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中文名称 英文名称 CAS号 化学式 结构式图片
—— (3S)-3-methoxy-N-[3-(2-methyl-1,3-thiazol-5-yl)-1H-indazol-5-yl]-1-[2-oxo-2-[4-(4-pyrimidin-2-ylphenyl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]pyrrolidine-3-carboxamide 1093062-95-3 C34H34N8O3S
(3S)-3-methoxy-N-[3-(2-methyl-1,3-thiazol-5-yl)-1H-indazol-5-yl]-1-[2-oxo-2-[4-(4-pyrimidin-2-ylphenyl)-3,6-dihydro-2H-pyridin-1-yl]ethyl]pyrrolidine-3-carboxamide
—— N-{2-chloro-5-[5-methanesulfonyl-1-(3-pyrrolidin-1-yl-propyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]-benzyl}-nicotinamide 1048036-60-7 C27H33ClN6O3S
N-{2-chloro-5-[5-methanesulfonyl-1-(3-pyrrolidin-1-yl-propyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]-benzyl}-nicotinamide
—— N-[(3R,4S)-3-{[4-(5-chloro-1,3-thiazol-2-yl)phenoxy]methyl}tetrahydro-2H-pyran-4-yl]cyclopropanesulfonamide 1402563-40-9 C18H21ClN2O4S2
N-[(3R,4S)-3-{[4-(5-chloro-1,3-thiazol-2-yl)phenoxy]methyl}tetrahydro-2H-pyran-4-yl]cyclopropanesulfonamide
—— 6-fluoro-4-(2-(4-tert-butylphenyl)-ethoxy)-quinazoline 158731-05-6 C20H21FN2O
6-fluoro-4-(2-(4-tert-butylphenyl)-ethoxy)-quinazoline
—— 2,3-difluoro-5-(2-methoxy-3-pyridinyl)phenyl 5-thio-β-D-xylopyranoside 1011721-24-6 C17H17F2NO5S
2,3-difluoro-5-(2-methoxy-3-pyridinyl)phenyl 5-thio-β-D-xylopyranoside
—— 3-Amino-1,8-dipropoxyanthracene-9,10-dione 1537900-57-4 C20H21NO4
3-Amino-1,8-dipropoxyanthracene-9,10-dione
—— 7-(4-ethyl-5-fluoropyridin-3-yl)-8-fluoro-1-methyl-4,5-dihydro-[1,2,4]triazolo[4,3-a]quinoline 1404366-80-8 C18H16F2N4
7-(4-ethyl-5-fluoropyridin-3-yl)-8-fluoro-1-methyl-4,5-dihydro-[1,2,4]triazolo[4,3-a]quinoline
—— 4-{cyclopropyl-[5-(2-fluoro-4-methanesulfonyl-phenyl)-[1,2,4]oxadiazole-3-carbonyl]-amino}-piperidine-1-carboxylic acid tert-butyl ester 1557031-48-7 C23H29FN4O6S
4-{cyclopropyl-[5-(2-fluoro-4-methanesulfonyl-phenyl)-[1,2,4]oxadiazole-3-carbonyl]-amino}-piperidine-1-carboxylic acid tert-butyl ester
—— 13-cyclohexyl-N-(dimethylsulfamoyl)-3-methoxy-6-(4-methyl-2-phenylpiperazine-1-carbonyl)-7H-indolo[2,1-a][2]benzazepine-10-carboxamide 1058130-82-7 C39H45N5O5S
13-cyclohexyl-N-(dimethylsulfamoyl)-3-methoxy-6-(4-methyl-2-phenylpiperazine-1-carbonyl)-7H-indolo[2,1-a][2]benzazepine-10-carboxamide
—— N-[5-(1-{2-hydroxy-3-[4-(1H-tetrazol-5-yl)-piperidin-1-yl]-propyl}-5-methanesulfonyl-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl)-2-trifluoromethyl-benzyl]-3-methyl-butyramide 1048034-73-6 C29H40F3N9O4S
N-[5-(1-{2-hydroxy-3-[4-(1H-tetrazol-5-yl)-piperidin-1-yl]-propyl}-5-methanesulfonyl-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl)-2-trifluoromethyl-benzyl]-3-methyl-butyramide
