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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-bromo-7-iodo-2-[4-(morpholin-4-ylmethyl)phenyl]-3H-imidazo[4,5-b]pyridine 1069131-89-0 C17H16BrIN4O
6-bromo-7-iodo-2-[4-(morpholin-4-ylmethyl)phenyl]-3H-imidazo[4,5-b]pyridine
—— [(2-(N,N-dimethylaminomethyl)phenyl)tin(IV)(phenyl)2(trifluoromethanesulfonate)] 1373498-91-9 C22H22F3NO3SSn
[(2-(N,N-dimethylaminomethyl)phenyl)tin(IV)(phenyl)2(trifluoromethanesulfonate)]
—— —— 1375896-03-9 C21H20ClF2N3O
—— —— 1378869-63-6 C20H12F9N5O3
—— —— 1312300-35-8 C16H24N2O5Si
—— (4S)-N-{(3S)-1-[2-cyano-4-(3-thienyl)phenyl]-3-pyrrolidinyl}-4-fluoro-L-prolinamide hydrochloride 1269409-25-7 C20H21FN4OS*ClH
(4S)-N-{(3S)-1-[2-cyano-4-(3-thienyl)phenyl]-3-pyrrolidinyl}-4-fluoro-L-prolinamide hydrochloride
—— 4-(2-(cyclohexylbutoxy))-3-nitrobenzaldehyde 1234323-32-0 C17H23NO4
4-(2-(cyclohexylbutoxy))-3-nitrobenzaldehyde
—— —— 1364522-98-4 C31H30Cl2N6O4
—— 2-(2,5-dimethoxyphenyl)-5,5-dimethyl-1,3,2-dioxaborinane 1188303-90-3 C13H19BO4
2-(2,5-dimethoxyphenyl)-5,5-dimethyl-1,3,2-dioxaborinane
—— 5-chloro-2-(3-ethylquinoxalin-2-yl)-N-(tetrahydro-2H-pyran-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine 1332728-28-5 C21H21ClN6O
5-chloro-2-(3-ethylquinoxalin-2-yl)-N-(tetrahydro-2H-pyran-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
—— N2-(2-chloro-benzyl)-N5-(3-pyridin-2-yl-propyl)-pyrido[4,3-d]pyrimidine-2,5-diamine 1228564-86-0 C22H21ClN6
N2-(2-chloro-benzyl)-N5-(3-pyridin-2-yl-propyl)-pyrido[4,3-d]pyrimidine-2,5-diamine
—— (±)-{4-chloro-2-[5-(2-fluoro-benzylcarbamoyl)-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridin-4-yl]-phenoxy}-acetic acid 1531634-51-1 C22H19ClFN3O4S
(±)-{4-chloro-2-[5-(2-fluoro-benzylcarbamoyl)-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridin-4-yl]-phenoxy}-acetic acid
—— methyl 4-(2-((R)-3,3-difluoro-5-((S,E)-3-hydroxyoct-1-en-1-yl)-2-oxopyrrolidin-1-yl)ethyl)benzoate 1544281-68-6 C22H29F2NO4
methyl 4-(2-((R)-3,3-difluoro-5-((S,E)-3-hydroxyoct-1-en-1-yl)-2-oxopyrrolidin-1-yl)ethyl)benzoate
—— (S)-2-((S)-3-(4-chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboximidamido)-3-hydroxypropanamide 1549792-46-2 C25H23Cl2N5O4S
(S)-2-((S)-3-(4-chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-4-phenyl-4,5-dihydro-1H-pyrazole-1-carboximidamido)-3-hydroxypropanamide
—— N-(3-methyl-1-((6-methylpyridin-2-yl)methyl)-1H-indazol-4-yl)-4-(4-(1-methylpiperidin-4-yl)phenylamino)thieno[3,2-d]pyrimidine-7-carboxamide 1527518-12-2 C34H34N8OS
