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中文名称 英文名称 CAS号 化学式 结构式图片
—— ethyl 2-amino-4-(5,7-dichloro-2,3-dihydro-1-benzofuran-4-yl)-5,7-dihydro-6H-pyrrolo[3,4-d]pyrimidine-6-carboxylate 1046860-53-0 C17H16Cl2N4O3
ethyl 2-amino-4-(5,7-dichloro-2,3-dihydro-1-benzofuran-4-yl)-5,7-dihydro-6H-pyrrolo[3,4-d]pyrimidine-6-carboxylate
—— 1-[4-chloro-3-(pyridin-2-ylethynyl)benzoyl]-4-(1,3-thiazol-2-yl)piperazine 1197358-22-7 C21H17ClN4OS
1-[4-chloro-3-(pyridin-2-ylethynyl)benzoyl]-4-(1,3-thiazol-2-yl)piperazine
—— 1-(4-fluorophenyl)-3-({[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino}carbonyl)imidazo[1,5-a]pyridin-2-ium trifluoroacetate 1039350-72-5 C2HF3O2*C23H18FN3O2
1-(4-fluorophenyl)-3-({[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]amino}carbonyl)imidazo[1,5-a]pyridin-2-ium trifluoroacetate
—— 4-[5-chloro-2-(1-cyclohexylmethyl-5,6-difluoro-1H-benzoimidazol-2-yl)-phenoxymethyl]-benzonitrile 1281980-94-6 C28H24ClF2N3O
4-[5-chloro-2-(1-cyclohexylmethyl-5,6-difluoro-1H-benzoimidazol-2-yl)-phenoxymethyl]-benzonitrile
—— N-(4-t-butoxycarbonylaminothiophen-3-yl)-5-[1-(2-dimethylaminoethyl)-3-(3-fluorophenyl)ureidomethyl]pyridine-2-carboxylic acid amide 1196982-84-9 C27H33FN6O4S
N-(4-t-butoxycarbonylaminothiophen-3-yl)-5-[1-(2-dimethylaminoethyl)-3-(3-fluorophenyl)ureidomethyl]pyridine-2-carboxylic acid amide
—— 4-{3-[(Z)-(6-hydroxy-3-oxo-1-benzofuran-2(3H)-ylidene)methyl]-5-methoxy-1H-indol-1-yl}butanenitrile 1200542-09-1 C22H18N2O4
4-{3-[(Z)-(6-hydroxy-3-oxo-1-benzofuran-2(3H)-ylidene)methyl]-5-methoxy-1H-indol-1-yl}butanenitrile
—— 4-(2,2,4-trimethyl-3-oxo-3,4-dihydro-2H-pyrido[3,2-b][1,4]oxazin-7-yl)-N-(3-fluoro-4-((1S,4S)-5-methyl-2,5-diazabicyclo[2.2.1]heptan-2-yl)phenyl)pyrimidin-2-amine 1182185-00-7 C26H28FN7O2
4-(2,2,4-trimethyl-3-oxo-3,4-dihydro-2H-pyrido[3,2-b][1,4]oxazin-7-yl)-N-(3-fluoro-4-((1S,4S)-5-methyl-2,5-diazabicyclo[2.2.1]heptan-2-yl)phenyl)pyrimidin-2-amine
—— ethyl 4-(6-{4-[(ethylamino)carbonyl]phenyl}-4H-1,3-benzodioxin-2-yl)piperidine-1-carboxylate 1200574-19-1 C25H30N2O5
ethyl 4-(6-{4-[(ethylamino)carbonyl]phenyl}-4H-1,3-benzodioxin-2-yl)piperidine-1-carboxylate
—— 4-[4-(2,6-Dimethylphenoxy)but-2-en-1-yl]morpholine hydrochloride 1185243-54-2 C16H24ClNO2
4-[4-(2,6-Dimethylphenoxy)but-2-en-1-yl]morpholine hydrochloride
—— 4-bromo-5-(4-fluorophenyl)-3-methyl-1-(2,2,2-trifluoroethyl)-1H-pyrazole 1221503-22-5 C12H9BrF4N2
4-bromo-5-(4-fluorophenyl)-3-methyl-1-(2,2,2-trifluoroethyl)-1H-pyrazole
—— N-ethyl-N'-(3-{[4-(3-isopropyl-2,4-dioxo-1,3,7-triazaspiro[4.5]dec-7-yl)piperidin-1-yl]carbonyl}-6-methylthieno[2,3-b]pyridin-2-yl)urea 1257424-19-3 C27H37N7O4S
