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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-(3-Isoquinolin-4-ylpyridin-2-yl)sulfanyl-2-methylpropanoic acid 1352794-02-5 C18H16N2O2S
2-(3-Isoquinolin-4-ylpyridin-2-yl)sulfanyl-2-methylpropanoic acid
—— N-(4-methoxyphenyl)-3-methyl-4-phenyl-2,4-dioxobutyramide 124982-26-9 C18H17NO4
N-(4-methoxyphenyl)-3-methyl-4-phenyl-2,4-dioxobutyramide
—— N'-hydroxy-1-[6-[5-(methylamino)pyrazin-2-yl]pyridin-3-yl]cyclobutane-1-carboximidamide 1369513-91-6 C15H18N6O
N'-hydroxy-1-[6-[5-(methylamino)pyrazin-2-yl]pyridin-3-yl]cyclobutane-1-carboximidamide
—— (1aS,5aS)-2-(2,4-difluoro-phenyl)-1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalene-4-carboxylic acid ((R)-1-ethyl-pyrrolidin-2-ylmethyl)-amide 1268877-16-2 C21H24F2N4O
(1aS,5aS)-2-(2,4-difluoro-phenyl)-1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalene-4-carboxylic acid ((R)-1-ethyl-pyrrolidin-2-ylmethyl)-amide
—— 4,4'-bis(tert-butyl)-2,2'-bipyridinedichloronickel(II)(H2O)2 1264222-58-3 C18H28Cl2N2NiO2
4,4'-bis(tert-butyl)-2,2'-bipyridinedichloronickel(II)(H2O)2
—— CgP-PPhob 1319714-13-0 C18H30O3P2
CgP-PPhob
—— —— 1350477-75-6 C20H15BrN2O5
—— —— 1447937-44-1 C25H27N3O2S2
—— 5-(5-(1-(2-(benzo[d]thiazol-2-yl)hydrazono)ethyl)furan-2-yl)-2-nitrobenzoic acid 1135868-81-3 C20H14N4O5S
5-(5-(1-(2-(benzo[d]thiazol-2-yl)hydrazono)ethyl)furan-2-yl)-2-nitrobenzoic acid
—— 5-cyclopropyl-8-fluoro-1-nicotinoyl-2,3,5,6-tetrahydrobenzo[b][1,5]diazocin-4(1H)-one 1307894-14-9 C19H18FN3O2
5-cyclopropyl-8-fluoro-1-nicotinoyl-2,3,5,6-tetrahydrobenzo[b][1,5]diazocin-4(1H)-one
—— N-[3-[2-tert-butyl-5-[2-(methylamino)pyrimidin-4-yl]-1,3-thiazol-4-yl]-2-chloro-5-fluorophenyl]propane-1-sulfonamide 1353574-34-1 C21H25ClFN5O2S2
N-[3-[2-tert-butyl-5-[2-(methylamino)pyrimidin-4-yl]-1,3-thiazol-4-yl]-2-chloro-5-fluorophenyl]propane-1-sulfonamide
—— cyclopropyl-[4-[[4-[3-(1H-indol-5-yl)-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]methyl]piperazin-1-yl]methanone 1351476-96-4 C30H29N5O
cyclopropyl-[4-[[4-[3-(1H-indol-5-yl)-1H-pyrrolo[2,3-b]pyridin-5-yl]phenyl]methyl]piperazin-1-yl]methanone
—— —— 188002-46-2 C27H29NO4
—— 6-amino-7,12-dioxo-4-phenyl-2-thioxo-2,3,4,4a,7,12,12a,15-octahydrobenzo[g]pyrimido[5',4':4,5][1,2]thiazino[2,3-a]quinoline-5-carbonitrile 1133972-28-7 C25H17N5O2S2
