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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-methyl-5-trifluoromethyl-2H-pyrazole-3-carboxylic acid [phenyl-(1-pyrrolidin-1-yl-cyclobutyl)-methyl]-amide 1208984-61-5 C21H25F3N4O
2-methyl-5-trifluoromethyl-2H-pyrazole-3-carboxylic acid [phenyl-(1-pyrrolidin-1-yl-cyclobutyl)-methyl]-amide
—— 3-[2-(3-fluorobenzyl)-2H-indazol-4-yl]-N-(2-hydroxyethyl)benzamide 1207964-23-5 C23H20FN3O2
3-[2-(3-fluorobenzyl)-2H-indazol-4-yl]-N-(2-hydroxyethyl)benzamide
—— 2-[1-[3-(3-fluorophenyl)propanoyl]piperidin-4-yl]-N-(2-piperidin-1-ylphenyl)-1,3-thiazole-4-carboxamide 1070190-66-7 C29H33FN4O2S
2-[1-[3-(3-fluorophenyl)propanoyl]piperidin-4-yl]-N-(2-piperidin-1-ylphenyl)-1,3-thiazole-4-carboxamide
—— (6S,9aS)-8-[[3-(3-aminophenyl)phenyl]methyl]-N-benzyl-6-[(4-hydroxyphenyl)methyl]-4,7-dioxo-2-prop-2-enyl-3,6,9,9a-tetrahydropyrazino[2,1-c][1,2,4]triazine-1-carboxamide 1145676-36-3 C37H38N6O4
(6S,9aS)-8-[[3-(3-aminophenyl)phenyl]methyl]-N-benzyl-6-[(4-hydroxyphenyl)methyl]-4,7-dioxo-2-prop-2-enyl-3,6,9,9a-tetrahydropyrazino[2,1-c][1,2,4]triazine-1-carboxamide
—— 3-((4-(4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-2-propylphenoxy)pyridin-2-yl)methyl)-5-(3-methoxyphenyl)-5-methylimidazolidine-2,4-dione 1198166-77-6 C29H27F6N3O5
3-((4-(4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)-2-propylphenoxy)pyridin-2-yl)methyl)-5-(3-methoxyphenyl)-5-methylimidazolidine-2,4-dione
—— (R)-3,3,3-trifluoro-2-hydroxy-N-(3-phenyl-2,2-bis(3-(trifluoromethoxy)phenyl)propyl)propanamide 1032187-63-5 C26H20F9NO4
(R)-3,3,3-trifluoro-2-hydroxy-N-(3-phenyl-2,2-bis(3-(trifluoromethoxy)phenyl)propyl)propanamide
—— N-((5-methoxy-1,3-dimethyl-1H-pyrazol-4-yl)methyl)-3-phenyl-2,2-bis(3-(trifluoromethoxy)phenyl)propan-1-amine 1032188-27-4 C30H29F6N3O3
N-((5-methoxy-1,3-dimethyl-1H-pyrazol-4-yl)methyl)-3-phenyl-2,2-bis(3-(trifluoromethoxy)phenyl)propan-1-amine
—— 2-aminocarbonylamino-6-(4-trifluoromethoxyphenyl)indole-3-carboxamide 1040167-80-3 C17H13F3N4O3
2-aminocarbonylamino-6-(4-trifluoromethoxyphenyl)indole-3-carboxamide
—— 2-(2-chloropyridin-3-yl)-5-(pyridin-3-yl)-1,3,4-oxadiazole 1033725-45-9 C12H7ClN4O
2-(2-chloropyridin-3-yl)-5-(pyridin-3-yl)-1,3,4-oxadiazole