N-(3-methyl-1-((6-methylpyridin-2-yl)methyl)-1H-indazol-4-yl)-4-(4-(1-methylpiperidin-4-yl)phenylamino)thieno[3,2-d]pyrimidine-7-carboxamide
—— (pivaloyloxy)methyl 6α-<1(R)-<<<(p-nitrobenzyl)oxy>carbonyl>oxy>ethyl>-1-oxopenicillanate 124093-84-1 C24H30N2O11S
(pivaloyloxy)methyl 6α-<1(R)-<<<(p-nitrobenzyl)oxy>carbonyl>oxy>ethyl>-1-oxopenicillanate
—— ((triphos)NiBr)(ClO4) 118084-01-8 C41H39BrNiP3*ClO4
((triphos)NiBr)(ClO4)
—— fac-[Re(CO)3(η(3)-Ph2P(CH2)2P(Ph)(CH2)2PPh2)]Cl 186667-59-4 C37H33O3P3Re*Cl
fac-[Re(CO)3(η(3)-Ph2P(CH2)2P(Ph)(CH2)2PPh2)]Cl
—— diethyl 3,3'-(1,3-phenylenebis(ethyne-2,1-diyl))dibenzoate 1276019-56-7 C28H22O4
diethyl 3,3'-(1,3-phenylenebis(ethyne-2,1-diyl))dibenzoate
—— (2-Formylphenyl) 4-chloro-3-nitrobenzenesulfonate 1334304-65-2 C13H8ClNO6S
(2-Formylphenyl) 4-chloro-3-nitrobenzenesulfonate
—— 1-[(2R,4S,5S)-4-[(2S)-2-[(3aR,4R,6S,6aS)-2,2-dimethyl-4-(5-methyl-2,4-dioxopyrimidin-1-yl)-3a,4,6,6a-tetrahydrofuro[3,4-d][1,3]dioxol-6-yl]-4-oxo-1,3-thiazolidin-3-yl]-5-(hydroxymethyl)oxolan-2-yl]-5-methylpyrimidine-2,4-dione 1330063-26-7 C25H31N5O10S
1-[(2R,4S,5S)-4-[(2S)-2-[(3aR,4R,6S,6aS)-2,2-dimethyl-4-(5-methyl-2,4-dioxopyrimidin-1-yl)-3a,4,6,6a-tetrahydrofuro[3,4-d][1,3]dioxol-6-yl]-4-oxo-1,3-thiazolidin-3-yl]-5-(hydroxymethyl)oxolan-2-yl]-5-methylpyrimidine-2,4-dione
—— 2-[1-[4,4-Bis(4-fluorophenyl)butyl]piperidin-4-yl]-1,3-dihydroisoindole 1347746-90-0 C29H32F2N2
2-[1-[4,4-Bis(4-fluorophenyl)butyl]piperidin-4-yl]-1,3-dihydroisoindole
—— (3S,4S)-1-[(2-methylpropan-2-yl)oxycarbonyl]-4-[[6-(2,2,2-trifluoroethoxy)-15,22-dioxa-3,5,7,9,29-pentazatetracyclo[21.2.2.14,8.110,14]nonacosa-1(26),4(29),5,7,10(28),11,13,23(27),24-nonaene-13-carbonyl]amino]pyrrolidine-3-carboxylic acid 1346651-09-9 C35H42F3N7O8
(3S,4S)-1-[(2-methylpropan-2-yl)oxycarbonyl]-4-[[6-(2,2,2-trifluoroethoxy)-15,22-dioxa-3,5,7,9,29-pentazatetracyclo[21.2.2.14,8.110,14]nonacosa-1(26),4(29),5,7,10(28),11,13,23(27),24-nonaene-13-carbonyl]amino]pyrrolidine-3-carboxylic acid
—— 9-Chloro-6-(2-pyrrolidin-1-ylethoxy)indeno[1,2-c]quinolin-11-one 1346622-27-2 C22H19ClN2O2
9-Chloro-6-(2-pyrrolidin-1-ylethoxy)indeno[1,2-c]quinolin-11-one
—— 1-(3-chloro-5-(trifluoromethyl)pyridin-2-yl)pyrrolidine-2-carboxylic acid 1188435-80-4 C11H10ClF3N2O2
1-(3-chloro-5-(trifluoromethyl)pyridin-2-yl)pyrrolidine-2-carboxylic acid
—— [2-cyclopropyl-5-methyl-6-[3-(trifluoromethyl)anilino]pyrimidin-4-yl]-[4-[[(3R,4R)-3-methoxyoxan-4-yl]amino]piperidin-1-yl]methanone 1349113-90-1 C27H34F3N5O3