6-amino-7,12-dioxo-4-phenyl-2-thioxo-2,3,4,4a,7,12,12a,15-octahydrobenzo[g]pyrimido[5',4':4,5][1,2]thiazino[2,3-a]quinoline-5-carbonitrile
—— (S)-[2-(diphenylphosphino)phenyl][(p-tolylsulfinyl)methyl]diphenylphosphonium hexafluorophosphate 1246638-48-1 C38H33OP2S*F6P
(S)-[2-(diphenylphosphino)phenyl][(p-tolylsulfinyl)methyl]diphenylphosphonium hexafluorophosphate
—— 2-{[2-(Hydroxymethyl)pyrrolidin-1-yl]methyl}cycloheptan-1-one hydrochloride 1909317-24-3 C13H24ClNO2
2-{[2-(Hydroxymethyl)pyrrolidin-1-yl]methyl}cycloheptan-1-one hydrochloride
—— 1-(2-methoxyethyl)-7-((N-(2-methoxymethylpyridin-3-ylmethyl)-N-(2-(2-methyl-4-oxo-4H-furo[3,2-c]pyridin-5-yl)ethyl)amino)methyl)-3,3-dimethyl-1,5-dihydrobenzo[b][1,4]diazepine-2,4-dione 1266561-35-6 C33H39N5O6
1-(2-methoxyethyl)-7-((N-(2-methoxymethylpyridin-3-ylmethyl)-N-(2-(2-methyl-4-oxo-4H-furo[3,2-c]pyridin-5-yl)ethyl)amino)methyl)-3,3-dimethyl-1,5-dihydrobenzo[b][1,4]diazepine-2,4-dione
—— 4-[[1-[[4-(1-methylethyl)-phenyl]sulfonyl]-5-trifluoromethyl-1H-indol-2-yl]methyl]-2-chlorobenzoic acid 1274942-39-0 C26H21ClF3NO4S
4-[[1-[[4-(1-methylethyl)-phenyl]sulfonyl]-5-trifluoromethyl-1H-indol-2-yl]methyl]-2-chlorobenzoic acid
—— 1-(4-(2,3-dimethylphenyl)piperazin-1-yl)-3-(9-(4-fluorophenyl)-8-methyl-9H-purin-6-ylamino)propan-2-ol 1307784-09-3 C27H32FN7O
1-(4-(2,3-dimethylphenyl)piperazin-1-yl)-3-(9-(4-fluorophenyl)-8-methyl-9H-purin-6-ylamino)propan-2-ol
—— methyl (Z)-2-(4H-indeno[1,2-b]thiophen-4-yl)-3-iodopropenoate 1022134-80-0 C15H11IO2S
methyl (Z)-2-(4H-indeno[1,2-b]thiophen-4-yl)-3-iodopropenoate
—— 4-(4-(tert-butyldimethylsilyloxy)phenyl)-2-methoxybutanenitrile 1015239-68-5 C17H27NO2Si
4-(4-(tert-butyldimethylsilyloxy)phenyl)-2-methoxybutanenitrile
—— 2-[2-(4-fluorophenyl)-6-oxopiperidin-1-yl]isoindoline-1,3-dione 1016971-32-6 C19H15FN2O3
2-[2-(4-fluorophenyl)-6-oxopiperidin-1-yl]isoindoline-1,3-dione
—— methyl (S)-1-(1-cyclopentyl-6-oxo-1,6-dihydropyridazin-3-yl)indoline-2-carboxylate 1187891-38-8 C19H21N3O3
methyl (S)-1-(1-cyclopentyl-6-oxo-1,6-dihydropyridazin-3-yl)indoline-2-carboxylate
—— 5-chloro-2-[[[3-[3-(trifluoromethyl)phenyl]imidazo[1,2-a]pyridin-8-yl]methyl]sulfonyl]-1H-benzimidazole 111477-10-2 C22H14ClF3N4O2S
5-chloro-2-[[[3-[3-(trifluoromethyl)phenyl]imidazo[1,2-a]pyridin-8-yl]methyl]sulfonyl]-1H-benzimidazole
—— US10266493, Example 5A 1352794-12-7 C14H14N2O2S