N-ethyl-N'-(3-{[4-(3-isopropyl-2,4-dioxo-1,3,7-triazaspiro[4.5]dec-7-yl)piperidin-1-yl]carbonyl}-6-methylthieno[2,3-b]pyridin-2-yl)urea
—— 2-(4-fluorophenyl)-5-[3-[2-(4-methoxyphenyl)propan-2-ylcarbamoyl]phenyl]-N-methyl-1-benzofuran-3-carboxamide 1217333-76-0 C33H29FN2O4
2-(4-fluorophenyl)-5-[3-[2-(4-methoxyphenyl)propan-2-ylcarbamoyl]phenyl]-N-methyl-1-benzofuran-3-carboxamide
—— 5-[6-chloro-5-(2-chloro-phenylethynyl)-1H-benzoimidazol-2-yloxy]-2-methyl-benzoic acid 1219738-26-7 C23H14Cl2N2O3
5-[6-chloro-5-(2-chloro-phenylethynyl)-1H-benzoimidazol-2-yloxy]-2-methyl-benzoic acid
—— 2'-(amino-acetyl)-1-(4-amino-2(S)-hydroxy-butyryl)-sisomicin 1154758-07-2 C25H47N7O10
2'-(amino-acetyl)-1-(4-amino-2(S)-hydroxy-butyryl)-sisomicin
—— tert-butyl {(3,5-dichloro-phenylsulphonyl)-[3-methyl-1-(6-methyl-pyridazin-3-yl)-1H-indol-5-yl]-amino}-acetate 1049024-48-7 C26H26Cl2N4O4S
tert-butyl {(3,5-dichloro-phenylsulphonyl)-[3-methyl-1-(6-methyl-pyridazin-3-yl)-1H-indol-5-yl]-amino}-acetate
—— N-1-adamantyl-2-amino-4-(4-bromo-2-chloro-5-methoxyphenyl)-5,7-dihydro-6H-pyrrolo[3,4-d]pyrimidine-6-carboxamide 1046858-84-7 C24H27BrClN5O2
N-1-adamantyl-2-amino-4-(4-bromo-2-chloro-5-methoxyphenyl)-5,7-dihydro-6H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
—— 4-fluoro-6-[(5-fluoro-1-methyl-2-oxopyridin-4-yl)methyl]-8-(2-oxo-1H-pyridin-3-yl)furo[2,3-e]indole-7-carboxylic acid 1037759-53-7 C23H15F2N3O5
4-fluoro-6-[(5-fluoro-1-methyl-2-oxopyridin-4-yl)methyl]-8-(2-oxo-1H-pyridin-3-yl)furo[2,3-e]indole-7-carboxylic acid
—— 2-(4-(((2-methoxy-6-phenylpyridin-3yl)methyl)amino)phenoxy)propanoic acid 1202162-74-0 C22H22N2O4
2-(4-(((2-methoxy-6-phenylpyridin-3yl)methyl)amino)phenoxy)propanoic acid
—— 2-[1-(2,3-dimethyl-phenyl)-1H-tetrazol-5-ylsulfanyl]-N-[2-(4-ethoxy-benzyl)-2H-pyrazol-3-yl]-acetamide 1200438-47-6 C23H25N7O2S
2-[1-(2,3-dimethyl-phenyl)-1H-tetrazol-5-ylsulfanyl]-N-[2-(4-ethoxy-benzyl)-2H-pyrazol-3-yl]-acetamide
—— (5R)-3-[(3',5'-dichlorobiphenyl-4-yl)methyl]-5-methyl-1,3-oxazolidin-2-one 1095986-81-4 C17H15Cl2NO2
(5R)-3-[(3',5'-dichlorobiphenyl-4-yl)methyl]-5-methyl-1,3-oxazolidin-2-one
—— (1R,2S)-2-(4-{[(2R)-2-benzylpiperazin-1-yl]carbonyl}-5-phenyl-1H-imidazol-1-yl)-1-{[2-(2-hydroxyethoxy)ethoxy]methyl}cyclohexanol 1083849-27-7 C32H42N4O5
(1R,2S)-2-(4-{[(2R)-2-benzylpiperazin-1-yl]carbonyl}-5-phenyl-1H-imidazol-1-yl)-1-{[2-(2-hydroxyethoxy)ethoxy]methyl}cyclohexanol
—— {5-fluoro-2-methyl-3-[4-(pyridine-2-sulfonyl)thiazol-5-ylmethyl]indol-1-yl}acetic acid methyl ester 1161865-83-3 C21H18FN3O4S2
{5-fluoro-2-methyl-3-[4-(pyridine-2-sulfonyl)thiazol-5-ylmethyl]indol-1-yl}acetic acid methyl ester
—— 1-{4-5-fluoro-4-(4-fluoro-3-methyl-phenylamino)pyrimidin-2-benzenesulphonyl}-4-((R)-2-methylpyrrolidin-1-ylmethyl)piperidin-4-ol 1049668-39-4 C28H34F2N6O3S
