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中文名称 英文名称 CAS号 化学式 结构式图片
—— tert-butyl 4-[4-(cyclopropylmethoxy)-3-(6-methyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-4-yl)phenyl]-3,6-dihydropyridine-1(2H)-carboxylate 1446235-60-4 C28H33N3O4
tert-butyl 4-[4-(cyclopropylmethoxy)-3-(6-methyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-4-yl)phenyl]-3,6-dihydropyridine-1(2H)-carboxylate
—— 4-(3-Chloroanilino)-1,3-dihydrothieno[3,4-c]pyridine-7-carbonitrile 1357187-39-3 C14H10ClN3S
4-(3-Chloroanilino)-1,3-dihydrothieno[3,4-c]pyridine-7-carbonitrile
—— 1-(2-Amino-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-d]azepin-6-yl)-2-[3-(4-methoxy-3-methylphenyl)-5-propan-2-ylpyrazol-1-yl]ethanone 1440952-39-5 C23H29N5O2S
1-(2-Amino-4,5,7,8-tetrahydro-[1,3]thiazolo[4,5-d]azepin-6-yl)-2-[3-(4-methoxy-3-methylphenyl)-5-propan-2-ylpyrazol-1-yl]ethanone
—— 2-[3-(4-Fluoro-3-methylphenyl)-5-methylpyrazol-1-yl]-1-(4-pyridin-2-ylpiperazin-1-yl)ethanone 1439303-03-3 C22H24FN5O
2-[3-(4-Fluoro-3-methylphenyl)-5-methylpyrazol-1-yl]-1-(4-pyridin-2-ylpiperazin-1-yl)ethanone
—— 6-[(2,6-difluoro-4-imidazo[1,2-a]pyridin-6-ylphenyl)methyl]-7H-pyrrolo[3,4-b]pyridin-5-one 1432438-12-4 C21H14F2N4O
6-[(2,6-difluoro-4-imidazo[1,2-a]pyridin-6-ylphenyl)methyl]-7H-pyrrolo[3,4-b]pyridin-5-one
—— {(S)-3-[1-(5-fluoro-6-methoxy-pyridin-3-yl)-2,3-dihydro-1H-pyrido[3,4-b][1,4]oxazin-7-yloxy]-pyrrolidin-1-yl}-(1-methyl-1H-imidazol-4-yl)-methanone 1446001-26-8 C22H23FN6O4
{(S)-3-[1-(5-fluoro-6-methoxy-pyridin-3-yl)-2,3-dihydro-1H-pyrido[3,4-b][1,4]oxazin-7-yloxy]-pyrrolidin-1-yl}-(1-methyl-1H-imidazol-4-yl)-methanone
—— 5-allyl-7-methoxy-5H-dibenzo[b,e][1,4]diazepin-11(10H)-one 1347035-39-5 C17H16N2O2
5-allyl-7-methoxy-5H-dibenzo[b,e][1,4]diazepin-11(10H)-one
—— 2-(2-Dimethylaminoethyl)-6,7-dimethyl-4-phenyl-1(2H)-isoquinolinone-3-carboxylic acid 159819-79-1 C22H24N2O3
2-(2-Dimethylaminoethyl)-6,7-dimethyl-4-phenyl-1(2H)-isoquinolinone-3-carboxylic acid
—— sodium;[chloro(nitro)methylidene]-dioxidoazanium 19282-07-6 CClN2O4*Na
sodium;[chloro(nitro)methylidene]-dioxidoazanium
—— 5-[[4-[(4-Fluorophenyl)-phenylmethyl]piperazin-1-yl]methyl]pyridine-3-carboxylic acid 1351371-29-3 C24H24FN3O2
5-[[4-[(4-Fluorophenyl)-phenylmethyl]piperazin-1-yl]methyl]pyridine-3-carboxylic acid
—— [3-(benzo[1,3]dioxol-5-yloxy)-2,4-difluoro-benzyl]-carbamic acid tert-butyl ester 1434723-48-4 C19H19F2NO5
[3-(benzo[1,3]dioxol-5-yloxy)-2,4-difluoro-benzyl]-carbamic acid tert-butyl ester
—— {7-[2-chloro-5-(trifluoromethoxy)phenyl]-1-oxo-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-4-yl}acetic acid 1429500-46-8 C16H12ClF3N2O4
