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中文名称 英文名称 CAS号 化学式 结构式图片
—— —— 1335556-53-0 C26H30FN3O7
—— —— 1335556-46-1 C28H35N3O8
—— —— 1208345-91-8 C20H12Cl3F7N4O
—— —— 1112120-39-4 C22H19N3O4
—— —— 1304433-54-2 C17H14ClF3N6
—— —— 1338581-52-4 C20H22N4OS
—— —— 1309982-94-2 Br*C10H13N2
—— N-EMK8-II-C 1315451-46-7 C42H76N10O13S4
N-EMK8-II-C
—— —— 1376938-64-5 C13H9ClO2
—— N2-(4-fluorobenzyl)-N4-{2-[1-(propan-2-yl)piperidin-4-yl]ethyl}-N6-[3-(trifluoromethyl)phenyl]-1,3,5-triazine-2,4,6-triamine 1174125-82-6 C27H33F4N7
N2-(4-fluorobenzyl)-N4-{2-[1-(propan-2-yl)piperidin-4-yl]ethyl}-N6-[3-(trifluoromethyl)phenyl]-1,3,5-triazine-2,4,6-triamine
—— N-(4-carbamoylphenyl)-5-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidine-3-carboxamide 1224940-45-7 C20H17N7O2
N-(4-carbamoylphenyl)-5-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (5R)-5-[2-[4-(5-amino-1H-pyrazol-4-yl)phenyl]ethynyl]-5-[(5-methoxy-3-oxo-1H-isoindol-2-yl)methyl]imidazolidine-2,4-dione 1226989-79-2 C24H20N6O4
(5R)-5-[2-[4-(5-amino-1H-pyrazol-4-yl)phenyl]ethynyl]-5-[(5-methoxy-3-oxo-1H-isoindol-2-yl)methyl]imidazolidine-2,4-dione
—— 5-amino-pyrazolo[1,5-a]pyrimidine-3-carboxylic acid [2-(2-ethyl-phenyl)-5-methyl-2H-pyrazol-3-yl]-amide 1224944-31-3 C19H19N7O
5-amino-pyrazolo[1,5-a]pyrimidine-3-carboxylic acid [2-(2-ethyl-phenyl)-5-methyl-2H-pyrazol-3-yl]-amide
—— 3-(2,2-dimethylpropanoyl)-2-(2-fluorophenyl)-4-hydroxy-1-[4-(1,2-oxazol-3-yl)phenyl]-2H-pyrrol-5-one 1067184-83-1 C24H21FN2O4
3-(2,2-dimethylpropanoyl)-2-(2-fluorophenyl)-4-hydroxy-1-[4-(1,2-oxazol-3-yl)phenyl]-2H-pyrrol-5-one
—— methyl 5-(N-(5-cyclopropyl-3-(methylcarbamoyl)-2-p-tolylfuro[2,3-b]pyridin-6-yl)methylsulfonamido)-2-methylenepentanoate 1345182-30-0 C27H31N3O6S
methyl 5-(N-(5-cyclopropyl-3-(methylcarbamoyl)-2-p-tolylfuro[2,3-b]pyridin-6-yl)methylsulfonamido)-2-methylenepentanoate
—— —— 1298098-49-3 C25H29FN6O2
—— sodium 3-(4-(5-(1-ethyl-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-3-yl)-1,2,4-oxadiazol-3-yl)-2,6-dimethylphenyl)propanoate 1233498-23-1 C24H29N4O3*Na
sodium 3-(4-(5-(1-ethyl-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-3-yl)-1,2,4-oxadiazol-3-yl)-2,6-dimethylphenyl)propanoate
—— N-(5-(2-amino-8-(trans-4-(2-hydroxyethoxy)cyclohexyl)-4-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)-2-methoxypyridin-3-yl)methanesulfonamide 1550189-72-4 C23H30N6O6S
N-(5-(2-amino-8-(trans-4-(2-hydroxyethoxy)cyclohexyl)-4-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)-2-methoxypyridin-3-yl)methanesulfonamide
—— [7-hydroxy-6-(6-methylamino-pyridine-3-carbonyl)-4,5-dihydro-benzothiazol-2-yl]-thiocarbamic acid S-ethyl ester 1187368-42-8 C17H18N4O3S2