—— ethyl (R,S)-formylamino-(1-methyl-4-S-nitrosomercapto-piperidin-4-yl)-acetate 1035695-81-8 C11H19N3O4S
ethyl (R,S)-formylamino-(1-methyl-4-S-nitrosomercapto-piperidin-4-yl)-acetate
—— 3-{1-[({2-[(cyclopentylmethyl)(ethyl)amino]-5-trifluoromethylphenyl}methyl){5-[2-(methylsulfonyl)ethoxy]pyrimidin-2-yl}amino]ethyl}-5-(trifluoromethyl)benzonitrile 1072907-13-1 C33H37F6N5O3S
3-{1-[({2-[(cyclopentylmethyl)(ethyl)amino]-5-trifluoromethylphenyl}methyl){5-[2-(methylsulfonyl)ethoxy]pyrimidin-2-yl}amino]ethyl}-5-(trifluoromethyl)benzonitrile
—— {5-[5-bromo-6-(4-methoxy-phenoxy)-pyridine-3-sulfonylamino]-5,6,7,8-tetrahydro-naphthalen-1-yloxy}-acetic acid 1208100-08-6 C24H23BrN2O7S
{5-[5-bromo-6-(4-methoxy-phenoxy)-pyridine-3-sulfonylamino]-5,6,7,8-tetrahydro-naphthalen-1-yloxy}-acetic acid
—— ethyl 8-chloro-1-cyclohexyl-4-oxo-4,5-dihydroimidazo-[1,5-a]quinoxaline-7-carboxylate 1033712-89-8 C19H20ClN3O3
ethyl 8-chloro-1-cyclohexyl-4-oxo-4,5-dihydroimidazo-[1,5-a]quinoxaline-7-carboxylate
—— 3-[1-[3-(5-fluoro-3-methyl-indol-1-yl)-5-pyrrolidin-1-yl-benzyl]-5-((S)-2-methylamino-propionylamino)-6-oxo-1,6-dihydro-pyridin-2-yl]-N,N-dimethyl-benzamide 1033124-61-6 C38H41FN6O3
3-[1-[3-(5-fluoro-3-methyl-indol-1-yl)-5-pyrrolidin-1-yl-benzyl]-5-((S)-2-methylamino-propionylamino)-6-oxo-1,6-dihydro-pyridin-2-yl]-N,N-dimethyl-benzamide
—— 2-(3-hydroxypropoxy)-N-(3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)-4-methylphenyl)pyridine-4-carboxamide 1025715-77-8 C25H24N6O3
2-(3-hydroxypropoxy)-N-(3-(4-(pyridin-3-yl)pyrimidin-2-ylamino)-4-methylphenyl)pyridine-4-carboxamide
—— methyl 4-(8-(5-chloro-6-methoxypyridin-3-yl)-[1,2,4]triazolo[1,5-a]pyridin-2-ylamino)benzoate 1202619-53-1 C20H16ClN5O3
methyl 4-(8-(5-chloro-6-methoxypyridin-3-yl)-[1,2,4]triazolo[1,5-a]pyridin-2-ylamino)benzoate
—— (RS)-1-benzenesulfonyl-3-(2-chloro-phenyl)-4-[4-(3-trifluoromethyl-pyridin-2-yl)-piperazine-1-carbonyl]-imidazolidin-2-one 1065143-99-8 C26H23ClF3N5O4S
(RS)-1-benzenesulfonyl-3-(2-chloro-phenyl)-4-[4-(3-trifluoromethyl-pyridin-2-yl)-piperazine-1-carbonyl]-imidazolidin-2-one
—— 2-(2-methoxyethoxy)-1,1-dimethylethyl 4-[(2,4-dichlorobenzoyl)amino]-1-(4-fluorophenyl)-2-methoxy-1H-imidazole-5-carboxylate 1072159-95-5 C25H26Cl2FN3O6
2-(2-methoxyethoxy)-1,1-dimethylethyl 4-[(2,4-dichlorobenzoyl)amino]-1-(4-fluorophenyl)-2-methoxy-1H-imidazole-5-carboxylate