{7-[2-chloro-5-(trifluoromethoxy)phenyl]-1-oxo-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-4-yl}acetic acid
—— (S)-N1-[7-((E)-3-methoxypropenyl)-2-pyridin-4-ylthieno[3,2-d]pyrimidin-4-yl]-3-phenylpropane-1,2-diamine 1438884-40-2 C24H25N5OS
(S)-N1-[7-((E)-3-methoxypropenyl)-2-pyridin-4-ylthieno[3,2-d]pyrimidin-4-yl]-3-phenylpropane-1,2-diamine
—— 4-[1-(3-Chlorophenyl)ethenyl]-6-methylidene-2-(4-methylphenyl)sulfonyl-1,3,5,6a-tetrahydrocyclopenta[c]pyrrole 1353956-87-2 C23H22ClNO2S
4-[1-(3-Chlorophenyl)ethenyl]-6-methylidene-2-(4-methylphenyl)sulfonyl-1,3,5,6a-tetrahydrocyclopenta[c]pyrrole
—— 5-{3-[4-(1-azabicyclo[2.2.2]oct-3-yl)piperazin-1-yl]-3-oxopropyl}-5-(4-bromophenyl)-5H-imidazo[2,1-a]isoindole 1227199-15-6 C30H34BrN5O
5-{3-[4-(1-azabicyclo[2.2.2]oct-3-yl)piperazin-1-yl]-3-oxopropyl}-5-(4-bromophenyl)-5H-imidazo[2,1-a]isoindole
—— 5-(4-(3,4-dichlorobenzyl)-4H-1,2,4-triazol-3-yI)-1Hbenzo[d]imidazole 1333405-69-8 C16H11Cl2N5
5-(4-(3,4-dichlorobenzyl)-4H-1,2,4-triazol-3-yI)-1Hbenzo[d]imidazole
—— 5-(4-(4-methylbenzyl)-4H-1,2,4-triazol-3-yI)-1H-benzo[d]imidazole 1333405-54-1 C17H15N5
5-(4-(4-methylbenzyl)-4H-1,2,4-triazol-3-yI)-1H-benzo[d]imidazole
—— ((R)-3-aminopiperidin-1-yl)-(4-{3-[1-(3-isopropyl-[1,2,4]oxadiazol-5-yl)-piperidin-4-yl]propoxy}-2-methylphenyl)methanone 1204309-63-6 C26H39N5O3
((R)-3-aminopiperidin-1-yl)-(4-{3-[1-(3-isopropyl-[1,2,4]oxadiazol-5-yl)-piperidin-4-yl]propoxy}-2-methylphenyl)methanone
—— 4-{4-fluoro-2-[(R)-(tetrahydro-pyran-3-yl)oxy]-phenylamino}-5-methyl-thieno[2,3-d]pyrimidine-6-carboxylic acid (3-pyrrolidin-1-yl-propyl)-amide 1332712-01-2 C26H32FN5O3S
4-{4-fluoro-2-[(R)-(tetrahydro-pyran-3-yl)oxy]-phenylamino}-5-methyl-thieno[2,3-d]pyrimidine-6-carboxylic acid (3-pyrrolidin-1-yl-propyl)-amide
—— N,N-dimethyl-4-[5-methyl-6-(1-methylsulfonylpiperidin-4-yl)oxypyrimidin-4-yl]oxypiperidine-1-sulfonamide 1233081-22-5 C18H31N5O6S2
N,N-dimethyl-4-[5-methyl-6-(1-methylsulfonylpiperidin-4-yl)oxypyrimidin-4-yl]oxypiperidine-1-sulfonamide
—— 3-[Diethoxy(oxido)phosphaniumyl]-1-methyl-1,8-naphthyridin-4-one 1350374-87-6 C13H17N2O4P
3-[Diethoxy(oxido)phosphaniumyl]-1-methyl-1,8-naphthyridin-4-one
—— N,N-diethyl(11R,12S,13E,15S)-9-butyryloxy-11,15-dihydroxy-7-thiaprosta-8,13-dienamide 170736-54-6 C27H47NO5S
N,N-diethyl(11R,12S,13E,15S)-9-butyryloxy-11,15-dihydroxy-7-thiaprosta-8,13-dienamide
—— N-[(1R,2R)-2-[[2-[2-methoxy-4-[4-(oxetan-3-yl)piperazin-1-yl]anilino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]-2,3-dihydro-1H-inden-1-yl]-N-methylmethanesulfonamide 1257258-99-3 C30H36F3N7O4S
N-[(1R,2R)-2-[[2-[2-methoxy-4-[4-(oxetan-3-yl)piperazin-1-yl]anilino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]-2,3-dihydro-1H-inden-1-yl]-N-methylmethanesulfonamide