—— [2-(Imidazol-1-yl)methyl-4-[[[4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl]carbonylamino]acetyl]phenyl]oxyacetic acid trifluoroacetate 197237-35-7 C2HF3O2*C22H22N4O5S
[2-(Imidazol-1-yl)methyl-4-[[[4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl]carbonylamino]acetyl]phenyl]oxyacetic acid trifluoroacetate
—— US10138229, Example 108 1558037-39-0 C21H20F3N5O3
US10138229, Example 108
—— N-methyl-N'-[(8-methyl-2-{methyl[2-(methylamino)ethyl]amino}quinolin-3-yl)methyl]cyclopropane-1,1-dicarboxamide 1365615-49-1 C21H29N5O2
N-methyl-N'-[(8-methyl-2-{methyl[2-(methylamino)ethyl]amino}quinolin-3-yl)methyl]cyclopropane-1,1-dicarboxamide
—— 1-benzyl-3-(4-chlorophenyl)-N-ethyl-4-methyl-N-(2-methylsulfonyl-ethyl)-5-(trifluoromethyl)-1H-pyrrole-2-carboxylic acid amide 1574113-25-9 C25H26ClF3N2O3S
1-benzyl-3-(4-chlorophenyl)-N-ethyl-4-methyl-N-(2-methylsulfonyl-ethyl)-5-(trifluoromethyl)-1H-pyrrole-2-carboxylic acid amide
—— [6-(2-methoxy-phenyl)-pyrimidin-4-yl]-[4-methoxy-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-phenyl]-amine 1569985-11-0 C23H24N4O2
[6-(2-methoxy-phenyl)-pyrimidin-4-yl]-[4-methoxy-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-phenyl]-amine
—— methyl N-[(1R)-2-[(1R,3S,5R)-3-[5-[13-[2-[(1R,3S,5R)-2-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]-2-azabicyclo[3.1.0]hexan-3-yl]-1H-imidazol-5-yl]-2,9-dioxatetracyclo[6.6.2.04,16.011,15]hexadeca-1(14),4(16),5,7,11(15),12-hexaen-6-yl]-1H-imidazol-2-yl]-2-azabicyclo[3.1.0]hexan-2-yl]-2-oxo-1-phenylethyl]carbamate 1377046-86-0 C47H48N8O8
methyl N-[(1R)-2-[(1R,3S,5R)-3-[5-[13-[2-[(1R,3S,5R)-2-[(2S)-2-(methoxycarbonylamino)-3-methylbutanoyl]-2-azabicyclo[3.1.0]hexan-3-yl]-1H-imidazol-5-yl]-2,9-dioxatetracyclo[6.6.2.04,16.011,15]hexadeca-1(14),4(16),5,7,11(15),12-hexaen-6-yl]-1H-imidazol-2-yl]-2-azabicyclo[3.1.0]hexan-2-yl]-2-oxo-1-phenylethyl]carbamate
—— (3S,4S)-3-Benzoyl-4-(4-methoxy-phenyl)-2-phenyl-5-((E)-styryl)-3,4-dihydro-2H-pyrazole-3-carbonitrile 129201-07-6 C32H25N3O2
(3S,4S)-3-Benzoyl-4-(4-methoxy-phenyl)-2-phenyl-5-((E)-styryl)-3,4-dihydro-2H-pyrazole-3-carbonitrile
—— NCHQ-I 1621233-63-3 C34H40N5O5
NCHQ-I
—— (+/-)-9-<(1'-tert-butyldiphenylsilyloxy-3',4'-methylenylbut-2'-oxy)methyl>adenine 141619-41-2 C27H33N5O2Si
(+/-)-9-<(1'-tert-butyldiphenylsilyloxy-3',4'-methylenylbut-2'-oxy)methyl>adenine
—— (3S,5R)-5-(tert-butyldimethylsilyloxy)-7-(4-methoxybenzyloxy)-hept-1-en-3-yl carbamate 1227514-63-7 C22H37NO5Si
(3S,5R)-5-(tert-butyldimethylsilyloxy)-7-(4-methoxybenzyloxy)-hept-1-en-3-yl carbamate
—— 1-(3-fluorophenyl)-3-(4-(4-(piperazin-1-ylmethyl)thiazol-2-yl)phenyl)urea 1387637-05-9 C21H22FN5OS
