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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-(cyclohexyloxy)-2-fluorobenzonitrile 1204182-23-9 C13H14FNO
3-(cyclohexyloxy)-2-fluorobenzonitrile
—— 2-(1-phenyl-1H-[1,2,3]triazol-4-yl)-5H-pyrrolo[2,3-b]pyrazine-7-carboxylic acid [(R)-2-(4-cyanopiperidin-1-yl)-1-cyclopropyl-2-oxoethyl]amide 1334674-28-0 C26H25N9O2
2-(1-phenyl-1H-[1,2,3]triazol-4-yl)-5H-pyrrolo[2,3-b]pyrazine-7-carboxylic acid [(R)-2-(4-cyanopiperidin-1-yl)-1-cyclopropyl-2-oxoethyl]amide
—— 6-[3-(Hydroxymethyl)phenoxy]-1-[(2,4,6-trifluorophenyl)methyl]-2,3-dihydroquinazolin-4-one 1276040-82-4 C22H17F3N2O3
6-[3-(Hydroxymethyl)phenoxy]-1-[(2,4,6-trifluorophenyl)methyl]-2,3-dihydroquinazolin-4-one
—— 2-(4-(1H-pyrazol-4-yl)phenyl)-1-(5-(4-bromo-3,5-dimethoxyphenyl)furan-2-yl)-2-methoxyethanone 1333471-43-4 C24H21BrN2O5
2-(4-(1H-pyrazol-4-yl)phenyl)-1-(5-(4-bromo-3,5-dimethoxyphenyl)furan-2-yl)-2-methoxyethanone
—— 2-[2-(3-Methylsulfanylphenyl)phenyl]acetamide 1226856-20-7 C15H15NOS
2-[2-(3-Methylsulfanylphenyl)phenyl]acetamide
—— 2-[2-(3-Chloro-4-fluorophenyl)phenyl]acetamide 1226855-92-0 C14H11ClFNO
2-[2-(3-Chloro-4-fluorophenyl)phenyl]acetamide
—— tert-butyl 4-amino-2,6-dimethylpiperidine-1-carboxylate 1801241-14-4 C12H24N2O2
tert-butyl 4-amino-2,6-dimethylpiperidine-1-carboxylate
—— 5-[4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl]quinolin-2(1H)-one 1609578-28-0 C23H16N2O3
5-[4-(furo[3,2-c]pyridin-4-yloxy)-2-methylphenyl]quinolin-2(1H)-one
—— N-{2-[2-(2-Nitro-phenylsulfanylmethyl)-cyclobut-1-enyl]-ethyl}-acetamide 137073-03-1 C15H18N2O3S
N-{2-[2-(2-Nitro-phenylsulfanylmethyl)-cyclobut-1-enyl]-ethyl}-acetamide
—— 1-methyl-2'-[(1R)-1-phenylethyl]spiro[3,4-dihydronaphthalene-2,3'-oxaziridine]-1-ol 131514-16-4 C19H21NO2
1-methyl-2'-[(1R)-1-phenylethyl]spiro[3,4-dihydronaphthalene-2,3'-oxaziridine]-1-ol
—— (R)-N-(1-(pyridin-4-yl)ethyl)-6-(5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl)pyridazin-3-amine 1441874-38-9 C14H11F3N6O
(R)-N-(1-(pyridin-4-yl)ethyl)-6-(5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl)pyridazin-3-amine
—— N-[1-[2-(dimethylamino)ethyl]pyrazol-3-yl]-8-methyl-9-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-5,6-dihydropyrazolo[3,4-h]quinazolin-2-amine 1448457-14-4 C29H37BN8O2
N-[1-[2-(dimethylamino)ethyl]pyrazol-3-yl]-8-methyl-9-[4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-5,6-dihydropyrazolo[3,4-h]quinazolin-2-amine
—— 13,26-Bis(2,4,6-trimethylphenyl)-5,18-dithiaheptacyclo[14.10.0.03,14.04,12.06,11.017,25.019,24]hexacosa-1(26),2,4(12),6,8,10,13,15,17(25),19,21,23-dodecaene 1443022-39-6 C42H32S2
13,26-Bis(2,4,6-trimethylphenyl)-5,18-dithiaheptacyclo[14.10.0.03,14.04,12.06,11.017,25.019,24]hexacosa-1(26),2,4(12),6,8,10,13,15,17(25),19,21,23-dodecaene