US10266493, Example 5A
—— 2-({[2-bromo-3,4-bis(methyloxy)phenyl]oxy}-methyl)-4-methylpyridine 1398697-16-9 C15H16BrNO3
2-({[2-bromo-3,4-bis(methyloxy)phenyl]oxy}-methyl)-4-methylpyridine
—— 3-{[5-(3-aminophenyl)-1H-pyrrolo[2,3-d]pyrimidin-4-yI]amino}-N-methylbenzenesulfonamide 1351090-55-5 C19H18N6O2S
3-{[5-(3-aminophenyl)-1H-pyrrolo[2,3-d]pyrimidin-4-yI]amino}-N-methylbenzenesulfonamide
—— rac-N-[2-{6-[3-(2-chloro-benzyl)-2-imino-7-methyl-2,3-dihydrobenzoimidazol-1-yl]-pyridazin-3-yl}-4-(1-hydroxy-ethyl)-phenyl]acetamide 1352873-58-5 C29H27ClN6O2
rac-N-[2-{6-[3-(2-chloro-benzyl)-2-imino-7-methyl-2,3-dihydrobenzoimidazol-1-yl]-pyridazin-3-yl}-4-(1-hydroxy-ethyl)-phenyl]acetamide
—— 2-Ethyl-1-propyl-8-[4-(4-trifluoromethyl-pyridin-2-yloxymethyl)-bicyclo[2.2.2]oct-1-yl]-1,7-dihydro-purin-6-one 1303955-33-0 C25H30F3N5O2
2-Ethyl-1-propyl-8-[4-(4-trifluoromethyl-pyridin-2-yloxymethyl)-bicyclo[2.2.2]oct-1-yl]-1,7-dihydro-purin-6-one
—— N-[4-methoxyphenylsulfonyl]-N'-[3-(3-methoxybenzyl)-1,2,4-thiadiazol-5-yl]propane-1,2-diamine 1029717-24-5 C20H24N4O4S2
N-[4-methoxyphenylsulfonyl]-N'-[3-(3-methoxybenzyl)-1,2,4-thiadiazol-5-yl]propane-1,2-diamine
—— methyl (1R,2R)-1-(3-acetyloxyphenyl)-2-(hydroxycarbamoyl)cyclopropane-1-carboxylate 1016164-74-1 C14H15NO6
methyl (1R,2R)-1-(3-acetyloxyphenyl)-2-(hydroxycarbamoyl)cyclopropane-1-carboxylate
—— 6-(8-(2,6-dichlorophenyl)-7H-purin-6-ylamino)nicotinonitrile 1334408-92-2 C17H9Cl2N7
6-(8-(2,6-dichlorophenyl)-7H-purin-6-ylamino)nicotinonitrile
—— 2-fluoro-3-(2-morpholin-4-yl-7-pyridin-4-yl-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-4-yl)-phenol trifluoroacetate 1007205-90-4 C2HF3O2*C21H20FN5O2
2-fluoro-3-(2-morpholin-4-yl-7-pyridin-4-yl-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-4-yl)-phenol trifluoroacetate
—— 7-[[[1(S)-1-(4-fluorophenyl)ethyl]methylamino]carbonyl]-3-phenyl-2-quinoxalinepentanoic acid 1383696-44-3 C29H28FN3O3
7-[[[1(S)-1-(4-fluorophenyl)ethyl]methylamino]carbonyl]-3-phenyl-2-quinoxalinepentanoic acid
—— N-((1S)-1-((1R)-2-((6'-(2,2-dimethylpropyl)-3,3-difluoro-3',4'-dihydrospiro[cyclobutane-1,2'-pyrano[2,3-b]pyridin]-4'-yl)amino)-1-hydroxyethyl)-3-buten-1-yl)-2-(methyloxy)acetamide 1091623-17-4 C25H37F2N3O4
N-((1S)-1-((1R)-2-((6'-(2,2-dimethylpropyl)-3,3-difluoro-3',4'-dihydrospiro[cyclobutane-1,2'-pyrano[2,3-b]pyridin]-4'-yl)amino)-1-hydroxyethyl)-3-buten-1-yl)-2-(methyloxy)acetamide