[2-cyclopropyl-5-methyl-6-[3-(trifluoromethyl)anilino]pyrimidin-4-yl]-[4-[[(3R,4R)-3-methoxyoxan-4-yl]amino]piperidin-1-yl]methanone
—— ethyl 7-({2-[3-(dimethylcarbamoyl)-4-({[6-methoxy-4'-(trifluoromethyl)biphenyl-2-yl]carbonyl}amino)phenyl]acetoxy}methyl)-6,7-dihydro-5H-cyclopenta[b]pyridine-7-carboxylate 1350469-35-0 C38H36F3N3O7
ethyl 7-({2-[3-(dimethylcarbamoyl)-4-({[6-methoxy-4'-(trifluoromethyl)biphenyl-2-yl]carbonyl}amino)phenyl]acetoxy}methyl)-6,7-dihydro-5H-cyclopenta[b]pyridine-7-carboxylate
—— 6-(2-(diethylamino)ethoxy)-2-9-dimethoxy-11H-indeno[1,2-c]quinolin-11-one 1346622-32-9 C24H26N2O4
6-(2-(diethylamino)ethoxy)-2-9-dimethoxy-11H-indeno[1,2-c]quinolin-11-one
—— 4-(furan-2-yl)-3-methyl-2H-pyrazolo[3,4-c]pyridine 1347758-94-4 C11H9N3O
4-(furan-2-yl)-3-methyl-2H-pyrazolo[3,4-c]pyridine
—— 2-{5-{[4-butyl-2-isopropyl-1-(5-methoxypyrimidin-2-yl)-6-oxo-1,6-dihydropyrimidin-5-yl]methyl}pyridin-2-yl}-N'-hydroxybenzimidamide 1283715-72-9 C29H33N7O3
2-{5-{[4-butyl-2-isopropyl-1-(5-methoxypyrimidin-2-yl)-6-oxo-1,6-dihydropyrimidin-5-yl]methyl}pyridin-2-yl}-N'-hydroxybenzimidamide
—— Allocernuin 15216-34-9 C16H26N2O
Allocernuin
—— 5-[5-Amino-6-[5-[4-(methylaminomethyl)phenyl]-1,3,4-oxadiazol-2-yl]pyrazin-2-yl]-1-(3-aminopropyl)pyridin-2-one 1349731-23-2 C22H24N8O2
5-[5-Amino-6-[5-[4-(methylaminomethyl)phenyl]-1,3,4-oxadiazol-2-yl]pyrazin-2-yl]-1-(3-aminopropyl)pyridin-2-one
—— Synthesis of 2-[5-[5-amino-6-[3-[4-[(cyclopropylamino)methyl]-2-fluoro-phenyl]isoxazol-5-yl]pyrazin-2-yl]-2-oxo-1-pyridyl]-2-ethyl-butanenitrile 1349733-44-3 C26H26FN7O2
Synthesis of 2-[5-[5-amino-6-[3-[4-[(cyclopropylamino)methyl]-2-fluoro-phenyl]isoxazol-5-yl]pyrazin-2-yl]-2-oxo-1-pyridyl]-2-ethyl-butanenitrile
—— [5-(4-Methylphenyl)pyridin-2-yl]methanol 1311151-83-3 C13H13NO
[5-(4-Methylphenyl)pyridin-2-yl]methanol
—— Methyl 5-(pyrrolidin-1-yl)pyridine-3-carboxylate 1414866-57-1 C11H14N2O2
Methyl 5-(pyrrolidin-1-yl)pyridine-3-carboxylate
—— 1-(4-(6-(N-(2-(piperazin-1-yl)ethyl)aminocarbonyl)-1H-indazol-4-yl)phenyl)-3-(3-(trifluoromethoxy)phenyl)urea 1285531-69-2 C28H28F3N7O3
1-(4-(6-(N-(2-(piperazin-1-yl)ethyl)aminocarbonyl)-1H-indazol-4-yl)phenyl)-3-(3-(trifluoromethoxy)phenyl)urea
—— 7-fluoro-5-(4-fluoro-phenyl)-3-methyl-1,3-dihydro-2,3,4-benzothiadiazepine-2,2-dioxide 1282510-52-4 C15H12F2N2O2S
7-fluoro-5-(4-fluoro-phenyl)-3-methyl-1,3-dihydro-2,3,4-benzothiadiazepine-2,2-dioxide
—— 2-chloro-6-(2-fluorophenyl)-7-hydroxy-1-(4-methylphenyl)-1,4-dihydro-5H-pyrrolo[3,2-b]pyridin-5-one 1272673-35-4 C20H14ClFN2O2