—— 3,3,3-trifluoro-N-(3-(5-methylisoxazol-3-yl)-2,2-bis(3-(trifluoromethoxy)phenyl)propyl)propan-1-amine 1032188-02-5 C24H21F9N2O3
3,3,3-trifluoro-N-(3-(5-methylisoxazol-3-yl)-2,2-bis(3-(trifluoromethoxy)phenyl)propyl)propan-1-amine
—— 3-chloro-4-ethyl-N-[3-(2-methyl-1,2,3,4-tetrahydro-isoquinolin-7-ylcarbamoyl)-benzyl]-benzamide 1038556-48-7 C27H28ClN3O2
3-chloro-4-ethyl-N-[3-(2-methyl-1,2,3,4-tetrahydro-isoquinolin-7-ylcarbamoyl)-benzyl]-benzamide
—— 2-aminocarbonylamino-6-[3-[1-(N-tert-butoxycarbonyl-N-cyclopropylamino)ethyl]phenyl]indole-3-carboxamide 1040168-99-7 C26H31N5O4
2-aminocarbonylamino-6-[3-[1-(N-tert-butoxycarbonyl-N-cyclopropylamino)ethyl]phenyl]indole-3-carboxamide
—— 2-aminocarbonylamino-6-(thiazol-2-yl)indole-3-carboxamide 1040168-70-4 C13H11N5O2S
2-aminocarbonylamino-6-(thiazol-2-yl)indole-3-carboxamide
—— 2-chloro-N-(2-methyl-4-phenylaminomethyl-cyclohexyl)-5-trifluoromethyl-benzamide 1207530-12-8 C22H24ClF3N2O
2-chloro-N-(2-methyl-4-phenylaminomethyl-cyclohexyl)-5-trifluoromethyl-benzamide
—— (6S,9aS)-N-benzyl-6-[(4-hydroxyphenyl)methyl]-8-[[1-(4-methylphenyl)sulfonylindol-6-yl]methyl]-4,7-dioxo-2-prop-2-enyl-3,6,9,9a-tetrahydropyrazino[2,1-c][1,2,4]triazine-1-carboxamide 1145674-40-3 C40H40N6O6S
(6S,9aS)-N-benzyl-6-[(4-hydroxyphenyl)methyl]-8-[[1-(4-methylphenyl)sulfonylindol-6-yl]methyl]-4,7-dioxo-2-prop-2-enyl-3,6,9,9a-tetrahydropyrazino[2,1-c][1,2,4]triazine-1-carboxamide
—— (R)-1-(2-oxo-tetrahydrofuran-3-yl)-3-(3-phenyl-2,2-bis(3-(trifluoromethoxy)phenyl)propyl)urea 1032187-73-7 C28H24F6N2O5
(R)-1-(2-oxo-tetrahydrofuran-3-yl)-3-(3-phenyl-2,2-bis(3-(trifluoromethoxy)phenyl)propyl)urea
—— 1-[4-[[2-Tert-butyl-5-[3-(trifluoromethyl)phenyl]sulfanylbenzimidazol-1-yl]methyl]piperidin-1-yl]ethanone 1067155-57-0 C26H30F3N3OS
1-[4-[[2-Tert-butyl-5-[3-(trifluoromethyl)phenyl]sulfanylbenzimidazol-1-yl]methyl]piperidin-1-yl]ethanone
—— 1-methyl-6-oxo-1,6-dihydro-pyridine-3-carboxylic acid 3-(2-methyl-1,2,3,4-tetrahydro-isoquinolin-7-ylcarbamoyl)-benzylamide 1038552-96-3 C25H26N4O3
1-methyl-6-oxo-1,6-dihydro-pyridine-3-carboxylic acid 3-(2-methyl-1,2,3,4-tetrahydro-isoquinolin-7-ylcarbamoyl)-benzylamide
—— 3-[[3-(cyclopentyloxy)-4-methoxyphenyl](1H-pyrazol-4-ylmethyl)amino]benzoic acid 1203592-49-7 C23H25N3O4
