— 8-(6-ethoxy-pyridin-3-yl)-3-methyl-1-(3-methyl-pyridin-2-yl)-1,3-dihydro-imidazo[4,5-c]quinolin-2-one 1257428-97-9 C24H21N5O2
8-(6-ethoxy-pyridin-3-yl)-3-methyl-1-(3-methyl-pyridin-2-yl)-1,3-dihydro-imidazo[4,5-c]quinolin-2-one
—— N-(4-Chloro-benzyl)-2-(3,4-dichloro-phenyl)-2-fluoro-4-(4-methanesulfonyl-amino-piperidin-1-yl)-N-methyl-butyramide 1131738-05-0 C24H29Cl3FN3O3S
N-(4-Chloro-benzyl)-2-(3,4-dichloro-phenyl)-2-fluoro-4-(4-methanesulfonyl-amino-piperidin-1-yl)-N-methyl-butyramide
—— 8-bromo-1-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-3-methyl-1,3-dihydroimidazo[4,5-c]quinolin-2-one 1257553-22-2 C17H16BrN5O
8-bromo-1-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-3-methyl-1,3-dihydroimidazo[4,5-c]quinolin-2-one
—— 6-(8-methylquinazolin-2-ylamino)-1H-indazole-3-carbonitrile 1169788-90-2 C17H12N6
6-(8-methylquinazolin-2-ylamino)-1H-indazole-3-carbonitrile
—— (R)-ethyl 3-(6-aminonicotinamido)-4-(biphenyl 4-yl)butanoate 1257443-76-7 C24H25N3O3
(R)-ethyl 3-(6-aminonicotinamido)-4-(biphenyl 4-yl)butanoate
—— (R)-4-(3'-chlorobiphenyl-4-yl)-3-[(2-methyloxazole-5-carbonyl)-amino]-butyric acid ethyl ester 1257444-51-1 C23H23ClN2O4
(R)-4-(3'-chlorobiphenyl-4-yl)-3-[(2-methyloxazole-5-carbonyl)-amino]-butyric acid ethyl ester
—— (1R,2R,4R)-4-(2-chloro-4-pyrazol-1-ylbenzenesulfonyl)-2-(3,3-difluoroazetidine-1-carbonyl)cyclopentanecarboxylic acid (1-cyanocyclopropyl)amide 1258446-75-1 C23H22ClF2N5O4S
(1R,2R,4R)-4-(2-chloro-4-pyrazol-1-ylbenzenesulfonyl)-2-(3,3-difluoroazetidine-1-carbonyl)cyclopentanecarboxylic acid (1-cyanocyclopropyl)amide
—— tert-butyl N-[[5-[4-[3-[(2R,3S,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydropyran-2-yl]phenyl]phenyl]-1,3,4-oxadiazol-2-yl]methyl]carbamate 1453852-89-5 C26H31N3O8
tert-butyl N-[[5-[4-[3-[(2R,3S,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydropyran-2-yl]phenyl]phenyl]-1,3,4-oxadiazol-2-yl]methyl]carbamate
—— N-(4-fluorophenyl)-3-[4-(hydroxymethyl)piperidin-1-yl]sulfonylbenzamide 1445785-06-7 C19H21FN2O4S
N-(4-fluorophenyl)-3-[4-(hydroxymethyl)piperidin-1-yl]sulfonylbenzamide
—— 2,5-dioxopyrrolidin-1-yl 4-[bis(4-chlorophenyl)methyl]-3-methylpiperazine-1-carboxylate 1460034-77-8 C23H23Cl2N3O4
2,5-dioxopyrrolidin-1-yl 4-[bis(4-chlorophenyl)methyl]-3-methylpiperazine-1-carboxylate
—— 1-(3-fluoro-3-methylbutyl)-3-(2-fluoro-5-(7-((2-hydroxyethyl)amino)-2-methyl-1,6-naphthyridin-3-yl)-4-methylphenyl)urea 1455031-89-6 C24H29F2N5O2
1-(3-fluoro-3-methylbutyl)-3-(2-fluoro-5-(7-((2-hydroxyethyl)amino)-2-methyl-1,6-naphthyridin-3-yl)-4-methylphenyl)urea
—— 5-[5-[1-[(1-methyl-1H-indol-3-yl)methyl]-(3R)-piperidinyl]-1H-1,3,4-oxadiazol-2-yl]-3-(1-ethyl-1H-pyrazol-4-yl)-1H-indazole 1374352-59-6 C29H30N8O
5-[5-[1-[(1-methyl-1H-indol-3-yl)methyl]-(3R)-piperidinyl]-1H-1,3,4-oxadiazol-2-yl]-3-(1-ethyl-1H-pyrazol-4-yl)-1H-indazole
—— 9-[5-(3-Oxo-2,4-dioxa-3-phosphaspiro[5.5]undecan-3-yl)pentyl]-N-(2,2,2-trifluoroethyl)-9H-fluorene-9-carboxamide 194214-16-9 C29H35F3NO4P
9-[5-(3-Oxo-2,4-dioxa-3-phosphaspiro[5.5]undecan-3-yl)pentyl]-N-(2,2,2-trifluoroethyl)-9H-fluorene-9-carboxamide