—— —— 1369397-79-4 C18H11Br2F2N3O
—— —— 1369395-97-0 C18H14BrClF2N2O2
—— —— 1370419-43-4 C21H20BrN5O5
—— (S)-N-(5,5-dimethylhexa-2,3-dien-1-yl)-N,4-dimethylbenzenesulfonamide 1431534-80-3 C16H23NO2S
(S)-N-(5,5-dimethylhexa-2,3-dien-1-yl)-N,4-dimethylbenzenesulfonamide
—— N-[(1S)-1-(aminocarbonyl)-2-methylpropyl]-1-(pyridin-2-ylmethyl)-1H-indazole-3-carboxamide 1185282-24-9 C19H21N5O2
N-[(1S)-1-(aminocarbonyl)-2-methylpropyl]-1-(pyridin-2-ylmethyl)-1H-indazole-3-carboxamide
—— N-[(1S)-1-(aminocarbonyl)-2,2-dimethylpropyl]-1-(4-cyanobenzyl)-1H-indazole-3-carboxamide 1185282-28-3 C22H23N5O2
N-[(1S)-1-(aminocarbonyl)-2,2-dimethylpropyl]-1-(4-cyanobenzyl)-1H-indazole-3-carboxamide
—— —— 1251929-74-4 C11H8BrN3S
—— —— 16437-26-6 C48H42N4O7
—— 2-(5-Methyl-isoxazol-3-yl)-2H-tetrazole-5-carboxylic acid hydrazide 18137-62-7 C6H7N7O2
2-(5-Methyl-isoxazol-3-yl)-2H-tetrazole-5-carboxylic acid hydrazide
—— —— 1369397-49-8 C18H15BrCl2N2O
—— 4-[[(3aR,5aR,5bR,7aR,9S,11aR,11bR,13aS)-3a-[5-(2-fluorophenyl)-1,3,4-oxadiazol-2-yl]-5a,5b,8,8,11a-pentamethyl-2-oxo-1-propan-2-yl-4,5,6,7,7a,9,10,11,11b,12,13,13a-dodecahydro-3H-cyclopenta[a]chrysen-9-yl]oxy]-2,2-dimethyl-4-oxobutanoic acid 1449798-55-3 C43H57FN2O6
4-[[(3aR,5aR,5bR,7aR,9S,11aR,11bR,13aS)-3a-[5-(2-fluorophenyl)-1,3,4-oxadiazol-2-yl]-5a,5b,8,8,11a-pentamethyl-2-oxo-1-propan-2-yl-4,5,6,7,7a,9,10,11,11b,12,13,13a-dodecahydro-3H-cyclopenta[a]chrysen-9-yl]oxy]-2,2-dimethyl-4-oxobutanoic acid
—— methyl {4-[3-fluoro-2-(3-quinolinyl)phenyl]-4-hydroxy-4-[(3R)-1-({4-[(methylamino)methyl]phenyl}carbonyl)-3-piperidinyl]butyl}carbamate 1070869-85-0 C35H39FN4O4
methyl {4-[3-fluoro-2-(3-quinolinyl)phenyl]-4-hydroxy-4-[(3R)-1-({4-[(methylamino)methyl]phenyl}carbonyl)-3-piperidinyl]butyl}carbamate
—— 1-(3-tert-butylphenyl)-N-(2,4-dichlorophenyl)-4,5-dihydro-1H-pyrrolo[1,2-a][1,4]diazepine-2(3H)-carboxamide 1126427-13-1 C25H27Cl2N3O
1-(3-tert-butylphenyl)-N-(2,4-dichlorophenyl)-4,5-dihydro-1H-pyrrolo[1,2-a][1,4]diazepine-2(3H)-carboxamide
—— 2-(3,4-dichloro-phenyl)-4-[4-(methanesulfonyl(methyl)amino)-piperidin-1-yl]-2-methyl-butyric acid methyl ester 1131739-25-7 C19H28Cl2N2O4S
2-(3,4-dichloro-phenyl)-4-[4-(methanesulfonyl(methyl)amino)-piperidin-1-yl]-2-methyl-butyric acid methyl ester
—— 1-(3,4-dichlorophenyl)-5-(trifluoromethyl)-1H-pyrazole-3-carboxylic acid 1105638-03-6 C11H5Cl2F3N2O2
1-(3,4-dichlorophenyl)-5-(trifluoromethyl)-1H-pyrazole-3-carboxylic acid
—— (S)-3-(2-(3-phenoxyphenyl)acetamido)-4-(4-(trifluoromethyl)phenyl)butanoic acid 1322600-41-8 C25H22F3NO4
(S)-3-(2-(3-phenoxyphenyl)acetamido)-4-(4-(trifluoromethyl)phenyl)butanoic acid