1-(3-fluorophenyl)-3-(4-(4-(piperazin-1-ylmethyl)thiazol-2-yl)phenyl)urea
—— tert-butyl 4-(2-(2-(2H-indazol-2-yl)thiazole-4-carboxamido)phenyl)piperazine-1-carboxylate 1026668-79-0 C26H28N6O3S
tert-butyl 4-(2-(2-(2H-indazol-2-yl)thiazole-4-carboxamido)phenyl)piperazine-1-carboxylate
—— Benz[a]anthracen-5-ol, 5,6-dihydro-6-methoxy-1-methyl-, cis- 120014-45-1 C20H18O2
Benz[a]anthracen-5-ol, 5,6-dihydro-6-methoxy-1-methyl-, cis-
—— Benzyl-(4,6-diiodo-pyrimidin-5-yl)-methyl-amine 1028303-49-2 C12H11I2N3
Benzyl-(4,6-diiodo-pyrimidin-5-yl)-methyl-amine
—— 3-{2-chloro-5-[5-methanesulfonyl-1-(3-morpholin-4-yl-propyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]-phenyl}-N-methyl-propionamide 1048036-90-3 C24H34ClN5O4S
3-{2-chloro-5-[5-methanesulfonyl-1-(3-morpholin-4-yl-propyl)-4,5,6,7-tetrahydro-1H-pyrazolo[4,3-c]pyridin-3-yl]-phenyl}-N-methyl-propionamide
—— 4-(2-isobutylamino-purin-9-yl)benzamide 1332368-98-5 C16H18N6O
4-(2-isobutylamino-purin-9-yl)benzamide
—— ethyl 2-[(5-chloro-2-thienyl)methyl]-3-oxo-butanoate 1335027-74-1 C11H13ClO3S
ethyl 2-[(5-chloro-2-thienyl)methyl]-3-oxo-butanoate
—— N-[2-methyl-4-(2-methyl-[1,3']bipyrrolidinyl-1'-yl)-phenyl]-4-morpholin-4-ylmethyl-benzamide trifluoroacetate 1146700-57-3 C2HF3O2*C28H38N4O2
N-[2-methyl-4-(2-methyl-[1,3']bipyrrolidinyl-1'-yl)-phenyl]-4-morpholin-4-ylmethyl-benzamide trifluoroacetate
—— methyl 3,5-diisopropylpyrrole-2-carboxylate 1116091-48-5 C12H19NO2
methyl 3,5-diisopropylpyrrole-2-carboxylate
—— (S)-1-ethyl-3-(4-(2-(3-methylmorpholino)-6-(1H-pyrazol-3-yl)pyrimidin-4-yl)phenyl)urea 1333108-33-0 C21H25N7O2
(S)-1-ethyl-3-(4-(2-(3-methylmorpholino)-6-(1H-pyrazol-3-yl)pyrimidin-4-yl)phenyl)urea
—— methyl 6-hydroxy-3-methyl-5-propylpyrazine-2-carboxylate 1332731-58-4 C10H14N2O3
methyl 6-hydroxy-3-methyl-5-propylpyrazine-2-carboxylate
—— 2-methyl-4-[3-[(5-methyl-3-{3-[4-(trifluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl}-1H-1,2,4-triazol-1-yl)methyl]phenoxy]butan-2-ol 1570498-31-5 C24H24F3N5O4
2-methyl-4-[3-[(5-methyl-3-{3-[4-(trifluoromethoxy)phenyl]-1,2,4-oxadiazol-5-yl}-1H-1,2,4-triazol-1-yl)methyl]phenoxy]butan-2-ol
—— 3-[2-Chloro-5-(oxolan-3-ylmethoxy)phenyl]-7-methyl-2,4,5,8,13-pentazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7,10,12-hexaene 1552286-69-7 C20H18ClN5O2
3-[2-Chloro-5-(oxolan-3-ylmethoxy)phenyl]-7-methyl-2,4,5,8,13-pentazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7,10,12-hexaene
—— 4-[(2-{4-[(2-cyano-ethyl)-methyl-carbamoyl]-3-fluoro-phenyl}-pyrimidine-5-carbonyl)-cyclopropyl-amino]-piperidine-1-carboxylic acid tert-butyl ester 1557036-56-2 C29H35FN6O4
4-[(2-{4-[(2-cyano-ethyl)-methyl-carbamoyl]-3-fluoro-phenyl}-pyrimidine-5-carbonyl)-cyclopropyl-amino]-piperidine-1-carboxylic acid tert-butyl ester
