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中文名称 英文名称 CAS号 化学式 结构式图片
—— [4-[[(3S,4S)-3-methoxyoxan-4-yl]amino]piperidin-1-yl]-[5-methoxy-6-[3-(trifluoromethyl)anilino]pyrimidin-4-yl]methanone 1349113-03-6 C24H30F3N5O4
[4-[[(3S,4S)-3-methoxyoxan-4-yl]amino]piperidin-1-yl]-[5-methoxy-6-[3-(trifluoromethyl)anilino]pyrimidin-4-yl]methanone
—— Tert-butyl 4-(2-methoxyethyl)-6-methyl-3-oxo-6,7,9,10-tetrahydro-[1,4]oxazino[2,3-h][3]benzazepine-8-carboxylate 1334434-33-1 C21H30N2O5
Tert-butyl 4-(2-methoxyethyl)-6-methyl-3-oxo-6,7,9,10-tetrahydro-[1,4]oxazino[2,3-h][3]benzazepine-8-carboxylate
—— 5-methoxy-N,N,2-trimethyl-4-[[4-[[4-methyl-2-[methyl(methylsulfonyl)amino]phenyl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamide 1226992-68-2 C26H31F3N6O4S
5-methoxy-N,N,2-trimethyl-4-[[4-[[4-methyl-2-[methyl(methylsulfonyl)amino]phenyl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamide
—— Ethyl 3-(5-cyano-2-phenylbenzimidazol-1-yl)benzoate 1106942-86-2 C23H17N3O2
Ethyl 3-(5-cyano-2-phenylbenzimidazol-1-yl)benzoate
—— 2-(4-fluorophenyl)-5-[2-methoxy-4-[[4-(trifluoromethyl)phenyl]methoxy]phenyl]-1H-imidazole 1239261-66-5 C24H18F4N2O2
2-(4-fluorophenyl)-5-[2-methoxy-4-[[4-(trifluoromethyl)phenyl]methoxy]phenyl]-1H-imidazole
—— Tert-butyl 7-(1,3-dimethoxy-1-oxopropan-2-yl)oxy-8-nitro-1,2,4,5-tetrahydro-3-benzazepine-3-carboxylate 1334434-93-3 C20H28N2O8
Tert-butyl 7-(1,3-dimethoxy-1-oxopropan-2-yl)oxy-8-nitro-1,2,4,5-tetrahydro-3-benzazepine-3-carboxylate
—— (S)-1-[(S)-3-methyl-2-((S)-2-methylaminopropionylamino)butyryl]-2,3-dihydro-1H-indole-2-carboxylic acid 5-fluoro-2-methylbenzylamide 1599453-72-1 C26H33FN4O3
(S)-1-[(S)-3-methyl-2-((S)-2-methylaminopropionylamino)butyryl]-2,3-dihydro-1H-indole-2-carboxylic acid 5-fluoro-2-methylbenzylamide
—— [(3R,4S,5S,6S)-5-methoxy-4-[(2R,3R)-2-methyl-3-(3-methylbut-2-enyl)oxiran-2-yl]-1-oxaspiro[2.5]octan-6-yl] methanesulfonate 132746-83-9 C17H28O6S
[(3R,4S,5S,6S)-5-methoxy-4-[(2R,3R)-2-methyl-3-(3-methylbut-2-enyl)oxiran-2-yl]-1-oxaspiro[2.5]octan-6-yl] methanesulfonate
—— (S)-5-Amino-3-(2,3-difluoro-5-((2-hydroxypyrido[3,4-b]pyrazin-5-yl)amino)phenyl)-3,6,6-trimethyl-3,6-dihydro-2H-1,4-thiazine 1,1-dioxide 1600507-16-1 C20H20F2N6O3S
(S)-5-Amino-3-(2,3-difluoro-5-((2-hydroxypyrido[3,4-b]pyrazin-5-yl)amino)phenyl)-3,6,6-trimethyl-3,6-dihydro-2H-1,4-thiazine 1,1-dioxide
—— 6-{4-[2-amino-6-methyl-5-propylpyrimidin-4-yl]-9-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}[1,3]thiazolo[5,4-b]pyridin-2-amine 1379578-81-0 C24H27N7OS
6-{4-[2-amino-6-methyl-5-propylpyrimidin-4-yl]-9-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}[1,3]thiazolo[5,4-b]pyridin-2-amine