3-[[3-(cyclopentyloxy)-4-methoxyphenyl](1H-pyrazol-4-ylmethyl)amino]benzoic acid
—— 4-[[3-(cyclopentyloxy)-4-(difluoromethoxy)phenyl](1,3-thiazol-5-ylmethyl)amino]benzoic acid 1203593-20-7 C23H22F2N2O4S
4-[[3-(cyclopentyloxy)-4-(difluoromethoxy)phenyl](1,3-thiazol-5-ylmethyl)amino]benzoic acid
—— 2,5-dimethyl-N-[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]-1,3-oxazole-4-carboxamide 1025714-17-3 C22H20N6O2
2,5-dimethyl-N-[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]-1,3-oxazole-4-carboxamide
—— 2-aminocarbonylamino-6-cyclopentylaminocarbonylindole-3-carboxamide 1040169-92-3 C16H19N5O3
2-aminocarbonylamino-6-cyclopentylaminocarbonylindole-3-carboxamide
—— 3-[3-[[4-(2-Chlorophenyl)-1,3-thiazol-2-yl]methylamino]phenyl]propanoic acid 1050507-01-1 C19H17ClN2O2S
3-[3-[[4-(2-Chlorophenyl)-1,3-thiazol-2-yl]methylamino]phenyl]propanoic acid
—— 5-(azepan-1-yl)-N-[5-[4-(trifluoromethyl)phenyl]-1H-pyrazol-3-yl]pentanamide 1040719-33-2 C21H27F3N4O
5-(azepan-1-yl)-N-[5-[4-(trifluoromethyl)phenyl]-1H-pyrazol-3-yl]pentanamide
—— 1-(5-tert-butyl-2-(4-isopropyl-2,2-dimethyl-3-oxopiperazine-1-carbonyl)thiophen-3-yl)-3-(4-methyl-3-(6-(morpholinomethyl)pyridin-3-yl)phenyl)urea 1207877-74-4 C36H48N6O4S
1-(5-tert-butyl-2-(4-isopropyl-2,2-dimethyl-3-oxopiperazine-1-carbonyl)thiophen-3-yl)-3-(4-methyl-3-(6-(morpholinomethyl)pyridin-3-yl)phenyl)urea
—— N-[6-[3-(2,2-dimethylpropanoylamino)phenoxy]imidazo[1,2-b]pyridazin-2-yl]-4-(trifluoromethyl)benzamide 1005783-83-4 C25H22F3N5O3
N-[6-[3-(2,2-dimethylpropanoylamino)phenoxy]imidazo[1,2-b]pyridazin-2-yl]-4-(trifluoromethyl)benzamide
—— (R)-3-[10-(2,3-difluoro-phenyl)-decanoylamino]-4-trimethylammonio-butyrate 1192177-93-7 C23H36F2N2O3
(R)-3-[10-(2,3-difluoro-phenyl)-decanoylamino]-4-trimethylammonio-butyrate
—— 3,5-di-tert-butyl-4-methoxy-N-(1-(4-methylpiperazine-1-carbonyl)cyclohexyl)benzamide 1191943-84-6 C28H45N3O3
3,5-di-tert-butyl-4-methoxy-N-(1-(4-methylpiperazine-1-carbonyl)cyclohexyl)benzamide
—— N-cyclohexylmethyl-2-(6-methoxy-1H-indol-3-yl)-2-oxo-N-({[(S)-1-(tetrahydro-furan-2-yl)methyl]-carbamoyl}-methyl)-acetamide 1192477-39-6 C25H33N3O5
N-cyclohexylmethyl-2-(6-methoxy-1H-indol-3-yl)-2-oxo-N-({[(S)-1-(tetrahydro-furan-2-yl)methyl]-carbamoyl}-methyl)-acetamide