—— 1-(3-methoxypropyl)-2-methyl-5-phenyl-N-[3-(trifluoromethyl)phenyl]pyrrole-3-carboxamide 1403944-93-3 C23H23F3N2O2
1-(3-methoxypropyl)-2-methyl-5-phenyl-N-[3-(trifluoromethyl)phenyl]pyrrole-3-carboxamide
—— 7-((R)-2-nitro-6,7-dihydro-5H-imidazo[2,1-b][1,3]oxazin-7-ylmethoxy)-1-[3-(4-trifluoromethoxyphenoxy)propyl]-2,3,4,5-tetrahydro-1H-benzo[b]azepine 1403318-35-3 C27H29F3N4O6
7-((R)-2-nitro-6,7-dihydro-5H-imidazo[2,1-b][1,3]oxazin-7-ylmethoxy)-1-[3-(4-trifluoromethoxyphenoxy)propyl]-2,3,4,5-tetrahydro-1H-benzo[b]azepine
—— N-(2-hydroxyethyl)-9-methyl-6-[4-(2-oxo-2,3-dihydro-1H-benzimidazol-1-yl)piperidin-1-yl]-9H-purine-8-carboxamide 1365605-56-6 C21H24N8O3
N-(2-hydroxyethyl)-9-methyl-6-[4-(2-oxo-2,3-dihydro-1H-benzimidazol-1-yl)piperidin-1-yl]-9H-purine-8-carboxamide
—— N-[2-[[5-[4-(4-cyanophenyl)piperidine-1-carbonyl]-2-methyl-phenyl]carbamoylamino]-2-methyl-propyl]pyridine-3-carboxamide 1034464-79-3 C31H34N6O3
N-[2-[[5-[4-(4-cyanophenyl)piperidine-1-carbonyl]-2-methyl-phenyl]carbamoylamino]-2-methyl-propyl]pyridine-3-carboxamide
—— 5'-O-acetyl-2',3'-O-isopropylidene-3-nitrouridine 162660-12-0 C14H17N3O9
5'-O-acetyl-2',3'-O-isopropylidene-3-nitrouridine
—— 4-((tert-butyldimethylsilyl)oxy)benzyl (7-nitrobenzo[c][1,2,5]oxadiazol-4-yl)carbamate 1579947-08-2 C20H24N4O6Si
4-((tert-butyldimethylsilyl)oxy)benzyl (7-nitrobenzo[c][1,2,5]oxadiazol-4-yl)carbamate
—— Li[B(Sal)(OH)2] 1258274-66-6 C7H6BO5*Li
Li[B(Sal)(OH)2]
—— 4-n-propyl-1-trimethylsilyloxy-1-cyclohexene 1003601-42-0 C12H24OSi
4-n-propyl-1-trimethylsilyloxy-1-cyclohexene
—— N-di-isopropyloxyphosphoryl-Ser-OMe 117286-91-6 C10H22NO6P
N-di-isopropyloxyphosphoryl-Ser-OMe
—— 2-bromo-1,3-bis(indazol-2-ylmethyl)benzene 1350625-00-1 C22H17BrN4
2-bromo-1,3-bis(indazol-2-ylmethyl)benzene
—— —— 133636-30-3 C18H20N6O
—— 2-benzyl-4-hydroxy-1-oxa-7-azacyclotetradecane-6,14-dione 1374151-64-0 C19H27NO4
2-benzyl-4-hydroxy-1-oxa-7-azacyclotetradecane-6,14-dione
—— 2-(2,4-dinitro-phenylsulfanyl)-5-isobutylsulfanyl-[1,3,4]thiadiazole 18905-55-0 C12H12N4O4S3
2-(2,4-dinitro-phenylsulfanyl)-5-isobutylsulfanyl-[1,3,4]thiadiazole
—— 1,2-dimethyl-4-p-bromophenyl-5-benzoyl-2-imidazoline 103518-44-1 C18H17BrN2O
1,2-dimethyl-4-p-bromophenyl-5-benzoyl-2-imidazoline
—— ethyl (4S)-2-amino-1',2'-dimethyl-5'-oxospiro[indeno[2,1-d][1,3]oxazole-4,4'-pyrrole]-3'-carboxylate 1217689-81-0 C18H17N3O4
ethyl (4S)-2-amino-1',2'-dimethyl-5'-oxospiro[indeno[2,1-d][1,3]oxazole-4,4'-pyrrole]-3'-carboxylate
—— 1-Naphthalen-2-ylsulfonylpyrrolidine-3-carboxylic acid 1394241-84-9 C15H15NO4S
1-Naphthalen-2-ylsulfonylpyrrolidine-3-carboxylic acid