—— 7-[[4-anilino-6-(4-hydroxyanilino)-1,3,5-triazin-2-yl]amino]-N-phenylheptanamide 1282038-06-5 C28H31N7O2
7-[[4-anilino-6-(4-hydroxyanilino)-1,3,5-triazin-2-yl]amino]-N-phenylheptanamide
—— 2-bromo-5-phenyl-(1,2,4)triazolo(1,5-a)pyrazine 1397287-44-3 C11H7BrN4
2-bromo-5-phenyl-(1,2,4)triazolo(1,5-a)pyrazine
—— US10485800, Cmpd ID GS 1351476-86-2 C30H31N5O
US10485800, Cmpd ID GS
—— 5-(4-benzhydryloxypiperidin-1-ylmethyl)pyridine-2-carboxylic acid 1351371-98-6 C25H26N2O3
5-(4-benzhydryloxypiperidin-1-ylmethyl)pyridine-2-carboxylic acid
—— 2-((4,6-difluoro-1-(3-(6-methoxypyridin-3-yl)benzyl)-1H-indol-3-yl)sulfonyl)-N-(pyridin-2-yl)acetamide 1353015-92-5 C28H22F2N4O4S
2-((4,6-difluoro-1-(3-(6-methoxypyridin-3-yl)benzyl)-1H-indol-3-yl)sulfonyl)-N-(pyridin-2-yl)acetamide
—— 6-amino-N-cycloheptyl-N-(2-morpholinoethyl)hexane-1-sulfonamide 1170232-31-1 C19H39N3O3S
6-amino-N-cycloheptyl-N-(2-morpholinoethyl)hexane-1-sulfonamide
—— 1-Ethyl-7-{[(3-hydroxy-benzyl)-(2-pyridin-3-yl-ethyl)-amino]-methyl}-3,3,5-trimethyl-1,5-dihydro-benzo[b][1,4]diazepine-2,4-dione 1266561-62-9 C29H34N4O3
1-Ethyl-7-{[(3-hydroxy-benzyl)-(2-pyridin-3-yl-ethyl)-amino]-methyl}-3,3,5-trimethyl-1,5-dihydro-benzo[b][1,4]diazepine-2,4-dione
—— 1-[4-{[(4-{[2-(methyloxy)ethyl]oxy}-2-pyridinyl)methyl]oxy}-3-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)phenyl] ethanone 1398696-38-2 C27H30N2O4
1-[4-{[(4-{[2-(methyloxy)ethyl]oxy}-2-pyridinyl)methyl]oxy}-3-(2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)phenyl] ethanone
—— 1-(2,4-dichloro-phenyl)-3-(3-oxo-1-propyl-2,3-dihydro-1H-indazol-5-yl)-urea 1160165-66-1 C17H16Cl2N4O2
1-(2,4-dichloro-phenyl)-3-(3-oxo-1-propyl-2,3-dihydro-1H-indazol-5-yl)-urea
—— 5-(4-fluoro-phenyl)-oxazole-4-carboxylic acid [2-(4-acetyl-thiazol-2-ylmethyl)-2H-[1,2,3]triazol-4-yl]-amide 1161778-32-0 C18H13FN6O3S
5-(4-fluoro-phenyl)-oxazole-4-carboxylic acid [2-(4-acetyl-thiazol-2-ylmethyl)-2H-[1,2,3]triazol-4-yl]-amide
—— (R,R)-benzoic acid (5-oxotetrahydrofuran-3-yl)phenylmethyl ester 1024594-76-0 C18H16O4
(R,R)-benzoic acid (5-oxotetrahydrofuran-3-yl)phenylmethyl ester
—— 3-(3-(but-3-yn-1-yl)-2,5-dioxo-2,5-dihydro-1H-pyrrol-1-yl)propanoic acid 1446684-84-9 C11H11NO4
3-(3-(but-3-yn-1-yl)-2,5-dioxo-2,5-dihydro-1H-pyrrol-1-yl)propanoic acid
—— (3R)-ethyl 3-<<4-<<4-(aminoiminomethyl)phenyl>amino>-1,4-dioxobutyl>amino>-4-pentynoate 169275-98-3 C18H22N4O4
(3R)-ethyl 3-<<4-<<4-(aminoiminomethyl)phenyl>amino>-1,4-dioxobutyl>amino>-4-pentynoate
—— [1R,2R,(S)R]-N-(4-(tert-butylsulfinyl)-1-(thiophen-2-yl)-2-methyl-3-oxobutyl)-4-methylbenzenesulfonamide 1215087-83-4 C20H27NO4S3