—— (S)-methyl 2-(2-(4-(3-(4-chloro-2-phenoxyphenyl)ureido)phenyl)thiazole-4-carboxamido)-3-methylbutanoate 1210761-79-7 C29H27ClN4O5S
(S)-methyl 2-(2-(4-(3-(4-chloro-2-phenoxyphenyl)ureido)phenyl)thiazole-4-carboxamido)-3-methylbutanoate
—— N-[2-(4-chlorophenylsulfonamido)ethyl]-7-methoxy-2-(thiophen-2-yl)-1H-benzo[d]imidazole-4-carboxamide 1207429-91-1 C21H19ClN4O4S2
N-[2-(4-chlorophenylsulfonamido)ethyl]-7-methoxy-2-(thiophen-2-yl)-1H-benzo[d]imidazole-4-carboxamide
—— (S)-(1-((2'-(1H-tetrazol-5-yl)biphenyl-4-yl)methyl)-2-butyl-4-chloro-1H-imidazol-5-yl)methyl 2,6-diaminohexanoate 1174759-40-0 C28H35ClN8O2
(S)-(1-((2'-(1H-tetrazol-5-yl)biphenyl-4-yl)methyl)-2-butyl-4-chloro-1H-imidazol-5-yl)methyl 2,6-diaminohexanoate
—— (RS)-4-(4-methoxy-phenyl)-4-(3-pyridin-3-yl-phenyl)-4,5-dihydro-oxazol-2-ylamine formate 1180017-07-5 CH2O2*C21H19N3O2
(RS)-4-(4-methoxy-phenyl)-4-(3-pyridin-3-yl-phenyl)-4,5-dihydro-oxazol-2-ylamine formate
—— 4-(4-(4-fluorophenyl)-6,7-dihydrothieno[3,2-c]pyridin-5(4H)-yl)-N-isopentyl-4-oxobutanamide 1224394-52-8 C22H27FN2O2S
4-(4-(4-fluorophenyl)-6,7-dihydrothieno[3,2-c]pyridin-5(4H)-yl)-N-isopentyl-4-oxobutanamide
—— 2-(3,4-Dichloro-phenyl)-4-(4-methanesulfonylamino-piperidin-1-yl)-2,N-dimethyl-N-(6-trifluoromethyl-pyridin-3-ylmethyl)-butyramide 1131737-74-0 C25H31Cl2F3N4O3S
2-(3,4-Dichloro-phenyl)-4-(4-methanesulfonylamino-piperidin-1-yl)-2,N-dimethyl-N-(6-trifluoromethyl-pyridin-3-ylmethyl)-butyramide
—— 1-(4-methoxyphenyl)-2-phenyl-1H-benzo[g]indole 1131891-12-7 C25H19NO
1-(4-methoxyphenyl)-2-phenyl-1H-benzo[g]indole
—— (R)-1-(3,4-difluoro-5-methoxyphenyl)-3-methylpiperazine 1095542-42-9 C12H16F2N2O
(R)-1-(3,4-difluoro-5-methoxyphenyl)-3-methylpiperazine
—— (S)-9-fluoro-1-{3-[(R)-2-oxo-3-(3-oxo-3,4-dihydro-2H-benzo[1,4]thiazin-6-yl)-oxazolidin-5-yl]-propylamine}-1,2-dihydro-pyrrolo[3,2,1-ij]quinolin-4-one 1220977-42-3 C25H23FN4O4S
(S)-9-fluoro-1-{3-[(R)-2-oxo-3-(3-oxo-3,4-dihydro-2H-benzo[1,4]thiazin-6-yl)-oxazolidin-5-yl]-propylamine}-1,2-dihydro-pyrrolo[3,2,1-ij]quinolin-4-one
—— (S,E)-N-(3,3-dimethyl-1-(methylamino)-1-oxobutan-2-yl)-3-(3,3-dimethylbut-1-enyl)-7-methyl-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-1-carboxamide 1094087-97-4 C21H35N5O2
(S,E)-N-(3,3-dimethyl-1-(methylamino)-1-oxobutan-2-yl)-3-(3,3-dimethylbut-1-enyl)-7-methyl-5,6,7,8-tetrahydroimidazo[1,5-a]pyrazine-1-carboxamide
—— N-(2'-ethyl-5'-(4-methyl-5-oxo-4,5-dihydro-1,3,4-oxadiazol-2-yl)-[1,1'-biphenyl]-4-yl)-4-methyl-1,2,3-thiadiazole-5-carboxamide 1373938-39-6 C21H19N5O3S
N-(2'-ethyl-5'-(4-methyl-5-oxo-4,5-dihydro-1,3,4-oxadiazol-2-yl)-[1,1'-biphenyl]-4-yl)-4-methyl-1,2,3-thiadiazole-5-carboxamide