1-{4-5-fluoro-4-(4-fluoro-3-methyl-phenylamino)pyrimidin-2-benzenesulphonyl}-4-((R)-2-methylpyrrolidin-1-ylmethyl)piperidin-4-ol
—— 2-amino-N-cyclobutyl-4-(2,4-dichloro-6-{[(2E)-3-phenylprop-2-en-1-yl]oxy}phenyl)-5,7-dihydro-6H-pyrrolo[3,4-d]pyrimidine-6-carboxamide 1046860-91-6 C26H25Cl2N5O2
2-amino-N-cyclobutyl-4-(2,4-dichloro-6-{[(2E)-3-phenylprop-2-en-1-yl]oxy}phenyl)-5,7-dihydro-6H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
—— 5-(5-biphenyl-4-yl-6-chloro-1H-benzoimidazol-2-yloxy)-2-ethyl-benzoic acid 1219739-20-4 C28H21ClN2O3
5-(5-biphenyl-4-yl-6-chloro-1H-benzoimidazol-2-yloxy)-2-ethyl-benzoic acid
—— 2-amino-N-cyclopropyl-4-[2,4-dichloro-6-(2-pyrrolidin-1-ylethoxy)phenyl]-5,7-dihydro-6H-pyrrolo[3,4-d]pyrimidine-6-carboxamide 1046859-70-4 C22H26Cl2N6O2
2-amino-N-cyclopropyl-4-[2,4-dichloro-6-(2-pyrrolidin-1-ylethoxy)phenyl]-5,7-dihydro-6H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
—— tert-butyl ((3,5-dichloro-phenylsulphonyl)-{1-[4-(tetrahydro-pyran-4-yloxy)-pyridin-2-yl]-1H-indol-5-yl}-amino)-acetate 1049023-95-1 C30H31Cl2N3O6S
tert-butyl ((3,5-dichloro-phenylsulphonyl)-{1-[4-(tetrahydro-pyran-4-yloxy)-pyridin-2-yl]-1H-indol-5-yl}-amino)-acetate
—— [4-({[1-(4-fluorophenyl)-1H-pyrazolo[3,4-c]pyridine-4-carbonyl]-amino}-methyl)-benzenesulfonylamino]-acetic acid methyl ester 1220026-20-9 C23H20FN5O5S
[4-({[1-(4-fluorophenyl)-1H-pyrazolo[3,4-c]pyridine-4-carbonyl]-amino}-methyl)-benzenesulfonylamino]-acetic acid methyl ester
—— 5-(3-fluoro-5-(propylcarbamoyl)phenyl)-2-(4-fluorophenyl)-N-methylbenzofuran-3-carboxamide 1217336-37-2 C26H22F2N2O3
5-(3-fluoro-5-(propylcarbamoyl)phenyl)-2-(4-fluorophenyl)-N-methylbenzofuran-3-carboxamide
—— tert-butyl (2S)-2-methyl-3-oxopyrrolidine-1-carboxylate 1030899-85-4 C10H17NO3
tert-butyl (2S)-2-methyl-3-oxopyrrolidine-1-carboxylate
—— 1,1-dimethylethyl (2S)-4-({6-[{[6-(3-fluorophenyl)-3-pyridinyl]carbonyl}(methyl)amino]-3-pyridinyl}methyl)-2-methyl-1-piperazinecarboxylate 1000813-19-3 C29H34FN5O3
1,1-dimethylethyl (2S)-4-({6-[{[6-(3-fluorophenyl)-3-pyridinyl]carbonyl}(methyl)amino]-3-pyridinyl}methyl)-2-methyl-1-piperazinecarboxylate
—— 2,3-dimethyl-1-oxo-1,2-dihydro-isoquinoline-4-carboxylic acid ((S)-1-phenyl-propyl)-amide 1215093-06-3 C21H22N2O2
2,3-dimethyl-1-oxo-1,2-dihydro-isoquinoline-4-carboxylic acid ((S)-1-phenyl-propyl)-amide
—— ethyl 3-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-5-(4,4,4-trifluorobutoxy)benzoate 1046861-38-4 C20H28BF3O5
ethyl 3-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-5-(4,4,4-trifluorobutoxy)benzoate
—— 2-phenyl-5-piperidin-1-yl-imidazo[1,2-c]pyrimidin-7-ylamine 1278407-67-2 C17H19N5