[7-hydroxy-6-(6-methylamino-pyridine-3-carbonyl)-4,5-dihydro-benzothiazol-2-yl]-thiocarbamic acid S-ethyl ester
—— —— 1181213-92-2 C16H27NO7
—— —— 1323985-20-1 C19H13ClF5NO2
—— 1-((1R,3s,5S)-3-(7-amino-3-(5-hydroxy-6-phenylpyridin-3-yl)-6-(methylsulfonyl)pyrazolo[1,5-a]pyrimidin-5-yl)-8-azabicyclo[3.2.1]octan-8-yl)-2-hydroxyethanone 1319250-58-2 C27H28N6O5S
1-((1R,3s,5S)-3-(7-amino-3-(5-hydroxy-6-phenylpyridin-3-yl)-6-(methylsulfonyl)pyrazolo[1,5-a]pyrimidin-5-yl)-8-azabicyclo[3.2.1]octan-8-yl)-2-hydroxyethanone
—— —— 1186105-13-4 C31H43N5O3
—— —— 1207332-13-5 C23H27N3O3
—— 7-({4-[(3-methoxybenzoyl)amino]piperidin-1-yl}methyl)-N-(2-methoxyethyl)-2-naphthamide hydrochloride 1018072-75-7 C28H33N3O4*ClH
7-({4-[(3-methoxybenzoyl)amino]piperidin-1-yl}methyl)-N-(2-methoxyethyl)-2-naphthamide hydrochloride
—— —— 1170069-32-5 C67H77Cl2N9O23
—— (±)-4-(2-allyloxy-5-chloro-phenyl)-6,7-dihydro-4H-thiazolo[5,4-c]pyridine-5-carboxylic acid tert-butyl ester 1531635-93-4 C20H23ClN2O3S
(±)-4-(2-allyloxy-5-chloro-phenyl)-6,7-dihydro-4H-thiazolo[5,4-c]pyridine-5-carboxylic acid tert-butyl ester
—— 1-(5-((1R,3s,5S)-8-(4H-1,2,4-triazole-3-carbonyl)-8-azabicyclo[3.2.1]octan-3-yl)-7-amino-3-(6-(4-ethoxyphenyl)pyridin-3-yl)pyrazolo[1,5-a]pyrimidin-6-yl)ethanone 1319249-00-7 C31H31N9O3
1-(5-((1R,3s,5S)-8-(4H-1,2,4-triazole-3-carbonyl)-8-azabicyclo[3.2.1]octan-3-yl)-7-amino-3-(6-(4-ethoxyphenyl)pyridin-3-yl)pyrazolo[1,5-a]pyrimidin-6-yl)ethanone
—— —— 1280182-58-2 C15H17N3O4S
—— 1-(5-((1R,3s,5S)-8-(4H-1,2,4-triazol-3-ylsulfonyl)-8-azabicyclo[3.2.1]octan-3-yl)-7-amino-3-(6-phenylpyridin-3-yl)pyrazolo[1,5-a]pyrimidin-6-yl)ethanone 1319248-68-4 C28H27N9O3S
1-(5-((1R,3s,5S)-8-(4H-1,2,4-triazol-3-ylsulfonyl)-8-azabicyclo[3.2.1]octan-3-yl)-7-amino-3-(6-phenylpyridin-3-yl)pyrazolo[1,5-a]pyrimidin-6-yl)ethanone
—— —— 1323984-36-6 C19H14F2N2O2
—— methyl 1-methyl-4-nitro-5-propyl-1H-pyrazole-3-carboxylate 1222955-90-9 C9H13N3O4
methyl 1-methyl-4-nitro-5-propyl-1H-pyrazole-3-carboxylate
—— N-(4-(2-(5-amino-7-(3-(methylamino)azetidin-1-yl)-2H-pyrazolo[4,3-d]pyrimidin-2-yl)ethyl)phenyl)acetamide 1222955-29-4 C19H24N8O
N-(4-(2-(5-amino-7-(3-(methylamino)azetidin-1-yl)-2H-pyrazolo[4,3-d]pyrimidin-2-yl)ethyl)phenyl)acetamide
—— —— 1532510-65-8 C27H22Cl2F4N2O4
—— 4',6'-O-p-dimethylaminobenzylideneparomomycin 1043874-59-4 C32H54N6O14
4',6'-O-p-dimethylaminobenzylideneparomomycin
—— α-(5-cyano-2,4-dioxo-3,4-dihydro-2<i>H</i>-pyrimidin-1-yl)-isovaleric acid 102495-42-1 C10H11N3O4
α-(5-cyano-2,4-dioxo-3,4-dihydro-2<i>H</i>-pyrimidin-1-yl)-isovaleric acid