—— (E)-N-(tert-butoxycarbonyl)-3-chloro-2-phenylprop-2-en-amine 1228964-38-2 C14H18ClNO2
(E)-N-(tert-butoxycarbonyl)-3-chloro-2-phenylprop-2-en-amine
—— —— 1058722-07-8 C12H18N2O2
—— —— 1013396-83-2 C19H25BF2N2O2
—— —— 1032401-36-7 C20H29NO2
—— —— 1236511-07-1 C43H64N12O12S
—— 1-((2R,3S)-3-Methyl-1,4-dioxa-spiro[4.5]dec-2-yl)-2-(pyridine-2-sulfinyl)-but-3-en-1-ol 107996-95-2 C18H25NO4S
1-((2R,3S)-3-Methyl-1,4-dioxa-spiro[4.5]dec-2-yl)-2-(pyridine-2-sulfinyl)-but-3-en-1-ol
—— —— 1314145-16-8 C12H9Br2Cl
—— 3-methyl-1-(4-methyl-1H-benzimidazol-2-yl)-4-(phenylmethyl)-1H-pyrazol-5-ol 1453097-14-7 C19H18N4O
3-methyl-1-(4-methyl-1H-benzimidazol-2-yl)-4-(phenylmethyl)-1H-pyrazol-5-ol
—— 3-(4-chlorophenyl)-2,3-dihydro-6-hydroxyinden-1-one 1274878-21-5 C15H11ClO2
3-(4-chlorophenyl)-2,3-dihydro-6-hydroxyinden-1-one
—— 2-(6-{4-[1-(propan-2-yl)piperidin-4-yl]-1,4-diazepan-1-yl}pyridine-2-yl)-1H-1,3-benzodiazole 1373269-80-7 C25H34N6
2-(6-{4-[1-(propan-2-yl)piperidin-4-yl]-1,4-diazepan-1-yl}pyridine-2-yl)-1H-1,3-benzodiazole
—— 1-[4,6-Bis(2,2,2-trifluoroethoxy)pyrimidin-2-yl]-3-(4-bromo-2,6-dichlorophenyl)urea 1138595-08-0 C15H9BrCl2F6N4O3
1-[4,6-Bis(2,2,2-trifluoroethoxy)pyrimidin-2-yl]-3-(4-bromo-2,6-dichlorophenyl)urea
—— ethyl N-[[4,6-bis(2,2,2-trifluoroethoxy)pyrimidin-2-yl]-(phenylmethoxymethyl)carbamoyl]-N-[4-(trifluoromethyl)phenyl]carbamate 1138591-94-2 C27H23F9N4O6
ethyl N-[[4,6-bis(2,2,2-trifluoroethoxy)pyrimidin-2-yl]-(phenylmethoxymethyl)carbamoyl]-N-[4-(trifluoromethyl)phenyl]carbamate
—— (2R)-N-(5-carbamoyl-2-fluorophenyl)-2-[4-[(4-chlorophenyl)methyl]-5-methyl-1,2,4-triazol-3-yl]pyrrolidine-1-carboxamide 1140491-74-2 C22H22ClFN6O2
(2R)-N-(5-carbamoyl-2-fluorophenyl)-2-[4-[(4-chlorophenyl)methyl]-5-methyl-1,2,4-triazol-3-yl]pyrrolidine-1-carboxamide
—— rac-{2-hydroxy-3-[1-(2-fluoro-5-trifluoromethylphenyl)cyclopropyl]-2-phenylethynylpropionic acid} (3,4-dichlorophenyl)amide 1100375-31-2 C27H19Cl2F4NO2
rac-{2-hydroxy-3-[1-(2-fluoro-5-trifluoromethylphenyl)cyclopropyl]-2-phenylethynylpropionic acid} (3,4-dichlorophenyl)amide
—— trimethyl-[3-[(2R,3S)-3-(phenylmethoxymethyl)oxiran-2-yl]-3-trimethylsilyloxyundec-1-en-2-yl]silane 112164-80-4 C27H48O3Si2
trimethyl-[3-[(2R,3S)-3-(phenylmethoxymethyl)oxiran-2-yl]-3-trimethylsilyloxyundec-1-en-2-yl]silane