—— (3R,3aR,6R,6aR)-6-[[6-chloro-5-[4-[4-(1H-1,2,4-triazol-5-yl)phenyl]phenyl]-1H-imidazo[4,5-b]pyridin-2-yl]oxy]-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-ol 1394372-35-0 C26H21ClN6O4
(3R,3aR,6R,6aR)-6-[[6-chloro-5-[4-[4-(1H-1,2,4-triazol-5-yl)phenyl]phenyl]-1H-imidazo[4,5-b]pyridin-2-yl]oxy]-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-3-ol
—— (S)-1-(3-(2-amino-5-methylphenoxy)piperidin-1-yl)-2,2,2-trifluoroethanone 1332712-48-7 C14H17F3N2O2
(S)-1-(3-(2-amino-5-methylphenoxy)piperidin-1-yl)-2,2,2-trifluoroethanone
—— 4-Methyl-2-pyridin-3-yl-5-[5-(trifluoromethyl)pyridin-2-yl]-1,3-thiazole 1204610-06-9 C15H10F3N3S
4-Methyl-2-pyridin-3-yl-5-[5-(trifluoromethyl)pyridin-2-yl]-1,3-thiazole
—— 2-Methoxy-2-(4-pyrazol-1-ylphenyl)-1-[5-(3,4,5-trimethoxyphenyl)furan-2-yl]ethanone 1333472-08-4 C25H24N2O6
2-Methoxy-2-(4-pyrazol-1-ylphenyl)-1-[5-(3,4,5-trimethoxyphenyl)furan-2-yl]ethanone
—— (R)-1-((S)-2,2,2-trifluoro-1-(3-(8-isopropoxyquinolin-2-yl)-[1,2,4]triazolo[4,3-a]pyridin-6-yl)ethyl)pyrrolidin-3-ol 1412247-21-2 C24H24F3N5O2
(R)-1-((S)-2,2,2-trifluoro-1-(3-(8-isopropoxyquinolin-2-yl)-[1,2,4]triazolo[4,3-a]pyridin-6-yl)ethyl)pyrrolidin-3-ol
—— (S)-tert-butyl 3-((6-(2,6-dichlorophenyl)-2-(3-fluoro-4-methoxybenzylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)methyl)piperidine-1-carboxylate 1190707-25-5 C31H34Cl2FN5O3
(S)-tert-butyl 3-((6-(2,6-dichlorophenyl)-2-(3-fluoro-4-methoxybenzylamino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)methyl)piperidine-1-carboxylate
—— N-((1S)-1-{5-[(hydroxyamino)carbonyl]-1,3-thiazol-2-yl}ethyl)-1-methyl-1H-benzimidazole-2-carboxamide 1332872-78-2 C15H15N5O3S
N-((1S)-1-{5-[(hydroxyamino)carbonyl]-1,3-thiazol-2-yl}ethyl)-1-methyl-1H-benzimidazole-2-carboxamide
—— 4-[1-({[(3,5-dichlorophenyl)amino]carbonyl}amino)ethyl]-N-hydroxybenzamide 1332893-17-0 C16H15Cl2N3O3
4-[1-({[(3,5-dichlorophenyl)amino]carbonyl}amino)ethyl]-N-hydroxybenzamide
—— Ethyl [8-methoxy-1-(2-methoxyethoxy)-2-oxo-3-(2,3,4-trimethylphenyl)-1,8-diazaspiro[4.5]dec-3-en-4-yl] carbonate 1228463-86-2 C24H34N2O7
Ethyl [8-methoxy-1-(2-methoxyethoxy)-2-oxo-3-(2,3,4-trimethylphenyl)-1,8-diazaspiro[4.5]dec-3-en-4-yl] carbonate
—— Methyl 6-(8-(benzo[d]thiazol-2-ylcarbamoyl)-3,4-dihydroisoquinolin-2(1H)-yl)-3-(3-(4-nitrophenoxy)phenyl)picolinate 1430752-46-7 C36H27N5O6S
Methyl 6-(8-(benzo[d]thiazol-2-ylcarbamoyl)-3,4-dihydroisoquinolin-2(1H)-yl)-3-(3-(4-nitrophenoxy)phenyl)picolinate
—— 1-[(4R)-7-chloro-2,2-bis(fluoromethyl)-3,4-dihydro-2H-chromen-4-yl]-3-(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-5-yl)urea 1444797-53-8 C22H22ClF2N3O3
1-[(4R)-7-chloro-2,2-bis(fluoromethyl)-3,4-dihydro-2H-chromen-4-yl]-3-(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-5-yl)urea
—— 6-(3,3-difluoropiperidin-1-yl)-2-methyl-3-nitropyridine 1435954-10-1 C11H13F2N3O2
6-(3,3-difluoropiperidin-1-yl)-2-methyl-3-nitropyridine