2-phenyl-5-piperidin-1-yl-imidazo[1,2-c]pyrimidin-7-ylamine
—— methyl 2-O-benzyl-3,4-dideoxy-4-(4-methylphenyl)sulfonyl-6-O-triphenylmethyl-α-D-erythro-hex-3-enopyranoside 1096364-46-3 C40H38O6S
methyl 2-O-benzyl-3,4-dideoxy-4-(4-methylphenyl)sulfonyl-6-O-triphenylmethyl-α-D-erythro-hex-3-enopyranoside
—— (E)-3-{2-[(R)-1-(9H-purin-6-yl)pyrrolidin-2-yl-methoxy]phenyl}acrylic acid 1201581-54-5 C19H19N5O3
(E)-3-{2-[(R)-1-(9H-purin-6-yl)pyrrolidin-2-yl-methoxy]phenyl}acrylic acid
—— (3-{2-[(benzoyl(ethyl)amino)-methyl]-4-trifluoromethyl-phenoxy}-phenyl)-acetic acid 1198281-92-3 C25H22F3NO4
(3-{2-[(benzoyl(ethyl)amino)-methyl]-4-trifluoromethyl-phenoxy}-phenyl)-acetic acid
—— (R)-3,5-dimethyl-N-(1methylpiperidin-3-yl)-1H-indole-2-carboxamide 1202242-35-0 C17H23N3O
(R)-3,5-dimethyl-N-(1methylpiperidin-3-yl)-1H-indole-2-carboxamide
—— 1,4,5,7-tetrahydro-3<i>H</i>-benzo[<i>b</i>][1,4]diazonine-2,6-dione 110460-07-6 C11H12N2O2
1,4,5,7-tetrahydro-3<i>H</i>-benzo[<i>b</i>][1,4]diazonine-2,6-dione
—— 5-(2',6',6'-trimethyl-2'-cyclohexen-1'-yl)benzoic acid 141885-42-9 C16H20O2
5-(2',6',6'-trimethyl-2'-cyclohexen-1'-yl)benzoic acid
—— tert-butyl ((S)-1-oxo-1-(((R)-1-(5-(2,2,2-trifluoroethoxy)pyridin-2-yl)ethyl)amino)-3-(3-(trifluoromethyl)phenyl)propan-2-yl)carbamate 1257117-61-5 C24H27F6N3O4
tert-butyl ((S)-1-oxo-1-(((R)-1-(5-(2,2,2-trifluoroethoxy)pyridin-2-yl)ethyl)amino)-3-(3-(trifluoromethyl)phenyl)propan-2-yl)carbamate
—— —— 1125889-67-9 C13H8F5N5O
—— tert-Butyl [3,5-dimethyl-1-(3-{[(4-methylphenyl)sulfonyl]amino}phenyl)-1H-pyrazol-4-yl]acetate 1379445-74-5 C24H29N3O4S
tert-Butyl [3,5-dimethyl-1-(3-{[(4-methylphenyl)sulfonyl]amino}phenyl)-1H-pyrazol-4-yl]acetate
—— 4-[(4-allyloxycarbonylamino-1-methyl-1H-pyrrole-2-carbonyl)-amino]-1-methyl-1H-imidazole-2-carboxylic acid 1152018-00-2 C15H17N5O5
4-[(4-allyloxycarbonylamino-1-methyl-1H-pyrrole-2-carbonyl)-amino]-1-methyl-1H-imidazole-2-carboxylic acid
—— —— 1012046-04-6 C25H31N3O5S
—— —— 1125887-25-3 C13H16N4O
—— (R)-N-((1R,2R,4S)-bicyclo[2.2.1]hept-2-yl)-1-(n-pentyl)-5-phenyl-4,5-dihydro-(1H)-pyrazole-3-carboxamide 1134632-45-3 C22H31N3O
(R)-N-((1R,2R,4S)-bicyclo[2.2.1]hept-2-yl)-1-(n-pentyl)-5-phenyl-4,5-dihydro-(1H)-pyrazole-3-carboxamide
—— —— 1125886-88-5 C13H16N4O
—— (R)-6-[(1R,2S)-2-((2S,3S)-2-tert-butoxycarbonylamino-3-methylpentanoyloxy)-1-hydroxypropyl]-2-(dimethylaminomethyleneamino)-4-oxo-4,6,7,8-tetrahydro-3H-pteridine-5-carboxylic acid tert-butyl ester 1041007-10-6 C28H47N7O8
(R)-6-[(1R,2S)-2-((2S,3S)-2-tert-butoxycarbonylamino-3-methylpentanoyloxy)-1-hydroxypropyl]-2-(dimethylaminomethyleneamino)-4-oxo-4,6,7,8-tetrahydro-3H-pteridine-5-carboxylic acid tert-butyl ester
—— —— 1190388-49-8 C25H27N3O2