2-chloro-6-(2-fluorophenyl)-7-hydroxy-1-(4-methylphenyl)-1,4-dihydro-5H-pyrrolo[3,2-b]pyridin-5-one
—— 2-(3-pyridin-3-ylphenyl)-N-[3-(trifluoromethyl)imidazo[5,1-b][1,3]thiazol-7-yl]acetamide 1279721-36-6 C19H13F3N4OS
2-(3-pyridin-3-ylphenyl)-N-[3-(trifluoromethyl)imidazo[5,1-b][1,3]thiazol-7-yl]acetamide
—— methyl 3-benzyl-3H-pyrrolo[1,2-a][1,2,3]triazolo[4,5-c]quinoline-10-carboxylate 1254221-63-0 C21H16N4O2
methyl 3-benzyl-3H-pyrrolo[1,2-a][1,2,3]triazolo[4,5-c]quinoline-10-carboxylate
—— methyl 3-hydroxy-4-(prop-2-yn-1-yloxy)benzoate 1356154-73-8 C11H10O4
methyl 3-hydroxy-4-(prop-2-yn-1-yloxy)benzoate
—— 5-[5-amino-6-[3-[4-(methylaminomethyl)phenyl]-1,2-oxazol-5-yl]pyrazin-2-yl]-3-cyclohexyl-1H-pyridin-2-one 1349733-14-7 C26H28N6O2
5-[5-amino-6-[3-[4-(methylaminomethyl)phenyl]-1,2-oxazol-5-yl]pyrazin-2-yl]-3-cyclohexyl-1H-pyridin-2-one
—— (S)-3-(2,5-difluoro-4-(methylsulfonyl)phenylamino)-1'-(5-(trifluoromethyl)pyridin-2-yl)-[1,4'-bipiperidin]-2-one 1351166-66-9 C23H25F5N4O3S
(S)-3-(2,5-difluoro-4-(methylsulfonyl)phenylamino)-1'-(5-(trifluoromethyl)pyridin-2-yl)-[1,4'-bipiperidin]-2-one
—— 5-(4-isopropylsulfonylphenyl)-3-[2-(2-thienyl)ethynyl]pyrazin-2-amine 1350351-20-0 C19H17N3O2S2
5-(4-isopropylsulfonylphenyl)-3-[2-(2-thienyl)ethynyl]pyrazin-2-amine
—— [[[4-(2-Methoxyphenyl)pyridin-2-yl]amino]-phosphonomethyl]phosphonic acid 1350451-99-8 C13H16N2O7P2
[[[4-(2-Methoxyphenyl)pyridin-2-yl]amino]-phosphonomethyl]phosphonic acid
—— 1-(n-butyl)-3-hydroxy-2-oxo-1,2-dihydro-4-quinolinecarboxylic acid 139094-87-4 C14H15NO4
1-(n-butyl)-3-hydroxy-2-oxo-1,2-dihydro-4-quinolinecarboxylic acid
—— 11-bromo-1,2,3,5,6,7,14,14a-octahydrobenzo[4,5]imidazo[1,2-a]pyrrolo[2,1-d][1,5]diazocine 1272321-45-5 C15H18BrN3
11-bromo-1,2,3,5,6,7,14,14a-octahydrobenzo[4,5]imidazo[1,2-a]pyrrolo[2,1-d][1,5]diazocine
—— 1-(1H-benzo[d]imidazol-5-yl)-5-(4-propoxyphenyl)pyrrolidin-2-one 1276024-12-4 C20H21N3O2
1-(1H-benzo[d]imidazol-5-yl)-5-(4-propoxyphenyl)pyrrolidin-2-one
—— 3-(N-ethyl-N-methylsulfamoylamino)-2,6-difluoro-N-(2-methoxypyrazolo[1,5-a]pyrimidin-6-yl)benzamide 1269515-83-4 C17H18F2N6O4S
3-(N-ethyl-N-methylsulfamoylamino)-2,6-difluoro-N-(2-methoxypyrazolo[1,5-a]pyrimidin-6-yl)benzamide
—— N-ethyl-4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]-N-[(2-propan-2-ylpyrimidin-4-yl)methyl]benzamide 1269614-88-1 C29H36N4O2
N-ethyl-4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]-N-[(2-propan-2-ylpyrimidin-4-yl)methyl]benzamide