[1R,2R,(S)R]-N-(4-(tert-butylsulfinyl)-1-(thiophen-2-yl)-2-methyl-3-oxobutyl)-4-methylbenzenesulfonamide
—— amide of laevorotatory o-phenoxyphenylsulfinylacetic acid 122993-08-2 C14H13NO3S
amide of laevorotatory o-phenoxyphenylsulfinylacetic acid
—— Alloc-Thr(tBu)-OH 1040744-62-4 C12H21NO5
Alloc-Thr(tBu)-OH
—— —— 1331756-38-7 C23H26ClNO3
—— methyl 3-amino-3-deoxy-α-D-lyxopyranoside 2-O,3-N-trichloroacetimidate 122204-80-2 C8H10Cl3NO4
methyl 3-amino-3-deoxy-α-D-lyxopyranoside 2-O,3-N-trichloroacetimidate
—— [2(S)-(2-{4-[3-(5-chloro-2-hydroxy-phenyl)-1H-pyrazol-4-ylethynyl]-phenylcarbamoyl}-piperidin-1-yl)-2-oxo-1(R)-phenyl-ethyl]-carbamic acid tert-butyl ester 1020840-33-8 C36H36ClN5O5
[2(S)-(2-{4-[3-(5-chloro-2-hydroxy-phenyl)-1H-pyrazol-4-ylethynyl]-phenylcarbamoyl}-piperidin-1-yl)-2-oxo-1(R)-phenyl-ethyl]-carbamic acid tert-butyl ester
—— 2,2,8,8-tetra(2-methoxyethylcarbamoyl)-3,4,6,7,8,9-hexahydro-2H-pyrimido[1,2-a]pyrimidine 1054553-39-7 C23H41N7O8
2,2,8,8-tetra(2-methoxyethylcarbamoyl)-3,4,6,7,8,9-hexahydro-2H-pyrimido[1,2-a]pyrimidine
—— ((4bS,8S,8aR)-3-Methoxy-8-methoxymethyl-4b,8-dimethyl-4b,5,6,7,8,8a,9,10-octahydro-phenanthren-1-ylamino)-oxo-acetyl chloride 160455-20-9 C21H28ClNO4
((4bS,8S,8aR)-3-Methoxy-8-methoxymethyl-4b,8-dimethyl-4b,5,6,7,8,8a,9,10-octahydro-phenanthren-1-ylamino)-oxo-acetyl chloride
—— (3S)-3-aminobutanoyl-D-histidine 1000578-31-3 C10H16N4O3
(3S)-3-aminobutanoyl-D-histidine
—— <2-Methoxy-6-(E)-(1-propenyl)phenoxy>acetic acid 144849-53-6 C12H14O4
<2-Methoxy-6-(E)-(1-propenyl)phenoxy>acetic acid
—— 2-chloro-4-methyl-phenyl lead triacetate 1154617-64-7 C13H15ClO6Pb
2-chloro-4-methyl-phenyl lead triacetate
—— N2-{2-[(5-fluoro-1,3-dihydro-2H-isoindol-2-yl)(methyl)amino]-2-oxoethyl}-N2-[2-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-N1-(2-aminoethyl)glycinamide hydrochloride 1190889-42-9 C25H30FN7O3*ClH
N2-{2-[(5-fluoro-1,3-dihydro-2H-isoindol-2-yl)(methyl)amino]-2-oxoethyl}-N2-[2-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-N1-(2-aminoethyl)glycinamide hydrochloride
—— ethyl N-[(3-cyclohexyl-2-phenyl-2H-indazol-6-yl)carbonyl]glycinate 1352083-48-7 C24H27N3O3
ethyl N-[(3-cyclohexyl-2-phenyl-2H-indazol-6-yl)carbonyl]glycinate
—— (2E)-N-[(2E)-3-phenylprop-2-en-1-yl]-3-(1H-pyrrolo[2,3-b]pyridin-3-yl)acrylamide 1160981-54-3 C19H17N3O
(2E)-N-[(2E)-3-phenylprop-2-en-1-yl]-3-(1H-pyrrolo[2,3-b]pyridin-3-yl)acrylamide
—— N-acetyl-1-acetoxymethyl-5-tosyloxy-7,8,9-trimethoxy-1,2-dihydro-3H-benzo[e]indole 1141759-05-8 C27H29NO9S
N-acetyl-1-acetoxymethyl-5-tosyloxy-7,8,9-trimethoxy-1,2-dihydro-3H-benzo[e]indole