—— (4-methoxyphenyl)methyl N-[2-(2-methoxyphenyl)-4-methyl-1,3-thiazol-5-yl]carbamate 1354397-06-0 C20H20N2O4S
(4-methoxyphenyl)methyl N-[2-(2-methoxyphenyl)-4-methyl-1,3-thiazol-5-yl]carbamate
—— N-(3-((2-((4-(1-ethylpiperidin-4-yl)phenyl)amino)thieno[3,2-d]pyrimidin-4-yl)oxy)phenyl)acrylamide 1353550-66-9 C28H29N5O2S
N-(3-((2-((4-(1-ethylpiperidin-4-yl)phenyl)amino)thieno[3,2-d]pyrimidin-4-yl)oxy)phenyl)acrylamide
—— N-[(1S)-1-[4-[1-(5-propan-2-yloxypyrimidin-2-yl)azetidin-3-yl]oxyphenyl]ethyl]acetamide 1443669-42-8 C20H26N4O3
N-[(1S)-1-[4-[1-(5-propan-2-yloxypyrimidin-2-yl)azetidin-3-yl]oxyphenyl]ethyl]acetamide
—— 1-(5-(5-(trifluoromethyl)pyridin-2-yloxy)pyrimidin-2-yl)ethanamine 1429182-23-9 C12H11F3N4O
1-(5-(5-(trifluoromethyl)pyridin-2-yloxy)pyrimidin-2-yl)ethanamine
—— (S)-1-(5-tert-butyl-3-((1-cyclopropyl-1H-tetrazol-5-yl)methyl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl)-3-methylpyrrolidin-3-ol 1433362-59-4 C18H26N10O
(S)-1-(5-tert-butyl-3-((1-cyclopropyl-1H-tetrazol-5-yl)methyl)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl)-3-methylpyrrolidin-3-ol
—— 3-{(1R)-1-[2-(3-ethyl-3-hydroxypent-1-yn-1-yl)phenyl]ethyl}-5-fluoro-2-oxo-N-1,2,4-thiadiazol-5-yl-2,3-dihydro-1,3-benzooxazole-6-sulfonamide 1432512-97-4 C24H23FN4O5S2
3-{(1R)-1-[2-(3-ethyl-3-hydroxypent-1-yn-1-yl)phenyl]ethyl}-5-fluoro-2-oxo-N-1,2,4-thiadiazol-5-yl-2,3-dihydro-1,3-benzooxazole-6-sulfonamide
—— (2S,4R)-N-[(6-chloropyridin-3-yl)methyl]-4-hydroxy-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]pyrrolidine-2-carboxamide 1448186-63-7 C17H19ClN4O4
(2S,4R)-N-[(6-chloropyridin-3-yl)methyl]-4-hydroxy-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]pyrrolidine-2-carboxamide
—— (S)-N1-[7-(2-methoxypyridin-3-yl)-6-methyl-2-pyridin-4-ylthieno[3,2-d]pyrimidin-4-yl]-3-phenylpropane-1,2-diamine 1438885-01-8 C27H26N6OS
(S)-N1-[7-(2-methoxypyridin-3-yl)-6-methyl-2-pyridin-4-ylthieno[3,2-d]pyrimidin-4-yl]-3-phenylpropane-1,2-diamine
—— Ethyl 3-[3-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]benzoate 1411993-05-9 C22H27BO4
Ethyl 3-[3-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]benzoate
—— N-[5-bromo-6-[1-(3,5-difluorophenyl)ethoxy]-2-methylpyridin-3-yl]-1-pyrrolidin-1-ylmethanimine 1404442-99-4 C19H20BrF2N3O
N-[5-bromo-6-[1-(3,5-difluorophenyl)ethoxy]-2-methylpyridin-3-yl]-1-pyrrolidin-1-ylmethanimine
—— [(1S,4R,6R,14S,18R)-4-(1-benzofuran-2-ylsulfonylcarbamoyl)-14-[(2-methylpropan-2-yl)oxycarbonylamino]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadecan-18-yl] 4-fluoro-1,3-dihydroisoindole-2-carboxylate 1078625-55-4 C40H48FN5O10S
[(1S,4R,6R,14S,18R)-4-(1-benzofuran-2-ylsulfonylcarbamoyl)-14-[(2-methylpropan-2-yl)oxycarbonylamino]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadecan-18-yl] 4-fluoro-1,3-dihydroisoindole-2-carboxylate