—— ((1R,3s,5S)-3-(7-amino-6-(methylsulfonyl)-3-(6-phenylpyridin-3-yl)pyrazolo[1,5-a]pyrimidin-5-yl)-8-azabicyclo[3.2.1]octan-8-yl)(4-aminopyrimidin-5-yl)methanone 1319251-74-5 C30H29N9O3S
((1R,3s,5S)-3-(7-amino-6-(methylsulfonyl)-3-(6-phenylpyridin-3-yl)pyrazolo[1,5-a]pyrimidin-5-yl)-8-azabicyclo[3.2.1]octan-8-yl)(4-aminopyrimidin-5-yl)methanone
—— 3-cyclobutyl-7-((3R)-3-(methylamino)pyrrolidin-1-yl)-2H-pyrazolo[4,3-d]pyrimidin-5-amine 1222954-03-1 C14H21N7
3-cyclobutyl-7-((3R)-3-(methylamino)pyrrolidin-1-yl)-2H-pyrazolo[4,3-d]pyrimidin-5-amine
—— —— 1323986-20-4 C19H14BrF4NO3
—— 3-endo-(8-{2-[(2-ethylbutyl)-((R)-2,3-dihydroxy-propionyl)amino]ethyl}-8-azabicyclo[3.2.1]oct-3-yl)-benzamide trifluoroacetate 1125454-05-8 C25H39N3O4
3-endo-(8-{2-[(2-ethylbutyl)-((R)-2,3-dihydroxy-propionyl)amino]ethyl}-8-azabicyclo[3.2.1]oct-3-yl)-benzamide trifluoroacetate
—— 2-(2-ethoxyphenyl)-N-(6-methyl-3-(3-sulfamoylphenyl)-1H-indazol-5-yl)acetamide 1338793-86-4 C24H24N4O4S
2-(2-ethoxyphenyl)-N-(6-methyl-3-(3-sulfamoylphenyl)-1H-indazol-5-yl)acetamide
—— rac-tert-butyl {1-[({8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridin-3-yl}-carbonyl)amino]propan-2-yl}carbamate trifluoroacetate 1609344-93-5 C2HF3O2*C25H30F2N4O4
rac-tert-butyl {1-[({8-[(2,6-difluorobenzyl)oxy]-2,6-dimethylimidazo[1,2-a]pyridin-3-yl}-carbonyl)amino]propan-2-yl}carbamate trifluoroacetate
—— —— 1340545-47-2 C59H39N3S
—— N-((4-(aminomethyl)cyclohexyl)methyl)-5-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidine-3-carboxamide 1224940-72-0 C21H27N7O
N-((4-(aminomethyl)cyclohexyl)methyl)-5-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidine-3-carboxamide
—— tert-butyl 4-[5-fluoro-4-(4-mesylbenzoyl)pyrrolo[2,3-d]pyrimidin-7-yl]piperidine-1-carboxylate 1236282-37-3 C24H27FN4O5S
tert-butyl 4-[5-fluoro-4-(4-mesylbenzoyl)pyrrolo[2,3-d]pyrimidin-7-yl]piperidine-1-carboxylate
—— 6-[3-(1,1,2,2-tetrafluoroethoxy)phenyl]-3[2H]pyridazinone 101975-09-1 C12H8F4N2O2
6-[3-(1,1,2,2-tetrafluoroethoxy)phenyl]-3[2H]pyridazinone
—— [6-[(7-methoxynaphthalen-2-yl)amino]-5-methylpyrimidin-4-yl]-[4-[[(3S,4S)-3-methoxyoxan-4-yl]amino]piperidin-1-yl]methanone 1349113-41-2 C28H35N5O4
[6-[(7-methoxynaphthalen-2-yl)amino]-5-methylpyrimidin-4-yl]-[4-[[(3S,4S)-3-methoxyoxan-4-yl]amino]piperidin-1-yl]methanone
—— N-((2R,3R)-3-methoxy-1-(pyrrolidin-1-yl)butan-2-yl)-N,3-dimethylbenzamide 1380100-58-2 C18H28N2O2
N-((2R,3R)-3-methoxy-1-(pyrrolidin-1-yl)butan-2-yl)-N,3-dimethylbenzamide
—— 2-(4-(Methoxycarbonyl)oxazol-5-yl)-4-phenoxybenzoic acid 1421312-31-3 C18H13NO6
2-(4-(Methoxycarbonyl)oxazol-5-yl)-4-phenoxybenzoic acid
—— —— 1277127-99-7 C16H17ClN2O5