—— N-[2-(2-hydroxyethoxy)ethyl]-1-(4-(3-[(2R)-2-methylpyrrolidin-1-yl]propoxy}phenyl)-1H-pyrazole-4-carboxamide 1152749-05-7 C22H32N4O4
N-[2-(2-hydroxyethoxy)ethyl]-1-(4-(3-[(2R)-2-methylpyrrolidin-1-yl]propoxy}phenyl)-1H-pyrazole-4-carboxamide
—— N-(4-isopropyl-2-(4-methoxyphenyl)oxazol-5-yl)furan-2-carboxamide 1151476-48-0 C18H18N2O4
N-(4-isopropyl-2-(4-methoxyphenyl)oxazol-5-yl)furan-2-carboxamide
—— H-c[Cys-Phe-DAgl(NMe,2naphthoyl)-IAmp-Tyr-Cys]-NH2 1150616-97-9 C51H59N9O8S2
H-c[Cys-Phe-DAgl(NMe,2naphthoyl)-IAmp-Tyr-Cys]-NH2
—— tert-butylN-[(1R)-1-(3-{[4-amino-3-(benzyloxy)phenyl]carbonyl}-4-chloro-2-fluorophenyl)propyl]carbamate 1433404-41-1 C28H30ClFN2O4
tert-butylN-[(1R)-1-(3-{[4-amino-3-(benzyloxy)phenyl]carbonyl}-4-chloro-2-fluorophenyl)propyl]carbamate
—— (1aR,5aR)-2-(2,4-difluoro-phenyl)-1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalene-4-carboxylic acid (1-pyridin-4-yl-cyclopropyl)-amide 1268877-82-2 C22H18F2N4O
(1aR,5aR)-2-(2,4-difluoro-phenyl)-1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalene-4-carboxylic acid (1-pyridin-4-yl-cyclopropyl)-amide
—— (2R,3R,4R,5R)-2-(5-fluoro-2,4-dioxopyrimidin-1-yl)-3,4-dihydroxy-5-(hydroxymethyl)-3-methyloxolane-2-carbonitrile 1402821-69-5 C11H12FN3O6
(2R,3R,4R,5R)-2-(5-fluoro-2,4-dioxopyrimidin-1-yl)-3,4-dihydroxy-5-(hydroxymethyl)-3-methyloxolane-2-carbonitrile
—— (S)-N-(4-cyclohexylbutyl)-2-(1-(5-methoxy-2-(3-oxo-3-(isopropylsulfonamido)propyl)benzyl)pyrrolidin-2-yl)oxazole-4-carboxamide 1403829-50-4 C32H48N4O6S
(S)-N-(4-cyclohexylbutyl)-2-(1-(5-methoxy-2-(3-oxo-3-(isopropylsulfonamido)propyl)benzyl)pyrrolidin-2-yl)oxazole-4-carboxamide
—— (1R,5S)-3-[5-(4-chloro-2,3-difluorophenyl)-2-ethylphenyl]-4-hydroxybicyclo[3.2.1]oct-3-en-2-one 1090512-09-6 C22H19ClF2O2
(1R,5S)-3-[5-(4-chloro-2,3-difluorophenyl)-2-ethylphenyl]-4-hydroxybicyclo[3.2.1]oct-3-en-2-one
—— (Z)-[4-[3,5-bis(trifluoromethyl)phenyl]-4-hydroxycyclohexyl]oxyimino-[tert-butyl(methyl)amino]-oxidoazanium 1407973-49-2 C19H25F6N3O3
(Z)-[4-[3,5-bis(trifluoromethyl)phenyl]-4-hydroxycyclohexyl]oxyimino-[tert-butyl(methyl)amino]-oxidoazanium
—— (2-methyl-6-methylideneocta-1,7-dien-3-yl) thiocyanate 124431-91-0 C11H15NS
(2-methyl-6-methylideneocta-1,7-dien-3-yl) thiocyanate
—— (2-Methyl-allyl)-(4,5,6,7-tetrahydro-1H-[1,3]diazepin-2-yl)-(2,4,6-trichloro-phenyl)-amine 120914-75-2 C15H18Cl3N3
(2-Methyl-allyl)-(4,5,6,7-tetrahydro-1H-[1,3]diazepin-2-yl)-(2,4,6-trichloro-phenyl)-amine
—— t-butyl [[5-cyano-6-[(cyclohexylmethyl)thio]-2-(1,1-dimethylethyl)-4-pyrimidinyl]oxy]acetate 119491-94-0 C22H33N3O3S
t-butyl [[5-cyano-6-[(cyclohexylmethyl)thio]-2-(1,1-dimethylethyl)-4-pyrimidinyl]oxy]acetate