—— 7-methyl-4-(2-methyl-5-pyrimidinyl)-6H-pyrrolo[1,2-a][1,4]benzodiazepine 1407992-72-6 C18H16N4
7-methyl-4-(2-methyl-5-pyrimidinyl)-6H-pyrrolo[1,2-a][1,4]benzodiazepine
—— (S)-tert-butyl 3-(3-aminopyridin-2-yloxy)piperidine-1-carboxylate 1332712-50-1 C15H23N3O3
(S)-tert-butyl 3-(3-aminopyridin-2-yloxy)piperidine-1-carboxylate
—— 2-[[3-(2-Methyl-5-pyridin-3-ylpyrazol-3-yl)pyrazol-1-yl]methyl]pyridine 1204610-74-1 C18H16N6
2-[[3-(2-Methyl-5-pyridin-3-ylpyrazol-3-yl)pyrazol-1-yl]methyl]pyridine
—— 5-(4-bromophenyl)-5-[3-(4,4-difluoropiperidin-1-yl)-3-oxopropyl]-5H-imidazo[2,1-a]isoindole 1227198-02-8 C24H22BrF2N3O
5-(4-bromophenyl)-5-[3-(4,4-difluoropiperidin-1-yl)-3-oxopropyl]-5H-imidazo[2,1-a]isoindole
—— phenyl 4-(5-(2-phenyl-5-(trifluoromethyl)oxazole-4-carboxamido)pyridin-2-yl)piperazine-1-carboxylate 1227860-69-6 C27H22F3N5O4
phenyl 4-(5-(2-phenyl-5-(trifluoromethyl)oxazole-4-carboxamido)pyridin-2-yl)piperazine-1-carboxylate
—— N-((1R)-1-{4-[(hydroxyamino)carbonyl]phenyl}butyl)-4-methoxybenzamide 1332890-74-0 C19H22N2O4
N-((1R)-1-{4-[(hydroxyamino)carbonyl]phenyl}butyl)-4-methoxybenzamide
—— 3-[[3-(isoquinolin-5-ylamino)piperidin-1-yl]methyl]-N-[2-(2-oxo-1,3-dioxolan-4-yl)ethyl]benzamide 1404375-44-5 C27H30N4O4
3-[[3-(isoquinolin-5-ylamino)piperidin-1-yl]methyl]-N-[2-(2-oxo-1,3-dioxolan-4-yl)ethyl]benzamide
—— 5-methyl-3-(4-(trifluoromethoxy)phenyl)isoxazol-4-carboxylic acid 1402881-82-6 C12H8F3NO4
5-methyl-3-(4-(trifluoromethoxy)phenyl)isoxazol-4-carboxylic acid
—— [(1R,2S,5S,6S,9S,10R)-21-cyano-1,5-dimethyl-12-oxo-16,17,18,19-tetrazahexacyclo[11.11.0.02,10.05,9.015,23.016,20]tetracosa-13,15(23),17,19,21-pentaen-6-yl] acetate 1364513-23-4 C25H27N5O3
[(1R,2S,5S,6S,9S,10R)-21-cyano-1,5-dimethyl-12-oxo-16,17,18,19-tetrazahexacyclo[11.11.0.02,10.05,9.015,23.016,20]tetracosa-13,15(23),17,19,21-pentaen-6-yl] acetate
—— 6-methyl-4-tosyl-1-oxa-4-azaspiro[4.5]deca-6,9-dien-8-one 1361991-55-0 C16H17NO4S
6-methyl-4-tosyl-1-oxa-4-azaspiro[4.5]deca-6,9-dien-8-one
—— tert-butyl 4-(1-cyanocyclobutyl)-4-hydroxypiperidine-1-carboxylate 1432493-43-0 C15H24N2O3
tert-butyl 4-(1-cyanocyclobutyl)-4-hydroxypiperidine-1-carboxylate
—— 5-fluoro-3-[(1R)-1-{2-[(1-hydroxycyclopentyl)ethynyl]phenyl}ethyl]-2-oxo-N-1,2,4-thiadiazol-5-yl-2,3-dihydro-1,3-benzooxazole-6-sulfonamide 1432512-94-1 C24H21FN4O5S2
5-fluoro-3-[(1R)-1-{2-[(1-hydroxycyclopentyl)ethynyl]phenyl}ethyl]-2-oxo-N-1,2,4-thiadiazol-5-yl-2,3-dihydro-1,3-benzooxazole-6-sulfonamide
—— 2-(1-((4-bromo-5-methyl-1H-pyrazol-1-yl)methyl)cyclohexyloxy)acetic acid 1430753-99-3 C13H19BrN2O3
2-(1-((4-bromo-5-methyl-1H-pyrazol-1-yl)methyl)cyclohexyloxy)acetic acid
—— 2-((S)-1-[1,4]dioxan-2-ylmethoxy)-9-(tetrahydro-pyran-4-ylmethoxy)-6,7-dihydro-pyrimido[6,1-a]isoquinolin-4-one 1445847-68-6 C23H28N2O6
2-((S)-1-[1,4]dioxan-2-ylmethoxy)-9-(tetrahydro-pyran-4-ylmethoxy)-6,7-dihydro-pyrimido[6,1-a]isoquinolin-4-one