—— 4-[3-(1-methylbutoxy)benzylidene]-N-pyridin-3-ylpiperidine-1-carboxamide 1191400-31-3 C23H29N3O2
4-[3-(1-methylbutoxy)benzylidene]-N-pyridin-3-ylpiperidine-1-carboxamide
—— 3-cyclohexyl-5-methyl-4-(4-phenylphenyl)-1H-imidazol-2-one 133259-86-6 C22H24N2O
3-cyclohexyl-5-methyl-4-(4-phenylphenyl)-1H-imidazol-2-one
—— 3-(2-cyanopropan-2-yl)-N-(1-(3-(trifluoromethyl)benzylcarbamoyl)cyclohexyl)benzamide 1191944-04-3 C26H28F3N3O2
3-(2-cyanopropan-2-yl)-N-(1-(3-(trifluoromethyl)benzylcarbamoyl)cyclohexyl)benzamide
—— 4-{3-[(3-methylcyclohexyl)oxy]benzylidene}-N-pyridin-3-ylpiperidine-1-carboxamide 1191400-29-9 C25H31N3O2
4-{3-[(3-methylcyclohexyl)oxy]benzylidene}-N-pyridin-3-ylpiperidine-1-carboxamide
—— cyclo[Abu-N(Me)Phe-D-Pro-Lys(Ac)] 1030273-91-6 C27H39N5O5
cyclo[Abu-N(Me)Phe-D-Pro-Lys(Ac)]
—— 2-(2-(1H-imidazol-4-yl)phenoxy)-N-phenylpropanamide 1300730-43-1 C18H17N3O2
2-(2-(1H-imidazol-4-yl)phenoxy)-N-phenylpropanamide
—— N-(4-(4-(4,6-dimethylpyridin-2-yl)piperazin-1-yl)phenyl)-2-(5-methyl-1-(2-methyloxazol-4-ylmethyl)-3-phenyl-1H-pyrrol-2-yl)-2-oxoacetamide 1192722-15-8 C35H36N6O3
N-(4-(4-(4,6-dimethylpyridin-2-yl)piperazin-1-yl)phenyl)-2-(5-methyl-1-(2-methyloxazol-4-ylmethyl)-3-phenyl-1H-pyrrol-2-yl)-2-oxoacetamide
—— N-[(3R)-1-cyano-3-pyrrolidinyl]-5-[(2,3-dihydroxypropyl)amino]-2-methylbenzenesulfonamide 1191409-27-4 C15H22N4O4S
N-[(3R)-1-cyano-3-pyrrolidinyl]-5-[(2,3-dihydroxypropyl)amino]-2-methylbenzenesulfonamide
—— 2-chloro-N-[(3R)-1-cyano-3-pyrrolidinyl]-5-[(1,3-thiazol-2-ylmethyl)amino]benzenesulfonamide 1191409-50-3 C15H16ClN5O2S2
2-chloro-N-[(3R)-1-cyano-3-pyrrolidinyl]-5-[(1,3-thiazol-2-ylmethyl)amino]benzenesulfonamide
—— 2,5-dibromo-N-[(3R)-1-cyano-3-pyrrolidinyl]-N-[(3,4-dichlorophenyl)methyl]benzenesulfonamide 1191925-75-3 C18H15Br2Cl2N3O2S
2,5-dibromo-N-[(3R)-1-cyano-3-pyrrolidinyl]-N-[(3,4-dichlorophenyl)methyl]benzenesulfonamide
—— N-{4-[5-(benzylsulfanyl)-1,3,4-thiadiazol-2-yl]phenyl}-1,4-benzodioxane-2-carboxamide 1608151-02-5 C24H19N3O3S2
N-{4-[5-(benzylsulfanyl)-1,3,4-thiadiazol-2-yl]phenyl}-1,4-benzodioxane-2-carboxamide
—— 1-methoxy-4-[2-methoxy-1-(4-methoxyphenyl)prop-1-enyl]benzene 101544-52-9 C18H20O3
1-methoxy-4-[2-methoxy-1-(4-methoxyphenyl)prop-1-enyl]benzene